Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
09/2000
09/12/2000US6118001 Anticancer agent; antiarthritic agent
09/12/2000US6117897 1/2 sulfate of a [(S) -1- [(S) -2- [(trans-4- aminocyclohexylmethyl) carbamoyl]pyrrolidine-1-carbonyl]- 2-isopropylthio-2-methylpropyl]carbamic acid propyl ester
09/09/2000CA2300412A1 Process for the preparation of 2-aryl-5-(perfluoro-alkyl) pyrrole compounds from n-[1-chloro-1-(perfluoroalkyl) methyl] arylimidoyl chloride compounds
09/08/2000WO2000052012A2 A method for synthesizing porphyrin compounds
09/08/2000WO2000051975A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors
09/08/2000CA2364878A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors
09/07/2000DE19909600A1 Catalytic preparation of cyclic and/or polymer compounds by educt metathesis is performed in the presence of one or more heterogeneous catalysts and ionic liquids
09/07/2000DE19908938A1 Übergangsmetallverbindung, Katalysatorsystem, Verfahren zu seiner Herstellung und seine Verwendung zur Polymerisation von Olefinen Transition metal compound catalyst system, to methods for its production and its use for the polymerization of olefins
09/06/2000EP1033371A1 Transition metal compound, catalyst system, process for the preparation thereof and its use for the polymerization of olefins
09/06/2000EP1032631A2 O-substituted n,n-diacylhydroxylamine bleach activators and compositions employing the same
09/06/2000EP1032560A1 Position-4 substituted 2-pyrrolidinone derivatives to reduce the level of extracellular glutamate
09/06/2000EP0824514B1 Dihalopropene compounds, insecticides containing them as active ingredients, and intermediates for their production
09/06/2000CN1265675A Benzyl compounds which inhibit leukocyte adhesion mediated by VLA-4
09/06/2000CN1265657A Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4
09/06/2000CN1265648A Conjugaes of dithiocarbamates with pharmacologically active agents and uses therefor
09/06/2000CN1265647A Acrylic metalloprotease inhibitor
09/06/2000CN1265645A Urokinase inhibitors
09/06/2000CN1265590A Substituted alkanohydroxamic acid and method of reducing TNF 'alpha' levels
09/05/2000US6114542 Ethers of polyalkyl or polyalkenyl N-hydroxyalkyl succinimides and fuel compositions containing the same
09/05/2000US6114541 Method for the preparation of α-Bromo-Lactam derivatives
09/05/2000US6114419 Fluorinated imides useful to impart repellency of low surface tension fluids to nonwoven fabrics, fibers, films and fabrics; melt extruding a filament of a dispersion of polymers and heterocyclic imide; molding materials
09/05/2000US6114393 Use of inhibitors of the sodium-hydrogen exchanger for the production of a pharmaceutical for the treatment of disorders which are caused by protozoa
09/05/2000US6114374 2-and 2,5-substituted phenylketoenols
09/05/2000US6114361 5-oxo-pyrrolidine-2-carboxylic acid hydroxamide derivatives
09/05/2000US6114335 Benzoylguanidine derivatives, process for their preparation their use in the preparation of medicines
08/2000
08/31/2000WO2000050470A2 Catalysts containing n-pyrrolyl substituted nitrogen donors
08/31/2000WO2000050386A1 Compounds and compositions for delivering active agents
08/31/2000WO2000050380A1 Monoamine reuptake inhibitors for treatment of cns disorders
08/31/2000WO2000040558A8 Aspartic protease inhibitors
08/31/2000WO2000012507A3 Pyrrolobenzodiazepines
08/31/2000CA2364849A1 Compounds and compositions for delivering active agents
08/31/2000CA2363628A1 Catalysts containing n-pyrrolyl substituted nitrogen donors
08/30/2000EP1031563A1 Sulfonyl derivatives
08/30/2000EP1030840A1 Cyclic amine derivatives and their use as drugs
08/30/2000CN1265097A Pyrrolidine carboxylic acid derivatives as endothelin antagonists
08/30/2000CN1265096A Hydrazine derivatives
08/29/2000US6110959 Carboxylic acid derivatives having fused rings
08/29/2000US6110958 Pyrrole compounds having parasiticidal properties
08/29/2000US6110947 An analgesic agent for treating stroke, abdominal pain; as antiinflammatory, diuretic, anesthetic or neuroprotective agents
08/29/2000US6110945 An antiinflammatory agent inhibiting the binding of integrins to their ligands; in the prophylaxis for treating immune or inflammatory disorders
08/29/2000US6110938 1-(arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-4-(heteroaryl)piperidines and related compounds useful as antipsychotics and analgesics
08/29/2000US6110933 Amino acid derivatives and their use as phospholipase A2 inhibitor
08/29/2000US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
08/29/2000US6110913 N-substituted azaheterocyclic carboxylic acids and esters thereof
08/29/2000US6110872 2,4,5-trisubstituted phenylketo-enols for use as pesticides and herbicides
08/29/2000US6110619 Electrochemical cells with cationic polymers and electroactive sulfur compounds
08/29/2000CA2012628C New fluoro-4 benzoic derivatives, process for their preparation and pharmaceutical compositions containing them
08/24/2000WO2000049007A1 Acetamido acetonitrile derivatives as inhibitors of cathepsin l and/or cathepsin s
08/24/2000WO2000048974A1 Stabilised compositions of o- and n-vinyl compounds and the use of ammonium salts as stabilisers
08/24/2000WO2000048584A2 Aroyl aminoacyl pyrroles for use in the treatment of neuropathic pain
08/24/2000WO1996012697A9 Calcium receptor-active compounds
08/24/2000CA2361390A1 Aroyl aminoacyl pyrroles for use in the treatment of neuropathic pain
08/23/2000EP1029872A1 Piperazine-cyclodextrin complexes
08/23/2000EP1029297A2 Method of virtual retrieval of analogs of lead compounds
08/23/2000EP1028961A1 Pleuromutilin derivatives as antimicrobials
08/23/2000EP1028942A2 Dipeptide nitriles
08/23/2000EP1028716A1 Method for treating and preventing heart failure and ventricular dilatation
08/23/2000EP0805795B1 Novel aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides
08/23/2000EP0763005B1 TETRAHYDROINDENO[1,2-d][1,3,2]OXAZABOROLES AND THEIR USE AS ENANTIOSELECTIVE CATALYSTS
08/23/2000EP0637297B1 Compounds having selectivity for retinoid x receptors
08/23/2000CN1264385A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and compositions containing same
08/23/2000CN1264300A Arylsubstituted piperazines useful in the threatement of bening prostatic hyperlasia
08/23/2000CN1055686C Substituted benzisoxazole and benzisothaazole herbicidal agents
08/22/2000US6107492 By optical resolution of a racemic mixture of alpha-ethyl-2-oxo-1-pyrrolidine acetamide by chromatography using silica gel supporting amylose tris(3,5-dimethylphenylcarbamate) as a packing material
08/22/2000US6107330 Inhibitor for narcotic analgesic dependence/resistance acquisition
08/22/2000US6107329 Hypotensive agents; cardiovascular disorders
08/22/2000US6107322 Pesticidal 1-polyarylimidazoles
08/22/2000US6107315 Nervous system disorders
08/22/2000US6107024 Using 1,2-dioxetane derivative substrate in enzyme-linked assay where enzyme is linked to antigen, antibody, hapten or nucleic acid; forms aryloxide intermediate when triggered, then releases energy to form light and two carbonyl compounds
08/22/2000CA2176973C Phenyl heterocycles as cyclooxygenase-2 inhibitors
08/17/2000WO2000047558A1 Amide compounds and medicinal use thereof
08/17/2000WO2000047547A2 Cycloalkyl amine compounds and uses thereof
08/17/2000WO2000047539A1 Fluorinating agent, process for producing the same, and use thereof
08/17/2000WO2000047207A1 LACTAM INHIBITORS OF FXa AND METHOD
08/17/2000WO2000047206A1 Use of pyrrolidine derivatives for the manufacture of a pharmaceutical composition for the treatment or prophylaxis of obesity or appetite regulation
08/17/2000WO2000012076A9 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
08/17/2000WO2000009109A3 Pipecolic acid derivatives for vision and memory disorders
08/17/2000DE19906316A1 Polymerizable vinyl compositions are stabilized by the addition of optionally substituted ammonium carbonate salts
08/17/2000CA2360305A1 Lactam inhibitors of fxa and method
08/16/2000EP1027339A1 Method and reagents for n-alkylating ureides
08/16/2000EP1027332A1 Novel lactam metalloprotease inhibitors
08/16/2000EP1027324A1 Optically active intermediates for the preparation of optically active substituted oximes, hydrazones and olefins useful as neurokinin antagonists
08/16/2000EP0738259B1 Phenyl acetic acid derivatives, process and intermediate products for their production and agents containing them
08/16/2000CN1263527A Cis-disubstituted aminocycloalykyl-pyrrolidine derivatives
08/16/2000CN1263524A Aromatic maleimides and their use as photoinitiators
08/16/2000CN1263523A A process for production of N-methyl pyrrolidone
08/16/2000CN1263464A Pharmaceutical preparations containing hydrosoluble ketoprofen salts and their application
08/16/2000CN1263089A Preparation of thiol-carbamate and sulfocyanic ester compound
08/16/2000CN1055464C Alkoxymethylationof pyrroles
08/15/2000US6103937 Producing unsaturated nitrogen containing compounds such as enamides, enamines and aryl amineslamides using as catalyst nickel and an organophosphine or carbene ligand
08/15/2000US6103910 D-proline derivatives
08/15/2000US6103899 Bicyclic aminoimidazoles
08/15/2000CA2192394C Thermosetting resin forming compositions, resins therefrom and methods for their preparation
08/10/2000WO2000046221A1 Sulfamato hydroxamic acid metalloprotease inhibitor
08/10/2000WO2000046194A1 Cyclic amine derivatives and uses thereof
08/10/2000WO2000046193A2 Ether derivatives having neuronal activity
08/10/2000WO2000046184A1 N2-phenylamidine derivatives
08/10/2000WO2000046183A1 N-substituted amino acids, antioxidant pharmaceutical compositions containing same and methods using same
08/10/2000WO1999063936A9 Novel therapeutic agents that modulate endothelin receptors
08/10/2000DE19905254A1 New ether compounds, useful for treating neurological diseases e.g. Parkinson's disease, amyotrophic lateral sclerosis and Alzheimer's disease