Patents
Sitemap › C07 - Organic chemistry › C07D - Heterocyclic compounds › C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868)
02/2011
02/03/2011CA2767285A1 2-amino-2-phenyl-alkanol derivatives, preparation thereof, and pharmaceutical compositions containing same
02/02/2011EP2278878A1 2-aryl glycinamide derivatives
02/01/2011US7879998 4-alkenyl-2-azetidinone derivatives, process for preparing 4-alkenyl-2-azetidinone derivatives and multicyclic compounds prepared using 4-alkenyl-2-azetidinone derivatives
02/01/2011US7879997 Tumor necrosis factor-alpha converting enzyme inhibitors such as (2S,3R)-4-oxo-3-[[4-[(2-phenylquinolin-4-yl)methoxy]phenyl]methyl]azetidine-2-carboxylic acid, useful for the treatment of diseases or conditions mediated by matrix Metalloproteinases and tumor necrosis factor-alpha
01/2011
01/27/2011WO2011010891A2 Novel post metallocene-type transition metal compound
01/27/2011US20110021779 Process for the preparation of 6-substituted-1-(2h)-isoquinolinones
01/27/2011US20110020324 Compound capable of binding s1p receptor and pharmaceutical use thereof
01/26/2011EP2277861A1 Cyclic amine-1-carboxylic acid ester derivative and pharmaceutical composition containing the same
01/26/2011EP2276753A1 Intermediates for the preparation of (3r, 4s) -1- (4-fluorophenyl) -3- [ (3s) -3- (4-fluorophenyl) -3-hydroxypropyl) ] -4- (4-hydroxyphenyl) -2-azetidinone
01/26/2011EP2276730A2 Carbamate and urea inhibitors of 11beta-hydroxysteroid dehydrogenase 1
01/26/2011CN101959855A Azetidine-derived compounds, preparation method therefor and therapeutic use of same
01/20/2011US20110015174 Cyclic inhibitors of carnitine palmitoyltransferase and treating cancer
01/19/2011EP2275395A2 Copper-catalyzed formation of carbon-carbon bonds
01/19/2011EP1581509B1 1-(amino)indanes as edg receptor agonists
01/19/2011CN101362731B Heterocyclic compounds and methods of use
01/18/2011US7871998 Diphenylazetidinone derivatives possessing cholesterol absorption inhibitory activity
01/18/2011CA2500964C Cyclohexyl sulphone derivatives as gamma-secretase inhibitors
01/13/2011US20110009617 Ruthenium Catalysts and Uses Thereof
01/13/2011US20110009377 Azetidine derivatives, their preparation and their application in therapy
01/12/2011EP2272826A1 2-mercaptopentancarboxylic acid derivatives, the method for preparing them and the pharmaceutical compositions containing them
01/12/2011EP2272813A2 Copper-catalyzed formation of carbon-oxygen bonds
01/12/2011CN101945852A Azetidine derivatives, their preparation and their application in therapy
01/12/2011CN101945851A Peptidyl nitriles and use thereof as dipeptidyl peptidase i inhibitors
01/11/2011US7868013 Cycloalkyl substituted pyrimidinediamine compounds and their uses
01/11/2011CA2456426C New mandelic acid derivatives and their use as thrombin inhibitors
01/06/2011WO2011000212A1 Preparation method for ezetimibe and intermediates thereof
01/06/2011WO2010129057A3 Tetracycline compounds
01/06/2011US20110002992 N-sulphonylated amino acid derivatives, method for the production and use thereof
01/05/2011CN101935309A Method for preparing ezetimibe and intermediate thereof
01/04/2011US7863333 asthma, multiple sclerosis, artherosclerosis, and rheumatoid arthritis; Azetidine-1-carboxylic acid {2-[({2-hydroxy-1-[(isopropyl-methyl-amino)-methyl]-pentylcarbamoyl}-methyl)-carbamoyl]-4-trifluoromethyl-phenyl}-amide
01/04/2011US7863317 Lactams of alkylated acyclic diamine derivatives as modulators of chemokine receptor activity
01/04/2011US7863265 N-{[4-((2R,3R)-1-(4-fluorophenyl)-3-{[(2R or S)-2-(4-fluorophenyl)-2-hydroxyethyl]thio}-4-oxoazetidin-2-yl)phenoxy]acetyl}glycyl-D-lysine, used as anticholesterol agents
12/2010
12/29/2010WO2010149888A1 Derivatives of 2-mercaptocyclopentane carboxylic acid, method for the preparation thereof, and pharmaceutical compositions containing the same
12/29/2010WO2010132670A3 Pentacycline compounds
12/29/2010EP2265578A1 Azetidine derivatives
12/29/2010CN201684437U Ortho-nitrotoluene drier
12/29/2010CN101928242A Method for preparing Imipenem intermediate
12/29/2010CN101928241A 2-mercaptopentancarboxylic acid derivatives, the method for preparing them and the pharmaceutical compositions containing them
12/28/2010US7858633 Cycloalkyl substituted pyrimidinediamine compounds and their uses
12/23/2010WO2010146299A1 Azetidine-derived esters, preparation thereof, and therapeutic use thereof as cannabinoid receptor modulators
12/22/2010EP2262766A2 Amide compounds, compositions and uses thereof
12/22/2010CN101264051B Modified release pharmaceutical formulation
12/21/2010US7855193 1-(4-(5-Phenylbenzofuran-2-yl)benzyl)azetidine-3-carboxylic acids; anticarcinogenic, antiinflammatory, antiarthritic, antidiabetic agents; transplant rejection, autoimmune diseases, lupus, multiple sclerosis, psoriasis, inflammatory bowel disease, Chron's disease
12/21/2010CA2464130C Mch antagonists for the treatment of obesity
12/21/2010CA2448896C Allylmercaptocaptopril compounds and uses thereof
12/16/2010WO2010142836A1 Synthesis of ttx intermediates
12/16/2010WO2010142650A1 Novel cyclopentane derivatives
12/16/2010WO2010142241A1 High penetration compositions or prodrugs of antimicrobials and antimicrobial-related compounds
12/16/2010CA2802316A1 Synthesis of ttx intermediates
12/16/2010CA2764376A1 High penetration compositions or prodrugs of antimicrobials and antimicrobial-related compounds
12/16/2010CA2762619A1 Novel cyclopentane derivatives
12/15/2010CN101141959B 2,5-disubstituted phenyl methanone derivatives as glycine transporter 1 (Glyt-1) inhibitors for the treatment of neurological and neuropsychiatric disorders
12/09/2010WO2010141494A2 Synthesis of ezetimibe
12/09/2010US20100311734 Spiro Compounds Useful as Antagonists of the H1 Receptor
12/08/2010EP2258682A2 Amino-substituted tricyclic derivatives and methods of use
12/08/2010EP1628685B1 Antiviral phosphonate analogs
12/08/2010CN101910123A Process for the preparation of 6-substituted-1-(2H)-isoquinolinones
12/07/2010US7846920 Bactericides; bacteriostats; therapy for bacteria infections
12/01/2010EP2254862A2 Azetidine-derived compounds, preparation method therefor and therapeutic use of same
12/01/2010CN101898990A Method for catalyzing and synthesizing chirality azetidine amide and carboxylic acid compound by microorganism system
11/2010
11/30/2010US7842684 Diphenylazetidinone derivatives possessing cholesterol absorption inhibitor activity
11/30/2010CA2460682C Ester compound and medical use thereof
11/25/2010WO2010113182A8 Intermediates in the preparation of 1,4-diphenyl azetidinone
11/25/2010US20100298556 Method for crystallization of azetidinonecarboxylic acid
11/25/2010US20100297077 Novel aryl potassium channel blockers and uses thereof
11/24/2010CN101891666A Preparation method of intermediate of beta methylcarbapenem antibiotics
11/24/2010CN101891665A (3S,4S)-4-acetyl-3-((R)-1-hydroxyethyl)-2-azetidinone and preparation method of same
11/24/2010CN101175722B Azetidine derivatives as ccr-3 receptor antagonists
11/18/2010US20100292206 Heterocyclic compound
11/18/2010US20100291299 Strontium and barium precursors for use in chemical vapor deposition, atomic layer deposition and rapid vapor deposition
11/17/2010EP1934175B1 Anti-hypercholesterolemic compounds
11/17/2010CN101888989A Novel aryl potassium channel blockers and uses thereof
11/16/2010US7834000 CGRP receptor antagonists
11/11/2010US20100286109 Amide derivatives as positive allosteric modulators and methods of use thereof
11/11/2010CA2761241A1 Tetracycline compounds
11/10/2010CN101475521B Method for synthesizing acetate of 1-benzhydryl-3-azetidine amidino acetic ester
11/04/2010US20100279998 Piperidinylalkylcarbamate derivatives, methods for their preparation and the therapeutic use thereof as fatty acid amido hydrolase enzyme inhibitors
11/04/2010US20100279997 Analgesic that binds filamin a
11/03/2010EP1963260B1 Process for the production of ezetimibe and intermediates used in this process
11/02/2010US7825109 Compound capable of binding S1P receptor and pharmaceutical use thereof
10/2010
10/28/2010WO2010124116A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
10/28/2010WO2010124114A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
10/28/2010WO2010124112A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
10/28/2010WO2010124108A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
10/28/2010WO2010124086A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
10/28/2010US20100273739 Aminotetraline Derivatives, Pharmaceutical Composition, Containing Them, and Their Use in Therapy
10/28/2010CA2759697A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
10/28/2010CA2759621A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
10/28/2010CA2759614A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
10/28/2010CA2759604A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
10/28/2010CA2759501A1 Azetidinyl diamides as monoacylglycerol lipase inhibitors
10/27/2010CN101870670A Synthesis method of cyclobutylamine-2-carboxylic acid
10/26/2010US7820645 Crystalline forms
10/21/2010WO2010121046A1 4-azetidinyl-1-phenyl-cyclohexane antagonists of ccr2
10/21/2010WO2010120935A1 Anti-viral compounds
10/21/2010US20100267689 4-azetidinyl-1-phenyl-cyclohexane antagonists of ccr2
10/21/2010US20100267669 Heterocyclic cetp inhibitors
10/21/2010CA2758934A1 4-azetidinyl-1-phenyl-cyclohexane antagonists of ccr2
10/21/2010CA2758484A1 Anti-viral compounds
10/20/2010EP2240441A1 Process for the preparation of 6-substituted-1-(2h)-isoquinolinones
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