Patents
Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868)
06/2005
06/15/2005EP1539744A2 N-hydroxyamide derivatives possessing antibacterial activity
06/15/2005EP1539690A2 Fluorinated monomers, fluorinated polymers having polycyclic groups with fused 4-membered heterocyclic rings, useful as photoresists, and processes for microlithography
06/15/2005EP1137634B1 Process for the synthesis of azetidinones
06/15/2005EP0991654B1 Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and compositions containing same
06/09/2005WO2005021497A3 Tethered dimers and trimers of 1,4-diphenylazetidn-2-ones
06/09/2005US20050124654 Compounds and methods of use
06/09/2005US20050124598 Antibiotic compounds
06/08/2005EP1538150A1 Novel pleuromutilin derivatives
06/08/2005CN1205187C New amidino derivatives and their use as thrombin inhibitors
06/08/2005CN1205184C Beta-lactan
06/08/2005CN1205183C New amidino derivatives and their use as thrombin inhibitors
06/07/2005US6903123 Antitussive agents, anxiolytic agents, analgesics for treating cough, anxiety and pain
06/02/2005WO2005049594A1 N-acylsulfonamide apoptosis promoters
06/02/2005WO2005049593A2 N-acylsulfonamide apoptosis promoters
06/02/2005WO2005049592A1 A novel process for ezetimibe intermediate
06/01/2005EP1534689A1 Novel carboxamide compounds having an mch-antagonistic effect, medicaments containing said compounds, and methods for the production thereof
06/01/2005EP1461315A4 Catalytic carbonylation of three and four membered heterocycles
06/01/2005EP1351959B1 Novel pleuromutilin derivatives
05/2005
05/31/2005US6900345 Antibiotics; mutilin 14-[N-(2-carbamoyloxyethoxycarbonyl)]carbamate; therapy for bacteria infections; chemical synthesis
05/31/2005US6900319 Carbo- and heterocyclic amidines
05/31/2005CA2158275C Taxanes having an amino substituted side-chain
05/26/2005WO2005047251A1 Melanocortin receptor agonists
05/26/2005WO2005047248A1 4-biarylyl-1-phenylazetidin-2-ones
05/26/2005WO2005047247A1 Novel1,3-disubstituted azetidine derivatives for use as 5ht2a receptor ligands
05/26/2005WO2005047246A1 Novel 1, 3-disubstituted azetidine deivatives for use as 5ht2a receptor ligands
05/26/2005US20050113450 method of sterilization, sanitation, antisepsis, and disinfection, includes applying antimicrobial compounds to a surface; e.g. 2-[(3-{[4-chloro(methyl)anilino]sulfonyl}benzoyl)amino]-5-(trifluoromethyl)benzoic acid
05/26/2005CA2545373A1 Novel 1,3-disubstituted azetidine derivatives for use as 5ht2a receptor ligands
05/26/2005CA2545058A1 4-biarylyl-1-phenylazetidin-2-ones
05/25/2005DE10348022A1 Neue Dipeptidylpeptidase IV-Inhibitoren zur funktionellen Beeinflussung unterschiedlicher Zellen und zur Behandlung immunologischer, entzündlicher, neuronaler und anderer Erkrankungen New dipeptidyl peptidase IV inhibitors for the functional influence of different cells and for the treatment of immunological, inflammatory, neuronal and other diseases
05/24/2005US6897323 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same
05/19/2005WO2005044256A1 2-azetidinones as anti-hypercholesterolemic agents
05/19/2005WO2005044195A2 Fused phenylalanine derivatives as dipeptidyl peptidase-iv inhibitors for the treatment or prevention of diabetes
05/19/2005US20050107605 Novel beta-lactams methods for the preparation of taxanes, and sidechain-bearing taxanes
05/19/2005US20050107444 E.g., 2-(3-{3-[(2-chloro-3-(trifluoromethyl)-benzyl)-(2,2-diphenylethyl)-amino]-propoxy}phenyl)-1-morpholin-4-yl-ethanone; agonists of the nuclear receptors, LXR alpha and LXR beta used to increase ABCA1, ABCG1, and apolipoprotein E expression and inhibiting cholesterol absorption
05/19/2005CA2543943A1 2-azetidinones as anti-hypercholesterolemic agents
05/19/2005CA2541212A1 Fused phenylalanine derivatives as dipeptidyl peptidase-iv inhibitors for the treatment or prevention of diabetes
05/18/2005CN1617718A N-aryl-N'-arylcycloalkyl-urea derivatives as MCH antagonists for the treatment of obesity
05/18/2005CN1616423A E-alpha-chloro alkyllene-beta-lactan compound synthetic method and its use
05/18/2005CN1202081C Amidino and guanidino bita-azetidinone tryptase inhibitors
05/17/2005CA2301967C Azetidinone derivatives for the treatment of hcmv infections
05/17/2005CA2301548C Azetidinone derivatives for the treatment of hcmv infections
05/17/2005CA2301543C Azetidinone derivatives for the treatment of hcmv infections
05/12/2005US20050101586 Novel 5-HT2A receptor ligands
05/06/2005WO2004096287A3 Inosine monophosphate dehydrogenase inhibitory phosphonate compounds
05/06/2005WO2004092116A8 Bicyclic compounds having bradykinin receptors affinity and pharmaceutical compositions thereof
05/05/2005US20050096357 Antibiotics; therapy for infections which is caused by drug-resistant Streptococcus, or bacteria infections
05/04/2005CN1612887A Phosphino-aminophosphines
04/2005
04/28/2005WO2005037779A2 Novel dipeptidyl peptidase iv inhibitors used for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases
04/28/2005WO2004100888A3 N-thiolated azetidinones and anti-cancer use thereof
04/28/2005CA2542807A1 Novel dipeptidyl peptidase iv inhibitors used for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases
04/27/2005CN1610663A Process for producing azetidinone compounds
04/27/2005CN1198839C Novel dipeptide amidines as thrombin inhibitors
04/26/2005CA2353981C Process for the synthesis of azetidinones
04/21/2005WO2005035492A1 3-SUBSTITUTED β-LACTAMYL VASOPRESSIN V1A ANTAGONISTS
04/21/2005WO2005034960A1 Treatment of diseases associated with the egr-1 enhancer element
04/21/2005WO2005020882A3 Compound capable of binding s1p receptor and pharmaceutical use thereof
04/21/2005CA2541590A1 Treatment of diseases associated with the egr-1 enhancer element
04/14/2005WO2005033100A1 Novel hypocholesterolemic compounds
04/14/2005WO2005016883A3 Acrylamide derivatives as vla-1 integrin antagonists and uses thereof
04/14/2005US20050080078 Such as [1-(4-chloro-phenyl)-cyclobutyl]-(3-hydroxymethyl piperidin-1-yl)-methadone for treating cocaine and/or methamphetamine addiction
04/14/2005US20050080071 Treatment methods
04/14/2005CA2541822A1 Novel hypocholesterolemic compounds
04/13/2005EP1522541A1 Novel hypocholesterolemic compounds
04/13/2005EP1521742A1 Diphenylazetidinone derivatives for treating disorders of the lipid metabolism
04/13/2005CN1196683C Amino-compound
04/12/2005US6878833 Tetraalkylammonium alkoxides
04/12/2005US6878732 5,7-diazaspiro(3.4)octane and -octene derivatives; treating diseases including emesis, depression, anxiety and cough
04/12/2005US6878700 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
04/07/2005US20050075367 Ester compound and medicinal use thereof
04/06/2005EP1077700B1 BENZIMIDAZOLE DERIVATIVES AS MODULATORS OF IgE
04/06/2005CN1604890A 取代的环己烷衍生物 Substituted cyclohexane derivatives
04/06/2005CN1195762C Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and compositions containing same
04/05/2005CA1341478C Therapeutic methods using catalytic antibodies
03/2005
03/31/2005US20050070719 Central nervous system disorders; antidiabetic agents; antiinflammatory agents; antiarthritic agents;obesity; osteoporosis ; anticancer agents
03/31/2005US20050070519 Cyclisation process for the preparation of c-2 beta-lactam compounds
03/30/2005EP1517892A1 Ring-substituted diphenyl azetidinones, method for the production thereof, medicaments containing said compounds, and use thereof
03/30/2005EP1517891A1 Diphenyl azetidinones substituted by acidic groups, method for their production, medicaments containing said compounds and use thereof
03/30/2005EP1517890A1 Cationically substituted diphenyl azetidinones, method for their production, medicaments containing said compounds and use thereof
03/30/2005CN1602206A Pharmaceutical compositions based on azetidine derivatives
03/29/2005US6872842 Butenyl substituted taxanes
03/29/2005US6872717 Pharmacological uses of azetidine derivatives
03/24/2005WO2005026113A1 1, 3-disubstituted azetidine derivatives for use as ccr-3 receptor antagonists in the treatment of inflammatory and allergic diseases
03/24/2005WO2004099132A3 Process for the preparation of trans-isomers of diphenylazetidinone derivatives
03/24/2005US20050065211 Ester derivatives
03/24/2005US20050065147 N-alkylated diaminopropane derivatives as modulators of chemokine receptor activity
03/24/2005US20050065142 Antidiabetic agents; therapy for insulin resistance
03/24/2005CA2539049A1 Quinazoline derivatives
03/23/2005EP1515726A1 Morpholine and tetrahydropyran derivatives and their use as cathepsin inhibitors
03/16/2005EP1513808A2 Fluorinated cyclic amides as dipeptidyl peptidase iv inhibitors
03/16/2005EP1513807A1 Pharmaceutical combination
03/16/2005EP1513806A1 New salts
03/16/2005EP1513496A1 Immediate release pharmaceutical formulation
03/16/2005EP1513495A1 Modified release pharmaceutical formulation
03/15/2005US6867298 Group IB compounds used as condensation, amination, amidation or arylation catalysts; catalysis; efficiency
03/15/2005US6867297 Process for synthesizing 4-substituted azetidinone derivatives
03/15/2005US6867203 Cinnamide derivatives with aryl sulfide functionality; cerebral vasospasm
03/10/2005WO2005021499A1 N-alkylated diaminopropane derivatives as modulators of chemokine receptor activity
03/10/2005WO2005021498A1 Lactams of alkylated acyclic diamine derivatives as modulators of chemokine receptor activity
03/10/2005WO2005021497A2 Tethered dimers and trimers of 1,4-diphenylazetidn-2-ones
03/10/2005WO2005020899A2 Substituted cycloalkyamine derivatives as modulators of chemokine receptor activity
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