Patents
Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868)
05/2012
05/10/2012US20120115840 Hemifumarate salt of 1-[4-[1-(4-cyclohexyl-3-trifluoromethyl-benzyloxyimino)-ethyl]-2-ethyl-benzyl]-azetidine-3-carboxylic acid
05/10/2012US20120115819 Pentacycline Compounds
05/09/2012EP2448919A2 Solubility and stability enchancing pharmaceutical formulation
05/09/2012CN102442934A Synthetic method of 6-oxo-2-azaspiro[3,3]heptane-2-t-butyl carboxylate
05/08/2012US8173634 Polymorphic form of 1-(4-{1-[(E)-4-cyclohexyl-3-trifluoromethyl-benzyloxyimino]-ethyl}-2-ethyl-benzyl)-azetidine-3-carboxylic
05/08/2012US8173631 Cyclic amine compounds
05/03/2012CA2814752A1 Diazeniumdiolate heterocyclic derivatives
05/02/2012CN102432514A Method for synthesizing 1-tert-butoxycarbonyl-3-fluoroazetidine
05/01/2012CA2698384C 3-pyridyl enantiomers and their use as analgesics
05/01/2012CA2623332C Carboxamide derivatives as muscarinic receptor antagonists
04/2012
04/26/2012WO2012054716A1 Piperidin-4-yl-azetidine diamides as monoacylglycerol lipase inhibitors
04/26/2012US20120101080 Composition for treatment of tuberculosis
04/24/2012US8163727 Biphenyloxyacetic acid derivatives for the treatment of respiratory disease
04/24/2012CA2524054C Immunosuppressant compounds and compositions
04/19/2012US20120094973 Catechol-based derivatives for treating or preventing diabetics
04/18/2012EP2441758A1 Synthesis of ttx intermediates
04/18/2012EP2440523A1 High penetration compositions or prodrugs of antimicrobials and antimicrobial-related compounds
04/18/2012EP2440521A1 Novel cyclopentane derivatives
04/17/2012US8158820 Compounds
04/12/2012US20120088749 S1P Receptor Modulating Compounds and Use Thereof
04/12/2012US20120088746 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same
04/05/2012WO2012020131A3 Aminoindane derivatives, pharmaceutical compositions containing them, and their use in therapy
04/05/2012US20120083601 Process for the synthesis of azetidinones
04/03/2012US8148422 Sulfonamides as TRPM8 modulators
04/03/2012CA2624481C Anti-hypercholesterolemic compounds
03/2012
03/21/2012CN102382026A Environmentally-friendly synthesis process of Aztreonam main ring (3S-trans)-3-amino-4-methyl-2-oxo-1-azetidinyl sulfonic acid
03/15/2012US20120064060 Compound having s1p receptor binding potency and use thereof
03/14/2012EP2427425A2 Tetracycline compounds
03/14/2012EP1169468B1 Stereoselective microbial reduction for the preparation of 1-(4-fluorophenyl)-3(r)-¬3(s)-hydroxy-3-(4-fluorophenyl)propyl) -4(s)-(4-hydroxyphenyl)-2-azetidinone
03/13/2012US8134014 Preparation of uretdione polyisocyanates
03/08/2012WO2012030907A1 Di-azetidinyl diamide as monoacylglycerol lipase inhibitors
03/08/2012CA2809991A1 Di-azetidinyl diamide as monoacylglycerol lipase inhibitors
03/01/2012WO2012025450A1 Phenylamidines having a high fungicidal activity and use thereof
03/01/2012US20120052040 Polymer compositions and methods for their use
02/2012
02/29/2012EP2421856A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
02/29/2012EP2421847A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
02/29/2012EP2421825A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
02/29/2012EP2421824A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
02/29/2012EP2421823A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
02/29/2012EP1667966B1 N-alkylated diaminopropane derivatives as modulators of chemokine receptor activity
02/23/2012US20120045390 Composition and Methods for the Diagnosis and Treatment of Tumor
02/22/2012EP2419419A1 4-azetidinyl-1-phenyl-cyclohexane antagonists of ccr2
02/22/2012EP2419404A1 Anti-viral compounds
02/22/2012EP0986384B1 Inhibitors of protein isoprenyl transferases
02/21/2012US8119625 Neurogenesis inducer or neuropathy therapeutic agent comprising alkyl ether derivative or salt thereof
02/21/2012CA2444031C 3,4-di-substituted cyclobutene-1,2-diones as cxc-chemokine receptor ligands
02/21/2012CA2400141C Pharmaceutical compositions containing azetidine derivatives, novel azetidine derivatives and preparation thereof
02/16/2012WO2012020130A1 Phenalkylamine derivatives, pharmaceutical compositions containing them, and their use in therapy
02/16/2012US20120040960 4-azetidinyl-1-phenyl-cyclohexane antagonists of ccr2
02/16/2012US20120040948 Aminoindane derivatives, pharmaceutical compositions containing them, and their use in therapy
02/16/2012US20120040947 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy
02/16/2012CA2806644A1 Aminoindane derivatives, pharmaceutical compositions containing them, and their use in therapy
02/16/2012CA2806643A1 Phenalkylamine derivatives, pharmaceutical compositions containing them, and their use in therapy
02/15/2012EP2417101A1 Indane derivatives
02/14/2012CA2463154C Heterocyclic compounds and methods of use
02/08/2012EP2414326A1 Intermediates in the preparation of 1,4-diphenyl azetidinone
02/08/2012EP2413701A1 Sulfonyl-azetidin-3-yl-methylamine amide analogs as glyt1 inhibitors, methods for making same, and use of same in treating psychiatric disorders
02/07/2012US8110678 Antibiotic-bound poly(caprolactone) polymer
02/02/2012US20120029185 Novel intermediates in the preparation of 1,4-diphenyl azetidinone
02/02/2012US20120028953 Azetidine Derivatives
02/02/2012US20120028937 Cyclic amine-1-carboxylic acid ester derivative and pharmaceutical composition containing the same
02/02/2012US20120028316 Enzymatic process for the preparation of (s)-5-(4-fluoro-phenyl)-5-hydroxy- 1morpholin-4-yl-pentan-1-one, an intermediate of ezetimibe and further conversion to ezetimibe
02/02/2012US20120028249 Anthraquinone based near ir emitting compounds and uses thereof
02/01/2012CN102336696A Intermediate for synthesizing 4-AA and preparation method and application thereof
01/2012
01/31/2012US8106191 Compounds based on N- acyl-pipecolyl and N-acyl-prolyl ligand moieties for multimerizing chimeric proteins containing immunophilin-derived domains
01/31/2012CA2550373C Anti-hypercholesterolemic compounds
01/26/2012US20120022263 3-aminoxalyl-aminobenzamide derivatives and insecticidal and miticidal agents containing same as active ingredient
01/26/2012US20120022248 B-lactam compounds
01/25/2012CN102329259A Preparation method for (1-benzydryl-3-azetidinol) cyanoacetate
01/24/2012CA2509159C Isophthalic acid derivatives
01/19/2012WO2012008435A1 Biaryl amide derivative or pharmaceutically acceptable salt thereof
01/18/2012CN102325750A Sulfonamides as trpm8 modulators
01/12/2012WO2012004382A1 New method for preparing ezetimibe
01/12/2012US20120010189 (3-(4-(aminomethyl)phenoxy or phenylthio)azetidin-1-yl)(5-phenyl-1,3,4-oxadiazol-2-yl)methanone compounds
01/05/2012WO2012003497A1 Napht- 2 -ylacetic acid derivatives to treat aids
01/05/2012WO2012003436A1 Methods for treating post traumatic stress disorder
01/05/2012CA2802308A1 Napht-2-ylacetic acid derivatives to treat aids
01/04/2012EP2402329A1 Analgetic phenylsulphonamides
01/04/2012CN102307852A Cyclic amine compounds
01/04/2012CN102304075A Inhibitors of viral replication
12/2011
12/29/2011WO2011120040A3 Thrombin inhibiting compositions
12/27/2011US8084607 Apoptosis promoters
12/22/2011WO2011158052A1 Nanostructured ezetimibe compositions, process for the preparation thereof and pharmaceutical compositions containing them
12/22/2011US20110312903 Fluorination of organic compounds
12/22/2011US20110311593 N-hydroxylated amidine-, guanidine- and/or aminohydrazone-type prodrugs for application on the skin
12/22/2011US20110311466 Novel 4-(azacycloalkyl)benzene-1,3-diol compounds as tyrosinase inhibitors, process for the preparation thereof and use thereof in human medicine and in cosmetics
12/21/2011EP2396300A1 New substituted tetrahydronapthalenes, method for the production thereof, and use thereof as drugs
12/21/2011EP2395992A2 Chemically programmed vaccination
12/21/2011EP1638551B1 Immunosuppressant compounds and compositions
12/21/2011CN102285907A 氨曲南单环母核的制备方法 Southern single aztreonam preparation ring nucleus
12/21/2011CN102285906A Process for preparation of ezetimibe and derivatives thereof
12/20/2011US8080542 S1P receptor modulating compounds and use thereof
12/20/2011US8080541 Carbocyclic GlyT-1 receptor antagonists
12/15/2011WO2011154953A1 Process for the preparation of iodides
12/14/2011CN102276511A 1-叔丁氧羰基-3-碘氮杂环丁烷的合成方法 1-tert-butoxycarbonyl-3-iodo-azetidine synthetic methods
12/08/2011WO2011151808A1 Hexafluoroisopropyl carbamate derivatives, their preparation and their therapeutic application
12/08/2011CA2801405A1 Hexafluoroisopropyl carbamate derivatives, their preparation and their therapeutic application
12/07/2011CN101367831B 用于制备碳青霉烯类抗生素的中间体及其制备方法 Intermediates and preparation method for preparing carbapenem antibiotic for
12/06/2011US8071788 Method and intermediates for the preparation of derivatives of N-(1-benzhydrylazetidin-3-yl)-N-phenylmethylsulfonamide
12/01/2011US20110294775 Novel compounds
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 ... 69