| Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868) |
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| 04/10/2013 | EP2576507A1 Hexafluoroisopropyl carbamate derivatives, their preparation and their therapeutic application |
| 04/09/2013 | US8415295 Heterocyclic boronic acid compounds |
| 04/04/2013 | WO2013047701A1 Phenyl derivative |
| 04/04/2013 | CA2849000A1 Phenyl derivative |
| 04/03/2013 | CN103012383A Ezetimibe intermediate and preparation method and application thereof |
| 04/03/2013 | CN101407486B Process for synthesizing 4-acetoxy-2-azetidinone |
| 04/02/2013 | US8410093 Cycloalkyl substituted pyrimidinediamine compounds and their uses |
| 04/02/2013 | CA2420652C Vertebrate intestinal protein which absorbs cholesterol, and the use of this protein for identifying inhibitors of intestinal cholesterol transport |
| 03/28/2013 | WO2013041480A1 New thio derivatives bearing lactams as potent hdac inhibitors and their uses as medicaments |
| 03/28/2013 | CA2843211A1 New thio derivatives bearing lactams as potent hdac inhibitors and their uses as medicaments |
| 03/27/2013 | CN103003233A Novel hydroxamic acid derivative |
| 03/27/2013 | CN102993077A Preparation method for Ezetimibe |
| 03/26/2013 | US8404671 Heterosubstituted N-thiolated beta-lactam compounds and methods of use |
| 03/21/2013 | US20130072677 Novel hydroxamic acid derivative |
| 03/20/2013 | CN102976993A Synthetic method of 3-hydroxyazetidine hydrochloride |
| 03/19/2013 | US8399454 Azetidinyl diamides as monoacylglycerol lipase inhibitors |
| 03/14/2013 | WO2013036015A2 Azetidine derivative and antidepressant composition containing same |
| 03/13/2013 | CN102971291A Novel amide derivative and use thereof as medicine |
| 03/12/2013 | US8394787 7-aza-spiro[3.5]nonane-7-carboxylate derivatives, preparation thereof and therapeutic use thereof |
| 03/06/2013 | CN1826344B (1S, 5S)-3-(5, 6-dichloro-3-pyridinyl)-3, 6-diazabicyclo[3.2.0]heptane is an effective analgesic agent |
| 03/06/2013 | CN102952055A Preparation method of ezetimibe and its intermediate |
| 03/06/2013 | CN101679236B Process for the preparation of ezetimibe and derivatives thereof |
| 03/05/2013 | US8389509 Substituted pyrazole compounds |
| 02/26/2013 | US8383810 Process for the synthesis of azetidinones |
| 02/21/2013 | WO2012173504A3 Method for synthesis of the substituted azetidinones and intermediates for their synthesis |
| 02/20/2013 | CN102936217A Preparation method of intermediate for penem |
| 02/20/2013 | CN102936216A Preparation method of 7,9-dioxo-2,6-aza-spiro[3.5]nona-2-tert-butyl formate and intermediate thereof |
| 02/20/2013 | CN101768101B Method for preparing 4-acetoxy-2-azetidinone |
| 02/14/2013 | WO2012116349A3 Novel cocrystals of ezetimibe |
| 02/14/2013 | US20130040932 Substituted aryl sulfone derivatives as calcium channel blockers |
| 02/14/2013 | US20130040926 Novel compound |
| 02/07/2013 | WO2013017548A1 1,4-diaryl-2-azetidinones with anti-tumoral activity |
| 02/06/2013 | CN101891665B (3S,4S)-4-acetyl-3-((R)-1-hydroxyethyl)-2-azetidinone and preparation method of same |
| 02/05/2013 | US8367654 8-AZA tetracycline compounds |
| 01/31/2013 | WO2013014604A1 Multicomponent crystalline system of ezetimibe and proline |
| 01/31/2013 | WO2013013505A1 9-aminomethyl substituted tetracycline compound |
| 01/31/2013 | WO2013013504A1 Tigecycline derivative |
| 01/31/2013 | CA2842838A1 9-aminomethyl substituted tetracycline compounds |
| 01/31/2013 | CA2841655A1 Multicomponent crystalline system of ezetimibe and proline |
| 01/29/2013 | US8362274 Arylalkylamine compound and process for preparing the same |
| 01/29/2013 | US8362000 Azetidinyl diamides as monoacylglycerol lipase inhibitors |
| 01/29/2013 | US8361998 Compounds and their use as IKACh blockers |
| 01/29/2013 | US8361994 Primary amine diazeniumdiolate heterocyclic derivatives |
| 01/17/2013 | WO2013008002A1 N- (6- ( (2r,3s) -3,4-dihydroxybutan-2-yloxy) -2- (4 - fluorobenzylthio) pyrimidin- 4 - yl) -3- methylazetidine- 1 - sulfonamide as chemokine receptor modulator |
| 01/17/2013 | CA2841859A1 N- (6- ( (2r,3s) -3,4-dihydroxybutan-2-yloxy) -2- (4 - fluorobenzylthio)pyrimidin- 4 - yl) -3- methylazetidine- 1 - sulfonamide as chemokine receptor modulator |
| 01/16/2013 | CN102884044A Derivatives of aminoindanes, their preparation and their application in therapeutics |
| 01/16/2013 | CN102875413A 免疫抑制剂化合物及组合物 Immunosuppressant compounds and compositions |
| 01/09/2013 | EP2542524A1 Derivatives of aminoindanes, their preparation and their application in therapeutics |
| 01/08/2013 | US8349825 Spirocyclic compounds |
| 01/08/2013 | CA2526530C (1s,5s)-3-(5,6-dichloro-3-pyridinyl)-3,6-diazabicyclo[3.2.0]heptane is an effective analgesic agent |
| 01/08/2013 | CA2525886C N-sulphonylated amino acid derivatives and their use as matriptase inhibitors |
| 01/03/2013 | US20130004518 Cyclic amine bace-1 inhibitors having a benzamide substituent |
| 01/02/2013 | CN101384532B Process for preparing optically active alcohols |
| 12/27/2012 | WO2012175962A1 COMPOUNDS FOR USE IN STABILISING p53 MUTANTS |
| 12/26/2012 | CN102108058B Cyclization reaction method of epoxy butyramide used in the synthesis of 4-AA |
| 12/25/2012 | US8338623 Compounds as cannabinoid receptor ligands |
| 12/20/2012 | WO2012173504A2 Method for synthesis of the substituted azetidinones and intermediates for their synthesis |
| 12/19/2012 | EP2534131A1 Methods of synthesizing and isolating n-(bromoacetyl)-3,3-dinitroazetidine and a composition including the same |
| 12/19/2012 | CN102827053A Aromatic amidine derivatives, and preparation method and pharmaceutical application thereof |
| 12/19/2012 | CN102827052A Method for synthesizing 3-hydroxy-azetidinehydrochloride |
| 12/19/2012 | CN102126999B Catalytic synthesis method of chiral azetidin-2-one-4-amide and carboxylic acid compounds in microorganism system |
| 12/19/2012 | CN101898990B Method for catalyzing and synthesizing chirality azetidine amide and carboxylic acid compound by microorganism system |
| 12/12/2012 | EP2531487A1 Aryl benzylamine compounds |
| 12/11/2012 | US8329749 Use of (−) (3-trihalomethylphenoxy) (4-halophenyl) acetic acid derivatives for treatment of hyperuricemia |
| 12/06/2012 | US20120309734 Combretastatin derivatives and uses therefor |
| 12/05/2012 | CN102807519A Preparation method of aztreonam side-chain small ring |
| 11/29/2012 | US20120302541 4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators |
| 11/29/2012 | US20120302539 Transglutaminase tg2 inhibitors, pharmaceutical compositions, and methods of use thereof |
| 11/28/2012 | EP2527317A1 Cyclic 11-beta hydroxysteroid dehydrogenase type I inhibitors |
| 11/28/2012 | CN102803236A Synthesis of TTX intermediates |
| 11/28/2012 | CN102803211A High penetration compositions or prodrugs of antimicrobials and antimicrobial-related compounds |
| 11/28/2012 | CN102803210A Azetidinyl diamides as monoacylglycerol lipase inhibitors |
| 11/22/2012 | WO2012157504A1 β-LACTAM COMPOUND AND METHOD FOR PRODUCING SAME |
| 11/22/2012 | WO2012155932A1 Improved process for the preparation of ezetimibe |
| 11/22/2012 | US20120295881 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy |
| 11/22/2012 | US20120295874 Coferons and methods of making and using them |
| 11/20/2012 | US8314087 Nitrogen-containing heterocyclyl ketones and methods of use |
| 11/14/2012 | CN102775366A Preparation method for 3-(5-methoxy-1,5-dioxopenyl)-(4S)-phenyloxazolidin-2-one |
| 11/13/2012 | US8309597 1,1′-diadamantyl carboxylic acids, medicaments containing such compounds and their use |
| 11/06/2012 | US8304403 Heterocyclic CETP inhibitors |
| 11/01/2012 | WO2012103456A3 Polycyclic beta lactam derivatives for the treatment of cancer |
| 10/31/2012 | CN102762535A Methods of synthesizing and isolating n-(bromoacetyl)-3,3-dinitroazetidine and a composition including the same |
| 10/31/2012 | CN101945851B Peptidyl nitriles and use thereof as dipeptidyl peptidase i inhibitors |
| 10/30/2012 | US8299067 5-demethoxyfumagillol and derivatives thereof |
| 10/30/2012 | US8299053 Cyclic nitro compounds, pharmaceutical compositions thereof and uses thereof |
| 10/30/2012 | US8299051 Beta-lactamase inhibitory compounds |
| 10/26/2012 | WO2012143337A1 Novel modulators of cortical dopaminergic- and nmda-receptor-mediated glutamatergic neurotransmission |
| 10/26/2012 | CA2832874A1 Novel modulators of cortical dopaminergic- and nmda-receptor-mediated glutamatergic neurotransmission |
| 10/24/2012 | EP2514743A1 Immunosuppressant Compounds and Compositions |
| 10/24/2012 | EP2513051A1 Combretastatin derivatives and uses therefor |
| 10/23/2012 | CA2566526C Naphthaline derivatives useful as histamine-3-receptor ligands |
| 10/18/2012 | WO2012142268A1 Phenyl bicyclic methyl azetidine derivatives as sphingosine-1 phosphate receptors modulators |
| 10/18/2012 | CA2833305A1 Phenyl bicyclic methyl azetidine derivatives as sphingosine-1 phosphate receptors modulators |
| 10/17/2012 | CN102741227A Aryl benzylamine compounds |
| 10/17/2012 | CN102741226A 4-substituted-2-phenoxy-phenylamine delta opioid receptor modulators |
| 10/17/2012 | CN102731362A Method for preparing 1-carboxylic acid tert-butyl ester-3-fluoro-azetidine derivative |
| 10/04/2012 | US20120252776 C4 Monomethyl Triterpenoid Derivatives and Methods of Use Thereof |
| 10/02/2012 | US8278341 Analogs of indole-3-carbinol and their use as agents against infection |
| 09/27/2012 | US20120245137 Aryl sulphone derivatives as calcium channel blockers |
| 09/26/2012 | CN1791395B 免疫抑制剂化合物及组合物 Immunosuppressive compounds and compositions |