Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
05/1995
05/11/1995WO1995012417A1 Alkyl, azido, alkoxy, and fluoro-substituted and fused quinoxalinediones and the use thereof as glycine receptor antagonists
05/11/1995DE4338397A1 N-Substituted bridged 4,7,8,9-tetrahydroisoindoline derivatives, their preparation and use
05/11/1995CA2175795A1 Alkyl, azido, alkoxy, and fluoro-substituted and fused quinoxalinediones and the use thereof as glycine receptor antagonists
05/11/1995CA2174235A1 Benzo-fused macrocycles promote release of growth hormone
05/10/1995EP0652216A2 Substituted Pyridyl salicylic aldehyde and salicylic acid derivatives, methods for preparing them and their use as herbicides
05/10/1995EP0651752A1 Novel chemiluminescent compounds and methods of use
05/10/1995EP0651750A1 Tetracyclic compounds process and intermediates for their preparation and their use as antitumour agents
05/09/1995CA1335502C Psychotropic bicyclic imides
05/04/1995WO1995011903A1 Tricyclic compounds having affinity for the 5-ht1a receptor
05/04/1995CA2174850A1 Tricyclic compounds having affinity for the 5-ht1a receptor
05/03/1995EP0650477A1 Light-activable 1-(2-nitrobenzyl)-substituted 1,4-dihydropyridines
05/02/1995US5412099 Intermediate benzothiazolyl- and benzoxazolyl-aldehyde compounds
05/02/1995US5412096 Treatment of senile dementia, Alzheimer*s disease, cholinergic activators
05/02/1995US5411970 Method of inhibiting lentivirus
05/02/1995US5411967 Carbamates of rapamycin
05/02/1995US5411960 Substituted pyrroloanthracenes and -diones
04/1995
04/27/1995WO1994027594A3 Stable copper(i) complexes and methods related thereto
04/26/1995EP0649847A2 Process and intermediates for the preparation of (+)- hydantocidin and analogs thereof
04/26/1995EP0649846A1 Galanthamine derivates, a process for their preparation and their use as medicaments
04/26/1995EP0649407A1 Dimeric piperidine, tetrahydropyridine and piperazine derivatives
04/26/1995EP0572437B1 2,4-diaminoquinazolines derivatives for enhancing antitumor activity
04/26/1995CN1101908A Angiotensin II antagonists
04/25/1995US5410055 Inotropic agent
04/22/1995CA2118469A1 Process and intermediates for the preparation of (+)- hydantocidin and analogs thereof
04/20/1995WO1995010519A1 Quinolizinone type compounds
04/20/1995WO1995010507A1 Phenylsulfonyl ureas, process for producing the same and their use as herbicides and plant growth regulators
04/20/1995CA2173459A1 Quinolizinone type compounds
04/19/1995EP0648771A1 Galanthamine derivatives, a process for their preparation and their use as medicaments
04/19/1995EP0648758A1 4-Arylamino-benzopyran and related compounds
04/19/1995EP0550635B1 Fused ring analogs of nitrogen containing nonaromatic heterocycles
04/18/1995US5407938 Certain 1-methyl-piperidine-4-spiro-4'-(1'-3'-oxazolines) and corresponding -(1',3' thiazolines)
04/18/1995US5407658 Analogs of cytochalasin B as radiopharmaceuticals for nuclear imaging of trans-membrane glucose transport
04/18/1995CA1335289C Piperidinyl benzisoxazole derivatives, their production and pharmaceutical use
04/12/1995EP0647641A1 Substituted heterocyclylisoquinolinium salts and compositions and methods of usethereof
04/12/1995EP0647228A1 Asymmetric hydrogenation of furoimidazole derivatives.
04/12/1995EP0647220A1 Ring-closed dihydropyridines and their use in the preparation of pharmaceutical compositions
04/12/1995EP0647137A1 Glycine receptor antagonists and the use thereof
04/11/1995US5405963 Reacting chiral cis dioxolanone having acid group with pyrrolo/3,4-b/quinoline having secondary amine function, converting to camptothecin analogue
04/11/1995US5405844 Tetracyclic antibiotics and processes for their preparation
04/08/1995CA2132766A1 4-arylamino-benzopyran and related compounds
04/06/1995WO1995009169A1 Process for the preparation of 9-amino camptothecin
04/06/1995WO1995009159A1 Quinoxaline derivative as antidiabetic agent
04/06/1995WO1995009152A1 Process for the preparation of sufentanil derivatives by carbene addition/aminolysis of 4-piperidone
04/06/1995CA2150345A1 Quinoxaline derivative as antidiabetic agent
04/05/1995EP0646126A1 Novel steroids with pregnane skeleton, pharmaceutical compositions containing them and process for preparing same
04/05/1995EP0646117A1 Methods and intermediates for the asymmetric synthesis of camptothecin and camptothecin analogs
04/05/1995EP0646115A1 Heterocyclic-cyclic amine derivatives
04/05/1995EP0387357B1 Indolenine derivatives
04/05/1995CN1101047A Intermediates useful in the preparation of pyranyl cyanoguanidine derivatives and methods of preparing same
04/05/1995CN1101039A 哌嗪衍生物 Piperazine derivatives
04/04/1995US5403931 (-)-(S)-2,8-dimethyl-3-methylene-1-oxa-8-azaspiro[4.5]decane L-tartrate
04/04/1995US5403843 Antitumor agents
04/04/1995US5403702 Crystals consisting of an indolinospirobenzopyran derivative
03/1995
03/29/1995EP0645391A2 Aminobenzoic acid derivatives
03/29/1995EP0644882A1 Novel piperzinyl-bis(alkylamino)pyrimidine derivatives and process for preparing same
03/29/1995CN1100725A 2-amino-4-heteroaryl-1,4-dihydropyridines, processes for their preparation and their use in medicaments
03/29/1995CN1027999C Process for preparation of heribicidal sulfonamides
03/28/1995US5401747 Antitumor agents or antileukemia agents and as inhibitors of topoisomerase
03/23/1995WO1995007918A2 Pyrimidine derivatives for labeled binding partners
03/23/1995WO1995007901A1 Substituted tetronic acids useful for treating hiv and other retroviruses
03/23/1995WO1995007894A1 Substituted pyridines and pyrimidines, process for producing them and their use as pesticides and fungicides
03/23/1995CA2168757A1 Substituted tetronic acids useful for treating hiv and other retroviruses
03/22/1995CN1100420A 2,6-disubstituted 4-quinolyl-dihydropyridines
03/22/1995CN1100419A 3-quinolyl-substituted dihydropyridines, process for their preparation and their use in medicaments
03/21/1995US5399725 Forming alcohol-amides by reacting a 7-oxabicycloheptane imide with a 2-/2-metallated phenyl/-1,3-dioxolane /metal is lithium or magnesium bromide/ and reducing the product
03/21/1995US5399707 Making salt of amino acid lysine, arginine or histidine with alpha-arylcarboxylic acid either by starting from second salt of anion and protonated cation of amino acid or by distilling water from amino acid-arylcarboxylic acid mixture
03/21/1995US5399582 Antiparasitic agents
03/16/1995WO1995007275A1 Photochromic compounds, methods and intermediates for producing them and their use
03/16/1995WO1995007269A1 Polar-substituted hydrocarbons
03/16/1995WO1995007262A1 Fused tricyclic heteroaromatic derivatives as dopamine receptor subtype ligands
03/16/1995WO1995007260A1 Tetrahydroisoquinolines as alpha-2 antagonists and biogenic amine uptake inhibitors
03/16/1995CA2171471A1 Polar-substituted hydrocarbons
03/16/1995CA2168738A1 Fused tricyclic heteroaromatic derivatives as dopamine receptor subtype ligands
03/15/1995EP0642516A1 Macrocyclic immunomodulators
03/15/1995EP0642502A1 Fungicidal imidazolinones
03/15/1995CN1100099A Quinolyl-dihydropyridine esters, processes for their preparation, and their use in medicaments
03/15/1995CN1100098A 2-amino-4-quinolyl-dihydropyridines, processes for their preparation, and their use
03/15/1995CA2131967A1 Substituted heterocyclylisoquinolinium salts and compositions and method of use thereof
03/14/1995US5397792 Process for trans-6-[2-(substituted-pyrrol-1-yl)alkyl]pyran-2-one inhibitors of cholesterol synthesis
03/14/1995US5397791 Fibrinogen receptor antagonists
03/14/1995US5397785 4-acylaminopyridine derivative
03/14/1995US5397783 Antidepressants, anxiolytic agents
03/14/1995CA1334755C Benzopyranopyridineacetic acid ester compounds and their pharmaceutical uses
03/14/1995CA1334754C 5-aryl-substituted-2,3-dihydro-imidazo¬1,2-a|furo and -thieno pyridines
03/09/1995WO1995006640A1 Carbocyclic and heterocyclic fused-ring quinolinecarboxylic acids useful as immunosuppressive agents
03/09/1995CA2170349A1 Carbocyclic and heterocyclic fused-ring quinolinecarboxylic acids useful as immunosuppresive agents
03/08/1995EP0641770A1 Novel compound with platelet aggregation inhibitor activity
03/08/1995EP0641345A1 Hypoglycemic n-sulfonyl-tetrahydro- 1,3]-dioxepino 5,6-b]azirines
03/08/1995EP0641343A1 4-mercaptoacetylamino- 2] benzazepinone(3) derivatives, and use as enkephalinase inhibitors
03/08/1995EP0641323A1 Carbostyril derivatives as matrix metalloproteinases inhibitors
03/08/1995EP0641304A1 Stereo-selective synthesis of 2-aryl-propionic acids of high optical purity by using chiral oxazolines
03/08/1995EP0641207A1 Enantiomeric cynemicin analogs, preparation and use thereof
03/08/1995EP0561845B1 Pyrido-anellated 4-oxo-4h-benzopyrans, a method of preparing them, and their use as antidotes
03/08/1995CN1099617A Antitussive
03/07/1995US5395952 Nonphytotoxic
03/07/1995US5395944 7-(aminomethyl-oxa-7-aza-bicyclo[3.3.0]oct-7-yl)quinolonecarboxylic and 7-(aminomethyl-oxa-7-aza-bicyclo[3.3.0]oct-7-yl)naphthyridone-carboxylic acid intermediates
03/07/1995US5395939 Dioxane intermediate
03/02/1995WO1995003303A3 Aza spiro compounds acting on the cholinergic system with muscarinic agonist activity
03/01/1995EP0640605A1 Spiropyran compound, optically active spiropyran compound, and use thereof
03/01/1995EP0640087A1 Use of tricyclic pyrimidine derivatives as anti-viral medicaments