| Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868) |
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| 04/19/2007 | WO2006135670A3 β-LACTAM SYNTHESIS |
| 04/19/2007 | WO2006135669A3 RESOLUTION OF ENANTIOMERIC MIXTURES OF β-LACTAMS |
| 04/19/2007 | CA2622755A1 Mek inhibitors and methods of their use |
| 04/18/2007 | CN1948312A Preparation method of meluopeinan |
| 04/17/2007 | US7205290 Diphenylazetidinone with improved physiological properties, process for its preparation, medicaments comprising this compound, and its use |
| 04/12/2007 | WO2006138230A3 The preparation and use of protease inhibitors |
| 04/11/2007 | EP1771410A1 Spirolactams and their synthesis |
| 04/11/2007 | CN1946685A Azetidine glycine transporter inhibitors |
| 04/11/2007 | CN1943786A Ester compound and its medicinal application |
| 04/10/2007 | US7202236 Salts of inhibitors of trypsin-like proteases such as thrombin, e.g., a sulfonate salt of Ph(3-Cl)(5-OCHF2) (R)CH(OH)C(O) (S)Aze-Pab(OMe), combined with a cellulose ether neutral gelling polymer for the treatment or prevention of thrombosis |
| 04/05/2007 | WO2007037743A1 Novel azetidine compounds useful in the treatment of functional gastrointestinal disorders, ibs and functional dyspepsia |
| 04/05/2007 | WO2007037518A1 Mutilin derivative and pharmaceutical composition containing the same |
| 04/05/2007 | WO2006138163A3 Anti-hypercholesterolemic compounds |
| 04/05/2007 | US20070078098 N-[3-(4-{(2S,3R)-2-(-(4-{[(2S, 5S, 3R, 4R, 6R)-3,4,5-trihydroxy-6-(hydroxymethyl)perhydro-2H-pyran-2-yl]ethyl-2-yl}phenyl)-3-[(3S)-3-(4-fluorophenyl)-3-hydroxypropyl]-4-oxoazetidin-1-yl}phenyl)propyl]-N-methylmethanesulfonamide; anticholesterol agent; low density lipoprotein; treating atherosclerosis |
| 04/05/2007 | CA2624491A1 Novel azetidine compounds useful in the treatment of functional gastrointestinal disorders, ibs and functional dyspepsia |
| 04/04/2007 | EP1768952A2 Preparation of beta-amino acids having affinity for the alpha-2-delta protein |
| 04/04/2007 | CN1942437A Substituted azetidine compounds as cyclooxygenase-1-cyclooxygenase-2 inhibitors, and their preparation and use as medicaments |
| 04/04/2007 | CN1939903A Mandelic acid derivatives and their use as throbin inhibitors |
| 04/04/2007 | CN1939902A Mandelic acid derivatives and their use as throbin inhibitors |
| 04/04/2007 | CN1307875C Compounds, compositions, and methods for controlling biofilms |
| 03/29/2007 | WO2007034325A1 Carboxamide derivatives as muscarinic receptor antagonists |
| 03/29/2007 | WO2007004028A3 Processes for the preparation of penems and its intermediate |
| 03/27/2007 | US7196099 Compounds and compositions as cathepsin inhibitors |
| 03/22/2007 | WO2007033039A2 Proteasome inhibiting beta lactam compounds |
| 03/22/2007 | WO2007031791A1 Biphenyl derivatives and their use in treating hepatitis c |
| 03/22/2007 | WO2006086562A3 Phenylazetidinone derivatives |
| 03/22/2007 | US20070066587 Substituted azetidine compounds, their preparation and use as medicaments |
| 03/22/2007 | CA2621364A1 Biphenyl derivatives and their use in treating hepatitis c |
| 03/21/2007 | EP1763514A2 Cycloalkyl substituted pyrimidinediamine compounds and their uses |
| 03/21/2007 | CN1931838A Azacyclo butanone derivative and its synthesis process |
| 03/20/2007 | US7192969 Ester derivatives |
| 03/20/2007 | US7192944 Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof |
| 03/15/2007 | WO2007030721A2 Processes for the preparation of (3r,4s)-4-((4-benzyloxy)phenyl)-1-(4-fluorophenyl)-3-((s)-3-(4-fluorophenyl)-3-hydroxypropyl)-2-azetidinone, an intermediate for the synthesis of ezetimibe |
| 03/15/2007 | US20070060561 Proteasome inhibiting beta-lactam compounds |
| 03/15/2007 | CA2616058A1 Processes for the preparation of (3r,4s)-4-((4-benzyloxy)phenyl)-1-(4-fluorophenyl)-3-((s)-3-(4-fluorophenyl)-3-hydroxypropyl)-2-azetidinone, an intermediate for the synthesis of ezetimibe |
| 03/08/2007 | WO2007026207A1 Direct aminolysis |
| 03/08/2007 | WO2006127893A3 Processes for production of 4-(biphenylyl)azetidin-2-one phosphonic acids |
| 03/08/2007 | US20070055065 3-amidinophenylalanine derivatives such as N-(2-aminoethyl)-1-[(2S)-3-(3-carbamimidoylphenyl)-2-[[2,4,6-tri(propan-2-yl)phenyl]sulfonylamino]propanoyl]piperidine-4-carboxamide, used as inhibitors of matriptase, for the prophylaxis of tumors |
| 03/08/2007 | US20070054891 e.g. 3-(2,4,4'-trichlorobenzhydryloxy)-N-(tert-butyl)azetidine-1-carboxamide; cannabinoid receptor antagonist; antidiabetic agent, antidepressant; eating disorders, obesity, nicotine addiction |
| 03/08/2007 | CA2616539A1 Direct aminolysis |
| 03/07/2007 | EP1758861A1 Dpp-iv inhibitors |
| 03/07/2007 | CN1925862A Treatment of diseases associated with the EGR-1 enhancer element |
| 03/07/2007 | CN1303067C Spiroheterocyclic nitriles useful as reversible inhibitors of cysteine proteases |
| 03/07/2007 | CN1302776C Peptide arginals and methods for treating disseminated intravascular coagulation |
| 03/01/2007 | WO2006122186A3 1,4-diphenyl-3-hydroxyalkyl-2-azetidinone derivatives for treating hypercholestrolemia |
| 03/01/2007 | US20070049748 Preparation of ezetimibe |
| 03/01/2007 | US20070049594 Novel compounds and compositions as cathepsin inhibitors |
| 02/28/2007 | EP1757582A1 Arylalkylamines and process for production thereof |
| 02/28/2007 | EP1756049A1 Method for producing 1,4-diphenyl azetidinone derivatives |
| 02/28/2007 | EP1755593A1 Naphthaline derivatives useful as histamine-3-receptor ligands |
| 02/28/2007 | EP1265606B9 Cell adhesion inhibitors |
| 02/28/2007 | CN1922135A 免疫抑制剂化合物和组合物 Immunosuppressant compounds and compositions |
| 02/28/2007 | CN1921858A Derivatives of piperidinylalkylcarbamates, preparation method thereof and use of same as faah enzyme inhibitors |
| 02/28/2007 | CN1301982C Compounds and method for preparing substituted 4-phenyl-4-cyanocyclohexanoic acids |
| 02/28/2007 | CN1301969C New mandelic acid derivatives and their use as thrombin inhibitors |
| 02/27/2007 | US7183304 Heterocyclic compounds and methods of use |
| 02/27/2007 | US7183270 Cyclic derivatives as modulators of chemokine receptor activity |
| 02/27/2007 | CA2432798C Sugar-substituted 2-azetidinones useful as hypocholesterolemic agents |
| 02/22/2007 | US20070043018 2"-Hydroxynicotianamine, process for producing the same and angiotensin converting enzyme inhibitor, hypotensive drug and health food |
| 02/22/2007 | US20070043017 Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use |
| 02/22/2007 | US20070043013 1,3 Disubstituted azetidine derivatives for use as ccr-3 receptor antagonists in the treatment of inflammatory and allergic diseases |
| 02/21/2007 | EP1753763A2 Indazole and indolone derivatives and their use as pharmaceuticals |
| 02/21/2007 | EP1753717A1 Method for producing diphenyl azetidinone derivatives |
| 02/21/2007 | EP1551797B1 Cyclohexyl sulphone derivatives as gamma-secretase inhibitors |
| 02/21/2007 | EP1425407A4 Enzymatic resolution of t-butyl taxane derivatives |
| 02/20/2007 | US7179907 3-amino-2-oxo-azetidin-1-yl) acetic acid derivatives with anti-PBP2a activity; providing a monobactam core alkyne,reacting monobactam alkyne under conditions that promote cyclotrimerization, performing a Diels-Alder reaction between the cyclotrimerization product of b) and a diene reactant |
| 02/15/2007 | US20070037971 Process for desilylation of carbapenem intermediates |
| 02/15/2007 | US20070037787 Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use |
| 02/15/2007 | US20070037785 Novel dipeptidyl peptidase IV inhibitors used for functionally influencing different cells and treating immunological, infammatory, neuronal, and other diseases |
| 02/13/2007 | US7176326 β-Lactams, methods for the preparation of taxanes, and sidechain-bearing taxanes |
| 02/13/2007 | US7176196 Bicyclic heterocycles as HIV integrase inhibitors |
| 02/13/2007 | US7176194 Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use |
| 02/13/2007 | US7176193 Antilipemic agents; therapy for insulin resistance |
| 02/13/2007 | CA2359744C Cephalosporins and homologues preparations and pharmaceutical compositions |
| 02/08/2007 | WO2007015533A1 Amidine compound and herbicide |
| 02/08/2007 | WO2007015161A1 Novel substituted azetidinones |
| 02/08/2007 | US20070032646 Novel taxanes and methods related to use and preparation thereof |
| 02/08/2007 | CA2615758A1 Novel substituted azetidinones |
| 02/07/2007 | CN1910141A Diamino alcohols and their use as renin inhibitors |
| 02/01/2007 | WO2007013592A1 Novel method for synthesis of intermediate in synthesis of carbapenem using sugar template |
| 01/31/2007 | EP1747197A1 Regioselective functionalisation and protection of spirolactams |
| 01/31/2007 | CN1906183A N-acylsulfonamide apoptosis promoters |
| 01/31/2007 | CN1905868A DPP-IV inhibitors |
| 01/31/2007 | CN1297546C Derivatives of N-(arylsulfonyl) beta-aminoacids comprising substituted aminomethyl group, prepn. method thereof and pharmaceutical compsns. contg same |
| 01/30/2007 | CA2226886C N-(4-substituted-benzyl)-2-aminolactam derivatives |
| 01/25/2007 | WO2006121861A3 Biphenylazetidinone cholesterol absorption inhibitors |
| 01/25/2007 | US20070021404 Novel aza-ring derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 01/25/2007 | US20070021403 Piperidinylalkylcarbamate derivatives, methods for their preparation and the therapeutic use thereof as fatty acid amido hydrolase enzyme inhibitors |
| 01/24/2007 | EP1745018A1 Azetidine glycine transporter inhibitors |
| 01/24/2007 | EP1539690A4 Fluorinated monomers, fluorinated polymers having polycyclic groups with fused 4-membered heterocyclic rings, useful as photoresists, and processes for microlithography |
| 01/24/2007 | CN1902169A 4-biarylyl-1-phenylazetidin-2-ones |
| 01/24/2007 | CN1902168A Novel1,3-disubstituted azetidine derivatives for use as 5ht2a receptor ligands |
| 01/24/2007 | CN1901971A Cyclopropane compounds and pharmaceutical use thereof |
| 01/18/2007 | WO2007007018A1 Piperazine heteroaryl derivates as gpr38 agonists |
| 01/18/2007 | WO2006124713A3 4-biarylyl-1-phenylazetidin-2-ones |
| 01/18/2007 | WO2006121822B1 USE OF β-LACTAMS FOR THE TREATMENTOF IBD AND GLAUCOMA |
| 01/17/2007 | CN1898203A Diphenylazetidinone derivates possessing cholesterol absorption inhibitory activity |
| 01/17/2007 | CN1898202A Anti-hypercholesterolemic compounds |
| 01/11/2007 | WO2007004028A2 Processes for the preparation of penems and its intermediate |
| 01/10/2007 | EP1741428A2 Cell adhesion inhibitors |