Patents
Patents for C07D 513 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (15,120)
03/2003
03/18/2003US6534506 Inhibitors of prenyl-protein transferase
03/18/2003US6534491 Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
03/13/2003US20030050300 Therapeutic 5-HT ligand compounds
03/12/2003EP1289965A1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists
03/12/2003EP0672031B1 Catechol diethers as selective pde iv inhibitors
03/12/2003CN1402730A Thiazolo (4,5-D) pyrimidine compounds
03/12/2003CN1402727A Bicyclic imidazo-3-yl-amine derivs. which are substd. on sixth ring
03/12/2003CN1402726A Bicyclic imidazo-5-yl-amine derivs.
03/11/2003US6531487 Water solubility; bioavailability
03/11/2003US6531484 Viricides for preventing infection by HIV, treating infection by HIV, delaying of the onset of AIDS, or treating AIDS
03/07/2003WO2002020531A2 Method for producing anellated tetrahydro-[1h]-triazoles
03/07/2003CA2421839A1 Method for producing anellated tetrahydro-[1h]-triazoles
03/06/2003WO2003018587A1 Helix mimetics and composition and methods related thereto
03/06/2003WO2002055507A8 1-dimercaptoalkylquinazolin-2,4(1h,3h)-diones as matrix metalloproteinase (mmp) inhibitors
03/06/2003US20030045545 Immunomodulators, induce cytokine biosynthesis, and antineoplastic agents
03/05/2003EP1287002A1 Crf receptor antagonists
03/05/2003EP1286994A1 Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity
03/05/2003EP0690863B1 Tetracyclic compounds as dopamine agonists
03/05/2003CN1400973A Novel biarylcarboxamides
03/05/2003CN1102596C 5H-thiazole [3,2-a] pyrmidine derivatives
03/05/2003CN1102595C Penems and their derivatives
03/05/2003CN1102593C N-[4(heteroarylmethyl)phenyl]-heteroarylamines compound
02/2003
02/27/2003WO2003016302A1 Diamine derivatives
02/27/2003WO2003016248A2 Bicyclic hydroxamates as inhibitors of matrix metalloproteinases and/or tnf-$g(a) converting enzyme (tace)
02/27/2003WO2003016245A1 Chromatographic separation of enantiomers of protected amino acids via smb-method
02/27/2003WO2003015773A2 2-amino-4,5-trisubstituted thiazolyl derivatives and their use against autoimmune diseases
02/27/2003WO2002089749A3 Arylsulfonamide ethers, and methods of use thereof
02/27/2003WO2002028865A3 Condensed pyridoindole derivatives
02/27/2003CA2456841A1 Cyclohexyl and piperidine diamine derivatives useful as activated blood coagulation factor x inhibitors
02/26/2003CN1399639A New oxabispidine compound useful in treatment of cardiac arrhythmias
02/25/2003US6525070 Bipiperidine derivatives as modulators of CCR3 activity and as H1 antagonists
02/25/2003US6525047 Which are growth hormone secretogogues and increase the level of endogenous growth hormone; treating osteoporosis, congestive heart failure, frailty associated with aging, obesity; accelerating bone fracture repair
02/25/2003US6525045 Positive allosteric AMPA receptor modulators
02/25/2003US6525042 Sulfonyl derivatives
02/25/2003US6525000 N-aminoureas are reacted with formaldehyde to give methyleneimino ureas, cyclizing these to give tetrahydro-4H-1,3,4-oxa(or thia)diazines, and cyclizing the fused triazoles using phosgene; herbicides
02/20/2003WO2003014125A1 Therapeutically useful tetracyclic ligands
02/20/2003WO2003014121A1 Compounds, derivatives, compositions, preparation and uses
02/20/2003WO2002072585A3 Substituted pyrazolopyrimidines and thiazolopyrimidines used as analgesics
02/20/2003WO2001079187A8 Substituted 1,4-thiazepine and analogs and their use as activators of caspases
02/20/2003US20030036543 Especially as inhibitors of Aurora-2 and GSK-3, for treating diseases such as cancer, diabetes and Alzheimer's disease.
02/20/2003CA2453219A1 Therapeutically useful tetracyclic ligands
02/19/2003EP1283834A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
02/19/2003EP1283833A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
02/19/2003EP1283832A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
02/19/2003EP1283831A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
02/18/2003US6521620 Suppressing tumors, especially breast cancers; antiproli-ferative agents; arthritis, vascular restenosis, psoriasis and angiogenesis; extremely low cytotoxicity
02/13/2003WO2003011870A1 Gonadotropin-releasing hormone receptor antagonists
02/13/2003WO2003011824A1 Bicyclic modulators of androgen receptor function
02/13/2003WO2003011286A1 Core modified porphyrins
02/13/2003WO2003011222A2 Thrombin inhibitors
02/13/2003US20030032652 Hydroxamic and carboxylic acid derivatives
02/13/2003US20030032647 Aromatic nitrogen-containing 6-membered cyclic compounds
02/13/2003US20030032642 Treating psoriasis, a disease in which angiogenesis is associated with raised CXCR2 chemokine levels, or COPD.
02/12/2003EP1282622A1 Crf receptor antagonists and methods relating thereto
02/12/2003EP0828488B1 Isothiazolones
02/12/2003CN1396923A 4-Pyridyl-and 2,4-pyrimidinyl-substituted pyrrole derivatives and their use in pharmacy
02/11/2003US6518423 Benzopiperidine derivatives
02/11/2003US6518422 Hydrogenation of 5,5-dioxo-2,3-dihydro-1H-pyrrolo-(2,1-c)(1,2,4)benzothiadiazine with a complex of ruthenium dichloride with 2,2'-bis(diphenylphosphine)-1,1'-binaphthyl and 1,2-diphenylethylenediamine as catalyst
02/11/2003US6518286 Compounds
02/11/2003US6518268 Telomerase inhibitors and methods of their use
02/11/2003CA2030715C Hexahydro-1h-quino¬4,3,2-ef|¬1,4|benzoxazepines and related compounds, a process and intermediates for their preparation and their use as medicaments
02/06/2003WO2003010138A2 Piperidine derivatives as antibacterial agents
02/06/2003WO2002059112A3 Pyrazole compounds useful as protein kinase inhibitors
02/05/2003CN1394857A Compound used as antiproliferative agent and glycinamide ribonucleotide transformylase inhibitor
02/04/2003US6515170 Enzymatic oxidative deamination process
02/04/2003US6515157 Ferrocenyldiphosphine-ruthenium complexes and a hydrogenation process of exocyclic double bond of d-thiophene to d-thiophane
02/04/2003US6514972 Heteropolycyclic inhibitors of protein kinases
01/2003
01/30/2003WO2003007958A1 Tetrahydroquinoxalines acting as bradykinin antagonists
01/30/2003WO2002059129A3 Substituted tetracyclic pyridoindoles as serotonin agonists and antagonists
01/30/2003US20030022914 Nitric oxide synthase inhibitors
01/30/2003US20030022905 Prevention and/or therapy of ischaemia and reperfusion damage; poly(ADP-ribose)-synthetase inhibitors
01/30/2003US20030022898 Methods of treating inflammatory and immune diseases using inhibitors of IkappaB kinase (IKK)
01/30/2003US20030022885 Pyrazole compounds useful as protein kinase inhibitors
01/30/2003CA2454007A1 Tetrahydroquinoxalines acting as bradykinin antagonists
01/29/2003EP1279674A2 Acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as TACE inhibitors
01/29/2003EP1278747A1 Pyrano, piperidino, and thiopyrano compounds and methods of use
01/29/2003EP1278744A1 Heterobicyclic sulfonamides and their use as platelet adp receptor inhibitors
01/29/2003EP1129097B1 Novel type condensed pyridazinone compounds
01/29/2003EP1104425B1 Novel thiazolopyrimidine compounds
01/29/2003EP0835243B1 Dialkyl phenyl halide-substituted keto-enols for use as herbicides and pesticides
01/29/2003CN1394203A Piperidine and piperazine derivatives which function as 5-HT2A receptor antagonists
01/29/2003CN1393449A Thienothiazine compound with anti-inflammatory and antalgic activity and its preparing process and usage
01/28/2003US6511977 For preventing or treating cardiac arrhythmia or atrial arrhythmia
01/28/2003CA2124375C Compounds containing a fused bicyclic ring and processes therefor
01/23/2003WO2003006471A1 Heteroaryl substituted fused bicyclic heteroaryl compounds as gabaa receptor ligands
01/23/2003WO2003006470A2 THIAZOLO [4,5-b]PYRIDINES AS FUNGICIDES
01/23/2003WO2003006447A2 Interaction inhibitors of tcf-4 with beta-catenin
01/23/2003WO2002085915A3 Novel insecticidal azoles
01/23/2003WO2002050066A3 Pyrazole compounds useful as protein kinase inhibitors
01/23/2003WO2002036562A3 1-aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands
01/23/2003US20030018032 Bicyclic imidazo-3-yl-amine derivatives
01/23/2003US20030018022 Antiinflammatory agents; antiallergens
01/23/2003CA2453554A1 Heteroaryl substituted fused bicyclic heteroaryl compounds as gabaa receptor ligands
01/23/2003CA2453175A1 Interaction inhibitors of tcf-4 with beta-catenin
01/22/2003EP1277741A1 Cyclic compounds
01/22/2003EP0646115B1 Heterocyclic-cyclic amine derivatives
01/16/2003WO2002051837A3 Heterocyclindazole and azaindazole compounds as 5-hydroxytryptamine-6 ligands
01/16/2003US20030013721 Antiinflammatory agents; immunology; cardiovascular disorders; rheumatic disorders
01/16/2003US20030013041 Write-once optical data carrier
01/15/2003EP1274709A1 Salts of bicyclic, n-acylated imidazo-3-amines and imidazo-5-amines
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