Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
07/2005
07/14/2005WO2005063771A1 Methods of preparing olanzapine
07/14/2005WO2005063742A2 Amidino compounds as cysteine protease inhibitors
07/14/2005WO2005063714A1 Analogs of benzoquinone-containing ansamycins for the treatment of cancer
07/14/2005WO2005062882A2 Rifamycin analogs and uses thereof
07/14/2005WO2005062748A2 Bicyclic carbohydrate compounds useful in the treatment of infections caused by herpesviridae
07/14/2005US20050153989 Pyrrolopyrimidine derivatives and analogs and their use in the treatment and prevention of diseases
07/14/2005US20050153942 Heterocyclic inhibitors of MEK and methods of use thereof
07/14/2005US20050152913 Process for preapring maytansinol
07/14/2005CA2551806A1 Methods of preparing olanzapine
07/14/2005CA2551611A1 Thiazole derivatives for treating or preventing parkinson's disease
07/14/2005CA2550729A1 Rifamycin analogs and uses thereof
07/13/2005EP1551849A1 Tricyclic tetrahydroquinoline antibacterial agents
07/13/2005EP1551822A2 Pentacyclic oxepines and derivatives thereof, process for their preparation and pharmaceutical compositions containing them
07/13/2005EP1551511A2 Heterocyclic aromatic compounds useful as growth hormone secretagogues
07/13/2005EP1551461A2 Azo compounds for type i phototherapy
07/13/2005EP1551412A1 Pharmaceutical compositions for the treatment of diseases related to neurotrophines
07/13/2005CN1639165A Purine derivatives as kinase inhibitors
07/13/2005CN1638769A Ophthalmic composition comprising ascomycin
07/13/2005CN1638633A Agonists and antagonists of 5h3-like receptors of invertebrates as pesticides
07/13/2005CN1637000A Imidazole ring-containing compound and organic electroluminescence display device
07/13/2005CN1636999A Benzobisazole-base compound
07/13/2005CN1210265C Phthalazine derivatives and remedies for erectile dysfunction
07/12/2005US6916809 Heterocyclic acridone inhibitors of IMPDH enzyme
07/07/2005WO2005061657A1 Single-layer organic el device
07/07/2005WO2005061483A2 Modulators of peripheral 5-ht receptors
07/07/2005US20050148769 Tricyclic compound having spiro union
07/07/2005US20050148623 HIV protease inhibiting compounds
07/07/2005US20050148603 Compositions useful as inhibitors of protein kinases
07/07/2005US20050148582 N-[1-butyl-4-piperidinylmethyl[3,4-dihydro-2 oxazino[3,2-a indole-10 carboxamide as drugs with Cahpo4 or Ca3/po4/2 fillers or binders for use in treatment of irritable bowel syndrome, urinry incontience or arrhythmias
07/07/2005US20050148578 1H-8-oxa-1-aza-dibenzo[e,h]azulene; dual inhibitors of tumour necrosis factor(alpha) and interleukin 1; antiinflammatory, analgesics
07/07/2005US20050148576 Dibenzo[b.f]oxazolo-azulines, -oxepines and -thiepines; antiinflammatories; analgesics
07/07/2005US20050147997 Blocking group(s) is released by reaction with trigger (phosphatase); optionally contains urea-containing group for attaching proteins, peptides or nucleic acids; rhodamine; kits
07/07/2005US20050145831 Antioxidants and antioxidant boosters capable of producing hydroperoxyl radicals
07/06/2005EP1550663A1 New crystalline forms of antiarrhythmic compounds
07/06/2005EP1549655A2 Substituted bicyclic thiophene derivatives, compostions containing such compounds and methods of use
07/06/2005EP1549626A1 Substituted (thiazol-2-yl) -amide or sulfonamide as glycokinase activators useful in the treatment of type 2 diabetes
07/06/2005EP1549624A2 Inhibitors of fatty acid amide hydrolase
07/06/2005EP1390370A4 Methods for preparation of cytotoxic conjugates of maytansinoids and cell binding agents
07/06/2005EP1315720B1 Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
07/06/2005CN1636005A Benzothiazinone and benzoxazinone compounds
07/06/2005CN1635979A IL-8 receptor antagonists
07/06/2005CN1635889A Isoxazolopyridinones and use thereof in the treatment of parkinson's disease
07/06/2005CN1635857A Medical devices containing rapamycin analogs
07/06/2005CN1634928A Camptothecin derivatives preparing process
07/05/2005US6914140 Asymmetric synthesis process
07/05/2005CA2220509C Fused polycyclic heterocycle derivatives
07/05/2005CA2183972C Oxazolidinone derivatives and pharmaceutical compositions containing them
06/2005
06/30/2005WO2005058913A1 Pyrido- and pyrimidopyrimidine derivatives as anti- proliferative agents
06/30/2005WO2005058912A1 Process for preparing amide acetals
06/30/2005WO2005058911A2 Substituted [1,4]oxazino[2,3-g]indazoles for the treatment of glaucoma
06/30/2005WO2005058888A2 Oxazolidinone-quinolone hybrid antibiotics
06/30/2005WO2005058327A1 Tricyclic 1-[(3-indol-3-yl)carbonyl] piperazine derivatives as cannabinoid cb1 receptor agonists
06/30/2005WO2005058318A1 3-cyano-quinoline derivatives with antiproliferative activity
06/30/2005WO2005058231A2 Rifamycin analogs and uses thereof
06/30/2005WO2005035533A8 Modulators of serotonin receptors
06/30/2005WO2002058698A8 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
06/30/2005US20050143436 N-acylamino with fused nitrogen heterocyclic ring compound; capase enzyme inhibitors; antiinflammatory agents; oral bioavailability; autoimmune diseases, destructive bone disorders, proliferative disorders, infectious diseases, degenerative diseases, and necrotic diseases
06/30/2005US20050143421 Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy
06/30/2005US20050143382 Heterocyclic compounds as pharmaceutically active compounds
06/30/2005US20050143374 Antimicrobial agents and uses thereof
06/30/2005US20050143372 Compounds, pharmaceutical compositions and methods of use therefor
06/30/2005US20050143338 1-(2,5'-Anhydro-lyxofuranosyl) thymines for the synthesis of radiomarked fluoro-3 deoxynucleotides
06/30/2005CA2549869A1 Pyrido- and pyrimidopyrimidine derivatives as anti- proliferative agents
06/30/2005CA2549728A1 3-cyano-quinoline derivatives with antiproliferative activity
06/30/2005CA2549001A1 Rifamycin analogs and uses thereof
06/30/2005CA2547519A1 Process for preparing amide acetals
06/29/2005EP1546369A2 Diagnosis and treatment of diseases arising from defects in the tuberous sclerosis pathway
06/29/2005EP1546151A1 Antidepressant cycloalkylamine derivatives of heterocycle-fused benzodioxans
06/29/2005EP1546150A1 Biologically active compounds
06/29/2005EP1545545A2 COMPOUNDS WITH THE BICYCLO 4.2.1 NONANE SYSTEM FOR THE TREATMENT OF i FLAVIVIRIDAE /i INFECTIONS
06/29/2005EP1545453A1 Methods and reagents for treating infections of clostridium difficile and diseases associated therewith
06/29/2005EP1359917B1 Thioxazinoquinolones useful for the treatment of viral infections
06/29/2005CN1633433A N-aroyl cyclic amines
06/28/2005US6911452 Central nervous system disorders, sleep disorders, eating disorders. sexual disorders, hypotensive agents
06/28/2005US6911445 For reatment of depression, childhood depression, dysthymia, anxiety, panic disorder, post-traumatic stress disorder, premenstrual dysphoric disorder, attention deficit disorder, obsessive-compulsive disorder, cocaine and alcohol addiction
06/28/2005US6911442 Has no toxicological effects; adapted for oral, topical or parenteral use and may be used for the treatment of bacterial infection in mammals
06/23/2005US20050137401 Process for the preparation of tetrahydrothieno [3,2-C] pyridine derivatives
06/23/2005US20050137189 For therapy of Gram-positive bacterial infection
06/22/2005EP1542674A1 Chondropsin-class antitumor v-atpase inhibitor compounds, compositions and methods of use thereof
06/22/2005EP1350794B1 Process for preparing substance gm-95
06/22/2005EP1268466B1 Decahydro-isoquinolines
06/22/2005CN1630655A Dual action antibiotics
06/22/2005CN1207294C Acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as TACE inhibitors
06/21/2005US6908932 Modulators of phosphoinositide 3-kinase
06/21/2005CA2250372C 6-phenylpyridyl-2-amine derivatives
06/21/2005CA2108068C Carbamates of rapamycin
06/16/2005WO2005054253A1 Process for the purification of macrolides
06/16/2005WO2005054242A1 Muscarinic agents as therapeutic compounds
06/16/2005WO2005054234A2 Substituted piperidino phenyloxazolidinones having antimicriobial activity with improved in vivo efficacy
06/16/2005WO2005026145A3 Quinolone antibacterial agents
06/16/2005WO2005025293A3 Fused ring heterocycles as potassium channel modulators
06/16/2005WO2005007658A3 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
06/16/2005US20050131226 Rearranged pentanols, a process for their production and their use as anti-inflammatory agents
06/16/2005US20050131164 Dehydration mixture of oxyamides; reacting acid or ester with dialkanolamine
06/16/2005US20050131043 Phenylethynyl and styryl derivatives of imidazole and fused ring heterocycles
06/16/2005US20050131008 42-O-alkoxyalkyl rapamycin derivatives and compositions comprising same
06/16/2005US20050131002 Anticholesterol agents; antilipemic agents; cardiovascular disorders; antiischemic agents; anticancer agents
06/16/2005US20050131001 Anticholesterol agents; antilipemic agents; antiischemic agents; cardiovascular disorders
06/16/2005US20050130979 2,3-dihydroxy-6-nitro-7-sulfamoyl-benzo(F)quinoxaline (NBQX) or the quinoxalinedione is 9-methyl-amino-6-nitro-hexahydro-benzo(F) quinoxalinedione (PNQX) for treating demyelinating disorders
06/16/2005US20050130976 Bicyclic inhibitors of MEK and methods of use thereof