Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
06/2002
06/11/2002US6403561 Disorders associated with the inactivation or excessive degradation of cholecystokinin; inhibiting the enzymatic hydrolysis of cholecystokinin 1-(2(s)-aminobutyryl)-2(s)-indolinecarboxylic acid
06/11/2002US6403555 Depsipeptide and congeners thereof for use as immunosuppressants
06/11/2002US6403112 Ectoin and ectoin derivatives as moisturizers in cosmetics
06/06/2002WO2002044324A2 Bile-acid derived compounds for enhancing oral absorption and systemic bioavailability of drugs
06/06/2002WO2002043773A2 Tissue specific prodrugs
06/06/2002WO2001079242A3 Process for preparing lipid ii and derivatives thereof
06/06/2002WO2001074768A3 Inhibitors of serine proteases, particularly hepatitis c virus ns3 protease
06/06/2002WO2001042225A8 4-pyrimidinyl-n-acyl-l-phenylalanines
06/06/2002US20020068747 Inhibitors of prenyl-protein transferase
06/06/2002US20020068697 Peptides blocking vascular endothelial growth factor (VEGF) -mediated angiogenesis, polynucleotides encoding said peptides and methods of use thereof
06/06/2002US20020068695 Peptido-mimetic compounds containing RGD sequence useful as integrin inhibitors
06/05/2002EP1211249A1 Novel thiazine or pyrazine derivatives
06/05/2002EP1210361A1 Stabilisation of freeze-dried cake
06/05/2002EP1210360A1 Compounds useful to mimic peptide beta-strands
06/05/2002EP1210355A2 Glycoconjugates, glycoamino, acids, intermediates thereto, and uses thereof
06/05/2002EP1141375A4 Metallopeptide combinatorial libraries and applications
06/05/2002EP1071442A4 Methods and compositions for peptide synthesis
06/05/2002EP0871443B1 Advanced glycation end-product intermediaries and post-amadori inhibition
06/05/2002CN1085980C Meta-guanidine, urea, thiourea or azacyclic amino benzoic and derivatives as integrin antagaonists
06/04/2002US6399629 Efflux pump inhibitors
06/04/2002US6399601 Antidiabetic agents; nervous system disorders; anticholesterol agents
06/04/2002US6399599 Substituted 2-oxo-1,4-diazacycloalkanes
06/04/2002US6399568 Anticancer agents
06/04/2002US6399132 Sweetener composition
06/04/2002US6399053 Methods of enhancing bioactivity of chemokines
06/04/2002CA2205198C Human neutrophil elastase inhibitors
06/04/2002CA2174097C Antithrombotic azacycloalkylalkanoyl peptides and pseudopeptides
05/2002
05/30/2002WO2002042462A2 Therapeutic agents and methods of use thereof for treating an amyloidogenic disease
05/30/2002WO2002042414A2 Amino acid conjugates providing for sustained systemic concentrations of gaba analogues
05/30/2002WO2002042412A2 Protease inhibitors and their pharmaceutical uses
05/30/2002WO2002042295A2 Peptides as met-ap2 inhibitors
05/30/2002WO2002042278A2 Imidazole and benzimidazole caspase inhibitors and uses thereof
05/30/2002WO2001096364A3 Peptides that stimulate cell survival and axon regeneration
05/30/2002WO2001042282A9 Depsipeptide and congeners thereof for use as immunosuppressants
05/30/2002WO2001037194A9 Crystallizable compositions comprising a caspase-7
05/30/2002WO2001016300A3 Method of identifying inhibitors of cdc25
05/30/2002US20020065416 Anti-inflammatory agents
05/30/2002US20020065391 Compound for use in the treatment of arthritis, inflammatory bowel disease, nervous system and cardiovascular disorders, arteriosclerosis, restenoses, diabetes, grafted organ damage, asthma, allergies, tumor metastasis and malaria
05/30/2002US20020065284 Dipeptide derivatives
05/30/2002US20020065228 Inhibition of biosynthesis of a digestive enzyme of blood-ingesting pests known to feed on humans and animals; insecticides; pesticides; miticides; beetles; moths; flies; fleas; mosquitoes; lice
05/30/2002US20020065219 Water soluble thiazolyl peptide derivatives
05/30/2002US20020064501 Determining peptide's therapeutic effect by administering to subject prone to showing signs of diabetes; determining development of diabetes
05/30/2002CA2429630A1 Imidazole and benzimidazole caspase inhibitors and uses thereof
05/29/2002EP1209167A1 Method of producing a biosensor protein capable of regulating a fluorescence property of the modified green fluorescent protein therein, and the biosensor protein produced by the method
05/29/2002EP1209147A1 Carboxylic acid derivatives and adhesion molecule inhibitors containing the same as the active ingredient
05/29/2002EP1208377A1 Melanocortin metallopeptide constructs, combinatorial libraries and applications
05/29/2002EP1208238A1 Methods of immobilizing ligands on solid supports and apparatus and methods of use therefor
05/29/2002EP1208103A2 Reverse-turn mimetics and methods relating thereto
05/29/2002EP1207897A2 Pharmaceutical compositions containing tripeptides
05/29/2002EP1207873A1 Methods of inhibiting osteoclast activity
05/29/2002CN1351609A Low-molecular inhibitors of complement proteases
05/29/2002CN1351587A Use of 2,4-diamino-3-hydroxycarboxylic acid derivatives as proteasome inhibitors
05/28/2002US6395763 Antitumor, anticancer agents; immunosuppressant
05/28/2002US6395532 Modified enzymes and their use for peptide synthesis
05/28/2002US6395474 Peptide nucleic acids
05/28/2002CA2054715C Process for the preparation of n-protected dialkyl(2s,3s)-3-ethylaspartates
05/23/2002WO2002040631A2 Dipeptide seryl-histidine and related oligopeptides cleave dna, protein, and a carboxyl ester
05/23/2002WO2002040508A2 Lactam dipeptide and its use in inhibiting beta-amyloid peptide release
05/23/2002WO2002040507A2 Novel compounds for uses in radioimmunoscintigraphy and/or radioimmunotherapy of cancers
05/23/2002WO2002040040A1 Camptothecin compounds with a sulfhydryl group
05/23/2002WO2002002596A3 Synthetic methods for aplidine and new antitumoral derivatives, methods of making and using them
05/23/2002WO2001085911A3 Chromosome 17p-linked prostate cancer susceptibility gene and a paralog and orthologous genes
05/23/2002WO2001027077A3 Hydroxysulfonylalkylene-, phosphonoalkylene- or difluoro(phosphononon)methyl- substituted benzene, or benzofuran derivatives as non-peptidic cdc25 inhibitors
05/23/2002US20020061909 Vitronectin receptor antagonist pharmaceuticals
05/23/2002US20020061874 Substituted lactam; gamma-secretase inhibitor; decreases production of beta-amyloid; treatment for Altzheimer's and Down's syndrome
05/23/2002US20020061844 Administering to the patient for inhibiting Fc receptor binding of immunoglobulin a compound selected from aromatic, heteroaromatic, cyclic, bicyclic and an amino acid derivative or salt
05/23/2002US20020061840 Tripeptide compounds useful as selective inhibitors of aminopeptidase A and corresponding pharmaceutical compositions
05/23/2002CA2428802A1 Camptothecin compounds with a sulfhydryl group
05/22/2002EP1206485A2 New effectors of dipeptidyl peptidase iv for topical use
05/22/2002EP1206484A2 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
05/22/2002EP1206449A1 Lactam inhibitors of hepatitis c virus ns3 protease
05/22/2002EP1206444A1 Compounds that inhibit tryptase activity
05/22/2002EP1206273A2 Peptides that block viral infectivity and methods of use thereof
05/22/2002EP1206272A1 Hybrid polypeptides with enhanced pharmacokinetic properties
05/22/2002CN1350548A Long lasting insulinotropic peptides
05/22/2002CN1350545A Spray drying of thrombin inhibitors
05/22/2002CN1350525A 1,3,4-oxadiazole derivatives and process for producing the same
05/21/2002US6392046 Aids therapy
05/21/2002US6391919 Aids therapy
05/21/2002US6391856 Method for treatment of allergic reaction using formyl peptide
05/21/2002US6391855 Compounds and methods for modulating junctional adhesion molecule-mediated functions
05/21/2002US6391305 Conjugates useful in the treatment of prostate cancer
05/21/2002CA2082636C Process for the preparation of sulfonylpristinamycin iib
05/21/2002CA2059909C Alkylation of azaglycine derivatives
05/21/2002CA2039706C Method for preparing amino acid derivatives and therapeutical applications of same
05/16/2002WO2002038796A2 Methods for determining protease cleavage site motifs
05/16/2002WO2002038591A1 Fap-activated anti-tumor compounds
05/16/2002WO2002038590A1 Fap-alpha-activated anti-tumor compounds
05/16/2002WO2002038540A2 Activity-dependent cysteine protease profiling reagent
05/16/2002WO2002038187A1 Fap-activated anti-tumour prodrug
05/16/2002WO2002038108A2 Methods of treating disorders related to apoe
05/16/2002WO2002038107A2 Stat modulators
05/16/2002WO2002007770A3 Polymeric conjugates of antitumor agents
05/16/2002WO2001081368A3 Blood-pressure reducing polypeptides containing vpp derived from microorganisms
05/16/2002WO2001081366A3 Purification of ace inhibiting polypeptides containing vpp from milk
05/16/2002WO2001079195A3 Pyridine and pyrazine derivatives as thrombin inhibitors
05/16/2002WO2001068678A3 Peptides that selectively bind to expanded polyglutamine repeat domains and methods of use thereof
05/16/2002US20020058784 Generation of preferential compound; obtain sample of diamino acid such as 2,3 diaminopropionic acid, incubate with compound with free amino group, recover urein
05/16/2002US20020058631 Dipeptide derivatives
05/16/2002US20020058629 S-nitrosothiols as agents for the treatment of circulatory dysfunctions