Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
04/1997
04/01/1997US5616775 Esterifying a n-protected methionine; oxidizing; reacting with an acid anhydride then an alkali metal hydroxide
04/01/1997US5616727 Process for purifying 1-[N2 -((S)-ethoxycarbonyl)-3-phenylpropyl)-N6 -trifluoroacetyl]-l-lysyl-l-proline (lisinopril (TFA) ethyl ester
04/01/1997US5616720 Treating 1,6-diphenyl- or dihetero-substituted 2,5-diaminohexanol/3-/ with tetraalkoxytitanium, then amidation of reaction product and acylation yield stable viricides
04/01/1997US5616714 Retroviral protease inhibiting compounds
04/01/1997US5616620 Amino acid derivatives, pharmaceutical compositions containing these compounds and their use in the treatment of obesity
04/01/1997US5616612 Therapy for cancer, aids, anemia, infections
04/01/1997US5616605 Peptide derivatives of collagenase inhibitor
03/1997
03/29/1997CA2186717A1 Substituted quinoline-2-carboxylic acid amides, their preparation and their use as medicaments and intermediate products
03/28/1997CA2186665A1 Sulfonamide derivatives
03/27/1997WO1997011366A1 Histone deacetylase as target for antiprotozoal agents
03/27/1997WO1997011091A1 Novel peptide compounds and medicinal compositions thereof
03/27/1997WO1997011068A1 Novel pyridonecarboxylic acid derivatives or their salts and antibacterial agent comprising the same as the active ingredient
03/27/1997WO1997010853A2 N2s2-type bi-functional nicotinamide chelating agents for radioactive isotopes
03/27/1997WO1997010838A1 Use of one or more peptides in a cosmetic composition or for the preparation of a medicament
03/27/1997WO1997002051A3 Cascade polymer complexes
03/27/1997DE19536783A1 Bifunktionelle Nicotinamid-Chelatbildner vom Typ N¶2¶S¶2¶ für radioaktive Isotope Bifunctional nicotinamide-type chelating agent N¶2¶S¶2¶ for radioactive isotopes
03/27/1997DE19536780A1 Bifunktionelle sulfidhaltige Sulfonamid-Chelatbildner vom Typ XSNY für radioaktive Isotope Bifunctional sulfide-containing sulfonamide-type chelating agent XSNY for radioactive isotopes
03/27/1997CA2232340A1 Bifunctional nicotinamide-chelating agents such as n2s2 for radioactive isotopes
03/27/1997CA2231251A1 Histone deacetylase as target for antiprotozoal agents
03/27/1997CA2186187A1 Process for separating amino acids and/or aminosulphonic acids by adsorbing the amino acids on zeolites
03/26/1997EP0764444A1 Use of at least one peptide in a cosmetic composition or for the preparation of a medicine
03/26/1997EP0764167A1 Bicycling lactam inhibitor of interleukin-1-beta converting enzyme
03/26/1997EP0764152A1 Substituted indolylmethylene-oxindole analogues as tyrosine kinase inhibitors
03/25/1997US5614649 Treatment of muscular disorders, substituted guanidines
03/25/1997US5614557 Method of controlling tumor growth rate
03/25/1997US5614547 Small molecule inhibitors of rotamase enzyme
03/25/1997US5614539 Urea compounds which are useful as platelet aggregation inhibitors
03/25/1997US5614531 Adhesion receptor antagonists
03/25/1997US5614522 Retroviral protease inhibitors
03/25/1997US5614499 Anticoagulants; treatment or prophylaxis of thrombosis
03/25/1997US5614498 Oligopeptides, bronchdilators
03/25/1997US5614497 Treatment of hypertension, cardiovascular disease and renal disease
03/20/1997WO1997010507A1 Molecules that home to a selected organ or tissue in vivo and methods of identifying same
03/20/1997WO1997010262A1 Peptide derivatives
03/20/1997WO1997010261A1 Peptide derivatives
03/20/1997WO1997010197A1 METHOD FOR PREPARING φ-AMINOALKANOIC ACID DERIVATIVES FROM CYCLOALKANONES
03/20/1997WO1997009995A1 Method for reducing the severity of gastro-intestinal damage
03/20/1997WO1997009993A1 Method for analyzing isomers of enalapril and enalaprilat
03/20/1997WO1997009981A1 Advanced glycation end-product intermediaries and post-amadori inhibition
03/20/1997CA2231220A1 Peptide derivatives
03/20/1997CA2231174A1 Peptide derivatives
03/20/1997CA2231043A1 Method for analyzing isomers of enalapril and enalaprilat
03/20/1997CA2205056A1 Method for reducing the severity of gastro-intestinal damage
03/19/1997EP0763537A2 Non-peptidyl Ras farnesyl transferase inhibitors
03/19/1997EP0763062A1 New opioid peptide analogs with mixed mu agonist/delta antagonist properties
03/19/1997EP0763055A1 Perfluoroalkyl ketone inhibitors of elastase and processes for making the same
03/19/1997EP0763051A1 3'-(4'-) nonradioactively tagged nucleosides and nucleotides with aminocarboxylic acid, peptide or carboxylic acid spacer
03/19/1997EP0762887A1 Acylated enol derivatives as prodrugs of elastase inhibitors
03/19/1997EP0754302A4 Methods and apparatus for synthesizing labeled combinatorial chemical libraries
03/19/1997CN1145369A Peptide useful as ligand
03/19/1997CN1145365A Camptothecin derivatives
03/18/1997US5612369 Treatment of arterial and venous thrombotic occlusive disorders, inflammation, cancer, and neurodegenerative diseases
03/18/1997US5612360 Aromatic n-heterocyclic compounds as hypotensive agents with acid groups, sulfonylcarboxamides or tetrazole groups
03/18/1997US5612002 Apparatus and method for multiple simultaneous synthesis
03/18/1997CA2031528C Radionuclide metal chelates for the radiolabeling of proteins
03/13/1997WO1997009344A2 Librairies of backbone-cyclized peptidomimetics
03/13/1997WO1997009303A1 Alpha-hydrazino acid derivatives and method for making same
03/13/1997WO1997008934A2 Aryl acrylic acid derivatives useful as protein tyrosine phosphatase inhibitors
03/13/1997CA2230861A1 Libraries of backbone-cyclized peptidomimetics
03/13/1997CA2224874A1 Aryl acrylic acid derivatives useful as protein tyrosine phosphatase inhibitors
03/12/1997EP0761681A2 Process for the preparation of substituted derivatives of N-ethylglycine
03/12/1997EP0761680A2 Tetrazole compounds having Interleukin-1beta converting enzyme inhibitory activity
03/12/1997EP0760813A1 Inhibitors of farnesyl-protein transferase
03/12/1997EP0662081B1 Ureido-acetamide derivatives, preparation thereof and drugs containing same
03/12/1997EP0583338B1 Method for synthesizing peptides, novel amino acid derivatives used therein, and methods for preparing same
03/12/1997CN1145075A Antagonist's of endothelin receptors
03/12/1997CN1145074A Carbamoylmethylurea derivative
03/11/1997US5610308 Process for preparing intermediates for thrombin inhibitors
03/11/1997US5610297 Inhibitors of serine protease and cysteine protease
03/11/1997US5610279 Human TNF receptor
03/11/1997US5610271 Kappa receptor selective opioid peptides
03/11/1997US5610190 Retroviral protease inhibitors
03/11/1997US5610183 Phenylglycine derivatives pharmaceutical compositions containing them and their use in therapy
03/11/1997US5610146 2,3-disubstituted isoxazolidines, a process for their preparation, agents containing them, and their use
03/11/1997US5610145 Carbamate stereoisomers
03/11/1997US5610144 Pyrrolidine and thiazolidine derivatives, their preparation and medicaments containing them
03/11/1997US5610143 Antibiotics GE 37468 A, B and C
03/11/1997US5609870 Antisecretory, immunology
03/06/1997WO1997008334A1 Cryptophycins from aberrant biosynthesis
03/06/1997WO1997008193A1 Acylated oligopeptide derivatives having cell signal inhibiting activity
03/06/1997WO1997008192A1 Tricyclic antidepressant derivatives and conjugated useful in immunoassays
03/06/1997WO1997008191A1 Polymorphs of the prodrug 6-n-(l-ala-l-ala)-trovafloxacin
03/06/1997WO1997008145A1 Meta-guanidine, urea, thiourea or azacyclic amino benzoic acid derivatives as integrin antagonists
03/06/1997WO1997008133A1 Amide compounds and use of the same
03/06/1997WO1997007798A1 Pharmaceutical compounds
03/06/1997CA2502764A1 Amide compounds
03/06/1997CA2246117A1 Cryptophycins from aberrant biosynthesis
03/06/1997CA2230540A1 Pharmaceutical compounds
03/06/1997CA2230209A1 Meta-guanidine, urea, thiourea or azacyclic amino benzoic acid derivatives as integrin antagonists
03/06/1997CA2230052A1 Tricyclic antidepressant derivatives and conjugated useful in immunoassays
03/06/1997CA2227516A1 Acylated oligopeptide derivatives having cell signal inhibiting activity
03/05/1997EP0759934A1 Neurotensin antagonist peptides
03/05/1997EP0759786A1 Somatostatin binding peptide-metal chelate conjugates
03/05/1997EP0759772A1 Tri-, tetra-, penta-, and polypeptides and their therapeutic use as an antidepressant agent
03/05/1997EP0759770A1 Cytokine regulatory agents and methods of use in pathologies and conditions associated with altered cytokine levels
03/05/1997EP0585300B1 Galanin antagonist
03/05/1997EP0505428B1 Chromogenic substrate
03/05/1997EP0504207B1 Peptide derivative, process for the preparation thereof, pharmaceutical preparation containing it
03/05/1997CN1144487A Hypocholesterolemic, antiatherosclerotic and hypotriglyceridemic aminoacetylmercapto derivatives
03/04/1997US5608078 Phosphonomethyldipeptides and process for preparation thereof