| Patents for C07D 513 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (15,120) |
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| 08/02/2000 | EP1023265A1 Azetidinone derivatives for the treatment of hcmv infections |
| 08/02/2000 | CN1055089C Intermediate of protein kinase C inhibitor and its preparation |
| 08/01/2000 | US6096763 Administering to the patients a2-oxo-1-benzimidazolinyl)piperidin-1-yl)alkyl)-1,2benzisothia zol-3-(2h)-one derivative as alpha-1a adrenergic receptor antagonist |
| 08/01/2000 | US6096755 N-substituted azabicycloalkane derivatives, their preparation and use |
| 08/01/2000 | US6096724 O(6)-alkylguanine-dna alkyltransferase (atase) enzyme inhibitors |
| 07/27/2000 | WO2000043398A2 Tricyclic benzodiazepines as vasopressin receptor antagonists |
| 07/27/2000 | WO2000043375A2 Substituted aryl heterocyclic compounds |
| 07/26/2000 | EP1022278A1 Tetracyclical derivatives from pyrimidine |
| 07/26/2000 | EP1021413A1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors |
| 07/26/2000 | EP1021173A1 Use of csaid?tm compounds for the management of uterine contractions |
| 07/26/2000 | CN1261366A Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha-1-blocking action |
| 07/25/2000 | US6093738 Imidazo(1,2-d)-thiadiazole compounds; peptic ulcer treatment |
| 07/25/2000 | US6093732 4-hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents |
| 07/25/2000 | US6093710 Benzothiophene derivatives, their preparation and use as urokinase inhibitors |
| 07/25/2000 | US6093709 Administering a therapeutic beta isozyme of protein kinase c inhibitor for inducing smooth muscle relaxation and vasodilation |
| 07/20/2000 | WO2000042031A2 Substituted 2-arylimino heterocycles and compositions containing them, for use as progesterone receptor binding agents |
| 07/20/2000 | DE19901846A1 New aryl-substituted aza-heterocyclic compounds, useful as pre- or post-emergence, total or selective herbicides, show defoliant, dessicant and especially weed-killing activity |
| 07/20/2000 | CA2359562A1 Substituted 2-arylimino heterocycles and compositions containing them, for use as progesterone receptor binding agents |
| 07/19/2000 | EP1020467A1 N-acylamino acid amide compounds and intermediates for preparation thereof |
| 07/19/2000 | EP1020448A2 Arylheterocycles with herbicidal activity |
| 07/19/2000 | EP1019408A1 1,2,3,4-TETRAHYDRO-BENZOFURO 3,2-c]PYRIDINE DERIVATIVES-- |
| 07/19/2000 | CN1260798A Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha 1-blocking action |
| 07/13/2000 | WO2000040228A2 Formulations comprising imiquimod or other immune response modifiers for treating mucosal conditions |
| 07/13/2000 | WO2000006597A9 Endogenous constitutively activated g protein-coupled orphan receptors |
| 07/12/2000 | EP1018514A1 NF-$g(k)B INHIBITORS CONTAINING INDAN DERIVATIVES AS THE ACTIVE INGREDIENT |
| 07/12/2000 | EP1017700A1 Macrocyclic porphyrazine-type compounds, metal derivatives thereof and process for their preparation |
| 07/12/2000 | EP1017695A1 Resolution of optically-active compounds |
| 07/12/2000 | EP0877734B1 Quinoline and quinazoline compounds useful in therapy |
| 07/12/2000 | EP0573659B1 Pyrazolothiazolopyrimidine derivative |
| 07/12/2000 | CN1259942A Novel guanidine mimics as factor Xa inhibitors |
| 07/12/2000 | CN1054377C New bicyclic derivatives of imidazole and their prepn. process, their use as medicaments and the pharmaceutical compositions containing them |
| 07/11/2000 | US6087380 Antithrombotic benzimidazoles; anticoagulants; 2-(n-(4-amidinophenyl)-aminomethyl)-benzimidazol-5-yl-carboxylic acids |
| 07/06/2000 | WO2000039108A1 Thrombin or factor xa inhibitors |
| 07/06/2000 | WO2000039102A1 THROMBIN OR FACTOR Xa INHIBITORS |
| 07/06/2000 | WO2000038683A1 THROMBIN OR FACTOR Xa INHIBITORS |
| 07/06/2000 | WO2000038680A1 Azabicycloalkanes as ccr5 modulators |
| 07/06/2000 | CA2349557A1 Thrombin or factor xa inhibitors |
| 07/06/2000 | CA2348740A1 Thrombin or factor xa inhibitors |
| 07/06/2000 | CA2320730A1 Thrombin or factor xa inhibitors |
| 07/05/2000 | EP1015479A1 Combinatorial libraries of peptidomimetic macrocycles and processes therefor |
| 07/05/2000 | EP1015451A1 Tetrahydro gamma-carbolines |
| 07/05/2000 | EP1015439A1 Prenyl transferase inhibitors |
| 07/05/2000 | EP1015434A2 Novel pyrimidin-4-one and pyrimidin-4-thione as fungicide |
| 07/05/2000 | CN1259132A Compounds |
| 07/04/2000 | US6084095 Including 6-amino-4-(3-bromoanilino)pyrido(3,2-d)pyrimidine; 4-(3-bromoanilino)-6-methylaminopyrido (3,2-d)pyrimidine; and 4-(3-bromoanilino)-6-methylaminopyrido(3,2-d)pyrimidine; useful in treating proliferative diseases such as cancer |
| 07/04/2000 | CA1341043C Piperazinyl derivatives of purines and isosteres thereof as hypoglycemic agents |
| 06/29/2000 | WO2000037474A1 Fused 1,2,4-thiadiazine derivatives, their preparation and use |
| 06/29/2000 | WO2000037461A1 4-(aminomethyl)-piperidine benzamides for treating gastrointestinal disorders |
| 06/29/2000 | WO2000037021A2 Products comprising trihydroxystilbenes and derivatives thereof and methods for their manufacture and use |
| 06/29/2000 | CA2394949A1 Products comprising trihydroxystilbenes and derivatives thereof and methods for their manufacture and use |
| 06/29/2000 | CA2353907A1 Fused 1,2,4-thiadiazine derivatives, their preparation and use |
| 06/28/2000 | EP1012145A1 Alkoxy-substituted compounds, methods, and compositions for inhibiting parp activity |
| 06/28/2000 | CN1258283A Cyclic diamine compounds and medicine contg. same |
| 06/28/2000 | CN1053908C Substd. thiazolo [3,2-a] azepine deriv. |
| 06/28/2000 | CN1053905C Oxadiazine derivs., their preparing process and use, intermediates for preparing same |
| 06/27/2000 | US6080868 As a quencher in a reporter-quencher energy-transfer dye pair for nucleic acid hybridization assays |
| 06/27/2000 | US6080855 2-isocephem and oxacephem derivatives and use as antibacterial agents |
| 06/27/2000 | US6080771 DC107 derivatives |
| 06/27/2000 | US6080764 Superoxide radical inhibitor |
| 06/22/2000 | WO2000035920A2 4,5-azolo-oxindoles |
| 06/21/2000 | EP1009739A2 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity |
| 06/21/2000 | EP1009738A1 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors |
| 06/20/2000 | US6077813 Substituted aromatic thiocarboxylic acid amides and their use as herbicides |
| 06/20/2000 | US6077812 Cycloimido-substituted benzofused heterocyclic herbicides |
| 06/20/2000 | CA1341035C Macrocyclic polyaza compounds containing 5 or 6 membered rings, process for producing them and pharmaceutical media containing them. |
| 06/15/2000 | WO2000034248A1 New benzimidazolone-, benzoxazolone-, or benzothiazolone derivatives as ion channel modulating agents |
| 06/15/2000 | CA2349616A1 New benzimidazolone-, benzoxazolone-, or benzothiazolone derivatives as ion channel modulating agents |
| 06/14/2000 | EP1007525A1 Aminometyl oxooxazolidinyl benzene derivatives |
| 06/14/2000 | CN1053448C Compound useful as antiproliferative agents and GARFT inhibitors |
| 06/13/2000 | US6075034 Spiro[piperidine-4,1'-pyrrolo [3,4-C] pyrrole]derivatives |
| 06/13/2000 | CA2014062C Pyridine derivatives |
| 06/07/2000 | EP1005468A1 Antibiotic oxazolidinone derivatives |
| 06/06/2000 | US6071906 Inhibits or modulates the inducible isoform of nitric oxide synthase over the the constitutive isoforms; antiarthritic, -diabetic, ischemic, thrombosis agents; cardiovascular disorders; toxic shock syndrome; autoimmune diseases |
| 06/06/2000 | US6071905 Treating tuberculosis, mycobacteriosis, viral and immune diseases, chlamydia infections, antitumor and -carcinogenic agents; microbiocides, in particular to mycobacteria resistant to isoniazide; stimulantes interferons |
| 06/02/2000 | WO2000031247A2 Recombinant methods and materials for producing epothilone and epothilone derivatives |
| 06/02/2000 | WO2000030639A1 Use of n-substituted azabicycloalkane derivatives for treating diseases of the central nervous system |
| 06/02/2000 | CA2352526A1 Use of n-substituted azabicycloalkane derivatives for treating diseases of the central nervous system |
| 06/02/2000 | CA2350189A1 Recombinant methods and materials for producing epothilone and epothilone derivatives |
| 05/31/2000 | EP1003751A1 Hydroxamic acid substituted fused heterocyclic metalloproteinase inhibitors |
| 05/31/2000 | EP1003721A1 Benzylidene-1,3-dihydro-indol-2-one derivatives as receptor tyrosine kinase inhibitors, particularly of raf kinases |
| 05/31/2000 | CN1255136A Substituted 4-arylmethylene-2-imino-2,3-dihydrothiazoles and derivatives and their pharmaceutical use |
| 05/31/2000 | CN1255042A Diaryl ethers and processes for their preparation and herbicidal and desiccant compositions containing them |
| 05/30/2000 | US6069144 N-heterocyclic compounds, intermediate products used to prepare them, agents containing them and their use in antifungal applications |
| 05/25/2000 | DE19854147A1 Control of cocaine addiction comprises administration of N-substituted azabicycloalkane derivative |
| 05/24/2000 | EP1001970A1 Dipeptide derivatives as growth hormone secretagogues |
| 05/24/2000 | EP1001782A1 5,6-HETEROARYL-DIPYRIDO 2,3-$i(b):3',2'-$i(f)]AZEPINES AND THEIR USE IN THE PREVENTION OR TREATMENT OF HIV INFECTION |
| 05/23/2000 | US6066658 For prevention and treatment of bone diseases such as osteoporosis, bone fractures, osteoarthritis and rheumatoid arthritis, arteriosclerosis, cancer metastasis, and diseases based on nerve degeneration |
| 05/23/2000 | US6066646 Insecticidal, acaricidal or nematicidal composition |
| 05/18/2000 | WO2000027852A1 Novel imidazo[5,1-b]thiazole derivatives and fungicides containing the same as the active ingredient |
| 05/18/2000 | WO2000027851A1 Novel type condensed pyridazinone compounds |
| 05/18/2000 | WO2000006597A3 Endogenous constitutively activated g protein-coupled orphan receptors |
| 05/17/2000 | EP1000946A2 Pesticidal and parasiticidal use of 2-(substituted thio)thiazolo-[4,5-b]pyridine compounds |
| 05/17/2000 | EP1000067A1 Thiazolobenzoheterocycles, preparation and medicines containing same |
| 05/17/2000 | EP1000066A1 Fused 1,2,4-thiadiazine derivatives, their preparation and use |
| 05/17/2000 | EP1000040A1 Il-5 inhibiting 6-azauracil derivatives |
| 05/17/2000 | EP1000028A1 Gastrokinetic monocyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives |
| 05/17/2000 | CN1253547A 1,4-substituted cyclic amine derivatives |
| 05/16/2000 | US6063918 Reacting a base with a 2-azetidinyl-3,4-dihalogeno-2-butenoic acid compound in an aqueous organic solvent to yield a cyclized isooxacephalosporin derivative; simplification |
| 05/16/2000 | CA2289363A1 Pesticidal and parasiticidal use of 2-(substituted thio) thiazolo-[4,5-b] pyridine compounds |
| 05/16/2000 | CA2011658C New 1,7-annelated 1h-indole-2-carboxylic acid-n-(1,4-benzodiazepin-3-yl) amides |