Patents
Patents for C07D 513 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (15,120)
10/2000
10/17/2000US6133445 Rigidized trimethine cyanine dyes
10/17/2000US6133270 Isothiazolones and pharmaceutical formulations
10/17/2000US6133254 Treatment of autoimmune diseases
10/17/2000CA2001205C Antimicrobial quinolonyl lactams
10/12/2000WO2000059913A1 Novel thiazolobenzimidazole derivatives
10/12/2000WO2000059510A1 Aminopyrimidines as sorbitol dehydrogenase inhibitors
10/12/2000WO2000059502A1 Pyrrolidine modulators of chemokine receptor activity
10/12/2000CA2484282A1 Pyrimidine derivatives intermediates for producing aminopyrimidines as sorbitol dehydrogenase inhibitors
10/12/2000CA2373717A1 Pyrrolidine modulators of chemokine receptor activity
10/12/2000CA2366858A1 Sorbitol dehydrogenase inhibitors
10/12/2000CA2365419A1 Novel thiazolobenzoimidazole derivatives
10/11/2000EP1042295A1 4-hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents
10/11/2000CN1269800A Tetrahydro Gamma-carbolines
10/05/2000WO2000058305A1 Novel compounds
10/05/2000WO2000058294A1 Antibacterial agents
10/05/2000CA2361366A1 Novel compounds
10/04/2000EP1039903A1 Il-8 receptor antagonists
10/04/2000CN1057088C Benzimidazole, prepn. method and use thereof
10/04/2000CN1057083C Tricyclic 1-aminoethylpyrrol derivative
10/03/2000US6127368 Anellated β-carbolines
09/2000
09/28/2000WO2000056738A1 Pyridine and pyrimidine derivatives and their use as inhibitors of cytokine mediated disease
09/28/2000WO2000056734A1 Bicyclic heterocycles, method for producing them and their use as herbicides and pharmaceutical agents
09/28/2000WO2000056710A1 3-(anilinomethylene) oxindoles as protein tyrosine kinase and protein serine/threonine kinase inhibitors
09/28/2000WO2000003981A3 Preparation of (s)-2-amino-6,6-dimethoxyhexanoic acid methyl ester via novel dioxolanes
09/28/2000CA2367866A1 Pyridine and pyrimidine derivatives and their use as inhibitors of cytokine mediated disease
09/27/2000EP1037633A1 Antiviral compounds
09/27/2000EP0773947B1 5H-THIAZOLO 3,2-a]PYRIMIDIN-5-ONE DERIVATIVES
09/27/2000CN1056844C Dioxide pyrrolo-pyrrolo derivatives
09/26/2000US6124331 Selective NPY (Y5) antagonists (tricyclics)
09/26/2000US6124330 N-[4-(Heteroarylmethyl)phenyl]-heteroarylamines
09/26/2000US6124243 Method of controlling graminaceous weeds
09/21/2000WO2000055159A2 Substituted aza-oxindole derivatives
09/21/2000WO2000055147A1 Fused 1,4-thiazine-2-carbonitrile derivatives, their preparation and use
09/21/2000WO2000054759A2 Lxr modulators
09/21/2000DE19912636A1 Bicyclische Heterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Herbizide und pharmazeutische Mittel Bicyclic heterocycles, process for their preparation and their use as herbicides and pharmaceutical compositions
09/21/2000CA2367595A1 Lxr modulators
09/20/2000EP0705816B1 Benzene derivative useful for ischemic diseases
09/19/2000US6121281 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
09/13/2000CN1266061A 2-mercapto-ethylamine cyclized hypocrellin and preparation process and usage thereof
09/13/2000CN1266057A Novel cyano-indole serotonin reextracted inhibitor compound, its preparation process and medicinal compositions having same
09/13/2000CN1056373C Process for preparation of fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles
09/12/2000US6117888 Thrombin inhibitors
09/08/2000WO2000052013A2 Thiazoloindolinone compounds
09/08/2000WO2000051996A1 Polycyclic thiazole-2-ylides amines, method for the production thereof and their utilization as medicaments
09/08/2000WO2000051602A1 Utilization of polycyclic 2-amino-thiazole systems in the production of medicaments for prophylaxis or treatment of obesity
09/08/2000WO2000037021A3 Products comprising trihydroxystilbenes and derivatives thereof and methods for their manufacture and use
09/08/2000WO2000018769A3 INDOLO[2,1-b]QUINAZOLE-6,12-DIONE ANTIMALARIAL COMPOUNDS AND METHODS OF TREATING MALARIA THEREWITH
09/08/2000CA2364902A1 Polycyclic thiazole-2-ylides amines, method for the production thereof and their utilization as medicaments
09/08/2000CA2362554A1 Utilization of polycyclic 2-amino-thiazole systems in the production of medicaments for prophylaxis or treatment of obesity
09/08/2000CA2361580A1 Thiazoloindolinone compounds
09/06/2000EP1033137A1 Diagnostics for complications of diabetes or renal insufficiency
09/06/2000EP1032574A2 INDOLO 2,1-b]QUINAZOLE-6,12-DIONE ANTIMALARIAL COMPOUNDS AND METHODS OF TREATING MALARIA THEREWITH
09/06/2000CN1265661A N-acylamino acid amide compounds and intermediates for preparation thereof
09/05/2000US6114537 Process for scavenging thiols
08/2000
08/31/2000WO2000050390A1 N-substituted arylsulfonylamino hydroxamic acids useful as inhibitors of c-proteinase and for treating or preventing disorders related to unregulated collagen production
08/31/2000DE19908537A1 Verwendung von polycyclischen 2-Amino-Thiazol Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas Use of 2-amino-thiazole polycyclic systems for the production of medicaments for the prophylaxis or treatment of obesity
08/31/2000DE19908536A1 Polycyclische Thiazol-2-yliden Amine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel Polycyclic thiazol-2-ylidene amines, process for their preparation and their use as medicaments
08/31/2000CA2364804A1 N-substituted arylsulfonylamino hydroxamic acids useful as inhibitors of c-proteinase and for treating or preventing disorders related to unregulated collagen production
08/30/2000EP1031563A1 Sulfonyl derivatives
08/30/2000EP1030840A1 Cyclic amine derivatives and their use as drugs
08/30/2000EP0836606B1 Condensed thiazole derivatives, having 5-ht receptor affinity
08/30/2000CN1265109A Thiazolobenzoheterocycles, prepn. and medicines containing same
08/29/2000US6110929 Immunomodulators which induce cytokine biosynthesis, including interferon and/or tumor biosynthesis, necrosis factor and inhibit t-helper-type 2 immune response; for treatment of viral and neoplastic diseases
08/29/2000CA2012628C New fluoro-4 benzoic derivatives, process for their preparation and pharmaceutical compositions containing them
08/24/2000WO2000049007A1 Acetamido acetonitrile derivatives as inhibitors of cathepsin l and/or cathepsin s
08/24/2000DE19906652A1 Processing of silver halide color photographic materials containing specified heterocyclic cyan couplers uses hydrazine derivatives as color developer to give new fast acid resistant cyan dyes
08/23/2000EP1029854A1 Oxazolidinones and their use as antibacterial agents
08/23/2000EP1028965A1 Cytotoxic pyridoacridine alkaloids
08/23/2000EP0698023B1 Fibrinogen receptor antagonists
08/23/2000EP0652882B1 Anellated (oxa)hydantoines and their use as herbicides
08/23/2000CN1264384A Fused 1,2,4-thiadiazine derivatives, their preparation method and use
08/23/2000CN1055699C Sulfomycin analogue
08/22/2000US6107310 Heteroarylcarboxamide derivatives for treating CNS disorders
08/22/2000US6107300 Arylamino fused pyrimidines
08/22/2000US6107294 Nervous system and psychological disorders
08/16/2000EP1028111A1 Amide derivatives or salts thereof
08/16/2000CN1055473C 1,9-bridged thiazolo (3,2-A) quinoline derivatives
08/15/2000US6103738 Quinoline and quinazoline compounds useful in therapy
08/15/2000US6103730 Amine substituted compounds
08/15/2000US6103724 Exhibit mainly antipsychotic effects, e.g., schizophrenia, organic mental disorders, affective disorders, anxiety, personality disorders; neuroleptic activitiy; atypical antipsychotics, cognition activators, antidepressants;
08/15/2000US6103658 Olefin polymerization catalysts containing group 8-10 transition metals, processes employing such catalysts and polymers obtained therefrom
08/10/2000WO2000046223A1 Tricyclic quinolonecarboxylic acid derivatives or salts thereof
08/10/2000DE19905278A1 Oxazolidinone und ihre Verwendung als antibakterielle Mittel Oxazolidinones and their use as antibacterial agents
08/09/2000EP1024810A1 Method for optimizing retinal and optic nerve health
08/09/2000CN1262679A IL-5 inhibiting 6-azauracil derivatives
08/09/2000CN1262674A Gatrokinetic monocyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives
08/09/2000CN1262621A Gastrokinetic bicyclc benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives
08/09/2000CN1262275A Substituted thiazol [3,2-alpha] azatropylidene derivatives
08/08/2000US6100271 Compounds which mediate intracellular signaling response to abnormal external stimuli characteristic of diseases; antiinflammatory agents, antifibrotic agents, antisclerotic agents, antitumor agents
08/08/2000US6100246 Spiro-piperidine derivatives as inhibitors of nitric oxide synthase
08/03/2000WO2000044756A1 Thiazolopyrimidine compounds, process for the preparation of the same and uses thereof
08/03/2000WO2000044749A1 Acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as tace inhibitors
08/03/2000WO2000044709A2 ACETYLENIC α-AMINO ACID-BASED SULFONAMIDE HYDROXAMIC ACID TACE INHIBITORS
08/03/2000WO2000044364A2 P53 inhibitors and their use for the treatment of cancer, hyperthermia, hypoxia, a burn, trauma to the central nervous system, a seizure, acute inflammation, tissue ageing, preservation of organs for transplant and preparation of a host for bone marrow transplant
08/03/2000CA2360671A1 P53 inhibitors and therapeutic use of the same
08/03/2000CA2359011A1 Thiazolopyrimidine compound, its production and use
08/03/2000CA2356299A1 Acetylenic .alpha.-amino acid-based sulfonamide hydroxamic acid tace inhibitors
08/03/2000CA2355735A1 Acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as tace inhibitors
08/02/2000EP1023898A1 Cyano-indoles as serotonine reuptake inhibitors and as 5-HT2c receptor ligands
08/02/2000EP1023269A1 Beta3-adrenoreceptor agonists, agonist compositions and methods of using