Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
11/1995
11/23/1995WO1995031464A1 New agonist compounds
11/23/1995WO1995031463A1 New antagonist compounds
11/23/1995CA2189139A1 New agonist compounds
11/22/1995EP0683166A1 3-Indolylpiperidines
11/22/1995EP0682657A1 9H-INDENO[1,2-b]PYRAZINE-3(4H)-ONES AND 9H-INDENO[1,2-b]PYRAZINE-2,3(1H,4H)-DIONES AND THEIR PREPARATION AND USE
11/22/1995CN1112116A Novel sulfonamidodioxepanes, methods of preparation, intermediates, salts and use thereof
11/21/1995US5468859 Process for asymmetric total synthesis of camptothecin analogues
11/21/1995US5468754 Anticarcinogenic agents
11/21/1995US5468748 Nervous system and psychological disorders; antagonize glycine binding site on N-methylaspartic acid receptor complex
11/16/1995WO1995030677A1 Substituted benzimidazoles for pest control
11/16/1995WO1995030642A1 Combinatorial dihydrobenzopyran library
11/16/1995WO1995030641A1 Nitro compounds and their compositions having anti-inflammatory, analgesic and anti-thrombotic acitivities
11/16/1995CA2189634A1 Combinatorial dihydrobenzopyran library
11/15/1995EP0681571A1 Spiro-substituted azacycles as tachykinin receptor antagonists
11/15/1995CN1111629A 5-vinyl- and 5-ethinyl-quinolone- and -naphthyridone-carboxyhic acids
11/14/1995US5466797 Intermediates for the preparation of cyclic urea
11/14/1995CA2045481C Immunosupressing agent and process of producing the same
11/09/1995WO1995029920A1 Khellactone derivatives and related compounds, process for their preparation and their use as antiviral and immunostimulating agents
11/09/1995WO1995029919A1 Preparation of a camptothecin derivative by intramolecular cyclisation
11/09/1995WO1995029918A1 Substituted (1,4)dioxino(2,3-f)benzoimidazole derivatives and their use in pest control
11/09/1995WO1995029917A2 Intermediates in pharmaceutical camptothecin preparation
11/09/1995WO1995029907A1 Benzofuran derivatives useful as inhibitors of bone resorption
11/09/1995DE4416116A1 Substituierte Benzimidazole Substituted benzimidazoles
11/09/1995DE4415435A1 Benzimidazol-Derivate Benzimidazole derivatives
11/08/1995EP0680953A1 1-[Styryl]- and 1-[2'-(heteroaryl)-ethenyl]-isoquinoline derivatives, a process for preparing them as well as medicaments containing them and the use of them
11/08/1995EP0680481A1 Derivates of azaanthraquinone and azaxanthone, herbicides and plant growth regulators containing the same
11/08/1995EP0680326A1 Pharmaceutical composition for treating nicotine dependence.
11/08/1995CN1111247A Protein kinase C inhibitors
11/08/1995CN1111245A Galanthamine derivatives, a process for their preparation and their use as medicaments
11/07/1995US5464859 Benzospiroalkene derivatives
11/07/1995US5464841 Use of delta opioid receptor antagonists to treat immunoregulatory disorders
11/04/1995CA2148412A1 1-¬styryl|- and 1-¬2'-(heteroaryl) -ethenyl| -isoquinoline derivatives, a process for preparing them as well as medicaments containing them and the use of them
11/02/1995WO1995029177A1 Tricyclic derivatives as 5ht2c and 5ht2b antagonists
11/02/1995EP0679640A1 Carboxylate and heat-sensitive recording material using same
11/02/1995EP0679396A1 Use of 3-substituted-2-oxidole-1-carboxamides for the manufacture of a medicament in the treatment and prevention of ischemia induced myocardial injury and cytokine mediated myocardial injury
10/1995
10/31/1995US5463076 Crosslinking phenylimide end caps condensed onto aromatic hub through ether linkages
10/31/1995US5463059 Process for the preparation of intermediates useful in the preparation of pyranyl cyanoguanidine derivatives
10/31/1995US5463054 Certain aryl fused pyrrolopyrimidines; a new class of GABA brain receptor ligands
10/31/1995US5463027 Fluorescence polarazation immunoassay for tetrahydrocannabinoids
10/31/1995US5463008 Polyorthocarbonates
10/31/1995US5462941 1-(cyclohexylalkylamino)-4-(phenyl, thienyl, or furyl) phthalazines; anti-platelet agglutination agents for treatment or prevention of cerebro- or cardiovascular disorders
10/26/1995WO1995028404A1 7,11 disubstituted camptothecin derivatives, formulations containing such derivatives and their use
10/26/1995WO1995028397A1 Alpha1c adrenergic receptor antagonists
10/26/1995WO1995028389A1 Spiro compound and medicinal composition thereof
10/26/1995CA2187767A1 Alpha1c adrenergic receptor antagonists
10/25/1995EP0678517A1 Spiropyrone compounds
10/25/1995EP0678507A1 Method for preparing homochiral maleimide intermediates, via silylation techniques, used in the enantioselective preparation of anti-thrombotic and anti-vasospastic compounds
10/25/1995EP0678025A1 Transdermal treatment of cancer with water-insoluble s-camptothecin of the closed lactone ring form
10/25/1995CN1110685A Nitrogen-containing spirocycles
10/25/1995CN1110680A Substituted 1H-3-aryl-pyrrolidine-2,4-diones derivative
10/24/1995US5461062 Condensed imidazopyridine derivatives
10/24/1995US5461061 Antidepressants
10/24/1995US5461050 Antiallergens
10/24/1995US5461026 Pyridine sulfonyl urea derivatives
10/24/1995US5461025 Benzenesulfonylurea derivatives
10/24/1995US5461024 Herbicides
10/24/1995CA1337423C 5(and/or 6)substituted 2-(2-imidazolin-2-yl)nicotinic acids, esters and salts, useful as herbicidal agents and novel intermediates for the preparation of said nicotinic acids, esters and salts
10/24/1995CA1337419C (2-imidazolin-2-yl) fused heteropyridine compounds, intermediates for the preparation of and use of said compounds as herbicidal agents
10/21/1995CA2146038A1 Method for preparing homochiral maleimide intermediates, via silylation techniques, used in the enantioselective preparation of anti-thrombotic and anti-vasospastic compounds
10/19/1995WO1995027914A1 Photochromic naphthopyran compounds
10/19/1995WO1995027715A2 Method of manufacture of (-)galanthamine in high yield and purity substantially free of epigalanthamine
10/19/1995WO1995027714A1 Active compounds
10/19/1995WO1995027713A1 Process for the resolution of etodolac using glucamine derivatives
10/19/1995WO1995027698A1 Herbicidal bicyclic and tricyclic imides
10/19/1995CA2187440A1 Herbicidal bicyclic and tricyclic imides
10/17/1995US5459269 Antitumor agents, antileukemic
10/17/1995US5459227 Aminoimides
10/17/1995US5459137 Muscle relaxants, anticonvulsants, neuroprotective agents
10/17/1995US5459129 Condensed heterocyclic compounds, their production and use
10/17/1995CA1337350C Herbicidal 2-(2-imidazolin-2-yl)-fluoroalkoxy-, alkenyloxy- and alkynyloxypyridines and quinolines
10/17/1995CA1337349C Dihydroimidazopyrrolopyridines, quinolines, thieno- and furopyridines
10/12/1995WO1995026954A1 Alkoxy-alkyl-substituted 1-h-3-aryl-pyrrolidine-2,4-diones used as herbicides and pesticides
10/12/1995WO1995021169A3 PROCESS FOR ISOMERIZATION OF SPIROCYCLIC COMPOUNDS WITH β-AMINOCARBOXYL AND/OR β-AMINOCARBONYL SYSTEMS
10/12/1995CA2187015A1 Alkoxy-alkyl-substituted 1-h-3-aryl-pyrrolidine-2,4-diones used as herbicides and pesticides
10/11/1995EP0676401A1 Annelated spirofluorene-2H-benzopyrans and their use in ophthalmic optics
10/11/1995EP0675889A1 Antiallergic triazolo(pyrrolo, thieno or furano)azepine derivatives
10/10/1995US5457119 A89271 factors and processes for their production
10/10/1995US5457111 Macrocyclic immunomodulators
10/10/1995US5457105 Quinazoline derivatives useful for treatment of neoplastic disease
10/05/1995WO1995026352A1 IMIDAZO[1,2-a]PYRAZINE-4-ONE DERIVATIVES, PREPARATION THEREOF AND DRUGS CONTAINING SAME
10/05/1995WO1995026351A1 1,2,4-TRIAZOLO[4,3-a]PYRAZINE-4-ONE DERIVATIVES, PREPARATION THEREOF AND DRUGS CONTAINING SAME
10/05/1995WO1995026349A1 INDENO[1,2-e]PYRAZINE-4-ONES, PREPARATION THEREOF AND DRUGS CONTAINING SAME
10/03/1995CA1337200C .beta.-carbolines, their bio-isosteric benzofuran and benzothiophene analogues having cytostatic properties
09/1995
09/28/1995WO1995025730A1 Nicotinic acid derivative and herbicide
09/28/1995WO1995025719A1 N-aryl and n-alkylsulphonylaminals as pesticides
09/28/1995DE4413659A1 N-Aryl- und N-Alkylsulfonylaminale N-aryl and N-Alkylsulfonylaminale
09/28/1995CA2185916A1 N-aryl and n-alkylsulphonylaminals as pesticides
09/27/1995EP0673928A1 Novel N-(3,4-dichlorophenyl-propyl)-piperidine derivatives as selective human NK3-receptor antagonists
09/27/1995EP0673380A1 Water soluble camptothecin derivatives
09/27/1995EP0673378A1 New triazolopyrimidones, their preparation and their use.
09/27/1995EP0673373A1 Bicyclic compounds with pharmaceutical activity
09/27/1995EP0673246A1 Use of alkylthiopyridines for controlling helicobacter bacteria
09/26/1995US5453471 Gas phase polymerization process
09/26/1995US5453424 Antiarrhythmia
09/26/1995US5453422 Animal growth promoters
09/21/1995WO1995025106A1 Oxazolidinone derivatives and pharmaceutical compositions containing them
09/21/1995WO1995024903A1 The use of amino hydrogenated quinazoline compounds and derivatives thereof for abstaining from drug dependence
09/20/1995EP0672660A2 Substituted cyclohexanol-esters, their use to treat illnesses and pharmaceutical preparations
09/20/1995EP0672047A1 ANTIALLERGIC IMIDAZO 1,2-a](PYRROLO, THIENO OR FURANO) 2,3-d]AZEPINE DERIVATIVES
09/20/1995EP0672046A1 Spirofuranone derivatives and their use in the treatment of neurodegenerative disorders