Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
08/1999
08/05/1999WO1999038844A1 Method for preparing an n-[(aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound
08/05/1999WO1999038838A1 Method for producing optically active amino alcohols
08/05/1999WO1999038508A1 Compounds, compositions and methods for treating or preventing pneumovirus infection and associated diseases
08/05/1999WO1995031429A8 Photocleavable agents and conjugates for the detection and isolation of biomolecules
08/05/1999DE19803892A1 Verfahren zur Herstellung von optisch aktiven Aminoalkoholen A process for preparing optically active amino alcohols
08/05/1999CA2319465A1 Compounds, compositions and methods for treating or preventing pneumovirus infection and associated diseases
08/05/1999CA2318601A1 Method for preparing an n-[(aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound
08/04/1999EP0933379A1 Novel peptide derivatives having thiazolyl-alanine residue
08/04/1999EP0933354A1 Calcium receptor-active compounds
08/04/1999EP0932658A2 Asymmetrical imide bleach activators and compositions employing the same
08/04/1999EP0932601A1 Process for preparing pharmaceutical compounds
08/04/1999EP0932598A1 ASPARTATE ESTER INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME
08/04/1999CN1225083A Calcium receptor-active compounds
08/04/1999CN1224714A N-(4-carbamimido-phenyl)-phenylglycinamid derivatives
08/03/1999US5932745 Process for converting propargylic amine-N-oxides to enaminones
08/03/1999US5932674 Crosslinked polymers
08/03/1999US5932598 Prodrugs of benzenesulfonamide-containing COX-2 inhibitors
08/03/1999US5932586 Prostaglandin synthase inhibitors
08/03/1999US5932575 Cardiac diseases improving agents
08/03/1999US5932559 Treatment of hyperandrogenic conditions
08/03/1999US5932550 Dipeptide compound or pharmaceutically acceptable salt thereof and medical use thereof
08/03/1999US5932296 Process for producing a surface coated with amino groups
07/1999
07/29/1999WO1999037618A1 Phenylalanine derivatives useful as pharmaceutical agents
07/29/1999WO1999037616A1 Piperidine and pyrrolidine derivatives comprising a nitric oxide donor for treating stress
07/29/1999WO1999037607A1 Potassium channel inhibitors
07/29/1999WO1999037307A1 Pharmaceutically active compounds and methods of use thereof
07/29/1999WO1999037306A1 Pharmaceutically active compounds and methods of use thereof
07/29/1999WO1999024537A3 O-substituted n,n-diacylhydroxylamine bleach activators and compositions employing the same
07/29/1999WO1999023587A3 Method of virtual retrieval of analogs of lead compounds
07/29/1999CA2318580A1 Pharmaceutically active compounds and methods of use thereof
07/29/1999CA2317457A1 Potassium channel inhibitors
07/28/1999EP0931064A1 Stabilised monomer composition
07/28/1999EP0931062A1 Conjugates and specific immunoassays for the methadone metabolite 2-ethylidine-1,5-dimethyl-3,3-diphenylpyrrolidine
07/28/1999EP0931060A1 Substituted n- (aminoiminomethyl or aminomethyl)phenyl]propyl amides
07/28/1999EP0643693B1 Reversal of multi-drug resistance by triphenyl-piperidine derivatives
07/28/1999CN1224004A Process for preparing enalaprol maleate
07/28/1999CN1044365C Alpha, omega-diarylalkane derivs., their preparation and their use in treatment and prevention of circulatory diseases and psychosis
07/27/1999US5929251 Reacting n-hydroxy-succinimide with carboxylic acid and a halophosphoric acid ester in presence of a base in a diluent to form a reaction mixture containing carboxylic acid succinimidyl ester, then reacting with a acylating agent
07/27/1999US5929232 Stereoselective ring opening reactions
07/27/1999US5929211 Carbohydrate-directed cross-linking reagents
07/27/1999US5929117 Immunotherapeutic agents
07/27/1999US5929114 Administering antiviral compound which extrudes zinc from nucleocapsid protein of human immunodeficiency virus
07/27/1999US5929077 Thioproline-containing inhibitors of farnesyl protein transferase
07/27/1999US5929067 N-acylating amine derivative of caprolactam compound with a carboxylic acid or derivatives to form amide derivative of caprolactam compound
07/27/1999CA2164804C Nk-1 receptor antagonists for the treatment of neuronal injury and stroke
07/22/1999WO1999036403A1 Novel dopamine re-uptake inhibitors and methods of synthesizing and using the same
07/22/1999WO1999036398A1 Aminosulphonylbenzamide derivatives as modulators of the activity of neuronal calcium channels
07/22/1999WO1999036393A1 INHIBITORS OF α4 MEDIATED CELL ADHESION
07/22/1999WO1999036068A1 Potassium channel activators
07/22/1999WO1999029309A3 2,2'-bi-1h-pyrrole derivatives useful in the treatment of leukemia brought on by htlv-i
07/22/1999CA2317536A1 Aminosulphonylbenzamide derivatives as modulators of the activity of neuronal calcium channels
07/22/1999CA2316853A1 Potassium channel activators
07/21/1999EP0930293A1 Process for the preparation of N-alkenyl carboxylic acid amide
07/21/1999EP0930075A1 Methods for preventing, inhibiting or treating graft rejection reactions in graft-versus-host disease (gvhd) and organ transplantation
07/21/1999EP0929538A1 O?2 -arylated or o?2 -glycosylated 1-substituted diazen-1-ium-1,2-diolates and o?2 -substituted 1- (2-carboxylato)pyrrolidin-1-yl]diazen-1-ium-1,2-diolates
07/21/1999EP0929530A1 Quinazoline derivatives and pharmaceutical compositions containing them
07/21/1999EP0929217A1 Sordarin derivatives
07/21/1999EP0759025B1 Amide derivatives and their therapeutic use
07/21/1999CN1223650A Piperidines and pyrrolidines
07/21/1999CN1223256A Biologically active ureido derivatives useful as antimetastatic agents
07/21/1999CN1044238C Method for preparing benzylidene derivatives
07/20/1999US5925787 Production of keto acids
07/20/1999US5925773 Chemical condensation of olefin with oxazole derivative to form pyrrole
07/20/1999US5925772 Cysteine protease inhibitors containing heterocyclic leaving groups
07/20/1999US5925762 Reacting primary phenyl carbamate or thiocarbamate with ammonia, a primary or secondary amine in dimethylsulfoxide
07/20/1999US5925667 Pyrrolidine derivative, anti-ulcer drug, and antibacterial drug
07/20/1999US5925616 Synergistic mixtures
07/20/1999US5925611 Cleaning process and composition
07/20/1999US5925597 Pre-emergence and post-emergence herbicides
07/20/1999CA1340665C Bifunctional coupling agents and radionuclide labeled compositions prepared therefrom
07/15/1999WO1999035129A1 Succinimide derivatives which inhibit retinoic acid metabolism
07/15/1999WO1999026584A3 Inhibitors of gap junction communication
07/14/1999EP0928787A1 Process for the preparation of 3-amino-pyrrolidine derivatives
07/14/1999EP0777649B1 N- 2-(pyrrolidinyl-1)-1-phenylethyl]acetamides as kappa receptor agonists
07/14/1999CN1222908A Polymerizable urea/ureido functional monomers
07/14/1999CN1222905A New synthetic catechol derivatives, method for production and use thereof
07/14/1999CN1222521A 1,3,8-triaza-spiro [4,5] decan-4-on derivatives
07/14/1999CN1044117C Compound for inhibition of HIV protease, its preparing method and its drug use
07/13/1999US5922892 Process to produce midazolam
07/13/1999US5922884 Pesticidal 1-polyarylpyrazoles
07/13/1999US5922881 Heterocyclic imino derivatives
07/13/1999US5922858 Misaminoacylated transfer ribonucleic acid with photocleavable marker; for incorporation of non-radioactive labels into nascent proteins by cellular or cell-free translation systems
07/13/1999US5922770 Novel compounds that stimulate the release of growth hormone from the pituitary
07/13/1999US5922763 Biphenyl derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
07/13/1999US5922717 Piperazine derivatives, medicaments comprising these compounds, their use and processes for their preparation
07/13/1999US5922589 Preparation of lactams from aliphatic α,ω-Dinitiles
07/13/1999CA2129144C Reversal of multi-drug resistance by triphenyl-azacycloalkane derivatives
07/12/1999CA2258166A1 Process for the preparation of 3-amino-pyrrolidine derivatives
07/08/1999WO1999033841A2 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha-1-blocking action
07/08/1999WO1999033840A2 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha1-blocking action
07/08/1999WO1999033797A1 NEW CRYSTALLINE POLYMORPHIC FORM OF 1-METHYL-5-p-TOLUOYLPYRROLE-2-ACETAMIDOACETIC ACID GUAIACYL ESTER (MED 15)
07/08/1999WO1999033796A1 5-arylpyrrole derivatives
07/08/1999WO1999033795A1 Prodrugs of aspartyl protease inhibitors
07/08/1999WO1999033789A1 SUBSTITUTED β-ALANINES
07/08/1999WO1999033460A1 Acyl guanidine sodium/proton exchange inhibitors and method
07/08/1999WO1999025686B1 Cyclic amine derivatives and their use as drugs
07/08/1999CA2316953A1 5-arylpyrrole derivatives
07/08/1999CA2316352A1 Acyl guanidine sodium/proton exchange inhibitors and method
07/08/1999CA2316235A1 Substituted .beta.-alanines
07/08/1999CA2282815A1 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha-1-blocking action