Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
04/2008
04/30/2008CN100384834C Epothilone derivatives
04/30/2008CN100384417C Pyranoindazoles and their use for the treatment of glaucoma
04/29/2008US7365201 Process for the preparation of the boron difluoride chelate of quinolone-3-carboxylic acid
04/29/2008US7365196 Sulphonamido-substituted bridged bicycloalkyl derivatives
04/29/2008US7365080 Pharmaceutical compositions comprising thieno[2,3-c]pyridine derivatives and use thereof
04/29/2008US7365079 2-(2-naphthyl)-4'-[3-oxospiro[6-azaisobenzofuran-1(3H),1-cyclohexan]-4'-yl]-1H-imidazole; metabolic, genitalor reproductive, gastro-intestinal, respiratory system disorders, antiinflammatory agent or glaucoma; cyclization
04/29/2008US7365078 Triaza-cyclopenta[cd]indene derivatives
04/29/2008US7365068 Hepatitis C virus infections; -(3-cyclopropyl-4-(pentyloxy)phenyl)-3-nicotinoylthiourea;methyl 2-oxo-2-(5-((3-(4-(pentyloxy)-3-(trifluoromethyl)phenyl)thioureido)carbonyl)pyridin-2-ylamino)acetate
04/24/2008WO2008047544A1 Diaryl ketimine derivative
04/24/2008WO2008021015A3 Methods of making esters of camptothecins
04/24/2008US20080097094 cis-6-(3-pyridinyl)-3,6-diazabicyclo[3.2.0]heptane; for controlling synaptic transmission, neurotransmitter release; Alzheimer's disease, Parkinson's disease, attention deficit disorder, depression, nicotinic withdrawal syndrome, Tourette's syndrome, schizophrenia and pain
04/24/2008US20080096952 Methods for the treatment of atherosclerosis, using substituted phenethylsulfones
04/24/2008US20080096876 Histamine receptor antagonists; 4-[3-(4-Piperidin-1-yl-but-1-ynyl)-benzyl]-thiomorpholine; antiallergens, antihistamines, antiepileptic agents; asthma, alzheimer's disease, narcolepsy, motion sickness, attention deficit disorder, schizophrenia
04/24/2008US20080096862 Lactam compounds and pharmaceutical use thereof
04/24/2008US20080096048 Thermally reversible; absorption ratio greater than 2.3
04/23/2008EP1913003A1 NEW PYRIDO[3',2':4,5]FURO[3,2-d]PYRIMIDINE DERIVATIVES
04/23/2008EP1913002A2 Method of acylating maytansinol with chiral amino acids
04/23/2008EP1912998A1 Pyrazole derivatives having tyrosinkinase activity
04/23/2008EP1912982A2 Novel heterocyclic nf- b inhibitors
04/23/2008EP1912980A2 Oxazolidinones bearing antimicrobial activity composition and methods of preparation
04/23/2008EP1912662A2 Peptide deformylase inhibitors
04/23/2008EP1912642A2 Synthesis and crystalline forms of npy5 antagonist
04/23/2008EP1534716B1 Heterobicyclic pyrazole derivatives as kinase inhibitors
04/23/2008EP1007033B1 Lymphocyte function antigen-1 antagonists
04/23/2008CN101166744A Spiroheterocyclic compounds and their uses as therapeutic agents
04/23/2008CN100383129C Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
04/22/2008US7361666 Ligands for cellular receptors, including opiate receptors; side effect reduction; base structure is a saturated nitrogen-containing ring substituted with a tertiary amide that is N-substituted with an arylalkyl group
04/22/2008CA2225807C Use of lamellarin-class alkaloids in methods of treatment
04/17/2008WO2008046084A2 Spiroheterocyclic compounds and their uses as therapeutic agents
04/17/2008WO2008046046A1 Tricyclic spiro-oxindole derivatives and their uses as therapeutic agents
04/17/2008WO2008044701A1 Method for producing piperidin-4-one derivative
04/17/2008WO2008044045A1 Pharmaceutical combinations
04/17/2008WO2008043791A2 Thiophene derivatives for treating hepatitis c
04/17/2008US20080091022 Reacting methscopolammonium bromide with potassium salt of tannic acid in water; antihistamines in the form of tannate salt are generally quite stable and may be administered in such form without untoward side effects
04/17/2008US20080090858 Condensed indoline derivatives and their use as 5HT, in particular 5HT2C, receptor ligands
04/17/2008US20080090846 Chemokine receptor binding heterocyclic compounds
04/17/2008US20080090831 Cytotoxic agents
04/17/2008US20080090803 Fatty alcohol drug conjugates
04/17/2008CA2666136A1 Tricyclic spiro-oxindole derivatives and their uses as therapeutic agents
04/17/2008CA2665605A1 New isocarbostyril alkaloid derivatives
04/16/2008EP1911753A1 Spiro-cyclic compound
04/16/2008EP1911350A1 Amidine compound and herbicide
04/16/2008EP1910377A2 Novel camptothecin analogues compounds, a method for the preparation thereof and pharmaceutical compositions containing said compounds
04/16/2008EP1910376A1 Novel camptothecin analogues compounds, a method for the preparation thereof and pharmaceutical compositions containing said compounds
04/16/2008EP1910375A1 Spirochromanone derivatives as acetyl coenzyme a carboxylase (acc) inhibitors
04/16/2008EP1910338A2 Heterotetracyclic compounds as tpo mimetics
04/16/2008EP1909788A2 Pharmaceutical compositions for the prevention and treatment of complex diseases and their delivery by insertable medical devices
04/16/2008EP1534334A4 Releasable polymeric conjugates based on aliphatic biodegradable linkers
04/16/2008CN101161654A Antineoplastic active canthardin derivative and method for preparing same
04/16/2008CN101161653A Method for preparing novel Pranoprofen key intermediates
04/16/2008CN101161641A Tricyclic steroid hormone nuclear receptor modulators
04/15/2008USRE40245 Gyrase inhibitors and uses thereof
04/15/2008US7358365 Process for the controlled increase in the molecular weight of polyethylenes
04/15/2008US7358263 Fused bicyclic-substituted amines as histamine-3 receptor ligands
04/15/2008US7358259 Tetrazoloquinoline, triazoloquinoline, and oxazoloquinoline compounds, e.g., 9-chloro-N-isopropoxytetrazolo[1,5-a]quinoline-4-carboxamide
04/15/2008US7358249 Heterocyclic compounds having inhibitory activity against HIV integrase
04/15/2008US7358246 5-(4,4-dimethyl-2-oxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1-methyl-1H-pyrrole-2-carbothioamide; contraceptive, menopause; reduces risk of uterine cancers coused by treating with estrogen receptor (ER) agonists
04/15/2008US7358244 Azabicycloalkane compounds
04/15/2008CA2337452C Process for the preparation of 4,5-diamino shikimic acid derivatives
04/10/2008WO2008042735A1 Tetrahydroquinoline, indoline, and related aniline derivatives of heterocycle-fused benzodioxan methylamines
04/10/2008WO2008028141A3 Raf inhibitor compounds and methods of use thereof
04/10/2008WO2008012361A3 Dimethano-[1,3] dioxocino [6,5-d] pyrimidine-spiro derivatives of tetrodotoxin, process for their synthesis and uses thereof in the treatment of pain
04/10/2008WO2007149451B1 Cycloalkanopyrrolocarbazole derivatives and the use thereof as parp, vegfr2 and mlk3 inhibitors
04/10/2008WO2007092535A3 4-acylaminopyridine derivative mediated neurogenesis
04/10/2008WO2007019180A3 Compounds for binding to eralpha/beta and gpr30, methods of treating disease states and conditions mediated through these receptors and identification thereof
04/10/2008US20080085925 Sulfonyltetrahydro-3H-benzo(e)indole-8-amine compounds as 5-hydroxytryptamine-6 ligands
04/10/2008US20080085469 Novel photoacid generators, resist compositions, and patterning process
04/09/2008EP1908755A1 Therapeutic agent for restenosis
04/09/2008EP1908752A1 Novel 2-quinolone derivative
04/09/2008EP1907395A1 Abca1 elevating compounds
04/09/2008EP1907394A1 Novel tetracyclic heteroatom containing derivatives useful as sex steroid hormone receptor modulators
04/09/2008EP1907371A1 Process for preparing 2-methoxycarbonylmethyl-6,6-dimethyl-2- tetrahydropyran carboxylic acid
04/09/2008EP1594867B1 Phenylacetamides and their use as glucokinase modulators
04/09/2008CN101160315A Cytoskeletal active compounds, composition and use
04/09/2008CN101160049A Spiroketal-substituted cyclic ketoenols
04/09/2008CN100379742C New tricyclic derivatives as LTD4 antagonists
04/08/2008US7355052 Melanocortin receptors; analgesivs; antiinflammatory agents; eating disorders; psycological disorders; anxiolytic agents; antidepressants; anticancer agents; aids; antiarthritic agents
04/08/2008US7354934 N1-(1H-Benzimidazol-2-ylmethyl)-N1-(5,6,7,8-tetrahydro-quinolin-8-yl)-butane-1,4-diamine; fusin and chemokine receptor antagonist; increase progenitor and stem cells in humans; HIV, antiinflammatory agent: rheumatoid arthritis, inflammatory bowel disease
04/08/2008US7354932 Chemokine receptor binding heterocyclic compounds with enhanced efficacy
04/08/2008US7354929 6-benzyl-3-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-2,6-dihydropyrazolo[3,4-c]pyridin-7-one; eating and psychological disorders; obesity, alcoholism
04/08/2008US7354927 6H-[1]benzopyrano[4,3-b]quinolines and their use as estrogenic agents
04/08/2008US7354925 Alpha aryl or heteroaryl methyl beta piperidino propanamide compounds as ORL1-receptor antagonists
04/08/2008US7354916 Tumor suppression agents with reduced side effects; anticancer; antibacterial and antiviral
04/08/2008US7354905 Thrombosis therapy; anticoagulants
04/08/2008CA2203183C Process for producing derivatives of 4a,5,9,10,11,12,-hexahydro-6h-benzofuro[3a,3,2-ef][2]benzazepine
04/08/2008CA2182504C Process for the preparation of a salt of clavulanic acid
04/03/2008WO2008038692A1 Diaryl ketimine derivative
04/03/2008WO2008038030A2 Dispiro tetraoxane compounds and their use in the treatment of malaria and/or cancer
04/03/2008US20080081910 5-HT1A receptor antagonists; modulating serotonin levels; central nervous system disorders; antidepressants; synthesis
04/03/2008US20080081902 Capping, polymerizing and separating failure sequences; kits for purifying oligonucleotides and polynucleotides
04/03/2008US20080081807 Arylphenyl-substituted cyclic keto-enols
04/03/2008US20080081803 Heterocyclic cyclopentyl tetrahydroisoquinoline and tetrahydropyridopyridine modulators of chemokine receptor activity
04/03/2008CA2665339A1 Dispiro tetraoxane compounds
04/03/2008CA2664358A1 Diarylketimine derivative
04/02/2008EP1905773A2 Compounds and methods for inhibiting mitotic progression by inhibition of aurora kinase
04/02/2008EP1904501A2 Chemical compounds
04/02/2008EP1904477A1 Indol-3-carbonyl-spiro-piperidine derivatives as v1a receptor antagonists
04/02/2008EP1904454A2 Process for the production of intermadiates for the preparation of tricyclic benzimidazoles
04/02/2008EP1453506B1 Topoisomerase poison agents
04/02/2008CN101155785A Novel adenosine a3 receptor modulators