Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
01/1996
01/16/1996US5484926 HIV protease inhibitors
01/16/1996US5484917 For treatment and prevention of gastrointestinal disorders, pain and anxiety
01/16/1996US5484772 Arginine aldehyde compounds as anticoagulants or treatment of thromboembolitic agents
01/16/1996US5484771 Ribonucleotide reductase inhibitors
01/16/1996US5484770 Peptide compounds which inhibit the proliferation of epidermal or epithelial stem cells
01/16/1996CA1337936C Vibriolysin coupling process
01/11/1996WO1996000738A1 Endothelin antagonists ii
01/11/1996WO1996000736A1 Histidine and homohistidine derivatives as inhibitors of protein farnesyltransferase
01/11/1996WO1996000581A1 Process to inhibit binding of the integrin alpha 4 beta 1 to vcam-1 or fibronectin
01/11/1996DE4425857A1 Kaskaden-Polymer-Komplexe, Verfahren zur ihrer Herstellung und diese enthaltende pharmazeutische Mittel Cascade polymer complexes, process for their preparation and pharmaceutical compositions containing them
01/11/1996CA2193828A1 Process to inhibit binding of the integrin alpha 4 beta 1 to vcam-1 or fibronectin
01/11/1996CA2190977A1 Histidine and homohistidine derivatives as inhibitors of protein farnesyltransferase
01/11/1996CA2190756A1 Endothelin antagonists ii
01/10/1996EP0691346A1 Novel aspartyldipeptide derivatives and sweetener
01/10/1996EP0691345A2 HIV protease inhibitor combinations
01/10/1996EP0690841A1 Synthetic matrix metalloprotease inhibitors and uses thereof
01/09/1996US5482947 Retroviral protease inhibitors
01/09/1996CA2153551A1 Aspartyldipeptide derivatives and sweetener
01/06/1996CA2153270A1 Hiv protease inhibitor combinations
01/03/1996EP0690070A1 Indole-containing peptide and process for preparing the same
01/03/1996EP0689588A1 Extracellular signal-regulated kinase, sequences, and methods of production and use
01/03/1996EP0689549A1 New urea derivates, their preparation and their use
01/03/1996CN1114321A Chemical compounds
01/02/1996US5481030 Phosphonic acid compounds
01/02/1996US5481021 Phenyl amidines derivatives useful as platelet aggregation inhibitors
01/02/1996US5480970 Radioactive materials for labels in diagnosis of tumors in tissues
01/02/1996US5480893 Antitumor
01/02/1996US5480871 Peptoid α-1 adrenergic receptor ligands
01/02/1996US5480668 N-substituted derivatives of aspartame useful as sweetening agents
12/1995
12/28/1995WO1995035316A1 New opioid peptide antagonists
12/28/1995WO1995035315A1 Gem-disubstituted amino acid derivatives
12/28/1995WO1995035314A1 Thiazolidine derivatives, their preparation and drugs containing same
12/28/1995WO1995035313A1 3-amino-2-oxo-1-piperidineacetic derivatives containing an arginine mimic as enzyme inhibitors
12/28/1995WO1995035312A1 Arginine mimic derivatives as enzyme inhibitors
12/28/1995WO1995035311A1 3-amino-2-oxo-1-piperidineacetic derivatives as enzyme inhibitors
12/28/1995WO1995035310A1 Pyrrolidine derivatives for the treatment of cholecystokinine and gastrine-related disorders
12/28/1995WO1995035309A1 New thrombin inhibitors, their preparation and use
12/28/1995WO1995035308A1 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME
12/28/1995WO1995035307A1 Peptide derivatives with metallopeptidase inhibitory activity
12/28/1995WO1995035297A1 Novel substituted purinyl derivatives with immunomodulating activity
12/28/1995WO1995035280A1 Methods of synthesis of peptidyl argininals
12/28/1995CA2193133A1 Novel thrombin inhibitors, the preparation and use thereof
12/28/1995CA2192697A1 Methods of synthesis of peptidyl argininals
12/28/1995CA2192686A1 Arginine mimic derivatives as enzyme inhibitors
12/28/1995CA2192484A1 New opioid peptide antagonists
12/28/1995CA2192211A1 3-amino-2-oxo-1-piperidineacetic derivatives containing an arginine mimic as enzyme inhibitors
12/28/1995CA2192210A1 3-amino-2-oxo-1-piperidineacetic derivatives as enzyme inhibitors
12/28/1995CA2165956A1 Novel substituted purinyl derivatives with immunomodulating activity
12/27/1995EP0688788A1 Boronic acid peptide derivatives having protease inhibiting activity, process for preparation thereof and pharmaceutical compositions comprising them
12/27/1995EP0688337A1 Compositions and methods for the treatment of immunomediated inflammatory disorders
12/27/1995EP0688315A1 New heterocyclic compounds, their preparation and their use
12/27/1995EP0688314A1 Prodrug derivatives of enzyme inhibitors with hydroxyl groups, methods of preparing them and their use
12/26/1995US5478811 Orally-active elastase inhibitors
12/26/1995US5478809 Blood disorders
12/26/1995US5478808 2-amino-6,7-dihydroxy-4-thiaheptanoic acid derivatives, production and use thereof
12/25/1995CA2126702A1 Indole-containing peptide and process for preparing the same
12/23/1995CA2152205A1 Boronic acid peptidic derivatives; process for preparing the same and pharmaceutical compositions containing them
12/22/1995WO1994029278A1 Compound for protective and anchor groups and its use
12/22/1995CA2164959A1 Compound for protective and anchor groups and its use
12/21/1995WO1995034817A1 Positive and positive/negative cell selection mediated by peptide release
12/21/1995WO1995034558A1 Chondramides, production methods, compositions comprising chondramides and cultures for chondramide production
12/21/1995WO1995034311A1 Piperazine compounds promote release of growth hormone
12/20/1995EP0687688A1 Antibodies against pneumolysine and their applications
12/20/1995EP0687675A2 Irreversible HIV protease inhibitors, intermediates, compositions and processes for the preparation thereof
12/20/1995EP0687270A1 Osteogenic growth oligopeptides and pharmaceutical compositions containing them
12/20/1995EP0687254A1 4-aminopyridines, their preparation and their use as antithrombotic agent
12/20/1995EP0394424B1 Peptides and polypeptides from the sub-maxilary gland of the rat, corresponding monoclonal and polyclonal antibodies, corresponding hybridomas and applications of said products to the diagnosis, detection or for therapeutical purposes
12/20/1995CN1113493A Boron containing derivative and preparation and medical application of same
12/19/1995US5476961 One-pot process for the preparation of α-L-aspartyl-L-phenylalanine methyl ester hydrochloride
12/19/1995US5476942 1-[2-amino-5-[1-(triphenylmethyl)-1H-imidazol-4-YL]-1-oxopentyl] piperidine derivatives, their preparation and their use as synthetic intermediates
12/19/1995US5476870 15-deoxyspergualin analogs, their method of preparation and their use in therapeutics
12/19/1995US5476841 Peptide
12/19/1995US5476766 Ligands of thrombin
12/14/1995WO1995033764A2 Oral compositions comprising a novel tripeptide
12/14/1995WO1995033763A1 Novel elastase inhibitors
12/14/1995WO1995033762A1 Perfluoroalkyl ketone inhibitors of elastase and processes for making the same
12/14/1995WO1995033751A1 Bicycling lactam inhibitor of interleukin-1-beta converting enzyme
12/14/1995WO1995033478A1 Acylated enol derivatives as prodrugs of elastase inhibitors
12/14/1995WO1995028426A3 Peptides for reducing or inhibiting bone resorption, angiogenesis and restenosis
12/13/1995EP0686642A2 Modified guanidino and amidino thrombin inhibitors
12/13/1995EP0506748B1 Amino acids, peptides or derivatives thereof coupled to fats
12/13/1995CN1113266A Enzymatic coupling of L-phenylalanine methyl ester and N-benzyloxycarbonyl-aspartic acid
12/12/1995US5475106 Agonist for cholecystokinin and gastrin receptors; nervous system, gastrointestinal disorders
12/12/1995US5475096 Binding to three-dimensional targets
12/12/1995US5475085 Unlimited array of peptides having reverse turn mimetics
12/12/1995US5475027 Retroviral protease inhibitors
12/12/1995US5475013 Inhibit human immunodeficiency virus protease
12/12/1995US5475006 Mixed oxidation products which cannot form Vitamin A
12/12/1995CA1337731C Inhibitory tetrapeptide of entry into cycle of hemopoietic stem cells, processes for its preparation and its uses
12/11/1995CA2151412A1 Modified guanidino and amidino thrombin inhibitors
12/07/1995WO1995032985A1 3'-(4'-) nonradioactively tagged nucleosides and nucleotides with aminocarboxylic acid, peptide or carboxylic acid spacer
12/07/1995WO1995025749A3 Eating suppressant peptides
12/07/1995CA2190982A1 3'-(4'-) nonradioactively tagged nucleosides and nucleotides with aminocarboxylic acid, peptide or carboxylic acid spacer
12/06/1995EP0685489A2 Tripeptide antithrombotic agents
12/06/1995EP0684944A1 Coupling product obtained from hystamine and an amino acid
12/06/1995EP0684843A1 TECHNETIUM-99m LABELED PEPTIDES FOR DIAGNOSTIC IMAGING
12/06/1995EP0684830A1 Inhibitors of thrombosis
12/06/1995EP0409962B1 Agent for inhibiting hiv-proteases
12/05/1995US5473097 Granules of α-L-aspartyl-L-phenylalanine methyl ester
12/05/1995US5473055 Antitumor agents; better water solubility, side effect reduction