Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
06/2000
06/21/2000EP1009770A1 Peptides containing an arginine mimetic for the treatment of bone metabolic disorders, their production, and drugs containing these compounds
06/21/2000EP1009737A2 Sulfonylamino substituted hydroxamic acid derivatives as metalloprotease inhibitors
06/21/2000EP1009405A1 Pyrrolidine and piperidine modulators of chemokine receptor activity
06/21/2000DE19952348A1 New bisphosphinyl-ferrocene ligand components for new metal complexes useful as catalysts in asymmetric hydrogenations
06/21/2000DE19858360A1 Verfahren zum Herstellen von 2,4-Dimethyl-pyrrol A method for the preparation of 2,4-dimethyl-pyrrole
06/21/2000DE19858352A1 Verfahren zum Herstellen von 2,4-Dimethyl-3,5-bis-alkoxycarbonyl-pyrrol A method for the preparation of 2,4-dimethyl-3,5-bis-alkoxycarbonyl-pyrrole
06/21/2000DE19858029A1 New substituted (hetero)aryl-alkanes, used as thrombin inhibitors, serine protease inhibitors, antithrombotic agents and intermediates
06/21/2000CN1257068A Process for preparation of condensed sulfamide
06/21/2000CN1053666C Benzoheterocylic compounds and process for preparing medicated salt thereof
06/21/2000CN1053657C Didepside phthaleins based internal parasite compositions, novel didepside phthaleins and preparation process thereof
06/20/2000US6077955 Preparation of lactams from aliphatic αω-dinitriles
06/20/2000US6077928 Bis(dialkylmaleimide) derivative and polyetherimide for optical communications formed therefrom
06/20/2000US6077863 2-aryl-4-halo-5-(trifluoromethyl)pyrrole-3-carbonitriles for the protection of wood, wood products and wooden structures from insect attack
06/20/2000US6077855 Hemoregulatory compounds
06/20/2000US6077813 Substituted aromatic thiocarboxylic acid amides and their use as herbicides
06/20/2000CA1341029C Peptidase inhibitors
06/17/2000CA2292246A1 New hydrazide derivatives, the procedure for preparing them and the pharmaceutical formulations that contain them
06/15/2000WO2000034268A1 Thiourea inhibitors of herpes viruses
06/15/2000WO2000034241A1 N-substituted 2-cyanopyrrolidines
06/15/2000WO2000034237A2 Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses
06/15/2000WO2000033788A2 Substituted nitrogen heterocyclic compounds and therapeutic uses thereof
06/15/2000WO2000010974A3 Process for the preparation of a maleimide compound, maleimide compound, radiation-curable compositions comprising said compound and coated products
06/15/2000WO2000009107A3 Sulfonamides of n-containing heterocyclic thioesters for vision and memory disorders
06/15/2000CA2355296A1 Substituted nitrogen heterocyclic compounds and therapeutic uses thereof
06/15/2000CA2350996A1 Thiourea inhibitors of herpes viruses
06/15/2000CA2350899A1 Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses
06/14/2000EP1008346A1 NF-$g(k)B INHIBITORS CONTAINING AS THE ACTIVE INGREDIENT PHENYLMETHYL BENZOQUINONE
06/14/2000EP1007729A1 COMPLEX FORMATION BETWEEN dsDNA AND OLIGOMER OF HETEROCYCLES
06/14/2000EP1007056A1 Method for the treatment of cystic fibrosis
06/14/2000EP1007033A1 Lymphocyte function antigen-1 antagonists
06/14/2000EP1007032A1 4-cyano-4-deformylsordaricin derivatives
06/14/2000EP1007025A1 Use of hydroxyguanidines
06/14/2000EP0777645B1 Oxime ethers and their use as pesticides
06/14/2000CN1256266A New method for preparing (S)-4-amino-hepta-5,6-dienoic acid and intermediate thereof
06/14/2000CN1053437C Synthetic method for lisinopril
06/13/2000US6075153 Catalytic hydrogenation of maleic anhydride, succinic anhydride or their acids in the presence of catalysts consisting of copper oxide, aluminum oxide and a graphite binder; for use in manufacturing n-methylpyrrolidone
06/13/2000US6075148 Carbamates and crop protection agents containing them
06/13/2000US6075126 Phenyldiboronic acid reagents and complexes
06/13/2000US6075052 Skin external preparation
06/13/2000US6075030 Fungicidal mixture
06/13/2000US6075026 Certain substituted 1-aryl-3-piperazin-1'-yl propanones
06/13/2000CA1341024C Benzo-fused cycloalkane and oxa- and thia-, cycloalkane trans-1, 2-diamine derivatives
06/13/2000CA1341023C Peptide derivatives
06/08/2000WO2000032649A1 Method of producing derivatized polymers
06/08/2000WO2000032588A2 Carboxylic acids and carboxylic acid isosteres of n-heterocyclic compounds
06/08/2000WO2000032582A1 Benzamide derivatives and their use as apob-100 secretion inhibitors
06/08/2000WO2000032575A1 β-ALANINE DERIVATIVES AS α4 INTEGRIN INHIBITORS
06/08/2000WO2000032188A2 Use of amtolmetin guacyl as an antiinflammatory drug
06/08/2000WO2000017228A3 Stereoselective process for enalapril
06/08/2000WO2000009103A9 N-linked sulfonamides of n-heterocyclic carboxylic acids or isosteres for vision and memory disorders
06/08/2000CA2634658A1 Use of amtolmetin guacyl for the production of anti-inflammatory drugs for intestinal inflammations
06/08/2000CA2353394A1 Benzamide derivatives and their use as apob-100 secretion inhibitors
06/08/2000CA2347701A1 .beta.-alanine derivatives as .alpha.4 integrin inhibitors
06/07/2000EP1005446A1 N-aroylphenylalanine derivatives
06/07/2000EP1005356A1 Novel antibacterial agents
06/06/2000US6071970 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
06/06/2000US6071950 N-substituted pyrrolidine derivatives and process for preparing the same
06/06/2000US6071948 Treatment of diseases caused by excessive blood vessel growth
06/06/2000US6071915 Arylsubstituted piperazines useful in the treatment of benign prostatic hyperplasia
06/06/2000US6071906 Inhibits or modulates the inducible isoform of nitric oxide synthase over the the constitutive isoforms; antiarthritic, -diabetic, ischemic, thrombosis agents; cardiovascular disorders; toxic shock syndrome; autoimmune diseases
06/06/2000US6071901 Treating pain, hyperalgesia and/or inflammatory conditions in which c-fibers play a pathophysiological role; inhibition of neurogenic inflammation involving the release of neuro-peptide from peripheral and central endings of sensory nerves
06/06/2000US6071895 Polar-substituted hydrocarbons
06/06/2000US6071510 Modified amino acids and compositions comprising the same for delivering active agents
06/02/2000WO2000031032A1 Pyrrolidine derivatives-ccr-3 receptor antagonists
06/02/2000WO2000030638A1 Drugs and reagents containing n-acyloxylated cycloalkyl compounds as the active ingredient
06/02/2000WO2000030624A2 Use of benzoylguanidines for the treatment of non-insulin-dependent diabetes mellitus
06/02/2000WO2000030445A1 Fungicides containing pyrrolidones as their active agents
06/02/2000WO2000009105A3 Small molecule carbamates or ureas for vision and memory disorders
06/02/2000CA2352196A1 Fungicides containing pyrrolidones as their active agents
06/02/2000CA2352154A1 Use of benzoylguanidines for the treatment of non-insulin-dependent diabetes mellitus
06/02/2000CA2350903A1 Pyrrolidine derivatives-ccr-3 receptor antagonists
05/2000
05/31/2000EP1004578A2 5-oxo-pyrrolidine-2-carboxylic acid hydroxamide derivatives
05/31/2000EP1004577A1 Process for preparing N-alkyl-2-pyrrolidones
05/31/2000EP1003758A2 Solution phase synthesis of oligonucleotides
05/31/2000EP1003740A2 Pyrrolidine-3-carboxylic acid derivatives and their use as endothelin antagoists
05/31/2000EP1003730A1 2-benzoyl-cyclohexane-1,3-diones
05/31/2000EP1003541A1 Inhibitors of hiv reverse transcriptase
05/31/2000EP1003540A1 $g(b)2-ADRENERGIC RECEPTOR AGONISTS
05/31/2000EP1003511A1 ALPHA 1aADRENERGIC RECEPTOR ANTAGONISTS
05/31/2000EP1003495A1 Pharmaceutical compounds
05/31/2000DE19955794A1 Pyrrolidin-Derivate-CCR-3-Rezeptor-Antagonisten Pyrrolidine derivatives-CCR-3 receptor antagonists
05/31/2000CN1255162A Protease inhibitors
05/31/2000CN1254596A Process for preparing composition to kill internal parasites
05/31/2000CN1052976C Substituted benzenesulfonylureas and -thioureas, preparation process and possible uses of pharmaceutical preparation therefor
05/30/2000US6069247 Reacting an acetylenecarboxy amide and an aryl or heterocyclyl halide or a group enhancing the electrophilicity of the atom to which it is attached for displacement; using a palladium compound catalyst, a base and an acid
05/25/2000WO2000029411A1 An improved process for the preparation of 7-azaindolyl-3-carboxylic acid
05/25/2000WO2000029376A1 Heteroarylthio compounds and cancer remedies containing the same
05/25/2000WO2000029375A1 Bisaryl compounds and cancer remedies containing the same
05/25/2000WO2000028983A1 Novel 4-dedimethy laminotetra cycline derivatives
05/25/2000WO2000028981A2 Methods for treating, preventing, and reducing the risk of the onset of alzheimer's disease using an hmg coa reductase inhibitor
05/25/2000WO2000018732A3 Disubstituted pyrrolidinones, medicaments containing these compounds, their use and the production thereof
05/25/2000WO2000018361A3 Method of treating hair loss using sulfonamides
05/25/2000CA2350420A1 Methods for treating, preventing, and reducing the risk of the onset of alzheimer's disease using an hmg coa reductase inhibitor
05/24/2000EP1001975A1 Benzyl compounds which inhibit leukocyte adhesion mediated by vla-4
05/24/2000EP1001932A1 Conjugates of dithiocarbamates with pharmacologically active agents and uses therefor
05/24/2000EP1001930A2 N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases
05/24/2000EP1001927A2 Novel polyamine analogues as therapeutic and diagnostic agents
05/24/2000EP1001766A1 Compounds and methods
05/24/2000EP0797386B1 Fungicidal mixture
05/24/2000CN1254337A N-hydroxy 4-sulfonyl butyramide compounds