Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
10/2001
10/04/2001WO2001072956A2 Compounds and methods for modulating desmosomal cadherin-mediated functions
10/04/2001WO2001072829A2 Peptides blocking vascular endothelial growth factor (vegf)-mediated angiogenesis, polynucleotides encoding said peptides and methods of use thereof
10/04/2001WO2001072770A1 Insulin potentiating peptides
10/04/2001WO2001072701A1 Ceramide derivatives and method of use
10/04/2001WO2001072324A1 Lactams as inhibitors of a-beta protein production
10/04/2001WO2001000663A3 Catalytically active recombinant memapsin and methods of use thereof
10/04/2001WO2000035941A3 Combinatorial process for preparing polyamines
10/04/2001EP1144434A3 Combinatorial process for preparing polyamines
10/04/2001EP1137763A1 Glucoamylases with n-terminal extensions
10/04/2001EP1137662A1 Pharmaceutical compositions comprising quinapril magnesium
10/04/2001EP1137661A1 Procollagen c-proteinase inhibitors
10/04/2001EP0853614B1 Substituted tetralylmethylen-oxindole analogues as tyrosine kinase inhibitors
10/04/2001EP0815123B1 Beta-sheet mimetics and use thereof as protease inhibitors
10/04/2001EP0802909B1 Substituted oxazolidine calpain and/or cathepsin b inhibitors
10/04/2001EP0688314B1 Prodrug derivatives of enzyme inhibitors with hydroxyl groups, methods of preparing them and their use
10/04/2001CA2404528A1 Peptides blocking vascular endothelial growth factor (vegf)-mediated angiogenesis, polynucleotides encoding said peptides and methods of use thereof
10/04/2001CA2404202A1 Compounds and methods for modulating desmosomal cadherin-mediated functions
10/04/2001CA2402769A1 Ceramide derivatives and method of use
10/04/2001CA2401120A1 Lactams as inhibitors of a-beta protein production
10/03/2001CN1315965A Hepatitis C inhibitor peptides
10/03/2001CN1315963A Benzodiazepines and benzothiazepines derivatives and HBSAG peptides binding to annexins, their compositions and use
10/03/2001CN1315959A N-Alkylaspartyldipeptide ester derivatives and sweeteners
10/03/2001CN1315958A Method for preparing crystal of aspartame derivative excellent in stability
10/03/2001CN1315957A Process for preparation of neotame
10/02/2001US6297380 Process and intermediates for growth hormone secretagogues
10/02/2001US6297217 Boronic ester and acid compounds, synthesis and uses
10/02/2001US6297216 Administering a dipeptide derivative to mammals
10/02/2001US6296850 Apoptosis-related compounds and their use
09/2001
09/27/2001WO2001070746A1 Furoisoquinoline derivatives, process for producing the same and use thereof
09/27/2001WO2001070672A2 Compounds and methods to treat alzheimer's disease
09/27/2001WO2001070337A1 Spiropiperidine derivatives as melanocortin receptor agonists
09/27/2001WO2001070275A2 Polyglutamic acid-camptothecin conjugates and methods of preparation
09/27/2001WO2001070049A1 Stability enhancement of sweeteners using salts containing divalent or trivalent cations
09/27/2001WO2001018232A3 Drug target isogenes: polymorphisms in the uncoupling protein 3 (mitochondrial, proton carrier) gene
09/27/2001WO2001000665A3 Inhibitors of memapsin 2 and use thereof
09/27/2001WO2000061541A3 Pharmaceutical compounds
09/27/2001DE10012120A1 New ligand, comprising therapeutic or diagnostic agent bonded non-covalently with substance having high affinity to transport molecule
09/27/2001CA2404226A1 Furoisoquinoline derivatives, process for producing the same and use thereof
09/27/2001CA2403631A1 Spiropiperidine derivatives as melanocortin receptor agonists
09/27/2001CA2402643A1 Polyglutamic acid-camptothecin conjugates and methods of preparation
09/27/2001CA2401749A1 Compounds and methods to treat alzheimer's disease
09/26/2001EP1136498A1 Inhibitors of serine proteases, particularly hepatitis c virus NS3 protease
09/26/2001EP1135406A1 Gamma-ketoacid tetrapeptides as inhibitors of caspase-3
09/26/2001EP1135151A1 Peptoid and nonpeptoid containing alpha-keto oxadiazoles as serine protease inhibitors
09/26/2001EP0802922B1 Novel amino acid derivatives, method of producing them and pharmaceutical compositions containing these compounds
09/26/2001EP0762887B1 Acylated enol derivatives as prodrugs of elastase inhibitors
09/26/2001EP0649426B1 Inhibitors of retroviral proteases
09/26/2001CN1314912A Tartrate salt of a sabstituted dipentide as growth hormone secretagogue
09/26/2001CN1314883A Amino acid derivatives and drug containing the same as the active ingredient
09/26/2001CN1071751C Reversible protease inhibitors
09/25/2001US6294686 Aspartame crystals and process for the preparation thereof
09/25/2001US6294534 Treatment of disorders responsive to the activation of melanocortin receptors, such as obesity, diabetes or male or female sexual dysfunction.
09/25/2001US6294525 Reverse-turn mimetics and methods relating thereto
09/25/2001US6294062 Method and device for electrochemical immunoassay of multiple analytes
09/25/2001CA1341296C 2-azabicycloalkane-3-carboxylic acid derivatives, processes for their preparation, agents containing these compounds and their use
09/20/2001WO2001068678A2 Peptides that selectively bind to expanded polyglutamine repeat domains and methods of use thereof
09/20/2001WO2001068655A2 Caprolactam derivatives and uses thereof
09/20/2001WO2001068145A2 Peptidase-cleavable, targeted antineoplastic drugs and their therapeutic use
09/20/2001WO2001068142A1 Therapeutic and diagnostic ligand systems comprising transport molecule binding properties and medicaments containing the same
09/20/2001WO2001068115A1 Process for producing peptide sequences possessing anti-hypertension activity
09/20/2001WO2001068114A1 Novel peptides with anti-hypertensive activity
09/20/2001WO2001068113A1 Anti-hypertensive peptides
09/20/2001WO2001047949A9 Aspartame derivative crystals
09/20/2001WO2001028579A3 Inhibitors of proteasomal activity for stimulating bone and hair growth
09/20/2001WO2001010456A3 Peptides that block viral infectivity and methods of use thereof
09/20/2001WO2000009537A3 Compounds having growth hormone releasing activity
09/20/2001US20010023301 By hydrogenating a mixture of 3,3-dimethylbutyraldehyde and N-benzyloxycarbonyl-L-alpha-aspartyl-L-phenylalanine-1-methyl ester in methanolic solvent, separating catalyst, desolventizing, adding water, separating solid neotame
09/20/2001US20010023244 Thrombin inhibitors
09/20/2001CA2401873A1 Peptidase-cleavable, targeted antineoplastic drugs and their therapeutic use
09/19/2001EP1133518A1 A METHOD FOR THE PREPARATION OF N-NEOHEXYL-$g(a)-ASPARTYL-L-PHENYLALANINE METHYL ESTER FROM IMIDAZOLIDIN-4-ONE INTERMEDIATES
09/19/2001EP0889901B1 Process and intermediates for the synthesis of lhrh antagonists
09/19/2001EP0802986B1 Methods of determining endogenous thrombin potential (etp) and thrombin substrates for use in said methods
09/19/2001EP0700302B1 Device for treating diabetes mellitus
09/19/2001EP0640099B1 Peptides having tachykinin antagonist activity
09/19/2001EP0600062B1 Polymer-bound paclitaxel derivatives
09/19/2001CN1313863A Inhibitors of urokinase and blood vessel fomation
09/19/2001CN1313855A Inhibitors of alpha4Betal mediated cell adhesion alpha Beta
09/19/2001CN1313846A C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cystenine proteases
09/18/2001US6291640 Peptidomimetic inhibitors of the human cytomegalovirus protease
09/18/2001US6291511 Biarylalkanoic acids as cell adhesion inhibitors
09/18/2001US6291452 Cholecystokinin antagonists.
09/18/2001US6291432 (r)-n-(2-methylbenzyl)-3-((2s, 3s)-3-(n-(2-chromonecarbonyl)-l-asparaginyl)amino-2-hydroxy-4-phenylbutano yl)-5,5-dimethyl-1,3-thiazolidine-4-carboxamide can be given as a typical example of this compound.
09/18/2001US6291004 Dipeptide sweeteners
09/13/2001WO2001066791A1 Method of screening inducible nitric oxide synthase activation inhibitor
09/13/2001WO2001066564A2 Gamma-secretase inhibitors
09/13/2001WO2001066147A2 Antimicrobial compounds and formulations
09/13/2001WO2001009169A3 Cysteine protease inhibitors
09/13/2001US20010021718 Antiscarring agent
09/13/2001US20010021713 Thromboresistant materials incorporating pyrazinone protease inhibitors
09/13/2001US20010021388 Cyclization of a triether with a diamine compound
09/13/2001CA2401525A1 Gamma-secretase inhibitors
09/13/2001CA2400410A1 Antimicrobial compounds and formulations
09/12/2001EP1132471A2 TNF-binding proteins
09/12/2001EP1132396A1 Physiologically active peptides
09/12/2001EP1132395A2 Process for the preparation of a pharmacologically active peptide
09/12/2001EP1132388A2 Hexahydropyrazolo[4,3-c]pyridine metabolites
09/12/2001EP1131636A1 Antibodies to peptides that target git receptors and related methods
09/12/2001EP1131634A2 Determining the mechanism of beta-amyloid peptide generation
09/12/2001EP1131351A2 Peptides that modulate the interaction of b class ephrins and pdz domains
09/12/2001EP1131341A1 Compound for inhibiting the influx of polymorphonuclear leukocytes (pmns) in a tissue, it's selection, pharmaceuticial compositions and use