Patents
Patents for C07D 513 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (15,120)
04/2001
04/11/2001CN1064354C Trilcyclic benzazepine vasopressin antagnonists
04/10/2001US6215016 Hematopoietic agents; preventing cytopenia
04/10/2001US6214853 Selective NPY (Y5) antagonists (bicyclics)
04/05/2001WO2001023375A2 Substituted pyridines and pyridazines with angiogenesis inhibiting activity
04/05/2001WO2000040228A3 Formulations comprising imiquimod or other immune response modifiers for treating mucosal conditions
04/04/2001EP1087981A2 Prenyl transferase inhibitors
04/04/2001EP1087770A1 Inhibitors of prenyl-protein transferase
04/04/2001EP0686636B1 Tricyclic benzazepine and benzothiazepine derivatives
04/04/2001CN1289766A Penicillene compounds and derivatives therefrom
04/03/2001US6211170 Azetidinone derivatives for the treatment of HCMV infections
03/2001
03/29/2001WO2000075139A3 Benzothiazinone and benzoxazinone compounds
03/28/2001EP1086108A1 Heterobicyclic and tricyclic nitric oxide synthase inhibitors
03/28/2001CN1289334A Benzothiadiazoles and derivatives
03/28/2001CN1063747C Quinotone and naphthyridonecarboxylic acid derivatives
03/27/2001US6207689 Polycyclic thiazol-2-ylidene amines, processes for their preparation and their use as medicaments
03/27/2001US6207664 Squalene synthetase inhibitor agents
03/22/2001WO2001019802A1 Aromatic nitrogenous six-membered ring compounds
03/22/2001WO2000001376A3 Pharmaceutical compositions and their uses for treatment of demyelinating disorders
03/21/2001EP1085011A1 Novel polyamine analogues as therapeutic and diagnostic agents
03/21/2001EP1084117A2 Novel herbicides
03/21/2001CN1063447C Condensed thiazine derivatives their production and use
03/20/2001US6204261 Inhibitors of interleukin-1β Converting enzyme inhibitors
03/15/2001WO2001017992A1 Inhibitors of prenyl-protein transferase
03/15/2001WO2000049007A8 Acetamido acetonitrile derivatives as inhibitors of cathepsin l and/or cathepsin s
03/15/2001CA2318004A1 Novel polyamine analogues as therapeutic and diagnostic agents
03/14/2001EP1082362A1 Supported group 8-10 transition metal olefin polymerization catalysts
03/13/2001US6200980 Method of treating a patient having precancerous lesions with phenyl purinone derivatives
03/13/2001US6200925 As polymerization catalyst
03/13/2001CA2146238C Novel mercaptoacetylamide bicyclic lactam derivatives useful as inhibitors of enkephalinase and ace
03/08/2001WO2001016139A1 Androgen receptor modulator compounds and methods
03/08/2001DE19942613A1 Preparation of condensed pyrroles, useful as 2- and 4-equivalent cyan couplers and coupler intermediate, involves reacting azolylacetic acid derivative with alpha-haloacetaldehyde and alkali cyanide and condensation
03/08/2001DE19942612A1 New cyan couplers, used in color photographic silver halide material, are 2- or 4-equivalent pyrrolo-oxadiazole, -thiadiazole or -triazole, compounds with 2 electron acceptor substituents
03/08/2001CA2383077A1 Androgen receptor modulator compounds and methods
03/07/2001EP1080095A1 Modulators of protein tyrosine phosphatases (ptpases)
03/07/2001EP1080094A1 G-csf mimetics
03/07/2001EP1080093A1 G-csf mimetics
03/07/2001EP1080068A1 Modulators of protein tyrosine phosphatases
03/07/2001EP1079763A2 Serotonergic 5ht 7? receptor compounds for treating ocular and cns disorders
03/07/2001CN1286683A Tetrahydrobenzindole derivs
03/06/2001US6197804 Kinase inhibitors; anticancer agents
03/06/2001US6197785 Cardiovascular disorders
03/01/2001WO2001014333A1 Substituted piperidine compounds useful as modulators of chemokine receptor activity
02/2001
02/28/2001CN1285821A Aryl Fused azapolycyclic compounds
02/27/2001US6194426 5,6,7,8 tetrahydroindolizines derivatives
02/21/2001EP1076656A2 N-heteroaryl-substituted pyridine derivatives and their use as herbicides
02/21/2001EP1076655A1 N-pyridonyl herbicides
02/20/2001US6191140 Potassium channel modulators; muscle relaxants; controlling cell membranes
02/20/2001US6191124 Methanol derivatives for treatment of retroviral infections especially HIV infections
02/20/2001CA2192289C Substituted heterocyclic derivatives
02/15/2001WO2001010842A2 Melanocortin-4 receptor binding compounds and methods of use thereof
02/15/2001WO2000054759A3 Lxr modulators
02/15/2001CA2381008A1 Melanocortin-4 receptor binding compounds and methods of use thereof
02/14/2001EP1076056A1 Novel spiro compounds or salts thereof and preventives/remedies for autoimmune diseases and ap-1 inhibitors containing the same
02/14/2001EP1075465A1 Arylphenyl-substituted cyclic keto enols
02/14/2001EP0815120B1 17-difluoromethylene-oestratrienes
02/14/2001CN1284075A Novel compounds having CGMP-PDE inhibitory effect
02/14/2001CN1283995A Antiviral compounds
02/13/2001US6187802 Substituted 4-arylmethylene-2-imino-2,3-dihydrothiazoles and derivatives and their pharmaceutical use
02/13/2001US6187774 Fused heterocyclic compounds and pharmaceutical applications thereof
02/13/2001US6187770 N-substituted azaheterocyclic compounds
02/13/2001CA2001203C Novel antimicrobial dithiocarbamoyl quinolones
02/08/2001WO2000068234A3 Process for the preparation of cefpodoxime acid
02/07/2001EP1073648A1 12,13-Modified epothilone derivatives
02/07/2001EP1073647A1 12,13-cyclopropane epothilone derivatives
02/07/2001EP0789702B1 Substituted tetracyclic oxazepine and thiazepine derivatives with 5-ht2 receptor affinity
02/07/2001CN1283198A Cytotoxic pyridoacridine alkaloids
02/07/2001CN1283114A Benzoxazine compounds for enhancing synaptic response
02/07/2001CN1061652C Endotheliomycine receptor antagonist
02/01/2001WO2001007467A1 Streptogramin derivatives, preparation and compositions containing same
01/2001
01/31/2001EP1071686A1 Novel heterocyclic compounds
01/31/2001EP1071426A2 Novel compounds and their use as positive ampa receptor modulators
01/31/2001CN1281854A Benzothiazine derivative
01/31/2001CN1061347C 抗真菌剂 Antifungal agents
01/30/2001US6180619 Prenyl transferase inhibitors
01/24/2001CN1281439A 4-Hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents
01/23/2001US6177442 Bicyclic amine derivatives
01/17/2001EP1069132A1 Bicyclic derivatives of amino-pyrazinones, process of preparation and pharmaceutical compositions comprising them
01/17/2001EP1068212A1 THIAZOLO 4,5-d]PYRIMIDINES AND PYRIDINES AS CORTICOTROPIN RELEASING FACTOR (CRF) ANTAGONISTS
01/17/2001CN1280568A Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and TACE inhibitors
01/17/2001CN1280496A Use of brinzolamide to prevent visual field loss
01/16/2001US6174839 As herbicide
01/11/2001WO2001002410A1 Novel process
01/11/2001WO2001002394A1 Substituted indole compounds and their use for the treatment of cancer
01/11/2001WO2001002379A1 Selective npy (y5) antagonists
01/11/2001WO2001002377A1 Telomerase inhibitors and methods of their use
01/11/2001WO2001002373A1 Dihydrobenzodiazepins and their use for treating dyslipidemia
01/11/2001WO2001001986A1 Method of reducing neuronal injury or apoptosis
01/11/2001WO2000043398A3 Tricyclic benzodiazepines as vasopressin receptor antagonists
01/11/2001CA2380866A1 Selective npy (y5) antagonists
01/11/2001CA2373883A1 Method of reducing neuronal injury or apoptosis
01/11/2001CA2341253A1 Telomerase inhibitors and methods of their use
01/10/2001CN1279241A Tetracydic fluoquinolone carboxylic acid, its preparing process and medicinal composition containing it as active component
01/10/2001CN1279240A Tetracyclic fluoquinolone carboxylic acid, its preparing process and medicinal composition containing it as active component
01/09/2001US6172076 Inhibitors of prenyl-protein transferase
01/09/2001US6172073 Benzimidazolyloxy alkanamines as serotonin reuptake inhibitors; nicotine and tobacco withdrawal; psychological, eating, brain, gastrointestinal, sleep, and sexual disorders
01/04/2001WO2001000583A1 Ucf116 derivatives as antitumor agents
01/04/2001WO2001000579A1 COMPOUNDS FOR THE MODULATION OF PPARη ACTIVITY
01/03/2001EP0708776B1 Antiallergic imidazoazepines
01/03/2001CN1278797A Oxo-substituted compouns, process of making, and compositions and methods for inhibiting parp activity
01/03/2001CN1278794A Substituted di-hydroxyl-indol derivatives as protein tyrosine kinase and as protein serine/threenine kinase inhibitors