Patents
Patents for C07D 513 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (15,120)
04/1999
04/22/1999WO1999011624B1 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity
04/22/1999CA2316296A1 Use of csaidtm compounds for the management of uterine contractions
04/21/1999EP0909760A1 New analogs of strobilurine having fungicidal properties, and their application for controlling phytopathogenous fungi
04/21/1999EP0369000B1 Macrocyclic complexes of yttrium, the lanthanides and the actinides having peripheral coupling functionalities
04/21/1999CN1214685A Inhibitors of farnesyl protein transferase
04/15/1999WO1999018076A1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
04/15/1999WO1999018073A1 Azetidinone derivatives for the treatment of hcmv infections
04/15/1999CA2303449A1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
04/14/1999EP0907650A1 N- 4-(heteroarylmethyl)phenyl]-heteroarylamines
04/14/1999EP0595924B1 Platelet activating factor antagonists
04/14/1999CN1214039A Carbamoyloxy derivatives of mutiline and their use as antibacterials
04/14/1999CN1042936C Substituted aminoquinolone compound, its application and medicinal compsns. containing same
04/13/1999CA1340493C Pyridone carboxylic acid derivatives and salts thereof, process for producing the same and antibacterial agents comprising the same
04/08/1999WO1999016769A1 Resolution of optically-active compounds
04/08/1999WO1999016752A1 β3-ADRENORECEPTOR AGONISTS, AGONIST COMPOSITIONS AND METHODS OF USING
04/08/1999WO1999016747A1 Sulfonyl derivatives
04/08/1999CA2304285A1 Sulfonyl derivatives
04/07/1999CN1213373A Pyrimidin-4-one-derivatives as pesticide
04/01/1999WO1999015533A1 Macrocyclic porphyrazine-type compounds, metal derivatives thereof and process for their preparation
04/01/1999WO1999015500A1 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
04/01/1999CA2302572A1 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
03/1999
03/31/1999EP0905136A1 Tetrahydro gamma-carbolines
03/30/1999US5889034 Antiinflammatory agent; antiatherosclerosis agent; viricides
03/30/1999US5889009 Method of inhibiting cell adhesion
03/30/1999US5889002 Fused 1,2,4-thiadiazine and fused 1,4-thiazine derivatives, their preparation and use
03/25/1999WO1999014202A2 Novel pyrimidin-4-one and pyrimidin-4-thione as fungicide
03/25/1999CA2301694A1 Novel pyrimidin-4-one and pyrimidin-4-thione as fungicide
03/24/1999EP0902684A1 Hexahydro-pyrido(4,3-b)indole derivatives as antipsychotic drugs
03/18/1999WO1999012926A1 Tetrahydro gamma-carbolines
03/18/1999CA2301807A1 Tetrahydro gamma-carbolines
03/17/1999EP0626962B1 Substituted phenylheterocyclic herbicides
03/11/1999WO1999011642A1 Aminometyl oxooxazolidinyl benzene derivatives
03/11/1999WO1999011628A1 Alkoxy-substituted compounds, methods, and compositions for inhi biting parp activity
03/11/1999WO1999011624A1 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity
03/11/1999CA2294118A1 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity
03/11/1999CA2294110A1 Alkoxy-substituted compounds, methods, and compositions for inhi biting parp activity
03/10/1999EP0900272A2 Tumor necrosis factor alpha convertase
03/10/1999CN1210531A Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
03/04/1999WO1999010346A1 Benzothiadiazinyl-indole derivatives and their use as serotonin receptor ligands
03/04/1999WO1999010342A1 Antibiotic oxazolidinone derivatives
03/04/1999WO1999010325A1 Benzylidene-1,3-dihydro-indol-2-one derivatives as receptor tyrosine kinase inhibitors, particularly of raf kinases
03/03/1999EP0745080B1 Novel mercaptoacetylamide disulfide derivatives useful as inhibitors of enkephalinase and ace
03/03/1999EP0724570B1 Amidino derivatives useful as nitric oxide synthase inhibitors
03/02/1999US5877313 Benzo-fused azepinone and piperidinone compounds useful in the inhibition of ACE and NEP
02/1999
02/25/1999WO1999009031A1 Nucleosides analogues, such as antivirals including inhibitors of retroviral reverse transcriptase and the dna polymerase of hepatitis b virus (hbv)
02/24/1999EP0897921A1 Benzothiadiazinyl-indole derivatives and their use as serotonin receptor ligands
02/24/1999EP0897912A1 Amidino derivatives useful as nitric oxide synthase inhibitors
02/24/1999CN1042228C Antiallergic imidazoazepines
02/23/1999US5874432 Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof
02/23/1999US5874429 Benzothiazine derivative
02/23/1999US5874382 Cyclic sulfonamide herbicides
02/22/1999CA2245331A1 Pharmaceutical compounds
02/18/1999WO1999007701A1 Tricyclic quinoxaline derivatives as protein tyrosine kinase inhibitors
02/18/1999WO1999007379A1 5,6-HETEROARYL-DIPYRIDO[2,3-b:3',2'-f]AZEPINES AND THEIR USE IN THE PREVENTION OR TREATMENT OF HIV INFECTION
02/18/1999CA2295620A1 5,6-heteroaryl-dipyrido¬2,3-b:3',2'-f|azepines and their use in the prevention or treatment of hiv infection
02/17/1999CN1208418A Pyrido-1,2,4-thiadiazine and pyrido-1,4-thiazine derivatives, their preparation and use
02/17/1999CN1208417A Fused 1,2,4-thiadiazine and fused 1,4-thiazine derivatives, their preparation and use
02/17/1999CN1208349A Composition for treating pain
02/17/1999CN1042133C N-substituted azabicycloheptane derivatives, the preparation and use thereof
02/16/1999US5872253 1-(3-heterocyclyphenyl)-s-triazine-2,4,6-oxo or thiotrione herbicidal agents
02/11/1999WO1999006410A1 Hydroxamic acid substituted fused heterocyclic metalloproteinase inhibitors
02/11/1999WO1999006402A1 N-acylamino acid amide compounds and intermediates for preparation thereof
02/11/1999WO1998040420A3 Catalyst compositions for the polymerization of olefins
02/11/1999CA2297988A1 Hydroxamic acid substituted fused heterocyclic metalloproteinase inhibitors
02/11/1999CA2297815A1 N-acylamino acid amide compounds and intermediates for preparation thereof
02/09/1999US5869659 Microbiocides
02/09/1999US5869655 Diamine compounds, methods of making same, method of use of same and intermediates
02/09/1999US5869650 Potentiate cytotoxicity of anticancer drugs
02/09/1999US5869492 Condensed thiazole derivatives, having 5-HT receptor affinity
02/09/1999US5869483 Tricyclic benzazepine vasopressin antagonists
02/09/1999US5869482 Dipyridio 2,3-b:3',2'-! azepines and their use in the prevention or treatment of HIV infection
02/09/1999US5869478 Administering as antiischemic agents
02/04/1999WO1999005147A1 Thiazolobenzoheterocycles, preparation and medicines containing same
02/03/1999EP0894003A1 N-formyl hydroxylamine containing compounds useful as ace inhibitors and/or nep inhibitors
01/1999
01/28/1999WO1999003861A1 Fused 1,2,4-thiadiazine derivatives, their preparation and use
01/28/1999WO1999003510A1 Diagnostics for complications of diabetes or renal insufficiency
01/28/1999CA2294830A1 Fused 1,2,4-thiadiazine derivatives, their preparation and use
01/27/1999EP0892797A1 Inhibitors of farnesyl protein transferase
01/27/1999EP0892780A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS
01/27/1999CN1206010A 5H-thiazole [3,2-a] pyrimidine derivatives
01/26/1999US5864043 Cardiovascular disorders and angiotensin antagonist
01/21/1999WO1999002505A1 Il-5 inhibiting 6-azauracil derivatives
01/21/1999WO1999002494A1 Gastrokinetic monocyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives
01/21/1999WO1999002156A1 Gastrokinetic bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivates
01/21/1999CA2294145A1 Il-5 inhibiting 6-azauracil derivatives
01/20/1999EP0891978A2 5H-Thiazolo (3,2-a) pyrimidine derivatives
01/20/1999EP0707579B1 Piperidinyl substituted methanoanthracenes as d1/d2-antagonists and 5ht2-serotanin-antagonists
01/19/1999US5861426 Nitro esters of aromatic compounds with amide or ester groups
01/13/1999CN1205004A Esters of 3-hydroxy-piperidinemethanol derivatives
01/12/1999US5859239 Mercaptoalkanoylamino and acylmercaptoalkanoylamino benzoxazepines and benzothiazepines
01/07/1999WO1999000133A1 Method for optimizing retinal and optic nerve health
01/07/1999EP0888359A1 Pyrimidin-4-one derivatives as pesticide
01/07/1999CA2294343A1 Method for optimizing retinal and optic nerve health
01/05/1999US5856564 Condensed benzazepine derivative and pharmaceutical composition thereof
01/05/1999US5856515 Electron-deficient porphyrins and processes and intermediates for preparing same
01/05/1999US5856478 Anellated (oxa)hydantoins and their use as herbicides
01/05/1999US5856477 Hypotensive agents; congestive heart failure
01/05/1999US5856476 Processes for preparing azepiones useful as intermediates in the preparation of inhibitors of angiotensin converting enzyme and neutral endopeptidase
01/05/1999US5856475 4-thia-1-azabicyclo/3.2.0/Heptane-3-Imino-2-isopropylidene-7-oxo-analogons of beta-lactams, processes for their preparation and the use thereof
12/1998
12/30/1998WO1998058947A1 Dipeptide derivatives as growth hormone secretagogues