Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
01/1997
01/28/1997US5597825 Aggregation inhibitors
01/28/1997US5597804 N-sulfonylarginine keto-amide compounds
01/23/1997WO1997002285A1 Macrolides
01/23/1997WO1997002284A1 New thrombin inhibitors, their preparation and use
01/23/1997WO1997002051A2 Cascade polymer complexes
01/23/1997WO1996040743A3 Inhibitors of factor xa
01/23/1997CA2225959A1 Cascade polymer complexes, process for their production and pharmaceutical agents containing said complexes
01/23/1997CA2224715A1 Macrolides
01/22/1997EP0754702A2 Cyclopentane-beta-amino acid-tripeptides
01/22/1997EP0754678A2 Improvement of physiological tolerance of pharmaceutical active beta-amino acids
01/22/1997EP0754302A1 Methods and apparatus for synthesizing labeled combinatorial chemical libraries
01/22/1997EP0528858B1 Inhibitors of dipeptidyl-aminopeptidase type iv
01/22/1997CN1141002A Labeled chemotactic peptides to image focal sites of infection or inflammation
01/22/1997CN1140709A Substituted N-(indole-2-carbonyl)-beta-alanimamides and derivatives as antidiabetic agents
01/21/1997US5596000 Amino acid derivatives, processes for the manufacture thereof and pharmaceutical compositions containing these compounds
01/21/1997US5595990 Treatment of cardiovascular disorders
01/21/1997US5595877 Methods of producing nucleic acid ligands
01/20/1997CA2181308A1 Improving the tolerability of pharmaceutically active beta-amino acids
01/16/1997WO1997001579A2 Somatostatin peptides
01/16/1997WO1997001576A2 Phenyl peptides, method for preparing same, and pharmaceutical compositions containing said peptides
01/16/1997WO1997001338A1 Pyridinone-thrombin inhibitors
01/16/1997WO1996034113A3 Methods for the identification of farnesyltransferase inhibitors
01/16/1997CA2224437A1 Pyridinone-thrombin inhibitors
01/16/1997CA2197861A1 Phenyl peptides, method for preparing same, and pharmaceutical compositions containing said peptides
01/15/1997EP0753526A1 Adipocyte differentiation inhibitor peptide and adipocyte differentiation inhibitor containing said peptide as active ingredient
01/15/1997EP0753059A1 Peptide production as fusion protein in transgenic mammal milk
01/15/1997EP0753004A1 Antagonists of endothelin receptors
01/15/1997EP0753003A1 Aziridine derivatives, their production and use
01/15/1997EP0752987A1 Pyrimidinyl derivatives as interleukin inhibitors
01/15/1997EP0752873A1 Labelled peptide compounds
01/15/1997EP0539484B1 Method for preparing sulphonylpristinamycin iib
01/15/1997CN1140455A Diastereomeric pure trifluoromethyl ketone peptide derivs. as inhibitors of human leukocyte elastase
01/15/1997CN1140454A Novel mercaptoacetylamido-1,3,4,5-tetrahydro-benzo|c¨ azepin-3-one disulfide derivs. useful as inhibitors of enkephalinase and ACE
01/14/1997US5594151 Phenylboronic acid complexing reagents derived from aminosalicylic acid
01/14/1997US5594106 Inhibitors of TNF-α secretion
01/14/1997US5593967 Cholecystokinin antagonists, their preparation and therapeutic use
01/14/1997US5593642 Containment of solid support within a gas dispersion tube
01/09/1997WO1997000894A1 Compounds with growth hormone releasing properties
01/09/1997WO1997000890A1 Peptide that inhibits blood triglyceride level rise and blood triglyceride level rise inhibitor containing said peptide as active ingredient
01/09/1997WO1997000889A1 Peptides binding to low-density lipoproteins
01/09/1997WO1997000886A1 Obesity protein intermediates and their preparation and use
01/09/1997DE19525924A1 Kaskaden-Polymer-Komplexe, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Mittel Cascade polymer complexes, process for their preparation and pharmaceutical compositions containing them
01/09/1997CA2224867A1 Obesity protein intermediates and their preparation and use
01/09/1997CA2224434A1 Compounds with growth hormone releasing properties
01/08/1997EP0752425A2 Peptide ligands for the constant region of immunoglobulins
01/08/1997EP0751961A1 Eating suppressant peptides
01/08/1997EP0751960A1 Synthetic inverso or retro-inverso t-cell epitopes
01/08/1997EP0751783A1 Hypocholesterolemic, antiatherosclerotic and hypotriglyceridemic aminoacetylmercapto derivatives
01/08/1997EP0751779A1 Selectively cleavable linkers based on iminodiacetic acid ester bonds
01/08/1997EP0751768A1 Anti-viral and anti-cancer agents
01/08/1997EP0579789B1 Method of separating a peptide from a resin
01/08/1997EP0558657B1 Retroviral protease inhibitors
01/08/1997EP0386044B1 Hypoglycaemic peptides
01/07/1997US5591891 N-[Mercaptoacyl (amino acid or peptide ) ] compounds and S-lipophiIic aliphatic carbonyl derivatives thereof as antihypertensives
01/07/1997US5591886 Process for the crystallizing L-α-aspartyl-L-phenylalanine methyl ester from the solution
01/07/1997US5591884 Dopamine agonists
01/07/1997US5591860 Retroviral protease inhibiting compounds
01/07/1997US5591739 2-substituted indane-2-carboxyalkyl derivatives useful as inhibitors of enkephalinase and ACE
01/07/1997US5591728 New phosphonic acid compounds
01/07/1997US5591711 Lysine-glycine-histidine tripeptide, fibroblast proliferation
01/07/1997US5591614 Process for the enzymatic preparation of macrolactone
01/07/1997US5591593 Peptide sequence which binds to a mucin expressed by an epithelial tumor
01/07/1997US5591591 Dioxetane compounds for the chemiluminescent detection of proteases, methods of use and kits therefore
01/07/1997CA2004606C Process for preparing optically active 2-oxoimidazolidine derivatives
01/03/1997WO1997000268A1 Process for preparing derivatives of azabicyclo naphthyridine carboxylic acid comprising a dipeptide
01/03/1997WO1997000241A1 New cationic and polycationic amphiphiles, reactives containing the same and their use
01/03/1997WO1997000071A1 Androgenic directed compositions
01/03/1997CA2225484A1 Androgenic directed compositions
01/03/1997CA2224566A1 New cationic and polycationic amphiphiles, reagents containing them and their use
01/02/1997EP0751146A1 Crystallization of alpha-L-aspartyl-l-phenylalanine methyl ester from aqueous solution
01/02/1997EP0750631A1 Novel mercaptoacetylamido 1,3,4,5-tetrahydro-benzo(c)azepin-3-one disulfide derivatives useful as inhibitors of enkephalinase and ace
01/02/1997EP0750610A1 Piperidyl-4-substituted thyrosine derivatives as scintigraphic imaging agents for the diagnosis of thrombosis
01/02/1997EP0750609A1 Isoprenyl transferase inhibitors
01/02/1997EP0750508A1 RETROPEPTIDES, ANTIBODIES THERETO, AND USES THEREOF FOR VACCINATION AND $i(IN VITRO) DIAGNOSIS
01/02/1997EP0750507A1 PROTEASOME REGULATION OF NF-$g(k)B ACTIVITY
01/02/1997EP0662145B1 Process for the selective increase of production of antibiotic ge 2270 factor a
01/01/1997CN1139427A Malarial aspartic protease inhibitors
01/01/1997CN1138983A Preparation of drug composition
12/1996
12/31/1996US5589579 Gene sequence and probe for a marker of non-small cell lung carinoma
12/31/1996US5589460 Modification of melanotrophic release inhibiting factor
12/31/1996US5589459 Synthetic peptides for detoxification of bacterial endotoxins and for the prevention and treatment of septic shock
12/31/1996US5589458 Compounds that inhibit T cell proliferation and methods for using the same
12/31/1996CA2180207A1 Crystallization of .alpha.-l-aspartyl-l-phenylalanine methyl ester from aqueous solution
12/27/1996WO1996041830A1 Cascade polymers with iodine-containing aromatic compounds
12/27/1996WO1996041640A1 Bradykinin analogs as selective thrombin inhibitors
12/27/1996WO1996041638A1 Calpain inhibitors for the treatment of neurodegenerative diseases
12/27/1996WO1996031525A3 Inhibitors of farnesyl-protein transferase
12/27/1996WO1996030395A3 Cysteine protease inhibitor
12/27/1996EP0749978A1 Method of separating and purifying trh analogs and process for producing solvates of trh analogs
12/27/1996EP0749494A1 Compositions for the inhibition of tnf formation and uses thereof
12/27/1996EP0749316A1 Antithrombotic agents
12/27/1996CA2224721A1 Calpain inhibitors for the treatment of neurodegenerative diseases
12/24/1996US5587514 Reacting enolate of alpha-n,n-di-protected-aminoalkyl methyl ketone with alpha-leaving group acetate or acetamide
12/24/1996US5587475 Derivatized virginiamycin M1
12/24/1996US5587388 Irreversible HIV protease inhibitors, intermediates, compositions and processes for the preparation thereof
12/24/1996US5587375 Azepinone compounds useful in the inhibition of ACE and NEP
12/19/1996WO1996041172A1 Functional surrogates of analytes of interest and methods of obtaining and using same
12/19/1996WO1996040752A1 Novel dolastatin derivatives, their preparation and use
12/19/1996WO1996040751A1 Novel dolastatin derivatives, their preparation and use
12/19/1996WO1996040748A1 Peptidyl heterocycles useful in the treatment of thrombin related disorders