Patents
Patents for C07D 513 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (15,120)
01/2002
01/23/2002EP1049744B1 Asymmetric cyanine dye quenchers
01/23/2002EP0711292B1 Aza spiro compounds acting on the cholinergic system with muscarinic agonist activity
01/23/2002CN1332743A Cell adhesion-inhibiting antinflammatory compounds
01/22/2002US6340752 Cleavage of thio group from carbonyl and conversion to lactam ester
01/22/2002US6340683 Selective NPY (Y5) antagonists (triazines)
01/17/2002WO2002004444A2 Heterocycle carboxamides as antiviral agents
01/17/2002WO2002004409A2 Tetrahydrobenzothiazole analogues as neuroprotective agents
01/17/2002US20020006944 Anticoagulants
01/17/2002US20020006941 p53 inhibitors and therapeutic use of the same
01/17/2002US20020006921 Dopaminergic agent
01/17/2002CA2415815A1 Tetrahydrobenzothiazole analogues as neuroprotective agents
01/16/2002EP1171442A1 Xanthine derivatives and analogs as cell signalling inhibitors
01/16/2002EP1171122A1 Pyrrolidine modulators of chemokine receptor activity
01/16/2002CN1331690A 4-(caminomethyl)-piperidine benzamides for treating gastrointestinal disorders
01/16/2002CN1331591A Piperidines as CCR5 modulators
01/16/2002CN1077886C Amidino derivatives useful as nitric oxide synthase inhibitors
01/15/2002CA2039826C Spiro bridged and unbridged heterocyclic compounds
01/10/2002WO2002002562A2 Heteropolycyclic inhibitors
01/10/2002WO2002002549A1 Tetrahydropyridino or piperidino heterocyclic derivatives
01/10/2002WO2002002512A2 Compounds to treat alzheimer's disease
01/10/2002WO2001036425A3 Imidazole compounds used as phosphodiesterase vii inhibitors
01/10/2002US20020004501 Therapy for muscular disorders, urogenital disorders, gastrointestinal disorders, respiratory system disorders
01/10/2002US20020004500 Drug mixture for cardiovascular disorders
01/10/2002DE10019714A1 Salze von bicyclischen, N-acylierten Imidazo-3-aminen und Imidazo-5-aminen Salts of bicyclic, N-acylated imidazo-3-amines and imidazo-5-amines
01/10/2002CA2414885A1 Heteropolycyclic inhibitors
01/10/2002CA2412287A1 Tetrahydropyridino or piperidino heterocyclic derivatives
01/10/2002CA2410651A1 Compounds to treat alzheimer's disease
01/09/2002EP1170273A1 Alkynic compounds, their use as monomers in vacuum deposition polymerisation, thin films formed from these polymers and their use in electroluminescent devices
01/09/2002CN1330655A Fused 1,2,4-thiadiazine derivatives, their preparation and use
01/09/2002CN1330654A 4,5-pyrrolo-oxindoles
01/08/2002US6337395 Selenium derivatives of porphryn
01/03/2002WO2002000658A1 Cyclic gmp-specific phosphodiesterase inhibitors
01/03/2002WO2002000612A1 Glucagon antagonists/inverse agonists
01/03/2002WO2002000223A1 Use of potassium channel agonists for reducing fat food comsumption
01/03/2002WO2002000222A1 Use of potassium channel agonists for the treatment of cancer
01/03/2002WO2001044247A3 Agents and methods for the treatment of proliferative diseases
01/03/2002US20020002173 E. g., 6-(3-chlorophenyl)-1,4-dihydro-4,4-dimethyl-2H-thieno-(2,3-d)(1,3)oxazine-2 -one; agonists and antagonists of the progesterone receptor; inducing contraception and treating or preventing benign or malignant neoplastic diseases
01/03/2002US20020002165 Growth hormone secretagogues useful for treatment/prevention of osteoporosis
01/03/2002CA2411552A1 Glucagon antagonists/inverse agonists
01/02/2002EP1167373A1 Ferrocenyldiphosphine-ruthenium complexes and a hydrogenation process of exocyclic double bond of d-thiophene to d-thiophane
01/02/2002EP1167369A1 Novel thiazolobenzimidazole derivatives
01/02/2002EP1165566A1 Pyridine and pyrimidine derivatives and their use as inhibitors of cytokine mediated disease
01/02/2002EP1165563A1 Bicyclic heterocycles, method for producing them and their use as herbicides and pharmaceutical agents
01/02/2002EP1165545A1 Novel compounds
01/02/2002EP1165532A1 Antibacterial agents
01/02/2002EP1165514A1 3-(anilinomethylene) oxindoles as protein tyrosine kinase and protein serine/threonine kinase inhibitors
01/02/2002EP0912553B1 BENZO[g]QUINOLINE DERIVATIVES
01/02/2002CN1329601A New benzimidazolone-benzoxazolone-, or benzothiazolone derivatives as ion channel modulating agents
01/02/2002CN1328824A Compound for curing female sexual disorder
12/2001
12/27/2001WO2001057042A3 4-pyridyl-and 2,4-pyrimidinyl-substituted pyrrole derivatives and their use in pharmacy
12/26/2001CN1328455A Use of N-substituted azabicycloalkane derivatives for treating diseases of central nervous system
12/25/2001US6333296 Diaryl ethers and processes for their preparation and herbicidal and desiccant compositions containing them
12/25/2001CA2209313C Heterocycle-fused thiazole derivatives
12/20/2001US20010053783 Central nervous system disorders
12/19/2001EP1164128A1 4-Cyanophenyliminoheterocycles
12/19/2001EP1163233A1 Fused 1,4-thiazine-2-carbonitrile derivatives, their preparation and use
12/19/2001EP0983063B1 Pharmaceutical composition containing uscharin
12/18/2001US6331623 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha-1-blocking action
12/18/2001US6331507 Substituted aromatic thiocarboxylic acid amides and their use as herbicides
12/13/2001WO2001025241A3 Fused 1-(2,6-dichloro-4-trifluoromethylphenyl)-pyrazoles, the synthesis thereof and the use thereof as pesticides
12/13/2001US20010051620 Tricyclic protein kinase inhibitors
12/13/2001DE10101324C1 New 1-(dimercaptoalkyl)-quinazoline-2,4(1H,3H)-diones, are stable matrix metalloproteinase inhibitors useful e.g. for treating rheumatism, tumor metastasis or sunburn
12/12/2001EP1161233A2 Lxr modulators
12/12/2001CN1326473A Supported group 8-10 transition metal olefin polymerization catalysts
12/11/2001US6329542 Preparation of (S)-2-amino-6,6-dimethoxyhexanoic acid methyl ester via novel dioxolanes
12/11/2001US6329375 Tricyclic quinoxaline derivatives as protein tyrosine kinase inhibitors
12/11/2001US6329367 Nervous system disorders and cardiovascular disorders
12/06/2001WO2001036426B1 Pyridinones to treat and prevent bacterial infections
12/05/2001EP1159280A2 Thiazoloindolinone compounds
12/05/2001EP0605493B1 THIADIAZOLO (4,3-a)PYRIDINE DERIVATIVES, METHODS OF PREPARING THEM AND DRUGS CONTAINING THEM
12/05/2001CN1325309A Compounds, compositions and method for treating or preventing viral infections and associated diseases
12/04/2001US6326378 Use of thiadiazolo[4,3-a]pyridine derivatives
11/2001
11/29/2001WO2001090101A1 Arylmethylamine derivatives for use as tryptase inhibitors
11/29/2001WO2001090094A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
11/29/2001WO2001090093A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
11/29/2001WO2001090092A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
11/29/2001WO2001090091A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
11/29/2001WO2001090090A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
11/29/2001WO2001090081A1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists
11/29/2001WO2001089526A1 Inhibition of inflammatory cytokine production by cholinergic agonists and vagus nerve stimulation
11/29/2001WO2000055159A3 Substituted aza-oxindole derivatives
11/29/2001US20010046989 Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and TACE inhibitors
11/29/2001CA2408791A1 Inhibition of inflammatory cytokine production by cholinergic agonists and vagus nerve stimulation
11/29/2001CA2408783A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
11/28/2001EP1157024A1 Acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as tace inhibitors
11/28/2001EP1157013A1 Polycyclic thiazole-2-ylides amines, method for the production thereof and their utilization as medicaments
11/28/2001EP0914129B1 Use of aspirochlorine or derivatives thereof as immunosuppressive agents
11/27/2001US6323201 Compounds for inhibition of ceramide-mediated signal transduction
11/27/2001US6323200 The compounds are immunomodulators and induce cytokine biosynthesis, including interferon and/or tumor biosynthesis, necrosis factor, and inhibit the t-helper-type 2 immune response.
11/27/2001US6323038 Diagnostic reagent for complications associated with diabetes or renal failure
11/22/2001WO2001087892A1 Crf receptor antagonists
11/22/2001WO2001087886A1 Crf receptor antagonists and methods relating thereto
11/22/2001WO2001087883A1 Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity
11/22/2001WO2001087844A1 Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity
11/22/2001WO2001030781A3 INHIBITORS OF αLβ2 MEDIATED CELL ADHESION
11/22/2001US20010044539 (2S,3Z)-2-amino-5-(6,7,8,9-tetrahydro-3-oxo-3H,5H -(1,2,4)oxadiazolo(4,3-a)azepin-5-yl)-3-pentenoic acid, for example
11/21/2001EP1156050A2 Substituted tricyclics useful in sPLA2 induced diseases
11/21/2001EP1155010A1 Acetamido acetonitrile derivatives as inhibitors of cathepsin l and/or cathepsin s
11/21/2001EP1154992A1 N-substituted arylsulfonylamino hydroxamic acids useful as inhibitors of c-proteinase and for treating or preventing disorders related to unregulated collagen production
11/21/2001EP0745081B1 indane-2-mercaptoacetylamide disulfide derivatives useful as inhibitors of enkephalinase