Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
09/2001
09/12/2001EP1131340A2 Hexapeptide with the stabilized disulfide bond and derivatives thereof regulating metabolism, proliferation, differentiation and apoptosis
09/12/2001EP1131317A1 Method for preparing (2s)-1- (2r,3s)-5- chloro-3-(2- chlorophenyl) -1-(3,4-dimethoxy benzenesulphonyl) -3-hydroxy-2, 3-dihydro-1h- indole-2-carbonyl] pyrrolidine-2- carboxamide
09/12/2001EP1131082A2 A method for treating tissue damaged from ischemia
09/12/2001EP1049481A4 Synthetic antineoplastic agents derived from dolastatin 15 and methods of making same
09/12/2001EP1047445A4 Modified enzymes and their use for peptide synthesis
09/12/2001EP0929572A4 Antithrombotic azacycloalkylalkanoyl peptides and pseudopeptides
09/12/2001EP0808326B1 Basic oxazoline-amide derivatives of ge 2270 and ge 2270-like antibiotics
09/12/2001EP0789585B1 A storage stable water solution for infusion containing a thrombin inhibitor
09/12/2001EP0586474B1 Peptide nucleic acids
09/12/2001CN1312818A Chemical synthesis of exochelins
09/12/2001CN1312817A Dolastatin 15 derivatives
09/12/2001CN1312805A Benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake
09/11/2001US6288231 Peptide-containing α-ketoamide cysteine and serine protease inhibitors
09/11/2001US6288077 2,3-methano-amino acid compounds
09/11/2001US6288072 Anticarcinogenic and antitumor agents; leukemia
09/11/2001US6288038 Accelerate apolipoprotein e production; nervous system disorders, alzheimer*s disease; antilipemic agents
09/11/2001US6288037 C-terminally modified pentapeptides containing valine and aspartic acid
09/11/2001US6287840 Peptidomimetics; coupling, deblocking; antiarthritic, antitumor, anticarcinogenic, and antimetastasis agents; muscular dystrophy, glomerulonephritis, malaria, alzheimer*s disease
09/11/2001US6287806 Method for producing a biologically active recombinant cysteine-free peptide
09/11/2001US6287794 Peptide having antithrombotic effect through reversible inhibition of blood coagulation factor; antiinflammatory agents; treatment of cardiovascular disorders
09/11/2001US6287761 Synthetic antigens for the detection of antibodies to hepatitis C virus
09/11/2001CA2125175C New peptide derivatives
09/07/2001WO2001064738A2 Heparin-binding amino acid sequences derived from human proteins facilitating penetration of a substance of interest into cells and/or cell nuclei
09/07/2001WO2001055329A8 Nucleic acids, proteins, and antibodies
09/07/2001WO2001016135A3 Reverse-turn mimetics and methods relating thereto
09/07/2001WO2001014395A3 Novel glycoconjugates, glycoamino, acids, intermediates thereto, and uses thereof
09/07/2001WO2000071571A3 Fap-activated anti-tumor compounds
09/07/2001CA2401613A1 Amino acids sequencing facilitating penetration of a substance of interest into cells and/or cell nuclei
09/06/2001US20010020006 Dipeptidyl peptidase; antidiabetic agents
09/05/2001EP1129112A2 Peptides containing a cholesterol recognition sequence and their uses
09/05/2001EP1129108A1 Caspases and apoptosis
09/05/2001EP1129107A1 Method for producing l-prolyl-l-m-sarcolysyl-l-p-fluorophenylalanine and derivatives thereof
09/05/2001EP0956029A4 Cyclic peptides having broad spectrum antimicrobial activity
09/05/2001CN1311793A Antipicornaviral compounds, their prepn. and use
09/04/2001US6284777 Carbohydrazide protease inhibitors
09/04/2001US6284454 Variant of LAV viruses
09/04/2001CA2224062C Substituted n-(indole-2-carbonyl)-glycinamides and derivatives as glycogen phosphorylase inhibitors
08/2001
08/30/2001WO2001062775A2 Novel antiarrhythmic peptides
08/30/2001WO2001062735A1 Novel malonic acid derivatives, processes for their preparation, their use as inhibitor of factor xa activity and pharmaceutical compositions containing them
08/30/2001WO2001010457A3 Pharmaceutical compositions containing tripeptides
08/30/2001US20010018423 Anticoagulant agents
08/30/2001US20010018422 Anticancer agents
08/29/2001EP1127884A1 Novel malonic acid derivatives, processes for their preparation, their use as inhibitor of factor XA activity and pharmaceutical compositions containing them
08/29/2001EP1127119A1 Compounds and methods for modulating claudin-mediated functions
08/29/2001EP1127071A1 Compounds with growth hormone releasing properties
08/29/2001CN1310626A Hybrid polypeptides with enhanced pharmacokinetic properties
08/28/2001US6281380 From aspartyl-phenylalanine methyl ester
08/28/2001US6281376 Therapeutic compound—fatty acid conjugates
08/28/2001US6281352 Antiinflammatory agents
08/28/2001US6281247 Salt forms of (2E)-5-amino-5-methylhex-2-enoic acid N-methyl-N-((1R)-1-(N-methyl-N-((1R)-1-(methylcarbamoyl)-2-phenylethyl)carbamoyl)-2-(2-naphthyl)ethyl)amide
08/28/2001US6281194 E.g., (s)-(1-((4-benzyloxy-benzyl)-(((1-phenyl-cyclobutylmethyl)-car bamoyl)-methyl)-carbamoyl)-2-(1h-imidazol-4-yl)-ethyl)-carbami c acid benzyl ester
08/28/2001US6280760 Peptide-coated implants and methods for producing same
08/28/2001CA2017252C Retroviral protease inhibiting compounds
08/25/2001CA2337923A1 Peptide antibiotics
08/23/2001WO2001061017A2 Modified cytokines for use in cancer therapy
08/23/2001WO2001060848A2 Conjugates targeted to target receptors
08/23/2001WO2001060843A1 Trh-like peptide derivatives as inhibitors of the trh-degrading ectoenzyme
08/23/2001WO2001060842A2 PROCESS FOR MAKING GRANULATED N-[N-(3,3-DIMETHYLBUTYL)-L-α-ASPARTYL]-L-PHENYLALANINE 1-METHYL ESTER
08/23/2001WO2001060813A1 Beta-alanine derivatives and their use as receptor antagonists
08/23/2001WO2001060416A2 Matrix metalloproteinase inhibitors as targeting components in diagnostic agents
08/23/2001US20010016570 Bone disorders
08/23/2001DE10005932A1 Peptide und Verfahren zur Diagnostik von Zöliakie und Dermatitis Peptides and methods for the diagnosis of celiac disease and dermatitis
08/23/2001CA2400631A1 Beta-alanine derivatives and their use as receptor antagonists
08/23/2001CA2400627A1 Trh-like peptide derivatives as inhibitors of the trh-degrading ectoenzyme
08/23/2001CA2398395A1 Conjugates targeted to target receptors
08/23/2001CA2395038A1 Matrix metalloproteinase inhibitors
08/22/2001CN1309566A Nocathiacin antibiotics
08/21/2001US6278000 Growth-hormone secretagogues
08/21/2001US6277863 Anticoagulant with reduced side effects
08/21/2001US6277827 Stability makes the novel species suitable for milling, compression and improved bioavailability; 2s-(4-(2, 5-dioxopyrrolidin-1-yl)-2s-mercaptobutyrylamino)-4-methylpenta noic acid (2,2-dimethyl-1s-methylcarbamoylpropyl)amide
08/21/2001CA2060652C N-substituted cycloalkyl and polycycloalkyl alpha-substituted trp-phe- and phenethylamine derivatives
08/16/2001WO2001058957A2 Enhancing the circulating half-life of antibody-based fusion proteins
08/16/2001WO2001058932A1 Cytostatic agent glycoconjugate
08/16/2001WO2001058928A1 N-terminal d(-)-penicillamine peptides as aldehyde sequestration agents
08/16/2001WO2001058868A1 Method for synthesis of perindopril and its pharmaceutically acceptable salts
08/16/2001WO2001058852A2 (r)-2-aryl-propionamides, useful in the inhibition of il-8-induced chemiotaxis of neutrophils
08/16/2001WO2001058471A2 Novel amino acid and peptide inhibitors of staphylococcus virulence
08/16/2001WO2001010893A3 Il-16 antagonists
08/16/2001WO2001010891A3 Il-16 antagonists
08/16/2001WO2001009173A3 Use of quinic, shikimic acids and their derivatives for preparing mannose receptor ligands
08/16/2001WO2001007033A3 Neuroprotective pharmaceutical reparations comprising p-fluoroselegiline
08/16/2001EP1123410A1 The enzyme-mediated synthesis of peptidomimetics
08/16/2001EP1123309A2 Cyclic tetrapeptides and their use as histone deacetylase inhibitor
08/16/2001EP1123308A1 Single morphic forms of known peptide metalloproteinase inhibitors
08/16/2001EP1123272A1 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
08/16/2001EP1011668A4 1,2,5-thiadiazolidin-3-one 1,1-dioxide derivatives
08/16/2001EP0839153B1 Process of preparation of peptides and n-carbamoyl protected peptides
08/16/2001EP0837877B1 L-aspartyl-l-thienylalanine methyl esters, process for producing them and their use as sweeteners
08/16/2001EP0805817B1 Thiol derivatives with metallopeptidase inhibitory activity
08/15/2001CN1308078A Camptothecin derivative and its preparation
08/14/2001US6274705 Antithrombotic azacycloalkylalkanoyl peptides and pseudopeptides
08/14/2001US6274556 Administering polypeptide derivative to treat inflammatory bowel disease and to prevent leukocyte infiltration into tissues
08/14/2001US6274336 Producing three-dimensional structure of active site using computer program, displaying and superimposing three-dimensional representation of test compound onto active site, preparing test compound, and testing in biological assay
08/09/2001WO2001056591A1 vMIP-II PEPTIDE ANTAGONISTS OF CXCR4
08/09/2001WO2001056560A1 Substituted amino acids as neutral sphingomyelinase inhibitors
08/09/2001DE10005275A1 Neuartige Glycokonjugate Novel glycoconjugates
08/09/2001CA2399792A1 Substituted amino acids as neutral sphingomyelinase inhibitors
08/09/2001CA2369056A1 Vmip-ii peptide antagonists of cxcr4
08/08/2001EP1122262A1 Neovascular-specific peptides
08/08/2001EP1121431A1 Non-endogenous, constitutively activated human g protein-coupled receptors