Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
08/1996
08/14/1996DE19504504A1 New orally active thrombin inhibiting peptide cpds.
08/14/1996CN1129000A New compound and its prepn.
08/14/1996CA2169335A1 Production of aldehyde derivatives
08/13/1996US5545838 Hypotensive agents
08/13/1996US5545750 Retroviral protease inhibiting compounds
08/13/1996US5545718 Synthetic peptides of the conjugate of ubiquitine and H2A histone
08/13/1996US5545662 Used to accelerate recovery from neutropenia accompanying radio or chemotherapy, bone marrow transplantation, or infections
08/13/1996US5545640 Viricides, hiv; aids
08/13/1996US5545621 Prodrug; controlling metabolism detoxification of cells
08/13/1996US5545568 Solid phase and combinatorial synthesis of compounds on a solid support
08/08/1996WO1996024061A1 Methods and apparatus for synthesizing labeled combinatorial chemical libraries
08/08/1996WO1996023812A1 Proline derivatives useful as inhibitors of human leukocyte elastase
08/08/1996WO1996023771A2 Platelet aggregation inhibitors
08/08/1996CA2210746A1 Platelet aggregation inhibitors
08/08/1996CA2209675A1 Proline derivatives useful as inhibitors of human leukocyte elastase
08/08/1996CA2186943A1 Methods and apparatus for synthesizing labeled combinatorial chemical libraries
08/07/1996EP0725075A1 Peptide derivatives comprising a phosphinic acid moiety as inhibitors of zinc depending endopeptidase 24-25
08/07/1996EP0724446A1 Electrophilic peptide analogs as inhibitors of trypsin-like enzymes
08/07/1996CN1128531A Therapeutic compound-fatty acid conjugates
08/06/1996US5543554 Exposing wet crystals of aspartame to a flow of air having a temperature of from 80 to 200 degree centigrade
08/06/1996US5543526 1-amino-4-(1H-imidazole)- aminobutaneboronic acid derivatives, their preparation and use as synthetic intermediates
08/06/1996US5543397 Glutamine source in culture medium
08/06/1996US5543396 Dipeptides as enzyme inhibitors of serine proteases; antiinflammatory and -tumor agents; anticoagulants; aids
08/01/1996WO1996022998A1 Thiol derivatives with metallopeptidase inhibitory activity
08/01/1996WO1996022997A1 Compounds with growth hormone releasing properties
08/01/1996WO1996022760A2 Antagonists of alpha-melanocyte stimulating hormone and methods based thereon
08/01/1996CA2210737A1 Antagonists of alpha-melanocyte stimulating hormone and methods based thereon
08/01/1996CA2210151A1 Thiol derivatives with metallopeptidase inhibitory activity
07/1996
07/31/1996EP0723974A1 Derivatives of mercaptoalkanoyldipeptides, their preparation and pharmaceutical compositions containing them
07/31/1996EP0723553A1 Compounds useful in anti-allergy treatment
07/31/1996EP0723552A1 Oligopeptides derived from c-reactive protein fragments
07/31/1996EP0723545A1 Quinolizinone type compounds
07/31/1996EP0723454A1 Novel tripeptides useful in immune and cns therapy
07/31/1996EP0723442A1 Lactone compounds for treating patients with precancerous lesions
07/31/1996EP0394326B1 Methods for the production of conformationally stabilized cell adhesion peptides
07/30/1996US5541334 Treating hiv
07/30/1996US5541290 Oligopeptide containing alpha-ketoamide group, treatment of alzheimer*s disease and other neurodegenerative disorders
07/30/1996US5541287 Diagnosis using cyclic tripeptides with nitrobenzyl 1,4,7,10-tetraazacyclododecane-n,n*,n**,n***tetraacetic acid biotin conjugate formed by alkylation and multistage process
07/30/1996US5541206 Retroviral protease inhibiting compounds
07/30/1996US5541162 Glutathione derivatives
07/25/1996WO1996022305A2 Modified peptides
07/25/1996WO1996022304A1 Conformationally constrained reverse-turn library and methods relating thereto
07/25/1996WO1996022303A1 Therapeutic compound - fatty acid conjugates
07/25/1996WO1996022106A1 Cd8 antagonists
07/25/1996WO1996022021A1 Protein hydroxylation inhibitors for fibroproliferative disorders
07/25/1996CA2210885A1 Protein hydroxylation inhibitors for fibroproliferative disorders
07/25/1996CA2210500A1 Therapeutic compound - fatty acid conjugates
07/25/1996CA2210349A1 Conformationally constrained reverse-turn library and methods relating thereto
07/24/1996EP0722459A1 Hemoregulatory penta- or hexapeptides
07/24/1996EP0722457A1 Compounds modifying serotoninergic transmission, diagnostic and therapeutic applications
07/24/1996EP0722456A1 Antifungal compositions
07/24/1996EP0722449A1 Boropeptide inhibitors of thrombin which contain a substituted pyrrolidine ring
07/24/1996EP0722439A1 Hiv protease inhibitors
07/24/1996EP0722431A1 Oxidized carotenoids, retinoids and related conjugated polyenes, and derived fractions and compounds useful as cell-differentiation inducers, cytostatic agents, and anti-tumor agents
07/24/1996EP0722321A1 Sulfoximine and sulfodiimine matrix metalloproteinase inhibitors
07/24/1996CN1127509A New peptide derivatives
07/24/1996CA2167763A1 Mercaptoalkyldipeptide derivatives; process for preparing the same and pharmaceutical compositions containing them
07/23/1996US5539122 Retroviral protease inhibiting compounds
07/23/1996US5539120 Arylalkyl-amines having anticonvulsant and neuroprotective properties
07/23/1996US5539104 1,4 Diazocines as fibrinogen antagonists
07/23/1996US5539082 Peptide nucleic acids
07/23/1996US5538951 Dipeptides of glutamic acid and tryptophan for immunology
07/23/1996US5538950 Endothelin antagonists and their preparation
07/23/1996CA1338484C 2,3-disubstituted isoxazolidines, a process for their preparation, agents containing them, and their use
07/18/1996WO1996021740A1 Methods of determining endogenous thrombin potential (etp) and thrombin substrates for use in said methods
07/18/1996WO1996021655A2 Substituted oxazolidine calpain and/or cathepsin b inhibitors
07/18/1996WO1996021464A1 Compositions for the delivery of antigens
07/18/1996WO1996021456A1 Inhibitors of prenyl transferases
07/18/1996CA2209492A1 Compositions for the delivery of antigens
07/18/1996CA2207252A1 Inhibitors of prenyl transferases
07/17/1996EP0721465A1 Glutathione s-transferase-activated compounds
07/17/1996EP0721449A1 INHIBITORS OF $g(b)-AMYLOID PROTEIN PRODUCTION
07/17/1996EP0721447A1 Anthracene derivatives for use as anticancer agent or dye
07/17/1996CN1126988A Difluoro statone analogs
07/17/1996CN1032308C Process for preparing optically active 2-oxoimidazolidine derivatives
07/16/1996US5536853 Opiate receptor ligands
07/16/1996US5536750 Antitumor
07/16/1996US5536716 Spiro piperidines and homologs which promote release of growth hormone
07/11/1996WO1996020949A1 Peptide and peptide analog protease inhibitors
07/11/1996WO1996020725A2 Peptide, peptide analog and amino acid analog protease inhibitors
07/11/1996CA2209234A1 Peptide and peptide analog protease inhibitors
07/10/1996EP0720988A1 Pseudopeptides containing trifluoromethyl substituted 2-azabicyclooctane
07/10/1996EP0720987A1 Acylated pseudopeptides containing trifluoromethyl substituted 2-azabicyclooctane
07/10/1996EP0720620A1 Glutathione analogs and paralog panels comprising glutathione mimics
07/10/1996EP0720619A1 Selectin binding glycopeptides
07/10/1996CN1126466A Nitrato amino acid disulphides for use in the therapy of disorders of the cardiovasculary system
07/10/1996CN1126207A Polysubstituted 3-acylamino-5-phenyl-1,4-benzodiazepin-2-one derivatives, process for their preparation and the pharmaceutical compositions containing them
07/10/1996CN1126203A Substituted heterocyclic carboxamides, their preparation and their use as pharmaceuticals
07/09/1996US5534538 High speed cleavage; artificial nutrition; cell cultures
07/09/1996US5534498 Trypsin inhibitors
07/09/1996US5534497 Radiopharmaceuticals; medical diagnosis
07/09/1996US5534496 Methods and compositions to enhance epithelial drug transport
07/09/1996US5534494 Polypeptide compounds having growth hormone releasing activity
07/05/1996CA2166374A1 Acylated pseudopeptides containing a trifluoromethyl-substituted 2-azabicyclooctane
07/05/1996CA2166372A1 Pseudopeptides having a trifluoromethyl-substituted 2-azabicyclooctane
07/03/1996EP0719790A2 Metal chelate forming peptides and use thereof
07/03/1996EP0719789A1 Process of producing alpha-L-aspartyldipeptide amide derivatives
07/03/1996EP0719779A1 Substituted thiazolo [3,2-alpha]azepine derivative
07/03/1996EP0719280A1 Process for the preparation of compounds having ace inhibitory action as well as novel compounds useful as starting materials or intermediates in said process
07/03/1996EP0719279A1 Process for purifying 1- n(2 -((s)-ethoxycarbonyl)-3-phenylpropyl)-n6 -trifluoroacetyl]-l-lysyl-l-prolin (lisinopril(tfa)ethylester)