Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
03/2001
03/21/2001EP1084133A1 Redox reversible bipyridyl osmium complex conjugates
03/21/2001EP1084132A1 Redox reversible imidazole-osmium complex conjugates
03/21/2001EP1083872A1 Pipecolic acid derivative hair growth compositions and uses
03/21/2001CN1288467A Compounds with growth hormone releasing properties
03/20/2001US6204406 Catalyst for asymmetric induction
03/20/2001US6204393 In aqueous solution; controlling ph; neutralization
03/20/2001US6204385 Reacting the corresponding nitrile with ammonia, amine or hydrazine in the presence of a mercaptocarboxylic acid
03/20/2001US6204361 Method of peptide synthesis
03/20/2001US6204279 Secondary amide containing benzoxazole derivatives
03/20/2001US6204268 Cyclic diaza compounds
03/20/2001US6204263 Thrombin inhibitors.
03/20/2001US6204261 Inhibitors of interleukin-1β Converting enzyme inhibitors
03/20/2001US6204035 Enzymatic protein associated with modulation of coagulation; for preparing tissues, and organs for grafting; anticoauglant; for diagnosis of defective coagulation in humans; for treating autoimmune and inflammatory diseases
03/20/2001US6204008 Bioprocess for production of dipeptide based compounds
03/20/2001CA2070169C Compounds with a sequence of three radicals, the central one being -aminoacidic and therapeutical applications thereof
03/20/2001CA1341206C Carboxyalkyl dipeptides, processes for their production and pharmaceutical compositions containing them
03/15/2001WO2001018232A2 Drug target isogenes: polymorphisms in the uncoupling protein 3 (mitochondrial, proton carrier) gene
03/15/2001WO2001018181A2 Enzyme inhibitors
03/15/2001WO2001018034A1 Process for producing aspartame derivative, method of purifying the same, crystals thereof and use of the same
03/15/2001WO2001018032A2 Dolastatin peptides
03/15/2001WO2001017563A2 Integrin-mediated drug targeting
03/15/2001WO2000061609A3 Prodrugs of thrombin inhibitors
03/15/2001WO2000053583A8 Inhibitors of protein tyrosine phosphatase
03/15/2001CA2383981A1 Integrin-mediated drug targeting
03/15/2001CA2383137A1 Method for producing aspartame derivative, method for purifying the same, crystals thereof and uses of the same
03/14/2001EP1082457A2 Nucleic acid encoding rate agouti related protein
03/14/2001EP1082314A1 New dipeptidyl peptidase iv effectors
03/14/2001EP1082126A1 Novel peptides
03/14/2001EP0812205B1 Antithrombotic azacycloalkylalkanoyl peptides and pseudopeptides
03/13/2001US6201103 Peptide nucleic acid incorporating a chiral backbone
03/13/2001US6200969 Contacting cells with reagent which suppresses protease activity of interleukin-1.beta.-converting enzyme (ice)/ced-3 family, inhibiting apoptosis in cell population to expanding or increasing survival of cell population
03/13/2001US6200967 Used as thrombin inhibitors, coagulation inhibitors and agents for the treatment of thromboembolic disorders
03/13/2001CA2146238C Novel mercaptoacetylamide bicyclic lactam derivatives useful as inhibitors of enkephalinase and ace
03/08/2001WO2001016372A1 Methods of immobilizing ligands on solid supports and apparatus and methods of use therefor
03/08/2001WO2001016300A2 Method of identifying inhibitors of cdc25
03/08/2001WO2001016211A1 Amphipathic compound having dendritic structure
03/08/2001WO2001016161A1 SYNTHESIS OF TEMPLATE-FIXED β-HAIRPIN LOOP MIMETICS
03/08/2001WO2001016135A2 Reverse-turn mimetics and methods relating thereto
03/08/2001WO2001016117A1 Processes for the preparation of oxo-oxazoline or alloamino acid derivatives
03/08/2001WO2000077184A9 Caspase-8 crystals, models and methods
03/08/2001WO2000038786A3 Use of cyclooxygenase 2 inhibitor and an integrin antagonist as a combination therapy in the treatment of neoplasia
03/08/2001CA2384126A1 Reverse-turn mimetics and methods relating thereto
03/08/2001CA2383603A1 Method of identifying inhibitors of cdc25
03/08/2001CA2382121A1 Methods of immobilizing ligands on solid supports and apparatus and methods of use therefor
03/07/2001EP1081158A1 Process for the purification of aspartame derivative
03/07/2001EP1080105A1 Phenylalanine derivatives having vla-4 antagonistic activity
03/07/2001EP1080104A1 Certain heteroaryl substituted thiol inhibitors of endothelin-converting enzyme
03/07/2001EP1079859A1 Bifunctional molecules and therapies based thereon
03/07/2001EP1079846A1 Hybrid polypeptides with enhanced pharmacokinetic properties
03/07/2001EP0641325B1 Retroviral protease inhibitors
03/07/2001CN1286695A Process for preparation of N2-(1 (s)-carboxy-3-phenylpropyl)-L-lysyl-L-proline
03/07/2001CN1286260A Crystal of methyl ester of alpha-L-asparaginyl-L-phenylalanine
03/06/2001US6197998 Adding dropwise to aqueous suspension of tyrosine two equivalents or more of haloacetyl halide and aqueous solution of inorganic base simultaneously to form n-haloacetyltyrosine, reacting with ammonium ion to form n-glycyltyrosine
03/06/2001US6197946 Nucleotide sequences coding hybrid albumin polypeptide; for production of heterologous polypeptide in hybrid animals
03/06/2001US6197794 Antiinflamamtory agents; immunology diseases
03/06/2001US6197750 C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases
03/06/2001US6197748 Ketoheterocyclic inhibitors of factor Xa
03/06/2001CA1341196C Process for the preparation of substituted imino diacids
03/01/2001WO2001014412A1 Compounds useful to mimic peptide beta-strands
03/01/2001WO2001014395A2 Novel glycoconjugates, glycoamino, acids, intermediates thereto, and uses thereof
03/01/2001WO2001014320A1 Compounds that inhibit tryptase activity
03/01/2001WO2001014318A2 New effectors of dipeptidyl peptidase iv for topical use
03/01/2001WO2000075365A3 COMPOUNDS AND METHODS TO ENHANCE rAAV TRANSDUCTION
03/01/2001DE19941062A1 Pure methyl 2-acetamido-3-chloropropionate preparation for use as intermediate for hypotensive agent ramipril, from methyl serinate hydrochloride by chlorination, acetylation and purification
03/01/2001DE19940130A1 Neue Effektoren der Dipeptidyl Peptidase IV zur topischen Anwendung New effectors of dipeptidyl peptidase IV for topical use
03/01/2001DE19939910A1 Neue Verbindungen, die Tryptase-Aktivität hemmen Novel compounds that inhibit tryptase activity
03/01/2001CA2381096A1 Compounds that inhibit tryptase activity
03/01/2001CA2379875A1 New effectors of dipeptidyl peptidase iv for topical use
03/01/2001CA2316767A1 Somatostatin antagonists and agonists that act at the sst subtype 2 receptor
02/2001
02/28/2001EP1077995A1 Antiangiogenic drug to treat cancer, arthritis and retinopathy
02/28/2001EP1077994A1 Imidazolidine derivatives, the production thereof, their use and pharmaceutical preparations containing the same
02/28/2001EP1077949A2 Combinations of protein farnesyltransferase and hmg coa reductase inhibitors and their use to treat cancer
02/28/2001CN1285356A Depeptide compound, its medical salt or ester, the medicinal composition using same as active component and the application for treating and preventing cell from dying
02/28/2001CN1062600C Process for preparation selenic antibody enzyme
02/27/2001US6194578 Growth hormone secretagogues; useful for prophylaxis and therapy of osteoporosis and/or frailty, insulin resistance in mammals, congestive heart failure, obesity, accelerating bone fracture repair reducing cachexia and protein loss
02/27/2001US6194429 Purification with a hydrophobic resin
02/27/2001US6194409 Heterocyclic derivatives and their use as antithrombotic agents
02/27/2001US6194386 Labelled peptide compounds
02/27/2001US6194380 Agents for promoting bone formation
02/27/2001US6194195 Pure culture; for production of hypotensive agents and therapies for asthma, cerebral apoplexy, angina pectoris, acute renal failure, cardiac infarction, and cerebral vasospasm
02/27/2001US6194143 Substrates for human cytomegalovirus protease
02/27/2001US6193981 Methods and compositions for impairing multiplication of HIV-1
02/27/2001CA2189526C Perfluoroalkyl ketone inhibitors of elastase and processes for making the same
02/22/2001WO2001013112A1 Melanocortin metallopeptide constructs, combinatorial libraries and applications
02/22/2001WO2001012653A1 Stabilisation of freeze-dried cake
02/22/2001WO2001012593A1 Arylsulfonanilide derivatives
02/22/2001WO2001012186A1 Cell adhesion inhibitors
02/22/2001WO2000071514A8 α-AMINO-β-SULFONYL HYDROXAMIC ACID COMPOUNDS
02/22/2001CA2380817A1 Cell adhesion inhibitors
02/22/2001CA2379647A1 Melanocortin metallopeptide constructs, combinatorial libraries and applications
02/21/2001EP1077218A2 Peptido-mimetic compounds containing RGD sequence useful as integrin inhibitors
02/21/2001EP1077217A2 Neuroactive peptides and their use
02/21/2001EP1077216A1 Crystallization of alpha-L-aspartyl-L-phenylalanine methyl ester from supersaturated solution
02/21/2001EP1076663A1 Functionalized alkyl and alkenyl side chain derivatives of glycinamides as farnesyl transferase inhibitors
02/21/2001EP1076645A1 Process for the preparation of methyl(2s)-2-[(3r)-3-(n-[tert-butyloxycarbonyl]-amino) -2-oxopyrr olidin-1-yl]propionate
02/21/2001EP1076563A1 Dipeptide caspase inhibitors and the use thereof
02/21/2001EP0835238B1 New cationic and polycationic amphiphiles, reactives containing the same and their use
02/21/2001CN1284964A Method for separating and purifying aspartame and aspartame derivative
02/21/2001CN1284943A Gamma-glutamyl and beta-aspartyl containing immunomodulator compounds and methods therewith
02/20/2001US6191282 Derivatives of 5-membered nitrogen containing heterocyclic ring is used as anticarcinogenic agent and anticoagulant