Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
07/1996
07/03/1996CN1032212C Process for preparing N-protected alpha-L-aspartyl-L-methyl phenylalaninate
07/02/1996US5532407 Adding l-aspartic acid or aqueous solution to side stream from production of alpha-l-aspartyl-l-phenylalanine methyl ester before or after mineral acid hydrolysis of side stream, adjusting ph of hydrolysis reaction mixture to 5-6
07/02/1996US5532366 Enzyme inhibitors
07/02/1996US5532359 Fungicides
07/02/1996US5532015 Drying wet crystals of l-aspartyl-l-phenylalanine methyl ester to adjust the water content
06/1996
06/29/1996CA2166246A1 Process of producing .alpha.-l-aspartyldipeptide amide derivatives
06/28/1996CA2165228A1 Metal chelate forming peptides and use thereof
06/27/1996WO1996019495A1 Methods and compositions for inhibition of membrane fusion-associated events, including hiv transmission
06/27/1996WO1996019494A1 Peptides having immunomodulatory activity
06/27/1996WO1996019493A1 N-SUBSTITUTED GLYCINE DERIVATIVES AS INHIBITORS OF FACTOR Xa
06/27/1996WO1996019492A1 Novel processes for preparing intermediates of inhibitors of enkephalinase and angiotensin converting enzyme and intermediates thereof
06/27/1996WO1996019491A1 Heterocyclic keto arginine peptides as thrombin inhibitors
06/27/1996WO1996019483A1 Low molecular weight bicyclic thrombin inhibitors
06/27/1996WO1996019473A1 New derivatives of pyroglutaminic acid, preparation process and applications
06/27/1996CA2208773A1 Heterocyclic keto arginine peptides as thrombin inhibitors
06/27/1996CA2208772A1 Low molecular weight bicyclic thrombin inhibitors
06/27/1996CA2207373A1 N-substituted glycine derivatives as inhibitors of factor xa
06/27/1996CA2206778A1 Peptides having immunomodulatory activity
06/26/1996EP0718307A2 Derivatives of 1-oxo-2-(phenylsulfonyl-amino)-pentylpiperidine, their preparation and therapeutic use
06/26/1996EP0718306A1 Crystallization of alpha-L-aspartyl-L-phenylalanine methyl ester from aqueous solution
06/26/1996EP0717751A1 Antibiotics 10381v, w, x, y, z1, z2, pre-b and t
06/26/1996EP0717736A1 Polar-substituted hydrocarbons
06/26/1996EP0717732A1 Polyamidic acid derivatives with antigastrin activity, a method for their preparation, and their pharmaceutical use
06/26/1996EP0717731A1 Difluoro statone antiviral analogs
06/25/1996US5530155 Crystallizing the amino acid by adding alkali to slurry, maintaining the ph at 3 to 8
06/25/1996US5530142 Process for the preparation of phosphorus-containing L-amino acids and their esters and N-derivatives
06/25/1996US5530097 Human cancer inhibitory peptide amides
06/25/1996US5529997 Administering for analgesic, hypotensive or diuretic effect or to treat congestive heart failure or irritable bowel syndrome
06/25/1996US5529996 2-substituted indane-2-mercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace
06/25/1996US5529995 Aminoacetylmercapto derivatives useful as inhibitors of enkephalinase and ACE
06/24/1996CA2166032A1 1-oxo-2-(phenylsulfonylamino)pentylpiperidine; process for preparing them and their use as therapeutic agents
06/20/1996WO1996018644A1 Aromatic heterocyclic derivatives as enzyme inhibitors
06/20/1996WO1996018643A1 Tachykinin antagonists
06/20/1996WO1996018627A1 Ahpba-containing tripeptide derivative
06/20/1996CA2206400A1 Aromatic heterocyclic derivatives as enzyme inhibitors
06/20/1996CA2204130A1 Tachykinin antagonists
06/19/1996EP0716658A1 Glycosyl amides of 2-aminoacylamino-2-deoxy sugars
06/19/1996EP0716609A1 METHODS AND COMPOSITIONS FOR STIMULATING AND INHIBITING TGF-$g(b) ACTIVITY
06/19/1996EP0535192B1 Novel dna gyrase inhibitors, process for their manufacture and pharmaceutical preparations containing same
06/19/1996CN1124964A Trifunctional antithrombin and antiplatelet peptides
06/19/1996CN1032058C A homogeneous compsn. for forming a film of precious metal and the process of firing such a film onto a substrate
06/18/1996US5527795 Mercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace
06/18/1996US5527770 Immunotherapeutic agent derived from bacteria
06/18/1996US5527689 Forming n-benzyloxycarbonyl-aspartyl-phenylalanine methyl ester in presence of protease and salt mixture
06/18/1996US5527610 Comprising tetrapeptide or pentapeptide repeating units containing proline and glycine with optional alanine residues
06/13/1996WO1996017942A1 Production of peptides using recombinant fusion protein constructs
06/13/1996WO1996017861A1 Substituted tetra- and pentapeptide inhibitors of protein:farnesyl transferase
06/13/1996WO1996017860A1 New dipeptide p-amidinobenzylamides with n-terminal sulfonyl or aminosulfonyl radicals
06/13/1996WO1996017838A1 Malonic acid based matrix metalloproteinase inhibitors
06/13/1996DE4443390A1 Neue dipeptidische p-Amidinobenzylamide mit N-terminalen Sulfonyl- bzw. Aminosulfonylresten New dipeptide p-Amidinobenzylamide with N-terminal sulfonyl or Aminosulfonylresten
06/13/1996CA2207874A1 Novel dipeptide p-amidinobenzylamides with n-terminal sulfonyl or aminosulfonyl radicals
06/13/1996CA2206848A1 Production of peptides using recombinant fusion protein constructs
06/13/1996CA2206665A1 Malonic acid based matrix metalloproteinase inhibitors
06/13/1996CA2204144A1 Substituted tetra- and pentapeptide inhibitors of protein:farnesyl transferase
06/12/1996EP0716150A1 DNA primer and a method for screening DNAs
06/12/1996EP0716086A1 Malonic acid based matrix metalloproteinase inhibitors
06/12/1996EP0715619A1 Inhibitors of tnf-alpha secretion
06/12/1996EP0715618A1 Hydroxyethylamino sulphonamides useful as retroviral protease inhibitors
06/12/1996EP0503044B1 Peptide compounds of laevorotatory amino acids and ring molecules, and therapeutical applications thereof
06/11/1996US5525727 Brain-specific drug delivery
06/11/1996US5525723 Inhibitors of angiotensin converting enzyme, neutral endopeptidase
06/11/1996US5525628 Salts of a glutathione alkylester and anaminoacids
06/11/1996US5525623 Compositions and methods for the treatment of immunomediated inflammatory disorders
06/11/1996US5525503 Signal transduction via CD28
06/11/1996US5525492 Polymerase chain reaction of nucleic acids
06/09/1996CA2137625A1 Process for the treatment of aspartame
06/06/1996WO1996016982A2 Ultraselective opioidmimetic peptides and pharmacological and therapeutic uses thereof
06/06/1996WO1996016981A2 Peptide compounds for prevention and/or treatment of no-mediated diseases
06/06/1996WO1996016950A1 Hiv protease inhibitors
06/06/1996WO1996016947A1 Novel 2,3-diketopiperazine derivative or salt thereof
06/06/1996WO1996016671A1 New antithrombotic formulation, process for its manufacturing, and use thereof
06/06/1996CA2206459A1 New antithrombotic formulation, process for its manufacturing, and use thereof
06/06/1996CA2206053A1 Novel 2,3-diketopiperazine derivatives or their salts
06/06/1996CA2164402A1 Dna primer and a method for screening dnas
06/05/1996EP0714903A1 New carbohydrate conjugates as cell adhesion inhibitors
06/05/1996EP0669935B1 Compounds useful as sweetening agents and process for their preparation
06/05/1996EP0577705B1 Method of enzymatic preparation of macrolactone
06/05/1996CN1124012A Arylating medicaments
06/05/1996CN1031948C Process for preparing antibiotic GE2270
06/04/1996US5523469 Reacting alkali metal sulfite on 1-(1-bromoethyl)-3-nitrobenzene; conversion to potassium salt; conversion to benzylquinium salt; then quaternization
06/04/1996US5523456 Anticarcinogenic agents
06/04/1996US5523313 Hypotensive agents; cardiotonic agents; inhibitors of neutral metalloendopeptidases; vasodilation; heart failure and renal insufficiency
06/04/1996US5523308 Peptidyl heterocycles useful in the treatment of thrombin related disorders
06/04/1996US5523289 Renin inhibitor
05/1996
05/30/1996WO1996016080A1 Human neutrophil elastase inhibitors
05/30/1996WO1996016079A2 Alpha-ketoamide derivatives as cathepsin l inhibitor
05/30/1996WO1996016078A1 Method of making a library of compounds
05/30/1996WO1996016027A1 Matrix metalloprotease inhibitors
05/30/1996WO1996015797A1 Pharmaceutical compositions comprising nitric oxide-releasing biopolymers
05/30/1996CA2205583A1 Method of making a library of compounds
05/30/1996CA2200964A1 Alpha-ketoamide derivatives as cathepsin l inhibitor
05/29/1996EP0713865A1 2-Aminobenzenesulphonic acid and 2-aminobenzenesulphonyl chloride derivatives, their preparation and their use as synthetic intermediates
05/29/1996EP0713859A2 Cinnamic acid derivatives, photocrosslinkable cinnamic acid-polymer derivative and crosslinked cinnamic acid polymer derivatives
05/29/1996EP0713495A1 Methods of enhancing bioactivity of chemokines
05/29/1996EP0471809B1 Method for preparing n-protected (2s,3s)-3-ethylaspartic acid dialkyl esters
05/29/1996CN1031880C Process for preparing novel analogs of peptidase substrates
05/28/1996US5521284 Human cancer inhibitory pentapeptide amides and esters
05/28/1996US5521179 Heterocyclic amides
05/28/1996US5521159 Partially modified and retro-inverted tetrapeptides analogues of C-reactive protein fragments
05/23/1996WO1996015148A2 Low molecular weight peptidomimetic growth hormone secretagogues