Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
06/1993
06/16/1993EP0546475A1 Biologically active pseurotin A and D, new metabolites from Aspergillus fumigatus, process for their preparation and their use as apomorphine antagonists
06/16/1993EP0546474A1 Pseurotin F1/F2, new metabolites from Aspergillus fumigatus, process for their preparation and their use as apomorphine antagonists
06/16/1993EP0546164A1 Indole derivatives, pharmaceutical compositions and methods of treating neurological and psychiatric disorders
06/15/1993US5219848 Cephem compounds
06/09/1993EP0545204A1 2-cyanobenzimidazoles, process for their preparation and their use in agriculture and new precursors
06/08/1993US5218121 Reacting protected 1-deoxynojirimycin with dialkyltin oxide, acylating, benzylating or allylating, oxidizing, reducing, fluorinating, deprotecting
06/08/1993US5218119 Process for preparing the octahydro-indolo[2,3-a] quinolizine diester derivatives
06/08/1993US5217975 Azabicyclic compounds for treating dementia
06/08/1993US5217961 Condensed quinoline system N-glycosides
06/08/1993CA1318874C Process for preparing optically active hydantoins
06/02/1993EP0543930A1 Arthropodicidal pyrazolines, pyrazolidines and hydrazines
06/02/1993EP0369000A4 Macrocyclic complexes of yttrium, the lanthanides and the actinides having peripheral coupling functionalities
06/02/1993CN1072683A 水溶性喜树碱衍生物 Water-soluble derivative of camptothecin
06/01/1993US5216175 Polyoxoheterocyclic tetracylic derivatives
06/01/1993US5216168 2- and 3- amino and azido derivatives of 1,5-iminosugars
06/01/1993US5216159 Certain cycloalkyl and azacycloalkyl pyrrolopyrimidines; a new class of GABA brain receptor ligands
06/01/1993US5216150 Muscle relaxant; enzyme inhibitor and platelet aggutination inhibitor
05/1993
05/27/1993WO1993010120A1 Marcfortine/paraherquamide derivatives useful as antiparasitic agents
05/27/1993CA2121234A1 Marcfortine/paraherquamide derivatives useful as antiparasitic agents
05/26/1993EP0543516A1 Hapalindole alkaloids as antifungal and antitumor agents
05/19/1993EP0542609A1 3-sulfonylamino-2-(1H)-quinolinones and 7-aza derivatives as excitatory amino acids antagonists
05/19/1993EP0542554A1 Substituted N-biphenylyl lactams
05/19/1993EP0542411A2 Tetrahydrothienopyridine derivatives, furo and pyrrolo analogs thereof and their preparation and uses for inhibiting blood platelet aggregation
05/18/1993US5212317 Methods and intermediates for the assymmetric synthesis of camptothecin and camptothecin analogs
05/18/1993US5212177 Indole and benzimidazole-substituted dihydropyrimidine derivatives
05/18/1993CA1317957C Process for the preparation of 1-alkyl-3-carboxy-4- cinnolones
05/18/1993CA1317940C Substituted n-(1-alkyl-3-hydroxy-4-piperidinyl)benzamides
05/18/1993CA1317938C Benzazapin derivatives
05/15/1993CA2082856A1 3-sulfonylamino-2-(1h)-quinoleinone derivatives, process for their preparation and pharmaceutical compositions containing them
05/14/1993CA2082787A1 Substituted n-biphenylyl lactams
05/13/1993WO1993009098A1 Novel 4-cinnolinone derivatives, their preparation and application in therapy
05/11/1993US5210213 Dimensional, crosslinkable oligomers
05/11/1993US5210088 Method of treatment and heterocyclic compounds used therein
05/11/1993CA1317590C 2-substituted-e-fused-¬1,2,4|triazolo¬1,5- c|pyrimidines, pharmaceutical compositions, and uses thereof
05/05/1993EP0540468A1 NIR-dyes, method for their preparation and their use
05/05/1993EP0540099A1 Water soluble camptothecin derivatives
05/05/1993EP0539372A1 Therapeutic agents
05/05/1993EP0502060A4 Spatially-addressable immobilization of anti-ligands on surfaces
05/04/1993US5208342 Conversion of pyridine-2,3-dicarboxylic acid esters to cyclic anhydrides
05/04/1993US5208330 Cognition activators
05/04/1993CA1317292C Derivatives of (1-hydroxy-2-piperidylalkyl)-indol-2-ones, 2-quinolinones, 2-benzo[b]azapinones, benzimidazol-2-ones, and quinazolin-2-ones, their preparation and their applicationin therapeutics
05/01/1993CA2081641A1 Nir dyes, methods of preparing them and their use
04/1993
04/30/1993CA2081580A1 Water soluble camptothecin derivatives
04/30/1993CA2081510A1 Alkaloids and processes for their production
04/29/1993WO1993008189A1 Chemical reactions on camptothecin or analogs
04/29/1993WO1993008170A1 Substituted heterocycles as angiotensin ii antagonists
04/29/1993CA2121816A1 Substituted heterocycles as angiotensin ii antagonists
04/28/1993EP0538534A1 Improved process for chemical reactions on camptothecin or analogs thereof
04/27/1993US5206387 Fused heteroalkylene quinolinamines
04/27/1993US5206382 Indole derivatives, pharmaceutical compositions and methods of treating neurological and psychiatric disorders
04/27/1993US5206365 Psychotropic heterobicycloalkylpiperazine derivatives
04/27/1993US5206258 Use of heteroaryl-3-oxo-propanenitrile derivatives in treating clinical wherein myelopoiesis suppression occurs
04/27/1993US5206251 Viricide
04/27/1993US5206240 Nitrogen-containing spirocycles
04/21/1993CN1071164A 含氮杂环化合物 Nitrogen-containing heterocyclic compounds
04/20/1993US5204473 Photostabilizers
04/20/1993US5204472 Quinoline and isoquinoline intermediates
04/15/1993WO1993007128A1 Cyclic ureas and analogues useful as retroviral protease inhibitiors
04/15/1993WO1993007125A1 2-substituted quinolines for treating leishmanioses
04/15/1993WO1993007124A1 Nitrogenous heterocyclic compound
04/15/1993DE4231565A1 Bis-imide(s) of halo-substd.-(di)oxy:di:phthalic acids
04/15/1993CA2120925A1 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors
04/15/1993CA2116336A1 Nitrogenous heterocyclic compound
04/14/1993EP0536119A1 Immunoregulatory agents
04/14/1993CN1070907A Process for preparation of 4-substituted-1, 4-dihydropydrines
04/13/1993US5202486 Tetrahydroethanonaphthaleneamine derivatives
04/13/1993US5202440 Cholinesterase inhibitors for treatment of alzheimer*s disease
04/13/1993US5202328 Substituted fused pyrimidinones
04/07/1993EP0535925A1 (Bicyclic-hetero-arylmethoxy)indoles as inhibitors of leukotriene biosynthesis
04/07/1993EP0535645A2 Carbamate derivatives of 4-amino-3-isoxazolidinones, 3-amino-1-hydroxypyrrolidin-2-ones and 1-amino-1-cyclopropanecarboxylic acid analogs, a process for their preparation and their use as medicaments
04/07/1993EP0535548A1 Inhibitor of atherosclerotic intimal thickening
04/06/1993US5200524 Camptothecin intermediates and method of making same
04/06/1993US5200420 2,6-dialkyl-4-(benzothiazol- or benzoxazol-4-yl-1,4-dihydropyridines
04/06/1993CA1315781C 1,4-diazepine derivatives having anti-ulcer activity
04/01/1993WO1993006105A1 Substituted phenserines and phenylcarbamates of (-)-eseroline, (-)-n1-noreseroline, and (-)-n1-benzylnoreseroline; as specific inhibitors of acetylcholinesterase
04/01/1993WO1993006082A1 Process for the preparation of 4-substituted-1,4-dihydropyridines
03/1993
03/31/1993EP0534859A1 Benzocyclobutyl- or indanyl-alkyl-amino-alkyl substituted 3-benzazepin-2-ones useful in the treatment of cardiovascular diseases
03/31/1993EP0534520A2 Process for the preparation of 4-substituted-1,4-dihydropyridines
03/31/1993EP0534443A1 3,6-Disubstituted pyridazine derivatives
03/30/1993US5198434 Angiotensin ii antagonizing fused pyridinyloxy containing derivatives
03/27/1993CA2078699A1 3,6-disubstituted pyridazine derivatives
03/24/1993EP0532531A1 Phenol and pyridinol derivatives as pharmaceuticals
03/23/1993US5196445 Heteroaryl-3-oxo-propanenitrile derivatives useful in the treatment of rheumatoid arthritis and other autoimmune diseases
03/23/1993US5196434 Antidepressants, anxiolytic agents
03/23/1993CA1314885C Tricyclic derivatives which are agonists of cholinergic receptors, and drugs in which they are present
03/23/1993CA1314881C Anti-anxiety agents
03/23/1993CA1314879C Anellated indole derivatives
03/18/1993WO1993005045A1 Spirocyclic benzopyran imidazolines
03/18/1993WO1993005043A1 Novel isatinoxime derivatives, their preparation and use
03/18/1993WO1993004682A1 Novel 4-arylpiperazines and 4-arylpiperidines
03/18/1993WO1993004680A1 Macrocyclic immunomodulators
03/18/1993CA2113818A1 Spirocyclic benzopyran imidazolines
03/18/1993CA2095847A1 Novel 4-arylpiperazines and 4-arylpiperidines
03/17/1993EP0532100A1 Benzodioxinopyrrole derivative as alpha 2-adrenoreceptor antagonist
03/17/1993CN1020103C 2,3,4,5,6,7-hexahydro-2,7-methylene-1,5-benzoxazonin and 1,4-benzoxazonin
03/14/1993CA2077919A1 Process for the preparation of 4- substituted-1, 4-dihydropydrines
03/12/1993WO1993004684A1 Novel 4-arylpiperazines and 4-arylpiperidines
03/12/1993CA2095826A1 4-arylpiperazines and 4-arylpiperidines
03/10/1993EP0530537A1 Condensed pyrimidine derivatives, their production and use as antitumor agents
03/10/1993EP0530264A1 Arthropodicidal tetrahydropyridazines.