Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
08/2008
08/06/2008EP1953165A1 Aza-substituted spiro derivative
08/06/2008EP1953147A1 Heterocyclic compound and medicinal application thereof
08/06/2008EP1953142A1 Process for the preparation of antihistaminic 4-diphenylmethyl piperidine derivatives
08/06/2008EP1951842A1 Use of rylene derivatives as photosensitizers in solar cells
08/06/2008EP1951725A1 N-sulfamoyl-n -benzopyranpiperidines as inhbitors of carbonic anhydrases
08/06/2008EP1951719A2 Certain chemical entities, compositions, and methods
08/06/2008EP1951690A1 Heterocyclic cetp inhibitors
08/06/2008EP1951235A2 Novel crystal forms of irinotecan hydrochloride
08/06/2008EP1951231A2 Camptothecin derivatives as chemoradiosensitizing agents
08/06/2008EP1660491B1 Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
08/06/2008CN101238133A Novel camptothecin analogues compounds, a method for the preparation thereof and pharmaceutical compositions containing said compounds
08/06/2008CN101238132A Spirochromanone derivatives as acetyl coenzyme A carboxylase(ACC) inhibitors
08/06/2008CN100408582C Homocamptoth-ecine compounds, their preparation process and use
08/06/2008CN100408573C Pyrazole compounds useful as protein kinase inhibitors
08/06/2008CN100408550C Method for synthesizing camptothecin-relating compounds
08/05/2008US7408062 Rigidized trimethine cyanine dyes
08/05/2008US7407972 e.g. 4,5-Dihydro-pyrazole-1,5-dicarboxylic acid 1-[(4-chloro-phenyl)-amide] 5-[(3-fluoro-2'-methanesulfonyl-biphenyl-4-yl)-amide]; anticoagulant, thrombolytic agent; thrombus formation within blood vessels; cardiovascular disease
08/05/2008US7407969 e.g. N-[1-(2-aminoethyl)-4-piperidinyl]-7-methyl-3-(8-quinolinylmethyl)-3H-imidazo[4,5-b]pyridin-2-amine tetrahydrochloride trihydrate; immunostimulant; lower respiratory tract illness during infancy and childhood, asthma, pneumonia
08/05/2008US7407968 Compounds
08/05/2008US7407967 Cyclopamine analogues and methods of use thereof
08/05/2008CA2331593C Metabolites of ecteinascidin 743
07/2008
07/31/2008WO2008005456A3 Fused heterocyclic inhibitors of d-amino acid oxidase
07/31/2008WO2007121453A3 2-hydroxy-1-oxo 1,2 dihydro isoquinoline chelating agents
07/31/2008US20080182990 Process for the Preparation of Irinotecan Hydrochloride Trihydrate
07/31/2008US20080182869 Method of Racemization of the R(-) Isomer of the (2-Chlorophenyl)-6,7-Dihydrothieno[3,2-C]Pyridine-5(4H)-Acetic Acid Methyl Ester
07/31/2008US20080182868 Novel chemical compounds
07/30/2008EP1950201A1 Substituted 3-cyanoquinolines as protein tyrosine kinases inhibitors
07/30/2008EP1950196A1 Method for manufacturing ammonium hexafluorphosphates
07/30/2008EP1948824A2 Fluorogenic probes for reactive oxygen species
07/30/2008CN101233140A Novel camptothecin analogues compounds, a method for the preparation thereof and pharmaceutical compositions containing said compounds
07/30/2008CN101233139A Alpha-(aryl-or heteroaryl-methyl)-beta-piperidinopropanoic acid compounds as ORL1-receptor antagonists
07/30/2008CN101233123A Process for preparing 2-methoxycarbonylmethyl-6,6-dimethyl-2- tetrahydropyran carboxylic acid
07/30/2008CN101233119A Novel heterocyclic nf-kb inhibitors
07/30/2008CN101232882A Percutaneously absorbable ophthalmic preparation
07/30/2008CN101230066A Antidepressant piperidine derivatives of heterocycle-fused benzodioxans
07/30/2008CN100406460C Novel derivative of camptothecine, preparing method and use
07/30/2008CN100406456C Process for preparing scopine esters
07/30/2008CN100406454C Pyrazole compounds useful as protein kinase inhibitors.
07/30/2008CN100406013C Camptothecin derivatives
07/29/2008US7405305 Pyrrole-2, 5dione derivatives and their used as GSK-3 inhibitors
07/29/2008US7405302 5-lipoxygenase-activating protein (FLAP) inhibitors
07/29/2008US7405295 Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of Bruton's tyrosine kinase by such compounds
07/29/2008US7405225 Substituted 3-amino-thieno[2,3-b]pyridine-2-carboxylic acid amide compounds and processes for preparing and their uses
07/29/2008US7405209 Protease inhibitors
07/29/2008US7405208 Benzoquinone ansamycins
07/29/2008CA2460939C Substituted pyrazolyl compounds for the treatment of inflammation
07/29/2008CA2432222C Pyrazole compounds useful as protein kinase inhibitors
07/29/2008CA2432132C Pyrazole compounds useful as protein kinase inhibitors
07/29/2008CA2401952C Pyranoindoles for treating glaucoma
07/24/2008WO2008089453A2 Inhibitors of d-amino acid oxidase
07/24/2008WO2008088689A1 Substituted spirochromanone derivatives as acc inhibitors
07/24/2008WO2008088688A1 Substituted spirochromanone derivatives as acc inhibitors
07/24/2008WO2008024497A3 INHIBITORS OF 11β -HYDROXYSTEROID DEHYDROGENASE TYPE 1
07/24/2008WO2008020269A3 A method of treating tumors with azaxanthones
07/24/2008WO2007149560A9 Fermentation and purification of actinomadura chromoprotein and related species
07/24/2008WO2007098462A3 Trans-fused chromenoisoquinolines, synthesis and methods for use
07/24/2008US20080176849 e.g. N-hydroxy-3-[4-[[(2-hydroxyethyl)[2-(1H-indol-3-yl)ethyl]-amino]methyl]phenyl]-2E-2-propenamide; histone deacetylase inhibitor; anticarcinogenic, antitumor, antiproliferative agents; improved stability
07/24/2008CA2676432A1 Inhibitors of d-amino acid oxidase
07/24/2008CA2674573A1 Substituted spirochromanone derivatives
07/23/2008EP1945647A2 Processes for preparation of maytansinol
07/23/2008EP1945646A1 Pyrimidine compounds for the treatment of inflammatory disorders
07/23/2008EP1412361B1 Substituted 5,6,6a,11b-tetrahydro-7-oxa-5-aza-benzo[c]fluorene-6-carboxylic acid derivatives serving as nmda antagonists
07/23/2008EP1342723B1 Indole derivatives and use thereof in medicines
07/22/2008US7402639 Narrow moleculae weight distribution; addition piolymers; process control
07/22/2008US7402593 (-)-5-methoxy-2-[[(4-methoxy-3,5-dimethyl-2-pyridyl)methyl]sulfinyl]imidazo[4,5-b]pyridine; proton pump inhibitor (PPI) to treat gastro-oesophageal reflux, digestive bleeding and dyspepsia; enantiomer; long duration of action; longer half-life in plasma; oxidation of sulfide followed by salt formation
07/22/2008CA2474511C Benzofuran and benzothiophene derivatives useful in the treatment of hyper-proliferative disorders
07/17/2008WO2008086409A1 5-furopyridinone substituted indazoles
07/17/2008WO2008085480A1 A novel and economical process for preparing (s,s)-2, 8-diazabicyclo[4.3.0]nonane and its enantiomer
07/17/2008WO2008084005A1 Spiropiperidine glycinamide derivatives
07/17/2008WO2008083729A1 Radiolabelling via fluorination of aziridines
07/17/2008WO2008060767A3 Macrocyclic benzofused pyrimidine derivatives
07/17/2008WO2008056257A3 Novel triazinedione derivatives as gaba-b receptor modulators
07/17/2008WO2007120648A3 Mono and di-substituted oxycodone compounds and compositions
07/17/2008US20080171888 Process for making spirolactone compounds
07/17/2008US20080171856 Antibodies; tissue-targeted therapy; for treatment of tumors, autoimmune diseases, graft rejections, graft versus host disease, viral infections, parasite infections
07/17/2008US20080171761 Substituted spirochromanone derivatives
07/17/2008US20080171760 e.g. N-[(4-Chlorophenyl)(phenyl)methyl]-2-oxo-2-(1'H,3H-spiro[2-indane-1,4'-piperidin]-1'-yl)ethanamine; vasopressin V1a receptor antagonist; antidepressant, anxiolytic, hypotensive agent; dysmenorrhea, chronic heart failure, liver cirrhosis, nephrotic syndrome, obsessive compulsive disorder
07/17/2008US20080171759 e.g. N-[(4-Chlorophenyl)(phenyl)methyl]-2-oxo-2-(1'H,3H-spiro[2-benzofuran-1,4'-piperidin]-1'-yl)ethanamine; vasopressin V1a receptor antagonist; antidepressant, anxiolytic, hypotensive agent; dysmenorrhea, chronic heart failure, liver cirrhosis, nephrotic syndrome, obsessive compulsive disorder
07/17/2008US20080171740 5,6,7,8-tetrahydro-8-quinolinamines as chemokine receptor CXCR4 antagonists such as N-(Imidazo[1,2-a]pyridin-2-ylmethyl)-N-(5,6,7,8-tetrahydro-8-quinolinyl)-1,4-butanediamine; HIV infection, rheumatoid arthritis; antiinflammatory, anticarcinogenic agent
07/17/2008US20080171733 Antiinflammatory agents, antidepressants, analgesics, purinergic receptor antagonists; neurodegenerative diseases, spinal cord injuries; 1-(2,3-dichlorophenyl)-N-[(2-methylphenyl)methyl]-1H-tetraazol-5-amine
07/17/2008US20080171040 Antibody-drug conjugates and methods
07/17/2008CA2674958A1 Spiropiperidine glycinamide derivatives
07/17/2008CA2674408A1 Radiolabelling via fluorination of aziridines
07/17/2008CA2673635A1 5-furopyridinone substituted indazoles
07/16/2008EP1944292A1 8-substituted-2,6-methano-3-benzazocines and 3-substituted morphinanes as opioid receptor binding agents
07/16/2008EP1944288A1 Radiolabelling via fluorination of aziridines
07/16/2008EP1944027A1 Pharmaceutical composition for treatment or prevention of nephritis and method for producing same
07/16/2008EP1943253A1 Novel crystalline forms
07/16/2008EP1943222A1 Antibacterial active 5-chinolin derivative
07/16/2008EP1942905A2 Niacin receptor agonists, compositions containing such compounds and methods of treatment
07/16/2008EP1073654B1 2,3-olefinic epothilone derivatives
07/16/2008CN101223175A Diazabenzo[de]anthracen-3-one compounds and methods for inhibiting PARP
07/16/2008CN101223146A Modulators of ATP-binding cassette transporters
07/16/2008CN101220037A 10-substitution homocamptothecin compounds and uses
07/16/2008CN101220036A Extraction of active ingredient such as betulinic acid from common camptotheca fruit with clean method
07/16/2008CN101220035A A kind of alkaloid, method for preparing the same and application in antineoplastic or antimicrobial aspects
07/16/2008CN100402499C 2-iminopyrrolidine derivatives
07/15/2008US7399861 side effects reduction; treating an obstructive disease of the respiratory tract or for treating overactive bladder; 3-oxa-9-azatricyclo(3.3.1.0(2,4)nonane derivatives
07/15/2008US7399765 Substituted diazabicycloalkane derivatives
07/10/2008WO2008083356A1 Substituted triazoles useful as axl inhibitors
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