Patents
Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868)
08/2014
08/21/2014US20140235611 Phenyl derivative
08/21/2014US20140235565 N-alkylthio beta-lactams, alkyl-coenzyme a asymmetric disulfides, and aryl-alkyl disulfides as anti-bacterial agents
08/19/2014US8809552 Azetidine compounds, compositions and methods of use
08/19/2014US8809316 Use of immunosuppressant compounds in a new indication
08/14/2014WO2014122222A1 Hydroxamate derivatives bearing amide-lactams as potent hdac inhibitors and their uses as medicaments
08/14/2014US20140228344 Alkene azetidine derivatives as sphingosine 1-phosphate (s1p) receptor modulators
08/14/2014US20140228341 Azetidine derivatives as sphingosine 1-phosphate (s1p) receptor modulators
08/14/2014US20140228339 Novel Compound
08/13/2014CN102448932B 氮杂环丁酮类化合物及医药应用 Azetidinone compounds and pharmaceutical applications
08/13/2014CN102015636B 作为组胺h3受体拮抗剂的氮杂环丁烷类和环丁烷类化合物 Azetidine as histamine h3 class and cyclobutane receptor antagonist compounds
08/13/2014CN101119966B 合成2-吖丁啶酮的方法 Synthesis of 2-azetidin-ketone
08/12/2014US8802659 Bicyclic aryl sphingosine 1-phosphate analogs
08/06/2014EP2762466A1 Phenyl derivative
08/06/2014CN103974936A 化学化合物 Chemical compounds
08/06/2014CN103965089A 一种立体选择性的合成降血脂药物依折麦布的方法 A stereoscopic selective synthesis of cholesterol-lowering drug ezetimibe methods
08/05/2014US8796245 C7-fluoro substituted tetracycline compounds
07/2014
07/30/2014EP2758371A1 New thio derivatives bearing lactams as potent hdac inhibitors and their uses as medicaments
07/30/2014CN103958465A 苯基衍生物 Phenyl derivatives
07/30/2014CN102741227B 芳基苄基胺化合物 Aryl benzyl amine compound
07/29/2014US8791159 Compound capable of binding S1P receptor and pharmaceutical use thereof
07/29/2014US8791100 Aryl benzylamine compounds
07/23/2014CN103936793A 含卡宾配体的催化剂及其制备方法与其在复分解反应中的应用 Catalyst and preparation method carbene ligand containing its metathesis reactions in the application
07/22/2014US8785669 Taxane compounds, compositions and methods
07/17/2014US20140200205 New thio derivatives bearing lactams as potent hdac inhibitors and their uses as medicaments
07/16/2014EP2754653A2 Azetidine derivative and antidepressant composition containing same
07/16/2014CN103922985A 一种氮杂环丁酮、合成方法及应用 One kind azetidinone, synthesis method and application
07/15/2014US8778628 Arylalkylamine compound and process for preparing the same
07/10/2014US20140194402 Pyruvate kinase activators for use in therapy
07/08/2014CA2650009C Il-8 receptor antagonists
07/08/2014CA2523083C Antiviral phosphonate analogs
07/03/2014US20140187533 Benzimidazole inhibitors of the sodium channel
07/03/2014US20140187532 4-(azacycloalkyl)benzene-1,3-diol compounds as tyrosinase inhibitors, process for the preparation thereof and use thereof in human medicine and in cosmetics
07/03/2014US20140187531 Apoptosis promoters
07/02/2014EP2749553A1 Process for preparation of enantiomerically pure S-(+)-N, N-dimethyl-a-[2-(naphthalenyloxy)ethyl] benzenemethanamine
07/02/2014CN101981003B 酰胺化合物、组合物及其应用 Amide compounds, compositions and use
06/2014
06/26/2014WO2014098098A1 Heterocyclic amide derivative, and medicine containing same
06/26/2014WO2014097257A1 A method of preparation of (1'r,3r,4r)-4-acetoxy-3-(1'-(tert-butyldimethylsilyloxy)ethyl)-2-azetidinone, a precursor for carbapenem antibiotics synthesis
06/26/2014US20140179665 Hepatitis b antiviral agents
06/26/2014US20140179661 N1-Cyclic Amine-N5-Substituted Biguanide Derivatives, Methods of Preparing the Same and Pharmaceutical Composition Comprising the Same
06/26/2014US20140179660 N1-Cyclic Amine-N5-Substituted Phenyl Biguanide Derivatives, Methods of Preparing the Same and Pharmaceutical Composition Comprising the Same
06/26/2014US20140179638 9-aminomethyl substituted tetracycline compounds
06/26/2014US20140179636 Liquid formulations
06/24/2014US8759387 Arylalkylamine compound and process for preparing the same
06/19/2014WO2014089810A1 METHOD FOR PREPARING CARBAPENEM INTERMEDIATE β-METHYL-ADC-8
06/19/2014US20140171649 Methods and Compositions for the Synthesis of Multimerizing Agents
06/19/2014US20140171402 Azetidine derivative and antidepressant composition including the same
06/18/2014CN103864658A Azacyclobutanone derivatives as well as preparation method and application thereof
06/18/2014CN102548962B Novel post metallocene-type transition metal compound
06/18/2014CN101506140B Cyclic 11-beta hydroxysteroid dehydrogenase type I inhibitors
06/17/2014US8753794 N-acyl-β-lactam derivative, macromolecular compound, and photoresist composition
06/12/2014WO2014087298A1 Novel selective androgen receptor modulators
06/10/2014CA2721815C Cyclic amine-1-carboxylic acid ester derivative and pharmaceutical composition containing the same
06/05/2014US20140155371 Multicomponent crystalline system of ezetimibe and proline
06/04/2014EP2738156A1 9-aminomethyl substituted tetracycline compound
06/04/2014CN103833544A 11-beta-hydroxysteroid dehydrogenase type i inhibitors
06/03/2014US8741261 Methods for carbon isotope labeling synthesis by transition metal-promoted carbonylation via isocyanate using azides and carbon-isotope monoxide
05/2014
05/30/2014WO2014081756A1 S1p and/or atx modulating agents
05/28/2014CN103819382A 一种依折麦布杂质的制备方法 A method for preparing ezetimibe ezetimibe impurities
05/28/2014CN102112430B 合成依泽替米贝的方法和用于该方法的中间体 Intermediate in the synthesis of ezetimibe method and the method used
05/21/2014EP2731945A1 N- (6- ( (2r,3s) -3,4-dihydroxybutan-2-yloxy) -2- (4 - fluorobenzylthio) pyrimidin- 4 - yl) -3- methylazetidine- 1 - sulfonamide as chemokine receptor modulator
05/21/2014CN102477008B 依泽替米贝的合成方法 Ezetimibe synthesis method
05/20/2014CA2591399C Aminocarboxylic acid derivative and medicinal use thereof
05/15/2014WO2014074848A1 Therapeutic compounds and compositions and their use as pkm2 modulators
05/15/2014WO2014072903A1 Novel aminomethyl-phenol derivatives as antimalarial agents
05/14/2014CN102137841B 邻位取代卤代烷基磺酰苯胺衍生物及除草剂 Ortho-substituted aniline derivatives and halogenated alkylsulfonyl herbicides
05/08/2014US20140128361 Cyclic amide bace-1 inhibitors having a benzamide substituent
05/08/2014US20140128360 Novel modulators of cortical dopaminergic- and nmda-receptor-mediated glutamatergic neurotransmission
05/07/2014CN103781781A 作为趋化因子受体调节剂的n-(6-((2r,3s)-3,4-二羟基丁-2-基氧基)-2-(4-氟苄基硫基)嘧啶-4-基)-3-甲基氮杂环丁烷-1-磺酰胺 As chemokine receptor modulators n- (6 - ((2r, 3s) -3,4- dihydroxybutan-2-yloxy) -2- (4-fluoro-benzyl thio) pyrimidin-4 - yl) -3-methyl-azetidine-1-sulfonamide
05/07/2014CN102432514B 1-叔丁氧羰基-3-氟氮杂环丁烷的合成方法 1-tert-butoxycarbonyl-3-fluoro-azetidine synthetic method
05/07/2014CN101945852B 氮杂环丁烷衍生物、其制备和其在治疗中的应用 Azetidine derivatives, their preparation and their use in therapy
04/2014
04/30/2014CN103755617A Method for preparing key impurity of ezetimibe
04/30/2014CN103755616A Method for preparing ezetimibe isomer
04/24/2014WO2014061693A1 Novel non-aromatic carbocyclic or non-aromatic heterocyclic derivative
04/23/2014CN103739537A New synthesis method of ezetimibe
04/22/2014US8703721 Arylalkylamine compound and process for preparing the same
04/16/2014CN103732577A New thio derivatives bearing lactams as potent HDAC inhibitors and their uses as medicaments
04/16/2014CN102477007B Novel method for preparing S-N-protective group-azetidine-2-carboxylic acid
04/16/2014CN102177134B C7-fluoro substituted tetracycline compounds
04/15/2014US8697888 Substituted (1-(methylsulfonyl)azetidin-3-yl)(heterocycloalkyl)methanone analogs as antagonists of muscarinic acetylcholine M1 receptors
04/15/2014US8697682 Salts
04/15/2014CA2653355C Substituted phenyl methanone derivatives
04/10/2014WO2014055548A1 Anti-fibrotic pyridinones
04/09/2014CN103709086A Preparation method for ezetimibe optical isomers and intermediate applied in preparation method
04/09/2014CN103709085A Pleuromutilin antibiotics
04/03/2014US20140094446 Cyclic Amino Acids for the Treatment of Pain
04/03/2014US20140094445 Substituted (e)-n'-(1-phenylethylidene)benzohydrazide analogs as histone demethylase inhibitors
04/03/2014US20140093518 Chemically Programmed Vaccination
03/2014
03/27/2014US20140088074 Fluorinated arylalkylaminocarboxamide derivatives
03/26/2014CN103665021A Synthetic method of biapenem drug intermediate 4-AA
03/26/2014CN103664877A Quinoline, preparation method and application of quinoline
03/20/2014US20140080802 Inhibitors of Histone Deacetylase
03/20/2014US20140080800 Inhibitors of Histone Deacetylase
03/20/2014US20140080770 Arylalkylamine compound and process for preparing the same
03/19/2014CN102731362B Method for preparing 1-carboxylic acid tert-butyl ester-3-fluoro-azetidine derivative
03/18/2014US8673901 Potassium channel blockers
03/13/2014WO2014036956A1 Crystal forms of azetidinone compounds and preparing methods thereof
03/13/2014WO2013190497A3 Compositions and methods for treatment of inflammatory diseases of the lung
03/11/2014US8669252 Prolylcarboxypeptidase inhibitors
03/06/2014US20140066420 Heterocyclic compound
03/05/2014CN103613526A Preparation method of meropenem intermediate cyclization compound
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