Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
12/1994
12/21/1994EP0629627A2 Bicyclic carboxylic acids and their derivatives as nep and aca inhibitors
12/21/1994EP0629612A1 Ureas derived from alpha, omega-diaminoacids and process for their preparation
12/21/1994EP0629211A1 4-oxo-2 thioxoimidazolidine derivates as inhibitors of blood platelet aggregation
12/21/1994EP0629210A1 Peptide linkage unit comprising methylene phosphinic acid
12/21/1994EP0629196A1 Heterocyclic compounds, processes for their preparation and pharmaceutical compositions containing them
12/21/1994EP0629133A1 Protein- and peptide-metal ion pharmaceutical applications
12/21/1994EP0624059A4 Combinatorial strategies for polymer synthesis.
12/21/1994CN1096515A New peptides
12/20/1994US5374736 L-4-(phosphinylethyl)-1,3-oxazolidin-5-one derivatives as intermediates for synthesis of phosphorus-containing L-amino acids
12/20/1994US5374733 Stability
12/20/1994US5374731 Amino acid derivatives with renin-inhibiting properties, a process for the preparation thereof, agents containing these, and the use thereof
12/20/1994US5374656 N-phenyl-n-alkoxycarbonylalkyl glycinamides, their preparation and the medicaments containing them
12/20/1994US5374623 Cysteine protease inhibitors effective for in vivo use
12/20/1994US5374622 Fibrinogen receptor antagonists
12/20/1994US5374618 Calcitonin peptides, and gene related pharmaceutical compositions
12/19/1994CA2125638A1 .alpha.,w-diaminoacid-derived ureins and process for their preparation
12/18/1994CA2126026A1 2-piperazinone compounds and their use
12/14/1994EP0627939A1 Conjugates of biotin and deferoxamine for radioimmunoimaging and radioimmunotherapy
12/14/1994EP0627929A1 Inhibitors of thrombosis
12/14/1994EP0627926A1 PEPTIDYL DERIVATIVES AS INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME
12/14/1994EP0627925A1 Trypsin inhibitors
12/14/1994CN1096300A Isosteric antiherpes peptide derivatives
12/14/1994CN1096299A Antiherpes peptide derivatives having a ureido N-terminus
12/08/1994WO1994028173A1 Association peptides
12/08/1994WO1994028012A1 Hydroxamate inhibitors of endothelin converting enzyme
12/08/1994WO1994027958A1 4-amidinophenylsulphonamides for the treatment of thrombo-embolitic conditions
12/08/1994WO1994027627A1 Hemoregulatory peptides
12/08/1994WO1994027584A2 Arylating medicaments
12/08/1994WO1994027444A2 A new bacterial toxin for use as a plant growth regulator and herbicide
12/08/1994CA2163459A1 Arylating medicaments
12/07/1994EP0627444A1 Monoacetic derivatives of the peptides leu-phe-ala and ala-leu-phe and their use in identifying and destroying tumour cells, viruses and virus-carrying cells
12/07/1994EP0416035B1 Amphiphilic peptides and use thereof
12/06/1994US5371269 Method for production of α-L-aspartyl-L phenylalanine methyl ester hydrochloride
12/06/1994US5371187 Crystalline N-(S-3-methylheptanoyl)-D-gamma-glutamyl-glycyl-D-alanine, and processes and intermediates therefor
12/06/1994US5371186 Synthetic peptides for detoxification of bacterial endotoxins and for the prevention and treatment of septic shock
12/06/1994US5371185 Theraputical agent
12/06/1994US5371072 Asp-Pro-Arg α-keto-amide enzyme inhibitors
12/06/1994CA1333441C Solid phase peptide synthesis
12/06/1994CA1333369C 3-propadienyl penicillin derivatives and intermediates
12/05/1994CA2125080A1 Peptidic phosphinyloxymethyl ketones as interleukin-1beta-converting enzyme inhibitors
12/04/1994CA2125021A1 Alpha-heteroaryloxymethyl ketones as interleukin-1 beta converting enzyme inhibitors
12/04/1994CA2124989A1 Endothelin antagonistic peptide
11/1994
11/30/1994EP0625987A1 Aminoacetylmercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace
11/30/1994EP0574545B1 Phenyl amidines derivatives useful as platelet aggregation inhibitors
11/30/1994CN1095724A Novel peptides the preparation and use thereof
11/30/1994CN1095709A 15-deoxyspergualin analogs, their method of preparation and their use in therapeutics
11/29/1994CA2124252A1 Method of reducing or preventing bone marrow hypoplasia
11/29/1994CA1333265C Coupling agents for radiolabeling proteins
11/24/1994WO1994026771A1 Process for the stereoselective preparation of l-alanyl-l-proline
11/24/1994WO1994026723A2 ras FARNESYL TRANSFERASE INHIBITORS
11/24/1994WO1994026719A1 Mercapto-amide derivatives useful as neutral endopeptidase and ace inhibitors
11/24/1994WO1994026718A1 3-aminoazepine compound and pharmaceutical use thereof
11/24/1994WO1994026311A1 Anthracycline conjugates, their preparation and their use as antitumor agents
11/24/1994WO1994026295A1 Metal chelates as spacer compounds in biologically active peptides
11/24/1994WO1994026294A1 Ligand precursors for incorporation into peptides
11/24/1994WO1994026272A1 3-[n-(2-mercapto-propionyl-amino-acetyl)]-tetrahydro-thiazolyl-4-carboxylic acid as antiinflammatory and immunostimulating agent
11/24/1994WO1994016073A3 Methods and reagents for inhibiting furin endoprotease
11/24/1994CA2162715A1 3-aminoazepine compound and pharmaceutical use thereof
11/24/1994CA2160786A1 Ras farnesyl transferase inhibitors
11/23/1994EP0625313A1 High-calorie, low-osmolarity solution for total parenteral nutrition via periperal-venous administration
11/23/1994EP0625263A1 Contrast agents useful for both x-ray and mri
11/23/1994EP0625145A1 3-phenylureido-azepin-2-ones and -benzazepin-2-ones useful as cholecystokinin antagonists
11/23/1994EP0531461B1 Biologically active peptides containing d-2-alkyltryptophan
11/22/1994US5366973 Mercaptoacetylamido pyridazo [1,2]pyridazine, pyrazolo[1,2]pyridazine pyrazolo[1,2]pyridazine, pyridazol[1,2-a][1,2]diazepine and pyrazolol[1,2-a][1,2]diazepine
11/22/1994CA1333208C Peptide boronic acid inhibitors of trypsin-like proteases
11/17/1994EP0624377A2 Lysosomal enzyme-cleavable antitumor drug conjugates
11/17/1994EP0624059A1 Combinatorial strategies for polymer synthesis
11/16/1994CN1095072A Difluoro pentapeptide derivative anti-inflammatory agents
11/15/1994US5364931 Phosphonate-containing pseudopeptides of the hydroxyethylamine and norstatin type
11/15/1994US5364851 Internal coupling/cyclization to form helical structures
11/15/1994US5364844 Renin-inhibitory oligopeptides, their preparation and use
11/15/1994US5364838 Method of administration of insulin
11/13/1994CA2123261A1 Urethanes and ureas that induce cytokine production
11/10/1994WO1994025573A1 Catalytic antibodies which hydrolyze primary amides and methods for eliciting such antibodies
11/10/1994WO1994025477A2 Novel peptide nucleic acids
11/10/1994WO1994025432A1 Amino acid amide derivative, agrohorticultural bactericide, and production process
11/10/1994WO1994025052A1 Use of glutathione diesters
11/10/1994WO1994025051A1 Thrombin inhibitors
11/10/1994WO1994025049A1 Amidino and guanidino substituted boronic acid inhibitors of trypsin-like enzymes
11/10/1994WO1994021781A3 Extracellular signal-regulated kinase, sequences, and methods of production and use
11/10/1994DE4315437A1 Novel amino acid derivatives, process for their preparation and pharmaceutical compositions containing these compounds
11/10/1994CA2161230A1 Novel peptide nucleic acids
11/10/1994CA2161216A1 Amidino and guanidino substituted boronic acid inhibitors of tryspin-like enzymes
11/10/1994CA2161114A1 Catalytic antibodies which hydrolyze primary amides and methods for eliciting such antibodies
11/10/1994CA2159834A1 Thrombin inhibitors
11/09/1994EP0623627A1 Sulfonamide derivatives
11/09/1994EP0623625A1 Aminophosphonic acid derivative
11/09/1994EP0623606A2 Peptidic ketones as interleukin-1beta-converting enzyme inhibitors
11/09/1994EP0623596A1 N-acylpyrrolidines or N-acylpiperidines having a guanidinyl- or amidinyl-substituted side chain as thrombin inhibitors
11/09/1994EP0623595A1 Guanidinyl- or amidinyl-substituted heterocyclic thrombin inhibitors
11/09/1994EP0623592A1 Peptide analogs as irreversible interleukin-1beta protease inhibitors
11/09/1994EP0623144A1 Synthetic peptides for detoxification of bacterial endotoxins and treatment of septic shock
11/09/1994CN1094731A 2-amino-6,7-dihydroxy-4-thiaheptanoic acid derivatives, production and use thereof
11/09/1994CN1094730A Peptides
11/09/1994CN1026498C Enzymatic membrane method for the synthesis and separation of peptides
11/08/1994US5362912 Process for the preparation of a substituted diaminodiol
11/08/1994US5362903 Diffusion dialysis of solution containing derivative and hydrochloric acid, basification, crystallization
11/08/1994US5362851 Tripeptides
11/08/1994US5362831 Polymer-bound paclitaxel derivatives
11/08/1994US5362727 Treatment of cardiovascular disorders