Patents
Sitemap › C07 - Organic chemistry › C07D - Heterocyclic compounds › C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
11/1999
11/02/1999US5977149 Dihydrotriazole compounds and their use for controlling fungal plant diseases
11/02/1999US5977140 N-[(4-Heteroaryl-1-Piperidinyl)Alkly] Phthalimides and related compounds and their therapeutic utility
11/02/1999US5977137 Sulfonamide inhibitors of aspartyl protease
11/02/1999US5977113 4-heteroaryl-1-piperazine alkylamines and their therapeutic utility
11/02/1999US5977075 N-aroylamino acid amides as endothelin inhibitors
11/02/1999US5977027 Pyrimidone isobutyric acid and herbicides containing the same
11/02/1999US5976812 Amphetamine linked to maleimide; for immunogens and conjugates; for production of antibodies and detection of drugs of abuse
11/02/1999US5976783 Crosslinking agent with enzyme cleavable portion for cyclization/deactivation of protein or enzyme; for analysis of specific enyzme in sample by determining cleavage of agent
10/1999
10/28/1999WO1999054321A1 Substituted diamines and their use as cell adhesion inhibitors
10/28/1999WO1999054320A1 Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
10/28/1999WO1999054314A1 Novel diphenyl-substituted 5-ring-heterocycles, method for producing them and their use as medicaments
10/28/1999WO1999054299A1 Pyrrolidines as inhibitors of neuraminidases
10/28/1999WO1999054298A1 Method for producing enantiomer-free n-methyl-n- [(1s)-1-phenyl- 2-((3s)- 3-hydroxypyrrolidine- 1-yl)ethyl]- 2,2-diphenyl acetamide
10/28/1999WO1999054284A1 Anthranilic acid derivatives as inhibitors of the cgmp-phosphodiesterase
10/28/1999WO1999053911A1 Antifungal agents
10/28/1999WO1999024460B1 Dipeptide nitriles
10/28/1999DE19818732A1 New aryl substituted cyclic ketoenol compounds useful for control of insects and as herbicides
10/28/1999DE19808261A1 Arylphenylsubstituierte cyclische Ketoenole Arylphenylsubstituierte cyclic ketoenols
10/28/1999CA2329422A1 Pyrrolidines as inhibitors of neuraminidases
10/28/1999CA2328720A1 Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
10/28/1999CA2328413A1 Anthranilic acid derivatives as inhibitors of the cgmp-phosphodiesterase
10/27/1999EP0952154A2 N-acyl and N-aroyl aralkyl amides
10/27/1999EP0951466A2 Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
10/27/1999CN1233256A Dipeptide benzamidine as a kininogenase inhibitor
10/27/1999CN1233237A Heteroaryl succinamides and their use as metalloproteinase inhibitors
10/26/1999USRE36359 Long chain carboxylic acid imide ester
10/26/1999US5973188 Anticoagulant; prevention cell, protein binding
10/26/1999US5973166 Subjecting n-maleimic acid in suitable reaction medium to aconditions sufficient to promote cyclodehydration using substituted amine or quaternaryammonium salt containing cation and anion as polarity modifier and an acid catalyst
10/26/1999US5973075 Methods for preparing rigid-rod macromonomers with reactive end groups
10/26/1999US5972982 Containing 5-to 9-membered heteroaryl mono- or bicyclic ring system having no more than 1 carbonyl carbon in the ring system; viricides, bactericides
10/26/1999US5972977 Ophthalmic pharmaceutical compositions comprising a nitrone compound and methods for treating ocular inflammation using such compositions
10/26/1999US5972719 Combinatorial hydroxy-amino acid amide libraries
10/21/1999WO1999053039A1 Treatment of parasitic diseases by inhibition of cysteine proteases of the papain superfamily
10/21/1999WO1999052876A1 Azacycloalkane derivatives, preparation and therapeutic application
10/21/1999WO1999052868A1 Substituted pyrrolidine hydroxamate metalloprotease inhibitors
10/21/1999WO1999052867A1 A process for the production of n-methyl pyrrolidone
10/21/1999WO1999052866A1 A process for the production of 2-pyrrolidone in a continous fashion, starting from gamma butyrolactone and ammonia
10/21/1999WO1999052528A1 Pharmaceutical preparations containing hydrosoluble ketoprofen salts and their application
10/21/1999WO1999043643A3 Metal-catalyzed arylations and vinylations of hydrazines, hydrazones, hydroxylamines and oximes
10/21/1999DE19827633A1 Production of N-methyl-N-(1-phenyl-2-(3-hydroxypyrrolidino)ethyl)-2,2-diphenylacetamide enantiomers, e.g. with antiinflammatory, analgesic and diuretic activity
10/21/1999DE19816880A1 New diaryl substituted heterocyclic compounds are AMPA receptor antagonists useful in treatment of neurodegenerative disorders and cerebral ischemia
10/21/1999DE19816479A1 Intermolecular preparation of enamines by catalytic reaction of alkynes with ammonia or primary or secondary amines
10/21/1999CA2328211A1 Substituted pyrrolidine hydroxamate metalloprotease inhibitors
10/21/1999CA2327282A1 Treatment of parasitic diseases by inhibition of cysteine proteases of the papain superfamily
10/21/1999CA2293605A1 Pharmaceutical preparations containing hydrosoluble ketoprofen salts and their application
10/21/1999CA2289497A1 A process for the production of n-methyl pyrrolidone
10/20/1999CN1232451A Substd. cyclic amine metalloprotease inhibitors
10/20/1999CN1232450A 2- and 2,5-substd. phenylketoenols
10/20/1999CN1232449A Process for preparing 2-phenyl-3-naphthylpropionic acid derivs.
10/20/1999CN1232399A Inhibitors of cysteine protease
10/20/1999CN1232388A Antimalarial and anti-babesiosis agent and pharmaceutical compositions contg. same
10/20/1999CN1232025A Pyrrolidine and piperidine derivatives
10/20/1999CN1045766C N-aminoalkylcarbonyloxyalkylpyrrole insecticidal, acaricidal and molluscicidal agents
10/19/1999US5969156 Crystalline [R- (R*,R*)]-2-(4-Dfluorophenyl)-β,δ-dihydroxy-5-(1-methylethyl)- 3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid hemi calcium salt (atorvastatin)
10/19/1999US5969138 Pyrrolidinone derivatives
10/19/1999US5969079 Heat resistant, high strength aerospace engineering thermoplastics
10/19/1999US5968963 PLA2 inhibitors and their use for inhibition of intestinal cholesterol absorption
10/19/1999US5968942 Inhibitors of hiv protease
10/16/1999CA2269049A1 N-acyl and n-aroyl aralkyl amides
10/14/1999WO1999051590A1 Substituted indolinones as kinase inhibitors
10/14/1999WO1999051573A2 Process for the preparation of a 2-oxopyrrolidine compound
10/14/1999WO1999033840B1 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha1-blocking action
10/13/1999EP0949242A1 Aromatic amine derivatives having nos inhibitory effect
10/13/1999EP0949238A1 Substituted propionyl derivatives
10/13/1999EP0948964A1 Novel n-substituted pyrrolidine derivatives and process for preparing the same
10/13/1999EP0936912A4 Inhibitors of cysteine protease
10/13/1999EP0783486B1 Novel prostaglandin synthase inhibitors
10/13/1999CN1231665A Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
10/13/1999CN1231662A Quinazoline derivatives and pharmaceutical compositions containing them
10/13/1999CN1231285A Process for preparing N-pyrrolidone acetate
10/13/1999CN1045595C Process for the preparation of the intermediates used in the synthesis of 3-aminopiperidine derivatives
10/12/1999US5965773 Process for the preparation of 2-aryl-5-(perfluoroalkyl) pyrrole compounds from N-(perfluoroalkylmethyl) arylimidoyl chloride compounds
10/12/1999US5965748 Succinimide derivative, process for production and use thereof
10/12/1999US5965747 Crystalline forms of antibiotic side chain intermediates
10/12/1999US5965746 Reacting an amino group-containing n-cyclic compound with maleic anhydride in acetic acid to obtain an n-cyclic maleamic acid, adding hexamethyldisilazane, cyclizing to form n-cyclic maleimide, use as a fluorescent dyes
10/12/1999US5965613 Fungicides for use in agriculture and horticulture; the compounds also have insecticidal and acaricidal activity
10/12/1999US5965556 Keto-acid amide derivatives, pharmaceutical compositions containing them and methods for inhibiting the activity of serine protease or thiol protease by administering the derivative to a mammal; alzheimer's disease
10/12/1999US5965546 1-[(2-pyrimidinyloxy)alkyl]4-(heteroaryl)piperazines and related compounds and their therapeutic utility
10/12/1999US5965539 Peptidomimetics; anti-cancer drugs
10/12/1999US5965121 Compounds and compositions for delivering active agents
10/07/1999WO1999050247A1 Compounds with activity on muscarinic receptors
10/07/1999WO1999050244A1 Nitroxide free radical dual indicator agents
10/07/1999WO1999050243A1 The use of derivatives of 2-oxopyrrole as crop protection agents and novel 2-oxopyrroles
10/07/1999WO1999050225A1 Aminocyclohexyl ether compounds and uses thereof
10/07/1999WO1999049856A2 Antagonists for treatment of cd11/cd18 adhesion receptor mediated disorders
10/07/1999DE3153481C2 New herbicides and intermediates
10/07/1999DE19815020A1 Neue substituierte Indolinone, ihre Herstellung und ihre Verwendung als Arzneimittel New substituted indolinones, their preparation and their use as medicaments
10/07/1999DE19812058C1 New 2-heterocyclyl-1,4-phenylenediamine derivatives
10/07/1999CA2325986A1 Antagonists for treatment of cd11/cd18 adhesion receptor mediated disorders
10/07/1999CA2325904A1 The use of derivatives of 2-oxopyrrole as crop protection agents and novel 2-oxopyrroles
10/06/1999EP0947505A2 Process for preparing optically active 4-hydroxy-2-pyrrolidone
10/06/1999EP0946570A1 Process for the preparation of an organozinc reagent
10/06/1999EP0946510A1 Novel compounds with analgesic effect
10/06/1999EP0946508A1 NITROGEN CONTAINING HETEROAROMATICS AS FACTOR Xa INHIBITORS
10/06/1999EP0946507A1 Substituted pyrrolyl compounds for the treatment of inflammation
10/06/1999EP0946501A1 Prevention of loss and restoration of bone mass by certain prostaglandin agonists
10/06/1999EP0946097A1 Composition and use
10/06/1999CN1230949A Stabilised monomer composition
10/06/1999CN1230539A Process for preparation of 2-aryl-5-(perfluoroalkyl) pyrrole compounds from N-(perfluoroalkyl-methyl) arylimidoyl chloride compounds
10/06/1999CN1230407A Method and compositions for treatment and prevention of tumors, tumor-related disorders and cachexia
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