Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
01/2001
01/30/2001US6180140 Modified amino acids for drug delivery
01/30/2001US6180116 Histidine derivatives, preparation process and uses
01/30/2001CA2124458C Technetium-99m labeled peptides for imaging
01/30/2001CA2101942C Technetium-99m labeled polypeptides for imaging
01/30/2001CA2052013C Tripeptide antithrombotic agents
01/25/2001WO2001005772A1 Pyrazinones, compositions containing such compounds
01/25/2001WO2000066587A3 Polyamines and their use in therapy
01/25/2001WO2000047605A3 Enterocyte growth factors and method for their isolation
01/25/2001DE19933861A1 New 2-aminomethyl-4-cyanothiazole, prepared from thioamide and bromopyruvate ester, used as intermediate for serine protease inhibitors, e.g. thrombin inhibitors
01/24/2001EP1070727A1 Low molecular weight peptide derivatives as inhibitors of the laminin/nidogen interaction
01/24/2001EP1070726A1 Aspartyl dipeptide ester derivatives and sweeteners
01/24/2001EP1070084A1 PIPERAZINES AS INHIBITORS OF FRUCTOSE-1,6-BISPHOSPHATASE (FBPase)
01/24/2001EP1070083A1 Crystalline forms of 1s- 1alpha (2s*,3r*), 9alpha]-6, 10-dioxo-n- (2-ethoxy-5 -oxo-tetrahydro-3 -furanyl) -9- (1-isoquinolyl) carbonyl]-amino] octahydro-6h -piridazino 1, 2-a] 1,2] diazepin- 1-carboxamide
01/24/2001EP1070060A1 Heterocyclic glycyl beta-alanine derivatives as vitronectin antagonists
01/24/2001EP1069906A1 Conjugates useful in the treatment of prostrate cancer
01/24/2001EP0712389B1 Therapeutic compound - fatty acid conjugates
01/24/2001EP0694039B1 1,5-benzodiazepine derivatives having cck antagonistic and or agonistic activity
01/24/2001CN1281346A Novel fluorescent reporter molecules and their applications, including assays for caspases
01/24/2001CN1281340A Mixed crystals comprising Aspartame and Aspartame derivative and process for producing same
01/24/2001CN1281339A Sweetener composition
01/24/2001CN1281338A Granular sweetener
01/23/2001US6177060 Nmr or x-ray lymphography images
01/23/2001CA2221767C A peptide inhibiting elevations of triglyceride levels in blood and an agent for inhibiting elevations of triglyceride levels in blood comprising the peptide as an active component
01/18/2001WO2001003723A1 Hybrid polypeptides with enhanced pharmacokinetic properties
01/18/2001WO2000063234A3 Pyrrolidincarbonylamino cyclic disulfides as vcam-vla4 antagonists
01/18/2001WO2000035492A3 Vitronectin receptor antagonist pharmaceuticals
01/18/2001WO2000019210A3 Determining the mechanism of beta-amyloid peptide generation
01/18/2001CA2377677A1 Hybrid polypeptides with enhanced pharmacokinetic properties
01/17/2001EP1069118A1 Process for producing 4-thiazolylmethyl derivative
01/17/2001EP1068295A1 Cell differentiation/proliferation and maintenance factor and uses thereof
01/17/2001EP1068218A2 Methods and compositions for the diagnosis and treatment of neuropsychiatric disorders
01/17/2001EP1067952A1 Methods for treatment and prevention of infections
01/17/2001EP1067894A2 Protease inhibitors
01/16/2001US6174915 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses
01/16/2001US6174887 Amide compounds and use of the same
01/16/2001US6174858 Conjugates useful in the treatment of prostate cancer
01/16/2001US6174691 Deactivating a preferential tumor glycoprotein or a cell expressing preferential glycoprotein; exposing preferential glycoprotein or cell expressing the preferential glycoprotein to a toxic substance
01/16/2001CA2200192C Amidino and guanidino substituted inhibitors of trypsin-like enzymes
01/16/2001CA2164707C Technetium-99m labeled peptides for imaging inflammation
01/16/2001CA2068324C Metal-peptide compositions and methods for stimulating hair growth
01/11/2001WO2001002601A2 Cell-based assay systems for examining hcv ns3 protease activity
01/11/2001WO2001002427A1 Streptogramin derivatives, preparation and compositions containing them
01/11/2001WO2001002426A1 A substantially crystalline form of melagatran
01/11/2001WO2001002424A2 Peptide boronic acid inhibitors of hepatitis c virus protease
01/11/2001WO2001002332A2 Process for the preparation of 3,3-dimethylbutanal
01/11/2001WO2001002018A2 Compounds that associate on the intermolecular level and aggregate bodies that contain them
01/11/2001WO2000063233A3 Peptides and the use thereof to control pests
01/11/2001WO2000061608A3 Low-molecular inhibitors of complement proteases
01/11/2001WO2000052019A3 Crystallization products of neotame and methods for producing same
01/11/2001DE19930177A1 Intermolekular assoziierende Verbindungen und diese umfassende Aggregate Inter-molecular compounds and associating this comprehensive aggregates
01/11/2001CA2376965A1 Peptide boronic acid inhibitors of hepatitis c virus protease
01/11/2001CA2376944A1 A substantially crystalline form of melagatran
01/11/2001CA2376698A1 Streptogramin derivatives, preparation and compositions containing them
01/10/2001EP1067138A1 Hydroxyproline derivatives
01/10/2001EP1067137A2 Granules of alpha-L-aspartyl-L-phenylalnine methyl ester
01/10/2001EP1067136A1 New peptide derivatives
01/10/2001EP1066316A1 Cinnamic acid derivatives having cell adhesion modulating activity
01/10/2001EP1066315A1 Use of inhibitors of mammalian asparaginyl endopeptidase for therapy of autoimmune disease
01/10/2001EP1056722A4 Bisulfate salt of hiv protease inhibitor
01/10/2001EP0742791B1 Macrocyclic difluorostatone derivatives useful as antiviral agents
01/10/2001CN1279236A Salt as thrombin inhibitor
01/09/2001US6172210 Nucleotide sequences which code enzymatic protein associated with phosphatides; for reduction and prevention of fibrin coagulation and vascular thrombosis; for diagnosing coagulation defects
01/09/2001US6172101 Treating human immunodeficiency virus infections
01/09/2001US6172082 α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
01/09/2001US6172044 Acylated enol derivative of α-ketoesters and α-ketoamides
01/09/2001US6171846 Culturing cells which are blocked in the synthesis of virginimycins; mutating genes in target microorganism and recovering cells with mutated target genes
01/09/2001US6171612 Gene therapy
01/09/2001US6171578 Glycoprotein iib/iiia receptor-binding benzodiazepine derivatives covalently linked to metal ion chelators.
01/09/2001US6171577 Accessible sulfhydryl group; and hexose moiety recognized by a mammalian liver receptor, wherein the hexose moiety is conjugated to the annexin.
01/04/2001WO2001001140A1 Epitopes formed by non-covalent association of conjugates
01/04/2001WO2001000665A2 Inhibitors of memapsin 2 and use thereof
01/04/2001WO2001000663A2 Catalytically active recombinant memapsin and methods of use thereof
01/04/2001WO2001000659A1 Benzimidazolone peptidomimetics as thrombin receptor antagonists
01/04/2001WO2001000658A1 C-terminal modified (n-substituted)-2-indolylcarbonyldipeptides as inhibitors of the ice/ced-3 family of cysteine proteases
01/04/2001WO2001000657A2 Novel indole peptidomimetics as thrombin receptor antagonists
01/04/2001WO2001000656A2 Novel indazole peptidomimetics as thrombin receptor antagonists
01/04/2001WO2001000622A1 Prodrugs of carbamate inhibitors of impdh
01/04/2001WO2001000247A1 Peptide-lipid conjugates, liposomes and liposomal drug delivery
01/04/2001WO2001000210A1 Reverse-turn mimetics and methods relating thereto
01/04/2001WO2000038715A3 Use of an integrin antagonist and radiation in the treatment of neoplasia
01/04/2001CA2376859A1 Peptide-lipid conjugates, liposomes and liposomal drug delivery
01/04/2001CA2375952A1 Reverse-turn mimetics and methods relating thereto
01/04/2001CA2374610A1 Catalytically active recombinant memapsin and methods of use thereof
01/04/2001CA2365341A1 C-terminal modified (n-substituted)-2-indolylcarbonyldipeptides as inhibitors of the ice/ced-3 family of cysteine proteases
01/03/2001EP1064354A1 Compositions and methods for gene-based vaccines to provoke t cell responses
01/03/2001EP1064300A1 Peptide turn mimetics
01/03/2001EP1064298A2 Inhibitors of caspases
01/03/2001EP1064021A1 Pharmaceutical composition containing a cysteine protease inhibitor for prophylaxis and therapy of brain tissue impairment
01/03/2001EP1064010A1 Peptide compositions and formulations and use of same
01/03/2001CN1278828A Sweetener salts of N-[N-3,3-dimethylbutyl)-L-&alpha,-aspartyl]-L-phenylalaning 1-methyl ester
01/03/2001CN1278827A Acid salts of N-[N-(3,3-dimethylbutyl)-L-alpha, -aspartyl]-L-phenylalanine 1-methyl ester
01/03/2001CN1278826A Metal complexes of N-[N-(3,3-dimethylbutyl)-L-alpha, -aspartyl]-L-phenylalanine 1-methyl ester
01/03/2001CN1278791A Process for the preparation of azacyclkylalkanoyl pseudotetrapeptides
01/03/2001CN1278790A Chemical compound
01/03/2001CN1278530A Novel peptide derivative
01/02/2001CA2184696C Hypocholesterolemic, antiatherosclerotic and hypotriglyceridemic aminoacetylmercapto derivatives
01/02/2001CA2114156C Elucidation and synthesis of selected pentapeptides
01/02/2001CA2086918C Biologically active compounds from blue-green algae
12/2000
12/28/2000WO2000078812A1 Method and compounds for inhibiting activity of serine elastases
12/28/2000WO2000078794A1 Cysteinyl protease inhibitors