Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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10/19/2005 | EP0983348B1 Polyketides and their synthesis and use |
10/19/2005 | CN1685232A Novel fluorescent label compounds |
10/19/2005 | CN1683374A Indole carbazole alkaloid and its preparing method and use |
10/18/2005 | US6956034 Oxazin(ethyl)one compounds used as fungicides |
10/13/2005 | WO2005095401A1 Alpha-trifluoromethyl alcohols or amines as glucocorticoid mimetics |
10/13/2005 | WO2005095384A1 Pyrazine derivatives and pharmaceutical use thereof as adenosine antagonists |
10/13/2005 | WO2005094833A1 Novel n-substituted dihydrobenzothiepino, dihydrobenzoxepino and tetrahydro benzocyclohepta indoles as selective estrogen receptor modulators |
10/13/2005 | US20050228179 Thionation of a carbonyl compound comprising a nitrile group, the presence of a decoy agent comprising a nitrile group |
10/13/2005 | US20050228012 Crystalline clopidogrel naphthalenesulfonate or hydrate thereof, method for preparing same and pharmaceutical composition containing same |
10/13/2005 | US20050228009 2-(4-benzo[b]thiophen-3-yl-3,6-dihydro-2H-pyridin-1-ylmethyl)-2,3-dihydro-7H -[1,4]dioxino[2,3-e]indole; serotonin reuptake and serotonin receptor inhibitor; antidepressant, anxiolytic agent; dysthymia, panic disorder, attention deficit disorder obsessive, obesity, drug abuse, sexual dysfunction |
10/13/2005 | US20050228003 Mitotic kinesin inhibitors |
10/13/2005 | US20050227971 Thioamide derivatives as progesterone receptor modulators |
10/13/2005 | US20050227963 Antiinflammatory agents |
10/13/2005 | US20050227955 Reduction of the benzoquinone moiety to form a hydroquinone, and salt formation, producing 17-ammonium hydroquinone ansamycin analogs with improved solubility and air stability; antiproliferative and anticarcinogenic agents |
10/13/2005 | CA2562126A1 Pyrazine derivatives and pharmaceutical use thereof |
10/13/2005 | CA2558019A1 Alpha-trifluoromethyl alcohols or amines as glucocorticoid mimetics |
10/12/2005 | EP1583972A2 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions |
10/12/2005 | EP1583757A1 Novel substituted nitrogen-containing heterobicycles and use thereof as factor xa inhibitors |
10/12/2005 | EP1583537A2 Piperidine compounds as antibacterials |
10/12/2005 | EP1015459B9 Tetrazole-containing rapamycin analogs with shortened half-lives |
10/12/2005 | CN1681822A Antidepressant arylpiperazine derivatives of heterocycle-fused benzodioxans |
10/12/2005 | CN1681821A Antidepressivt virkende cykloalkylaminderivater AV heterocykle-kondenserte benzodioksaner |
10/12/2005 | CN1681820A Antidepressant piperidine derivatives of heterocycle-fused benzodioxans |
10/12/2005 | CN1681817A Biologically active compounds |
10/12/2005 | CN1679583A Pharmaceutical composition comprising condensed indole compound |
10/12/2005 | CN1679559A Cancer treatment |
10/12/2005 | CN1222529C Water soluble rapamycin esters |
10/12/2005 | CN1222528C Process for purification of salt of clavulanic acid |
10/11/2005 | US6953791 Dipeptide derivatives |
10/06/2005 | WO2005092864A1 Imidazole compounds for the treatment of neurodegenerative disorders |
10/06/2005 | US20050222425 Process for making amide acetals |
10/06/2005 | US20050222409 Preparation of levofloxacin and forms thereof |
10/06/2005 | US20050222244 Synthesis of UDP-glucose: N-acylsphingosine glucosyltransferase inhibitors |
10/06/2005 | US20050222176 Piperidinylamino-thieno[2,3-D] pyrimidine compounds |
10/06/2005 | US20050222175 New piperidinylamino-thieno[2,3-D] pyrimidine compounds |
10/06/2005 | US20050222159 2,3-dihydropyridazin-3-ones e.g. 3-amino-6-(1-isopropyl-6-oxo-1,6-dihydro-3-pyridazinyl)-5-phenyl-2-pyrazinecarboxamide; adenosine antagonists; depression, dementia, Parkinson's disease, anxiety, pain, hypertension, obesity, gout, bronchial asthma |
10/06/2005 | US20050222143 Helix mimetics and composition and methods related thereto |
10/06/2005 | US20050222139 Non-peptide gnrh antagonists |
10/06/2005 | US20050222125 For therapy of depression, anxiety and body weight disorders |
10/06/2005 | US20050220823 Ophthalmic composition comprising ascomycin |
10/05/2005 | EP1581521A1 Fused heterocyclic derivatives as ppar modulators |
10/05/2005 | EP1581518A2 Substituted 1-piperidin-4-yl-4-pyrrolidin-3-yl-piperazine derivatives and their use as neurokinin antagonists |
10/05/2005 | EP1581491A1 Indole derivatives as ppar modulators |
10/05/2005 | EP1373273B1 Process for preparing maytansinol |
10/05/2005 | CN1678372A Heterocyclic aromatic compounds useful as growth hormone secretagogues |
10/05/2005 | CN1678312A Use of CCI-779 as an antineoplastic agent |
10/05/2005 | CN1678310A Medicament containing disorazoles and derivatives thereof for the treatment of benign and malignant tumoral diseases |
10/04/2005 | US6951938 Aryl fused azapolycyclic compounds |
10/04/2005 | US6951863 Pyridoarylphenly oxazolidinone antibacterials, and related compositions and methods |
10/04/2005 | US6951850 Dipeptide derivatives |
10/04/2005 | CA2245539C Condensed 2,3-benzodiazepine derivatives and their use as ampa-receptor inhibitors |
09/29/2005 | WO2005090357A1 Tricyclic benzopyran compound as anti-arrhythmic agents |
09/29/2005 | WO2005090294A2 PROCESS OF MAKING α-AMINOOXYKETONE/α-AMINOOXYALDEHYDE AND α-HYDROXYKETONE/α-HYDROXYALDEHYDE COMPOUNDS AND A PROCESS OF MAKING REACTION PRODUCTS FROM CYCLIC α,ß-UNSATURATED KETONE SUBSTRATES AND NITROSO SUBSTRATES |
09/29/2005 | WO2005089754A1 (indol-3-yl)-heterocycle derivatives as agonists of the cannabinoid cb1 receptor |
09/29/2005 | WO2005089118A2 Novel bicyclic compounds as modulators of androgen receptor function and method |
09/29/2005 | WO2005070940A3 Rifamycin derivatives effective against drug-resistant microbes |
09/29/2005 | WO2005054234A3 Substituted piperidino phenyloxazolidinones having antimicriobial activity with improved in vivo efficacy |
09/29/2005 | WO2005025507A3 Dihydropyridine compounds for treating or preventing metabolic disorders |
09/29/2005 | WO2005009398A3 Tetracyclic benzamide derivatives and methods of use thereof |
09/29/2005 | US20050215610 Such as 3-(4-(2-[2-(3,5-Difluoro-phenyl)-acetylamino]-pentanoylamino)-imidazol-1-yl)-butyric acid methyl ester; secretase, A beta -peptide inhibitor; neurogenerative and neurological diseases: Alzheimer's disease; Notch signaling pathway inhibitor; antiinflammatory agent, asthma, autoimmune diseases |
09/29/2005 | US20050215556 Macrocyclic kinase inhibitors |
09/29/2005 | US20050215547 Optically active pyridine derivative and a medicament containing the same |
09/29/2005 | CA2557054A1 (indol-3-yl)-heterocycle derivatives as agonists of the cannabinoid cb1 receptor |
09/28/2005 | EP1580187A1 Apoptogenic and antiproliferative analogs of ceramide |
09/28/2005 | EP1578752A1 Method for producing pyridoxine or an acid addition salt thereof |
09/28/2005 | EP1578743A2 Antibacterial agents |
09/28/2005 | EP1578705A2 Medical devices containing rapamycin analogs |
09/28/2005 | EP1183260B1 Triphendioxazine compounds |
09/28/2005 | CN1675225A Macrocyclic pyrimidines, their production and use as pharmaceutical agents |
09/28/2005 | CN1675224A Fused heterocyclic isoxazoline derivatives and their use as anti-depressants |
09/28/2005 | CN1675223A C6- and C9-substituted isoxazoline derivatives and their use as anti-depressants |
09/28/2005 | CN1675222A C-substituted tricyclic isoxazoline derivatives and their use as anti-depressants |
09/28/2005 | CN1675187A Co-surfactants based on aldehydes |
09/28/2005 | CN1673221A Isoxazoline derivative and herbicide comprising the same as active ingredient |
09/27/2005 | US6949578 useful in selectively inhibiting or antagonizing the alpha v beta 3 and/or alpha v beta 5 integrins; treatment of osteoporosis, humoral hypercalcemia of malignancy, Paget's disease, tumor metastasis, solid tumor growth (neoplasia), angiogenesis |
09/27/2005 | US6949562 Heterocyclic compounds as ligands of the GABAA receptor |
09/22/2005 | WO2005087769A1 Fused ring azadecalin glucocorticoid receptor modulators |
09/22/2005 | WO2005087232A1 Bicyclic modulators of androgen receptor function |
09/22/2005 | US20050209276 Etherification, dehalogenation; filtration, crystallization; bactericides |
09/22/2005 | US20050209266 nitrosated 42-deoxy-42-(1H-tetrazol-1-yl)-rapamycin; endothelium-derived relaxing factor (EDRF) agonist; anticoagulant and platelet inhibition agents; restenosis, atherosclerosis, thrombosis; stent coating; minimize interaction between blood and artificial surfaces; mix with nitric oxide donor compound |
09/22/2005 | US20050209262 Process for producing optically active sulfoxide |
09/22/2005 | US20050209225 Substituted indoles and their use as integrin antagonists |
09/22/2005 | US20050209224 N4-(4H-5-pyrid[1,4]oxazin-6-yl)-2,4-pyrimidinediamine derivatives; for treating rheumatoid arthritis |
09/22/2005 | US20050209210 Having activity against both rifampin and ciprofloxacin-resistant microorganisms |
09/22/2005 | US20050209191 1-Aza-dibenzoazulenes as inhibitors of tumour necrosis factor production and intermediates for the preparation thereof |
09/22/2005 | US20050208598 Biotin recognition sensors and high-throughput assays |
09/22/2005 | CA2558899A1 Fused ring azadecalin glucocorticoid receptor modulators |
09/21/2005 | EP1577301A1 Diamine derivatives |
09/21/2005 | EP1575952A1 Synthesis of heteroaryl acetamides |
09/21/2005 | EP1140091B1 Formulations comprising imiquimod or other immune response modifiers for treating cervical dysplasia |
09/21/2005 | CN1671800A Fibre-reactive azo dyes, their preparation and their use |
09/21/2005 | CN1671711A Calcitonin gene related peptide receptor antagonists |
09/21/2005 | CN1671690A Antimicrobial aza-bicyclic derivates, their compositions and uses |
09/20/2005 | US6946473 4-((4-But-2-ynyloxy-benzenesulfonyl)-methyl-amino)-1,3-dimethy l-1H- pyrazolo(3,4-b)and dericatives; bioavailability; no pharmacokinetic problems; bioselectiveity; rheumatoid arthritis, osteoarthritis, sepsis, AIDS, ulcerative colitis |
09/15/2005 | WO2005085257A1 Macrolides and methods for producing same |
09/15/2005 | WO2005051300A3 Bicyclic inhibitors of mek and methods of use thereof |
09/15/2005 | WO2005049604A3 Antithrombotic aromatic ethers |
09/15/2005 | US20050203296 Piperazine substituted aryl benzodiazepines and their use as dopamine receptor antagonists for the treatment of psychotic disorders |
09/15/2005 | US20050203154 Novel tetracyclic arylsulfonyl indoles having serotonin receptor affinity useful as therapeutic agents, process for their preparation and pharmaceutical compositions containing them |
09/15/2005 | US20050203122 Benzenesulfonic acid salts of clopidogrel, methods for preparing same, and pharmaceutical formulations thereof |