Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
09/2006
09/20/2006CN1835749A 有丝分裂驱动蛋白抑制剂 Mitotic kinesin inhibitors
09/20/2006CN1275966C Pyrido-pyrido-pyrrolo pyrrolo-indole and pyrido-pyrrolo pyrrolo carbazole derivatives, method for prodn. thereof and pharmaceutical compsns. contg. said derivatives
09/19/2006US7109377 Synthesis of combinatorial libraries of compounds reminiscent of natural products
09/19/2006US7109340 Substituted tetrahydro-1H-pyrazolo [3,4-c] pyridines, compositions comprising them, and use
09/19/2006US7109338 For use in the prophylaxis and the treatment of Picornavirus and human rotavirus infections.
09/19/2006US7109235 Microtubule stabilizing compounds
09/19/2006US7109228 Pyrazole derivatives
09/19/2006CA2232195C Isoxazolidine derivatives
09/14/2006WO2006096325A1 Oxepane isomer of 42-o-(2-hydroxy)ethyl-rapamycin
09/14/2006WO2006095185A1 39-desmethoxy derivatives of rapamycin
09/14/2006WO2006094934A1 Substituted oxa-diaza-spiro-[5.5]-undecanone derivatives and their use as neurokinin antagonists
09/14/2006WO2006094682A1 Benzothiazole, thiazolopyridine, benzooxazole and oxazolopyridine derivatives as antidiabetic compounds
09/14/2006WO2006094662A1 New polymorphous forms of rifaximin, processes for their production and use thereof in the medicinal
09/14/2006US20060205769 Piperidine or 8-aza-bicyclo[3.2.1]oct-3-yl derivatives useful as modulators of chemokine receptor activity
09/14/2006US20060205766 Process for making crystalline form I of clopidogrel hydrogen sulphate
09/14/2006US20060205765 1-{1-[4-(3-amino-5-phenyl-1H-pyrazolo[3,4-b]pyridin-6-yl)benzyl]piperidin-4-yl}-1,3-dihydro-2H-benzimidazol-2-one; anticarcinogenic agents
09/14/2006US20060205757 39-desmethoxyrapamycin, compositions and methods of use thereof
09/14/2006US20060205756 Antitussives
09/14/2006US20060205744 Fused heterocyclic derivatives as ppar modulators
09/14/2006US20060205742 Heterocyclic compounds and cerebral function improvers containing the same as the active ingredient
09/14/2006US20060205718 Benzothiazole, thiazolopyridine, benzooxazole and oxazolopyridine derivatives
09/14/2006US20060205710 Spiroazacyclic compounds as monoamine receptor modulators
09/14/2006US20060205707 adenosine triphosphate inhibitors used for the treatment of cancer; anticarcinogenic agents
09/14/2006US20060205676 I kappa B kinase beta inhibitors that are 2-amino-4,6-disubstituted nicotinic acid ester analogs; antiinflammatory, antitumor and antiischemic effects; asthma; nuclear factor kappa B inhibitors; 7-(2-hydroxyphenyl)-5-(3-piperidinyl)-1,4-dihydro-2H-pyrido[2,3-d][1,3]oxazin-2-one
09/14/2006CA2602010A1 Oxepane isomer of 42-o-(2-hydroxy)ethyl-rapamycin
09/14/2006CA2600640A1 39-desmethoxy derivatives of rapamycin
09/14/2006CA2599250A1 Benzothiazole, thiazolopyridine, benzooxazole and oxazolopyridine derivatives as antidiabetic compounds
09/14/2006CA2598530A1 Substituted oxa-diaza-spiro-[5.5]-undecanone derivatives and their use as neurokinin antagonists
09/13/2006CN1832938A N-heterocyclyl phenyl-substituted cyclic ketoenols
09/12/2006US7105675 Analgesics with use of treating pain and as immunomodulators and for treatment of drug dependence
09/12/2006US7105667 Fused heterocyclic compounds and use thereof
09/12/2006US7105663 Derivatives of pyrimido[6,1-a]isoquinolin-4-one
09/12/2006US7105535 Such as n-{4-[4-(1,3-benzoxazol-2-yl)pyrazol-3-yl]phenyl}-n'-methyl urea; synthesis; cancer, cell proliferative disorders, viral infections, autoimmune diseases, neurodegenerative disorders
09/12/2006US7105529 A novel compound for treating alopecia induced by cancer chemotherapy or radiotherapy
09/12/2006US7105492 Antitumor agents
09/08/2006WO2006094236A1 N-phenyl benzamide derivatives as sirtuin modulators
09/08/2006WO2006093745A1 Purification of rapamycin
09/08/2006WO2006093743A1 Recovery of cci-779 from mother liquors
09/08/2006WO2006093514A2 Aryl and arylalkylenyl substituted thiazoloquinolines and thiazolonaphthyridines
09/08/2006WO2006008091A3 Oxidative degradation products of atorvastatin calcium
09/08/2006CA2599989A1 N-phenyl benzamide derivatives as sirtuin modulators
09/08/2006CA2599582A1 Purification of rapamycin
09/08/2006CA2599580A1 Recovery of cci-779 from mother liquors
09/07/2006US20060199956 Bicyclic heterocycles as HIV integrase inhibitors
09/07/2006US20060199836 Novel thienopyridine compounds, and methods of use thereof
09/07/2006US20060199833 Novel chemiluminescent compounds and their use
09/07/2006US20060199815 NK1 antagonists
09/07/2006US20060199814 Chemical Intermediate
09/07/2006US20060199812 Method of conjugating aminothiol containing molecules to vehicles
09/07/2006US20060199794 avoid the adverse side effects associated with non-selective receptor interactions; 1-(4-Fluorobenzyl)-2-(4-methoxybenzyl)-8-methyl-1,2,8-triaza-spiro[4.5]decan-3-one; 1-oxa-4,9-diaza-spiro[5.5]undecan-3-one compounds as monoamine receptor modulators; schizophrenia, psychosis, migraine, hypertension
09/07/2006US20060198870 Medical devices containing rapamycin analogs
09/06/2006EP1698630A1 New polymorphous forms of rifaximin, processes for their production and use thereof in the medicinal preparations
09/06/2006EP1698627A1 Pyrazole compounds useful as protein kinase inhibitors
09/06/2006EP1697384A1 Pyrido- and pyrimidopyrimidine derivatives as anti-proliferative agents
09/06/2006EP1697383A1 Process for the purification of macrolides
09/06/2006EP1697382A2 Rifamycin analogs and uses thereof
09/06/2006EP1697377A1 Polycyclic agents for the treatment of respiratory syncytial virus infections
09/06/2006EP1697359A1 Muscarinic agonists as therapeutic compounds
09/06/2006EP1697355A2 Amidino compounds as cysteine protease inhibitors
09/06/2006EP1696930A1 Tricyclic 1-((3-indol-3-yl)carbonyl)piperazine derivatives as cannabinoid cb1 receptor agonists
09/06/2006EP1696914A1 3-cyano-quinoline derivatives with antiproliferative activity
09/06/2006CN1829722A Regioselective synthesis of CCI-779
09/06/2006CN1829721A Spiro '1-azabicyclo' 2.2.2! octan-3,5'-oxazolidin - 2'-one! derivatives with affinity to the alpha7 nicotinic acetylcholine receptor
09/06/2006CN1829718A Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
09/06/2006CN1273472C Garland chrysanthemum analogue, its synthesis method and use
09/05/2006US7101908 Nontoxic treatment for infections from cytomegalovirus
09/05/2006US7101891 Compounds and pharmaceutical compositions for inhibiting MRP1
09/05/2006US7101428 stability of gamma-quinacridone pigment during milling by addition of 2,9-dichloroquinacridone
08/2006
08/31/2006WO2006060614A9 Methods for preparing pimecrolimus
08/31/2006US20060194823 Sulfonamido-macrocycles as Tie2 inhibitors and the salts thereof, a pharmaceutical composition comprising these compounds, the method of preparing and the use thereof
08/31/2006US20060194819 Activation specific inhibitors of nf-kb and method of treating inflammatory processes in cardio-vascular diseases
08/31/2006US20060194794 oxadiazoles such as 2-({[5-(3,4,5,6-Tetrahydro-2H-[1,2']bipyridinyl-4-yl)-[1,3,4]oxadiazol-2-ylmethyl]-amino}-methyl)-phenylamine exhibiting vasopressin antagonistic activity and can be used in the treatment of dysmenorrhea
08/31/2006US20060194294 Process for the recovery of staurosporine from a fermentation broth
08/30/2006CN1826333A Diamine derivatives
08/29/2006US7098330 Pyrazolylamine substituted quinazoline compounds useful as protein kinase inhibitors
08/29/2006US7098234 Indole derivatives, process for preparation of the same and use thereof
08/29/2006CA2396738C Thiazole derivatives as active superoxide radical inhibitors
08/24/2006WO2006089100A1 Benzoxazole carboxamides for treating cinv and ibs-d
08/24/2006WO2006078891A3 Imidazolylmethyl and pyrazolylmethyl heteroaryl derivatives
08/24/2006WO2006020561A3 Antibacterial agents
08/24/2006US20060189666 Alzheimer's disease; bridged bicycloalkyl sulphonamide and sulphamide derivatives; [9-endo]2',3', 4',5'-Tetrahydro-5'-(2.2.2-trifluoroethyl)spiro[3-{(E)-2-[5-(4-fluorophenyl)-1-methyl-1H-pyrazol-3-yl]ethenyl}-4-methyl bicyclo[4.2.1]non-3-ene]-9,3'-[1,2,5]thiadiazol-1',1'-dioxide
08/24/2006US20060189652 7-oxo-6-(sulphooxy)-1,6-diazabicyclo[3,2,1]octane-2-carboxamide; reacting nitrogen heterocyclic compound with carbonylation agent selected from phosgene, diphosgene, triphosgene, aryl chloroformates, aralkyl chloroformates, alkyl chloroformates, cyclization
08/24/2006US20060189643 Novel heterocyclic compounds having anti-HBV activity
08/24/2006US20060189639 Antagonists of the mGlu receptor and uses thereof
08/24/2006US20060189604 Gramnegative and Grampositive bacterial infections; substituted Piperidine derivatives specially optionally substituted pyrido [3,2, -b][1,4] thiazin-yl; 6-({(3R,4S)-3-Fluoro-1-[(R)-2-hydroxy-2-(2-methoxy-quinolin-8-yl)-ethyl]-piperidin-4-ylamino }-methyl)-4H-pyrido[3,2-b][1,4]thiazin-3-one; nontoxic
08/24/2006US20060189602 Antiviral agent especially to treat hepatitis C virus infections; 5-Hydroxy-4-(7-methoxy-1,1-dioxo-1,2-dihydro-1 lambda 6-benzo[1,2,4]thiadiazin-3-yl)-2-(3-methyl-butyl)-6-thiophen-2-yl-2H-py-ridazin-3-one; side effects reduction
08/24/2006US20060189601 Antibacterial agents
08/24/2006US20060189597 Lactam compounds and pharmaceutical use thereof
08/24/2006DE102004046142B4 Neue selektiv wirksame Substanzen zur Behandlung von Krankheiten, die durch Mykobakterien hervorgerufen werden, Verfahren zu ihrer Herstellung und ihre Verwendung Selectively new active substances for the treatment of diseases which are caused by mycobacteria, processes for their preparation and their use
08/24/2006CA2597962A1 Benzoxazole carboxamides for treating cinv and ibs-d
08/23/2006EP1692142A1 Process for preparing amide acetals
08/23/2006EP1692140A1 Compositions useful as inhibitors of protein kinases
08/23/2006EP1539133B1 Aminocyclohexene quinolines and their azaisosteric analogues with antibacterial activity
08/23/2006EP1368358B1 Isoxazoline derivatives as anti-depressants
08/23/2006CN1823081A Rapamycin carbohydrate derivatives
08/23/2006CN1823073A CCI-779 isomer C
08/23/2006CN1823072A Inhibitors of P38 and methods of using the same
08/23/2006CN1823069A Process for synthesizing beta-lactamase inhibitor intermediates
08/22/2006US7094780 3-aminoquinazolin-2,4-dione antibacterial agents
08/22/2006US7094516 Benzobisazole compound and optical recording medium containing the compound