Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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12/08/2005 | WO2004093805A3 Selective spirocyclic glucocorticoid receptor modulators |
12/08/2005 | WO2004078682A3 Cyclic compounds and compositions as protein kinase inhibitors |
12/08/2005 | US20050272768 Process for preparation of amorphous form of a drug |
12/08/2005 | US20050272762 Thienopyridines as IKK inhibitors |
12/08/2005 | US20050272754 Polymorphic forms of rifaximin, processes for their production and uses thereof |
12/08/2005 | US20050272730 Thienopyridazines as IKK inhibitors |
12/08/2005 | US20050272721 Stable salts of olanzapine |
12/08/2005 | US20050272720 Process for making olanzapine Form I |
12/08/2005 | US20050272133 A C9-deoxomeridamycin, used as a neuroregenerative agent |
12/08/2005 | US20050272132 For therapy of a fungal infection |
12/08/2005 | US20050269556 Polymer matrix and a compound of a photochromic moiety and an oligomer of polyether, polyalkylene polyfluoroalkylene, polyfluoroalkylenyloxy, polydi(C1 to C10 hydrocarbyl)siloxane, polysilicene acid; the photochromic adduct does not become covalently tethered to the polymer matrix |
12/08/2005 | CA2565065A1 Therapeutic compounds: pyridine as scaffold |
12/07/2005 | EP1601678A2 Fused pyrrole compounds |
12/07/2005 | EP1601673A1 Novel fused heterocycles and uses thereof |
12/07/2005 | EP1601354A2 Oxadiazoline ligands for modulating the expression of exogenous genes via an ecdysone receptor complex |
12/07/2005 | EP1296987B1 Compounds for treating impaired fundic relaxation |
12/07/2005 | EP1199306B1 Biarylurea derivatives |
12/07/2005 | CN1705672A New benzodioxino-isoindole derivatives, useful for treatment of cancer, are inhibitors of cell cycle |
12/07/2005 | CN1705671A Chemical intermediate |
12/07/2005 | CN1705670A 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles |
12/07/2005 | CN1230437C Synthetic process for intermediate for ecteinascidin and phthalascidin compounds |
12/06/2005 | US6972299 Phenylethynyl and styryl derivatives of imidazole and fused ring heterocycles |
12/06/2005 | US6972296 Antichoelsterol agents; cardiovascular disorders; antihistamines; multiple sclerosis; antihistamines |
12/06/2005 | US6972193 dimerization or oligomerization of intracellular proteins to activate genetic transcription; signal transduction and activators of transcription |
12/04/2005 | CA2568914A1 Therapeutic agents, and methods of making and using the same |
12/01/2005 | WO2005113562A1 Hiv integrase inhibitors: cyclic pyrimidinone compounds |
12/01/2005 | WO2005113536A2 Tri- and bi-cyclic heteroaryl histamine-3 receptor ligands |
12/01/2005 | WO2005113509A1 Novel 4-oxoquinoline compound and use thereof as hiv integrase inhibitor |
12/01/2005 | WO2005052542A3 Method and composition useful for determining fk 506 |
12/01/2005 | US20050267303 Cyclic indole and heteroindole derivatives and methods for making and using as pharmaceuticals |
12/01/2005 | US20050267115 Melanin-concentrating hormone (MCH); for the treatment of metabolic disorders and/or eating disorders, such as obesity and diabetes, also drug dependencies, and urinary incontinence |
12/01/2005 | US20050267105 Bicyclic heterocycles as HIV integrase inhibitors |
12/01/2005 | US20050267099 Reacting a des-piperazine olanzapine with an N-formyl piperazine to form an N-formyl olanzapine |
12/01/2005 | US20050267048 Bicyclic carbohydrate compounds useful in the treatment of infections caused by herpesviridae |
12/01/2005 | CA2566755A1 Hiv integrase inhibitors: cyclic pyrimidinone compounds |
11/30/2005 | EP1600180A2 Antiproliferative drug and delivery device |
11/30/2005 | EP1599486A1 Preparation of k-252a |
11/30/2005 | EP1599461A1 Thiolactones |
11/30/2005 | EP1599206A2 Aminocyclopentyl fused heterotricylicamide modulators of chemokine receptor activity |
11/30/2005 | EP1392702B1 Compounds and methods for inhibiting mrp1 |
11/30/2005 | CN1703408A Substituted (thiazol-2-yl) -amide or sulfonamide as glycokinase activators useful in the treatment of type 2 diabetes |
11/30/2005 | CN1703407A Inhibitors of fatty acid amide hydrolase |
11/30/2005 | CN1701814A F1K-1 is a receptor for vascular endothelial growth factor |
11/30/2005 | CN1229381C Macrolides compound |
11/30/2005 | CN1229377C Spiro [Piperidine-4,1'-pyrrolo[3,4-c] pyrrole] |
11/30/2005 | CN1229111C Sustained release preparations |
11/29/2005 | US6969711 Cyclic diamine compounds and medicine containing the same |
11/24/2005 | WO2005111039A2 Compounds and methods for inhibiting mitotic progression by inhibition of aurora kinase |
11/24/2005 | WO2005111030A1 Quinolone antibacterial agents |
11/24/2005 | WO2005111015A1 Substituted pyrrolidine derivative |
11/24/2005 | WO2005110992A1 Amido compounds and their use as pharmaceuticals |
11/24/2005 | WO2005110971A1 Heteroaryl substituted cyclohexyl-1,4-diamine derivatives |
11/24/2005 | WO2005110416A2 4,5-disubstituted-2-aryl pyrimidines |
11/24/2005 | WO2005110410A2 Kinase inhibitors as therapeutic agents |
11/24/2005 | WO2005079192A3 Novel treatment |
11/24/2005 | US20050261496 3-(Morpholin-4-ylsulfonyl)-5-(1,3-thiazol-2-yl)-1H-indole-2-carboxamide; inhibiting, modulating and/or regulating signal transduction of both receptor and non-receptor tyrosine kinases; anticarcinogenic, -diabetic, -arhtritic, -inflammatory agents; psoriasis; angiogenesisinhibitors; liver cirrhosis |
11/24/2005 | US20050261494 Process for synthesis of dinitrotetraoxadiazaisowurzitane (DTIW) |
11/24/2005 | US20050261493 Methods for the isolation and purification of ansamitocins |
11/24/2005 | US20050261322 HIV integrase inhibitors |
11/24/2005 | US20050261284 Diazinopyrimidines |
11/24/2005 | US20050261277 Pentacyclic oxepines and derivatives thereof, compositions and methods |
11/24/2005 | US20050261262 Rifamycin derivatives effective against drug-resistant microbes |
11/24/2005 | CA2566212A1 Heteroaryl-substituted cyclohexyl-1,4-diamine derivatives |
11/24/2005 | CA2566158A1 Kinase inhibitors as therapeutic agents |
11/24/2005 | CA2565238A1 Amido compounds and their use as pharmaceuticals |
11/24/2005 | CA2563607A1 4,5-disubstituted-2-aryl pyrimidines |
11/24/2005 | CA2508065A1 Antiproliferative drug and delivery device |
11/23/2005 | EP1598359A1 Process for synthesis of dinitrotetraoxadiazisowursitane (DTIW) |
11/23/2005 | EP1597264A2 Antiparasitic terpene alkaloids |
11/23/2005 | EP1597260A1 Triazole compounds useful in therapy |
11/23/2005 | CN1701075A Antidepressant indolealkyl derivatives of heterocycle-fused benzodioxan methylamines |
11/23/2005 | CN1699367A Process for synthesis of dinitrotetraoxadiazaisowurzitane (dtiw) |
11/22/2005 | US6967205 Compounds with antibacterial and antiparasitic properties |
11/22/2005 | US6967198 Tricyclic compounds protein kinase inhibitors for enhancing the efficacy of anti-neoplastic agents and radiation therapy |
11/22/2005 | US6967079 Pyrimidine derivatives for labeled binding partners |
11/17/2005 | WO2005107760A1 Compounds and compositions as inducers of keratinocyte differentiation |
11/17/2005 | WO2005095401A8 Alpha-trifluoromethyl alcohols or amines as glucocorticoid mimetics |
11/17/2005 | WO2005051906A3 Heterocyclic inhibitors of mek and methods of use thereof |
11/17/2005 | US20050256313 Co-surfactants based on aldehydes |
11/17/2005 | US20050256310 Therapeutic compounds |
11/17/2005 | US20050256309 Tri-and bi-cyclic heteroaryl histamine-3 receptor ligands |
11/17/2005 | US20050256154 4-Amino-thieno[3,2-c]pyridine-7-carboxylic acid amides |
11/17/2005 | US20050256153 Thienopyridinone compounds and methods of treatment |
11/17/2005 | US20050256152 Salt of a sulfonic acid containing clopidogrel and use thereof for the production of pharmaceutical formulations |
11/17/2005 | US20050256140 Condensed pyridines and pyrimidines with tie2 (tek) activity |
11/17/2005 | US20050256124 Melanin-concentrating hormone receptor antagonists and compositions and methods related thereto |
11/17/2005 | US20050256119 selective serotonine (5-HT) reuptake inhibitor activity in combination with additional alpha 2-adrenocptor antagonist activity; To treat anxiety, movement disorders, psychosis, Parkinson's disease and body weight disorders including anorexia nervosa and bulimia without being sedative |
11/17/2005 | US20050256109 HIV integrase inhibitors: cyclic pyrimidinone compounds |
11/17/2005 | US20050256108 avoid the adverse side effects associated with non-selective receptor interactions; 1-(4-Fluorobenzyl)-2-(4-methoxybenzyl)-8-methyl-1,2,8-triaza-spiro[4.5]decan-3-one; 1-oxa-4,9-diaza-spiro[5.5]undecan-3-one compounds as monoamine receptor modulators; schizophrenia, psychosis, migraine, hypertension |
11/17/2005 | US20050256102 Inhibit Aurora kinase; cancer; 4-[9-Chloro-7-(2-fluoro-phenyl)-5H-benzo[c]pyrimido[4,5-e]azepin-2-ylamino]-N-(2-methylamino-ethyl)-benzamide; 9-Chloro-N-(4-{[3-(dimethylamino)azetidin-1-yl]carbonyl}phenyl)-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-amine |
11/17/2005 | US20050256099 Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions |
11/17/2005 | US20050256096 Having another functional group or pharmacophore covalently attached through a carbamate linkage, e.g., 25-O-Desacetyl-N-(1-carbonyl-4-methyl-piperazine) 3-morpholino rifamycin S; dual-function antibiotic mechanism provides for reduced frequency of resistance. |
11/17/2005 | US20050255465 Novel fluorescent label compounds |
11/16/2005 | EP1595884A2 Salt of sulfonic acid containing clopidogrel and use thereof for the production of pharmaceutical formulations |
11/16/2005 | EP1594865A2 Antibacterial agents |
11/16/2005 | EP1594495A1 Oxazolidinone derivates n-substituted by a tricyclic ring, for use as antibacterial agents |
11/16/2005 | EP1421634B1 Organic electroluminescent device based on 2,5-diaminoterephthalic acid derivatives |
11/16/2005 | EP1363631A4 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same |
11/10/2005 | WO2005106007A1 Labeling of rapamycin using rapamycin-specific methylases |
11/10/2005 | WO2005105814A1 Tetracyclic inhibitors of janus kinases |