Patents for C07D 515 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (877) |
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07/20/2010 | US7759345 ecteinascidins used for treating lung, colon, kidney, prostate, ovarian, breast and pancreatic cancers, leukaemia or melanoma |
06/24/2010 | WO2010071213A1 Resin composition containing cyclic carbodimide |
06/24/2010 | CA2745989A1 Resin composition comprising a cyclic carbodiimide |
06/23/2010 | CN101754970A Macrocyclic indole derivatives for the treatment of hepatitis c infections |
06/22/2010 | US7741325 Benzo[b]chromeno-naphthyridin-7-one and pyrano[2′,3′:7,8]quino[2,3-b]quinoxalin-7-one compounds |
06/15/2010 | US7737159 such as 2-(3-(aminomethyl)pyrrolidin-1-yl)-4-(4-methoxybenzyl)-7-oxo-4,7-dihydro[1,3]thiazolo[4,5-b]pyridine-6-carboxylic acid, used for treating drug-resistant bacterial infections |
06/09/2010 | CN101730692A Pyridazinone derivatives useful as glucan synthase inhibitors |
05/18/2010 | US7718669 Triazolopyridine derivatives as inhibitors of lipases and phospholipases |
05/14/2010 | WO2010017093A3 Dopamine receptor ligands with enhanced duration of action |
05/11/2010 | US7714133 alpha-(2-chlorophenyl)-6,7dihydrothieno[3,2-c]pyridine-5(4H)-acetic acid methyl ester (clopidogrel hydrogen sulphate); separating crystalline form out of a solution of clopidogrel in the form of the free base in a 2-propanol or n-butyl acetate solvent by adding sulphuric acid |
05/11/2010 | CA2503663C Novel quinoxalinone derivatives |
04/28/2010 | EP2178886A1 Macrocyclic indole derivatives for the treatment of hepatitis c infections |
04/28/2010 | EP2178885A1 Macrocyclic indole derivatives for the treatment of hepatitis c infections |
04/27/2010 | US7705014 e.g. 2-{4-[(3-hydroxy-4,7-dihydroisoxazolo[5,4-c]pyridin-6(5H)-yl)methyl]phenyl}-3-phenyl-1,6-naphthyridin-5(6H)-one; serine/threonine kinase (Akt) suppression; increased cellular potency or solubility, greater selectivity, enhanced pharmacokinetic properties, lack of off target activity; cancer |
04/06/2010 | US7691877 Pharmaceuticals |
04/01/2010 | WO2010037069A2 Dithienopyrrole dyes for imaging and therapy |
04/01/2010 | CA2738035A1 Dithienopyrrole dyes for imaging and therapy |
03/18/2010 | WO2010031054A1 Compositions and methods for treating epilepsy |
03/18/2010 | US20100069374 Tricyclic benzopyrane compound |
03/11/2010 | WO2010028116A1 Macrocyclics pyrimidines as aurora kinase inhibitors |
03/11/2010 | WO2010027567A2 Tricyclic spirocycle derivatives and methods of use thereof |
03/11/2010 | CA2735420A1 Macrocyclic pyrimidines as protein kinase inhibitors |
03/02/2010 | US7671068 N-(alkoxyalkyl) carbamoyl-substituted 6-phenyl-benzonaphthyridine derivatives and their use as PDE ¾ inhibitors |
02/23/2010 | US7666879 enzyme inhibitor; 2-{2-Fluoro-4-[7-(2-methyl-pyridin-4-yl)-imidazo[1,2-a]pyridin-3-yl]-phenyl}-N-(3-trifluoromethyl-phenyl)-acetamide; angiogenesis inhibitor; antitumor agent; treating hyperglycemia, psoriasis, rheumatoid arthritis, Kaposi's sarcoma, autoimmune diseases, inflammation, and eye disorders |
02/23/2010 | US7666876 Buprenorphine formulations for intranasal delivery |
02/18/2010 | WO2010018233A1 Macrocyclic indole derivatives useful as hepatitis c virus inhibitors |
02/18/2010 | CA2733762A1 Macrocyclic indole derivatives useful as hepatitis c virus inhibitors |
02/16/2010 | CA2406095C Synthetic process for the manufacture of an ecteinaschidin compound |
02/11/2010 | WO2010017093A2 Dopamine receptor ligands with enhanced duration of action |
01/26/2010 | US7652010 Azabicyclic aryl derivatives and their medical use |
01/26/2010 | US7652008 Tricyclic benzopyran compound as anti-arrhythmic agents |
01/21/2010 | WO2009069147A4 Improved process for preparation of triazol-benzodiazepine derivatives |
01/14/2010 | WO2010003658A1 Macrocyclic indole derivatives useful as hepatitis c virus inhibitors |
01/14/2010 | CA2729307A1 Macrocyclic indole derivatives useful as hepatitis c virus inhibitors |
01/12/2010 | US7645766 Method for treatment of depression and depressive mood disorders |
01/05/2010 | US7642247 1,3,5-triazines for treatment of viral diseases |
12/31/2009 | US20090326221 New oxabispidine compunds useful in the treatment of cardiac arrhythmias |
12/24/2009 | US20090318412 Tricyclic heterocyclic compound and use thereof |
12/22/2009 | US7635394 Composition for the dyeing of keratin fibers comprising at least one 3-amino-pyrazolopyridine derivatives |
12/03/2009 | WO2009069147A3 Improved process for preparation of triazol-benzodiazepine derivatives |
12/01/2009 | US7625924 Nicotinic alpha-7 receptor ligands and preparation and uses thereof |
12/01/2009 | US7625892 Pharmaceutical compositions for the treatment of diseases related to neurotrophines |
10/21/2009 | CN101563352A Antiviral indoles |
10/14/2009 | CN100548988C Metabolites of ecteinascidin 743 |
10/14/2009 | CN100548296C Mitotic kinesin inhibitors |
10/06/2009 | US7598389 Silylated carboxamides |
10/06/2009 | US7598254 Substituted 1,3-thiazolo[5,4-d]pyrimidines as xanthine oxidase inhibitors |
10/06/2009 | US7598237 7-aryl 1,5-dihydro-4,1-benzoxazepin-2(3H)-one derivatives and their use as progesterone receptor modulators |
10/01/2009 | US20090247533 Ecteinascidins |
09/29/2009 | US7595400 Synthesis of antitumor agents including camptothecin derivative 9-ethyl-9-hydroxy-1-pentyl-1H,12H-pyrano[3'',4'':6',7']-indolizino[1',2':6,5]pyrido[4,3,2-de]quinazoline-10,13(9H,15H)-dione |
09/01/2009 | US7582652 Kinase inhibitors |
08/25/2009 | US7579472 Efficient synthesis of 4,5-dihydro-pyrazolo[3,4-c]pyrid-2-ones |
08/25/2009 | US7579360 Triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors |
08/25/2009 | US7578856 [2-(3-Aminopyrazolo[1,5-a]pyridin-2-ylamino)ethyl]tri-;methylammonium salt; for keratinous fibers, hair; for multi-compartment devices |
08/18/2009 | US7576198 A hydroxy compound containing substituted orpyridine, pyrazine, pyrimidine, oxazole, thiadiazole, quinoline, isoquinoline etc. as anti HIV agent, for treating AIDS |
08/12/2009 | CN101506199A Azetidine compounds as orexin receptor antagonists |
08/06/2009 | US20090198051 Chemical intermediates for sulfiding under mild conditions forming ring compounds for use as marine alkaloids; connecting reaction of 4 components, transforming c22-tert-butyltriphenylsilyl to acety group, cyclization, hydroxy group to methanesulonyl group, reduction of amide, dehydration,Heck reaction |
08/05/2009 | EP1805144A4 Heterocyclical chromophore architectures |
07/30/2009 | WO2009093009A1 Fused tricyclic thiophene derivatives as mek inhibitors |
07/28/2009 | US7566707 For example, 2-[3-(Tert-butyloxycarbonylamino)-piperidin-1-yl]-3-(2-butyn-1-yl)-5-[(dibenzo[b,f][1,4]-oxazepin-11-yl)methyl]-3,5-dihydro-imidazo[4,5-d]pyridazin-4-one; inhibiting effect on activity of the enzyme dipeptidylpeptidase-IV; use in treatment of diabetes mellitus, arthritis, obesity |
07/22/2009 | EP2079704A2 Therapeutic compounds |
07/07/2009 | US7557121 Tetrahydronaphthyridine derivatives |
07/07/2009 | US7557114 Heterocyclic-substituted phenyl methanones |
06/25/2009 | US20090163507 Synthesis of naturally occuring ecteinascidins and related compounds |
06/17/2009 | EP2069332A2 Azetidine compounds as orexin receptor antagonists |
06/16/2009 | US7547782 Met kinase inhibitors |
06/16/2009 | US7547709 Prevent free radical cellular damage; oxidation resistant additive for fuels, lubricants, rubbers, polymers, solvents, chemical and foodstuff; lipid and water soluble vitamin c, vitamin e |
06/09/2009 | US7544697 Pyrazolopyridines and analogs thereof |
06/02/2009 | US7541367 3-benzoimidazolyl-pyrazolopyridines useful in treating kinase disorders |
05/28/2009 | US20090137597 Novel quinoxalinone derivatives |
05/13/2009 | CN101429200A Tricyclic benzopyran compound as anti-arrhythmic agents |
05/05/2009 | US7528148 Pyrazolo[3,4-B]pyridine compounds, and their use as phosphodiesterase inhibitors |
05/05/2009 | US7528147 e.g. 2 {5,6-dimethoxy-1-[2-(4-methylpiperazin- 1 -yl)ethyl]-1H-indol-3 -yl}-1H-pyrrolo[2,3- b]pyridine; Insulin Growth Factor-1 (somatomedin) antagonist; antiproliferative, antitumor agent; solid tumor; prostate, lung and breast cancer |
04/30/2009 | WO2008140420A3 Pyrimidine derivatives |
04/28/2009 | US7524956 Hemisynthetic method and new compounds |
04/28/2009 | US7524864 Methods of treating sleep disorders |
04/28/2009 | US7524860 Antibacterial agents |
04/23/2009 | WO2009052288A1 Spiro-condensed 1, 3, 4-thiadiazole derivatives for inhibiting ksp kinesin activity |
04/23/2009 | CA2702922A1 Spiro-condensed 1,3,4-thiadiazole derivatives for inhibiting ksp kinesin activity |
04/21/2009 | US7521460 e.g. 3-[(2,4-Difluorophenyl)amino]-2-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]carbonyl}-7-phenylthieno[2,3-b]pyridin-6(7H)-one; autoimmune, neurodegenerative disorders, antiinflammatory agent; p38 MAP kinase inhibitor |
04/15/2009 | CN100477993C Compositions and uses of et743 for treating cancer |
04/08/2009 | CN100475822C Synthesis method for producing ecteinascidin compound |
04/07/2009 | US7514448 Azaindoles useful as inhibitors of rock and other protein kinases |
04/01/2009 | CN101400684A Thiazole compound |
03/31/2009 | US7511057 Triazolopyridinylsulfanyl derivatives as p38 MAP kinase inhibitors |
03/24/2009 | US7507746 Enantiomer of tenatoprazole and the use thereof in therapy |
03/19/2009 | US20090076017 Deuterium-enriched trabectedin |
03/17/2009 | US7504412 Melanin concentrating hormone receptor antagonists; such as n-(2-cyclopropyl-3-methylimidazo[1,2-a]-pyridin-6-yl)-4-(2-pyridyl)benzamide; central nervous system, cardiovascular and metabolic disorders; synthesis |
03/17/2009 | US7504390 Benzoxazepine derivatives and their use as AMPA receptor stimulators |
03/10/2009 | US7501438 1-(3-naphthalen-1-yl-imidazo[1,5-a]pyridin-1-yl)-butan-1-one; chronic pain, an inflammatory disorder, rheumatoid arthritis, multiple sclerosis, osteoporosis and osteoarthritis; cannabinoid receptor ligands |
03/03/2009 | US7498342 Compounds modulating c-kit activity |
02/24/2009 | US7495009 Imidazopyridine derivatives as melancortin receptor agonists |
02/24/2009 | US7494991 For microbial infections specially Gram-positive bacterial infection; atherosclerosis-associated disease |
02/19/2009 | WO2007095389A3 Treatment of hyperproliferative diseases with camptothecine n-oxide and analogs |
02/05/2009 | US20090036673 Ecteinascidin 743; 5-(1,2-diaminoethyl-), 3,4-methylenedioxyphenol intermediate, of which the amine group cyclizes |
01/27/2009 | US7482452 intermediates for p38 MAP kinase inhibitors; industrial scale; 3-cyano-6-oxo-2-thio-1,6-dihydropyridines or pyrimidine, 2,4-diones as starting reactants and 2-cyano-N-phenylthioacetamide; cyclization; diazotization of 3-amino-7H-thieno[2,3-b]pyridin-6-ones, halide displacement |
01/27/2009 | US7482338 Non-amide nonanes |
01/22/2009 | WO2009010785A1 Macrocyclic indole derivatives for the treatment of hepatitis c infections |
01/22/2009 | WO2009010783A1 Macrocyclic indole derivatives for the treatment of hepatitis c infections |
01/22/2009 | CA2693537A1 Macrocyclic indole derivatives for the treatment of hepatitis c infections |