| Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726) |
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| 05/22/2008 | WO2008060476A2 Nitrogen-containing heterocyclic compounds and methods of use thereof |
| 05/22/2008 | WO2008059867A1 Novel 1,2-dihydroquinoline derivative having (substituted phenyl or substituted heterocyclic) carbonyloxy lower alkyl group and ester-introduced phenyl group as substituents |
| 05/22/2008 | WO2008059866A1 Novel 1,2-dihydroquinoline derivative having substituted phenylamino lower alkyl group and ester-introduced phenyl group as substituents |
| 05/22/2008 | WO2008059865A1 Novel 1,2-dihydroquinoline derivative having substituted phenylchalcogeno lower alkyl group and ester-introduced phenyl group as substituents |
| 05/22/2008 | WO2008059046A1 Macrocyclic inhibitors of hepatitis c virus |
| 05/22/2008 | WO2008058990A1 7,7-disubstituted pyrano-[2,3-c]-imidazo-[1,2-a]-pyridine derivatives and their use as gastric acid secretion inhibitors |
| 05/22/2008 | WO2008021926A3 Modulators of glucocorticoid receptor, and/or ap-1, and/or nf-kb activity and use thereof |
| 05/22/2008 | WO2007104557A3 Novel heterocyclic nf-kb inhibitors |
| 05/22/2008 | US20080119520 Disorders related to memory and cognition processes, neurological processes, cardiovascular function, and body weight; benzoxazole, benzimidazole, and indole compounds substituted with pyrrole, azepane, piperidine or azetidine e.g. 4-{2-[2-(2-methyl-pyrrolidin-1-yl)-ethyl]-benzooxazol-5-yl}-benzonitrile |
| 05/22/2008 | US20080119505 (4aR,10bR)-6-(2,6-Dimethoxy-pyridin-3-yl)-8,9-dimethoxy-1,2,3,4,4a,10b-hexahydro-phenanthridine; phosphodiesterase inhibitor; airway obstructions, antiinflammatory agent, antidepressant; dermatoses, eczema, lupus, rheumatoid arthritis, osteoarthritis, AIDS, multiple sclerosis, graft versus host reaction |
| 05/22/2008 | US20080119460 {2-Amino-4-[(4-(4-chlorophenyl)piperidin-1-yl)methyl]thiophen-3-yl}(4-chlorophenyl)methanone; analgesic, antidepressant; cardiac disease or disorder, neurological disease or injury, sleep disorder, epilepsy, neuropathic pain, angina |
| 05/22/2008 | CA2669670A1 Nitrogen-containing heterocyclic compounds and methods of use thereof |
| 05/22/2008 | CA2669607A1 Novel 1,2-dihydroquinoline derivative having (substituted phenyl or substituted heterocyclic) carbonyloxy lower alkyl group and ester-introduced phenyl group as substituents |
| 05/22/2008 | CA2668596A1 Novel 1,2-dihydroquinoline derivative having substituted phenylamino lower alkyl group and ester-introduced phenyl group as substituents |
| 05/22/2008 | CA2668592A1 Novel 1,2-dihydroquinoline derivative having substituted phenylchalcogeno lower alkyl group and ester-introduced phenyl group as substituents |
| 05/22/2008 | CA2661338A1 Macrocyclic inhibitors of hepatitis c virus |
| 05/21/2008 | EP0911334B1 Quinolinomorphinane derivatives and medicinal use thereof |
| 05/21/2008 | CN101184760A Heterocyclic spiro-compounds |
| 05/21/2008 | CN101184759A Novel substituted tetracyclic tetrahydrofuran, pyrrolidine and tetrahydrothiophene derivatives and their use as a medicament |
| 05/21/2008 | CN101184756A Isoflavonoid dimers |
| 05/21/2008 | CN101184485A Fused imidazole derivatives and use thereof as aldosterone synthase inhibitors |
| 05/20/2008 | US7375225 4-cyanocoumarin derivatives and uses thereof |
| 05/20/2008 | US7375222 anti-dementia agent which uses a BEC 1 potassium channel inhibitor as the active ingredient; to improve learning disorder |
| 05/20/2008 | US7375204 reporter system reflecting the transport process that transports GPI-anchored proteins to the cell wall was constructed and compounds inhibiting this process were discovered; antifungal agents; inhibiting expression of cell wall glycoproteins and preventing pathogens from showing pathogenicity; DNA |
| 05/20/2008 | US7375101 N-(7-chloro-2,3-dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl)-N'-(5isoquinolinyl)-thiourea; bradykinin receptor B2 antagonists;analgesic; septic shock, pancreatitis, edema, rhinitis, asthma, colitis, arthritis, hepatorenal syndrome, cancer, bacterial and viral infections, ulcerative colitis |
| 05/20/2008 | CA2432223C Pyrazole compounds useful as protein kinase inhibitors |
| 05/20/2008 | CA2416976C Treatment of estrogen receptor positive carcinoma with a rapamycin and an antiestrogen |
| 05/20/2008 | CA2395717C Fused imidazolium derivatives |
| 05/20/2008 | CA2205664C Indole derivatives and medicinal use thereof |
| 05/15/2008 | WO2008056687A1 Novel spiropiperidine derivative |
| 05/15/2008 | WO2008056657A1 Lyophilized preparation comprising phenanthridine derivative |
| 05/15/2008 | WO2008056150A1 Heterocyclyc sulfonamides having edg-i antagonistic activity |
| 05/15/2008 | WO2008038030A3 Dispiro tetraoxane compounds and their use in the treatment of malaria and/or cancer |
| 05/15/2008 | WO2007064914A8 5-(arylsulfonyl)-pyrazolopiperidines |
| 05/15/2008 | US20080114153 Potent, durable cytotoxic agents; tissue targeted therapy; tumors, autoimmune diseases, graft versus host disease, viral and parasite infections |
| 05/15/2008 | US20080114048 Novel tetracyclic heteroatom containing derivatives useful as sex steroid hormone receptor modulators |
| 05/15/2008 | US20080114020 Difluoro-Substituted Imidazopyridines |
| 05/15/2008 | US20080114018 Condensed indoline derivatives and their use as 5HT, in particular 5HT2C, receptor ligands |
| 05/15/2008 | US20080113994 For example, 6-chloro-9-methyl-9-(3,4,5-trimethoxyphenyl)-4,9-dihydro-3H-furo[3,4-b]quinolin-1-one; for controlling animal pests, in particular insects, arachnids and mites, which are found in enclosed spaces such as dwellings |
| 05/15/2008 | US20080113972 Enzyme inhibitors of cGMP-metabolizing phosphodiesterases, for TREATMENT OF CARDIOVASCULAR DIORDERS, CEREBROVASCULAR DISORDERS, UROGENITAL DISORDERS AND ERECTILE DYSFUNCTION; chemical synthesis |
| 05/15/2008 | US20080113963 Prepared by submitting benzimidazole compound to a cyclization reaction; gastric secretion inhibiting and gastric and intestinal protective action properties; for gastrointestinal disorders; for example, 2,3-Dimethyl-8-phenyl-3,6,7,8-tetrahydro-chromeno[7,8-a]imidazole-5-carboxylic acid dimethylamide |
| 05/15/2008 | US20080113962 Condensed Tricyclic Benzimidazoles For the Treatment of Gastrointestinal Disorders |
| 05/15/2008 | CA2668853A1 Novel triazinedione derivatives as gaba-b receptor modulators |
| 05/15/2008 | CA2668785A1 Heterocyclyc sulfonamides having edg-i antagonistic activity |
| 05/14/2008 | EP1920773A1 Compositions for inhibition of anglogenesis |
| 05/14/2008 | EP1919920A2 Pentacyclic kinase inhibitors |
| 05/14/2008 | EP1465900B1 Rho-kinase inhibitors |
| 05/14/2008 | CN100387602C Chelerythrine compound and its preparing method |
| 05/14/2008 | CN100387601C Process for preparing hexahydro-2H-pyranyl [3,2-c] quinoline derivatives |
| 05/14/2008 | CN100387127C Fungicides |
| 05/13/2008 | US7371875 Compounds based on 3,7-dioxo-2-aza-6-oxabicyclo(3.2.0)heptane; proteosome inhibitors for treating proliferative or inflammatory disorders with better stability, toxicity and/or oral bioavailability |
| 05/13/2008 | US7371864 3-(1-hydroxy-1-methyl-ethyl)-1-(4-methoxy-phenyl)-6-[4-(2-oxo-2H-pyridin-1-yl)-phenyl]-1,4,5,6-tetrahydro-pyrazolo[3,4-c]pyridin-7-one for treating thromboembolic disorders |
| 05/13/2008 | US7371863 Method for manufacture of THIP |
| 05/13/2008 | US7371778 Spiro and dispiro 1,2,4-trioxolane antimalarials |
| 05/13/2008 | US7371761 Lactam-containing compounds and derivatives thereof as factor Xa inhibitors |
| 05/13/2008 | US7371757 Fused heterocycles as inhibitors of glutamate racemase(MURI) |
| 05/13/2008 | US7371748 Benzothiazole derivatives |
| 05/08/2008 | WO2008053031A1 Compounds which potentiate ampa receptor and uses thereof in medicine |
| 05/08/2008 | WO2008052444A1 Compounds with a six-membered heterocyclic ring, their preparing method and pharmaceutical use |
| 05/08/2008 | WO2008052352A1 Substituted quinone indoleamine 2,3-dioxygenase (ido) inhibitors and syntheses and uses therefor |
| 05/08/2008 | WO2008028021A3 Pyranoindazole cyclic carbonates and their use |
| 05/08/2008 | WO2007147480A3 Polymorphic forms and process |
| 05/08/2008 | WO2007120752A3 4, 5-dihydro- [1, 2, 4] triazolo [4, 3-f] pteridines as protein kinase plk1 inhibitors for the treatment of proliferative disorders |
| 05/08/2008 | WO2007117591A3 Total synthesis of salinosporamide a and analogs thereof |
| 05/08/2008 | US20080108689 Octahydropyrano[3,4-C]Pyrrole Tachykinin Receptor Antagonists |
| 05/08/2008 | US20080108645 Dihydrotetrabenazines And Pharmaceutical Compositions Containing Them |
| 05/08/2008 | US20080108619 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses |
| 05/08/2008 | US20080108591 2-amino-3,6-dihydro-4-dimethyl-amino-6-ethyl-1,3,5-triazine hydrochloride; advanced glycosylation end-products inhibitor;antidiabetic, insulin resistance, neurodegenerative disorders, renal complications, atherosclerosis, angiopathy |
| 05/07/2008 | EP1917964A1 Percutaneously absorbable ophthalmic preparation |
| 05/07/2008 | EP1917267A1 Crystal form of asenapine maleate |
| 05/07/2008 | CN101175759A Nitrogen-containing heterocyclic compounds and methods of use thereof |
| 05/07/2008 | CN101175741A Intermediate compounds for the prepation of trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oxepino[4,5-C]pyrrole |
| 05/07/2008 | CN101175738A Apoptosis promoters |
| 05/07/2008 | CN101175565A Manufacture of lactones |
| 05/07/2008 | CN101172979A Antineoplastic activity canthardin derivant and method of preparing the same |
| 05/07/2008 | CN101172978A Six-member heterocyclic compounds, prepare method and medical uses of the same |
| 05/07/2008 | CN101172967A Method for preparation of 10,11-dihydro-10-hydroxy-5h-dibenz/b,f/azepine-5-carboxamide and 10,11-dihydro-10-0x0-5h-dibenz/b,f/azepine-5-carboxamide |
| 05/07/2008 | CN101172930A 2.4-dihalogen-6-(C2-C3-alkyl)-phenyl substituted tetramic acid derivatives |
| 05/07/2008 | CN100386328C Bicyclic pyridine and pyrimidine P38 kinase inhibitors |
| 05/06/2008 | US7368569 Combining a strong base with a phenyl isonicotinamide in aprotic solvents to form a solutions, then reacting with a cyclohexanone carboxylic acid or ester and water, and acidifying the solution to obtain chemical intermediates for neuropeptide Y antagonists used for treating bulimia, obesity or diabetes |
| 05/06/2008 | US7368564 Bridged macrocyclic module compositions |
| 05/06/2008 | US7368455 2-(4-fluorophenyl)-3-[2-(2-methoxy-1-methylethylamino)pyrimidin-4-yl]-6,7-dihydro-5H-pyrazolo[1,2-a]pyrazol-1-one; cytokines (interleukin-1, 6, 8 and Tumor Necrosis Factor- alpha) inhibitor; antiinflammatory and antiarthritic agents; osteoporosis, rheumatic diseases; antidiabetic |
| 05/06/2008 | CA2258949C Novel heterocyclic compounds process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases |
| 05/02/2008 | WO2008051523A2 Carbazole derivatives useful as medicaments in cancer therapy |
| 05/02/2008 | WO2008051475A2 Hcv ns3 protease inhibitors |
| 05/02/2008 | WO2008011611A3 Compounds and compositions as itpkb inhibitors |
| 05/02/2008 | WO2008008882A3 Glucocorticoid receptor modulator and methods of use |
| 05/01/2008 | US20080103309 preparation method of 7-ethyl-10-hydroxycamptothecin from 4-ethyl-7,8-dihydro-4-hydroxy-1H-pyrano[3,4-f]indolizine-3,6,10(4H)-trione and 1-(2-amino-5 -hydroxyphenyl)-propan-1-one using higher reaction temperature and faster heating to that temperature in the presence of catalyst |
| 05/01/2008 | US20080103135 Histamine H3 antagonists; do not contain imidazolyl moiety; such as 1-[4-(4-piperidin-1-ylmethyl-phenyl)-but-3-ynyl]-piperidine |
| 05/01/2008 | US20080102031 4-[(4-N,N-diethylaminocarbonyl)phenyl]-spiro[2H,1-benzopyran-2,4'-piperidine; ligands of delta opioid receptor; analgesic, anxiolitic, antidepressant, analgesic; gastrointestinal disorders, neurodegenerative diseases; side effect reduction |
| 04/30/2008 | EP1915378A1 Viral polymerase inhibitors |
| 04/30/2008 | EP1915371A2 Bridged n-bicyclic sulfonamido inhibitors of gamma secretase |
| 04/30/2008 | DE102006050148A1 New trifluoromethoxy-phenyl substituted tetramic acid-derivatives useful to combat parasites including insects, arachnid, helminth, nematode and mollusk and/or undesirable plant growth and in hygienic sectors |
| 04/30/2008 | CN101171252A Tetracyclic azapyrazinoindolines as 5-HT2 ligands |
| 04/30/2008 | CN101171249A Method for producing indole derivative having piperidine ring |
| 04/30/2008 | CN101171222A Terrylene and quaterrylene derivatives |
| 04/30/2008 | CN100384850C Galantamine derivative and its preparation process and use |
| 04/30/2008 | CN100384849C Quinoline 3-amino chroman derivatives |
| 04/30/2008 | CN100384838C Novel benzylpiperidine compound |
| 04/30/2008 | CN100384836C Novel cyclic amide derivatives |