Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
02/1996
02/04/1996CA2155092A1 Benzoxazolyl- and benzothiazolyloxazolidinones
02/01/1996WO1996002546A1 Water-soluble esters of camptothecin compounds
02/01/1996WO1996002545A1 Heterocycle-condensed morphinoid derivatives
02/01/1996WO1996002536A1 4-hydroxy-3-phenyl-indeno(1,2-b)pyridine-2(1h)-one derivatives as nmda antagonists
02/01/1996WO1996002524A1 Phenylcarbamate derivatives suitable to the use as anticholinesterase substances
02/01/1996CA2194877A1 Heterocycle-condensed morphinoid derivatives
01/1996
01/31/1996EP0694035A1 Water-soluble camptothecin derivatives, process for their preparation and their use as antitumor agents
01/31/1996CN1115759A Tricyclic carboxylate
01/30/1996US5488054 Treatment of restenosis
01/25/1996WO1996001827A1 Tetracyclic derivatives and their use as antitumour agents
01/24/1996EP0693283A1 Heart failure remedy
01/24/1996EP0693069A1 Novel polycyclic systems, and derivatives thereof, as neurotransmitter release enhancer useful in the treatment of cognitive disorders
01/23/1996US5486615 Method of making asymmetric DE ring intermediates for the synthesis of camptothecin analogs
01/23/1996US5486532 Adrenergic agonist
01/23/1996US5486524 Restenosis
01/23/1996US5486523 Antiinflammatory
01/23/1996US5486522 Carbamates of rapamycin
01/23/1996US5486516 Furopyrimidine derivatives
01/23/1996US5486512 Learning enhancement
01/21/1996CA2154097A1 N-(substituted amino)imide derivatives, preparation process thereof, and herbicidal composition
01/18/1996WO1996001113A1 Method and medicine for alleviating jet lag
01/18/1996CA2193473A1 Method and medicine for alleviating jet lag
01/17/1996EP0691972A1 FURO 3,2-b]PYRIDINES AND THIENO 3,2-b]PYRIDINES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS
01/17/1996EP0691971A1 7-azabicyclo- 2.2.1]-heptane and -heptene derivatives as analgesics and anti-inflammatory agents
01/17/1996EP0691965A1 Photochromic naphthopyran compounds
01/17/1996EP0537313B1 Arylalkyl esters of 4,5-dihydroxy-9,10-dihydro-9,10-dioxo-2-anthracenecarboxylic acid having therapeutical activity
01/17/1996CN1115181A Process for the preparation of 9-amino camptothecin
01/16/1996US5484925 Synthesis of (-)-swainsonine and intermediate compounds employed in such synthesis
01/16/1996US5484923 Process of making spirocycles and analogs thereof
01/16/1996US5484791 Carbamates of rapamycin
01/16/1996US5484790 Carbamates of rapamycin
01/16/1996CA1337937C Tricyclic 3-oxo-propanenitrile derivatives and process for their preparation
01/11/1996WO1996000730A1 Vitronectin receptor antagonists
01/11/1996WO1996000728A1 Processes and intermediates for the preparation of cyclic urea hiv protease inhibitors
01/11/1996WO1996000574A1 Vitronectin receptor antagonists
01/11/1996CA2193966A1 Vitronectin receptor antagonists
01/10/1996EP0691342A1 Benzopyrane derivatives, process for their preparation and pharmaceutical compositions containing them
01/10/1996EP0690863A1 Tetracyclic compounds as dopamine agonists
01/10/1996EP0690843A1 Indoletetralins having dopaminergic activity
01/10/1996EP0613470B1 Novel 4-cinnolinone derivatives, their preparation and application in therapy
01/10/1996CN1114834A Quinoxaline derivative as antidiabetic agent
01/10/1996CN1114651A 3-indolylpiperidine
01/10/1996CN1114650A MDR reversal agents
01/09/1996US5482960 Nonpeptide endothelin antagonists
01/09/1996US5482867 Spatially-addressable immobilization of anti-ligands on surfaces
01/04/1996WO1996000219A1 Pyrimidinyl- and triazinyl-oxy and thio-3-haloalkyl-propionic acid derivatives as herbicides
01/03/1996EP0553130B1 Pyrrolidine dione derivatives
01/02/1996US5480989 Carbamates of rapamycin
01/02/1996US5480988 Carbamates of rapamycin
01/02/1996US5480892 (N-phthalimidoalkyl)piperidines
01/02/1996US5480887 Protease inhibitors
12/1995
12/28/1995WO1995035303A1 Synthesis of conduritol epoxides and aziridines and methods of using such to synthesize higher disaccharides
12/28/1995WO1995029917A3 Intermediates in pharmaceutical camptothecin preparation
12/27/1995EP0688320A1 Tricyclic benzodiazepins, their use and preparation
12/27/1995EP0688211A1 Methods and compositions for inhibition of angiogenesis
12/26/1995US5478949 Reacting the starting carbazolone with dialkyl oxalate, then formaldehyde and 2-methylimidazole
12/26/1995US5478943 Reacting 2-bromo- or 2-iodo-3-hydroxymethylquinoline with 7-oxopyrido(5,4-c)-2-oxo-3-alkyl-3-hydroxy-3,6-dihydropyran by Mitsunobu reaction
12/26/1995US5478937 Chemical intermediates for antiarrhythmia agent, antilipemic agent, vasodilator and hypotensive agent
12/26/1995US5478845 Piperidine derivatives
12/26/1995US5478835 Tricyclic compounds and intermediates thereof
12/26/1995CA1337817C Heterocyclic spiro compounds and methods for preparing the same
12/21/1995WO1995034547A1 C-4 amide substituted compounds and their use as therapeutic agents
12/21/1995WO1995034546A1 Benzopyrans and their use as therapeutic agents
12/21/1995DE4421347A1 High purificn. of perylene-tetra:carboxylic anhydride imide(s)
12/20/1995CN1113491A Novel hydroxylamines with hypoglycemic activity
12/20/1995CN1113490A New acronycine analogues, a process for their preparation and pharmaceutical compositions containing them
12/19/1995US5476859 Antiviral compounds
12/14/1995WO1995033720A1 Novel fused-ring carboxylic acid compound or salt thereof, and medicinal use thereof
12/14/1995WO1995033491A1 Biotin compounds for targetting tumors and sites of infection
12/14/1995CA2192384A1 Biotin compounds for targetting tumors and sites of infection
12/14/1995CA2168858A1 Novel fused-ring carboxylic acid compound or salt thereof, and medicinal use thereof
12/13/1995EP0686637A1 Tetracyclic 1,4-oxazine derivatives, process for their preparation and pharmaceutical compositions containing them
12/13/1995EP0686158A1 Methods for purifying 20(s)-camptothecin
12/13/1995CN1113384A Process for the preparation of 9-amino camptothecin
12/13/1995CN1113228A A process for preparing the intermediate of the derivatives of monocycle beta-lactam antibiotics
12/12/1995US5475110 Treating nervous system disorders and inflammation, inhibiting protein and tyrosine kinases, inhibiting cell growth
12/12/1995US5475108 Camptothecin intermediates and method of making camptothecin and comptothecin analogs
12/12/1995US5475092 Deliver cytotoxic drugs to specific cell population in targeted fashion
12/12/1995US5474998 Arthropodicidal pyrazolines, pyrazolidines and hydrazines
12/07/1995WO1995032985A1 3'-(4'-) nonradioactively tagged nucleosides and nucleotides with aminocarboxylic acid, peptide or carboxylic acid spacer
12/07/1995CA2190982A1 3'-(4'-) nonradioactively tagged nucleosides and nucleotides with aminocarboxylic acid, peptide or carboxylic acid spacer
12/06/1995EP0685465A1 Butine- or hexadiine linked hindered amines as stabilizer
12/06/1995EP0684949A1 Chemical compounds
12/06/1995CN1112926A 1,3 substituted condensed pyrazole compound, the application and prepn. method
12/06/1995CN1112919A Pharmaceutical agents for the treatment of myocardial reperfusion injury and myocardial stunning
12/05/1995US5472974 Benzimidazole derivatives, agricultural and horticultural fungicides containing the same as an active ingredient and intermediate compounds thereof
12/05/1995US5472964 Diaryl 5,6-fused heterocyclic acids as leukotriene antagonists
12/03/1995CA2150644A1 Butyne-linked or hexadiyne-linked hindered amines as stabilisers
11/1995
11/30/1995WO1995032207A1 Method for the preparation of 9-amino camptothecin
11/30/1995WO1995032206A1 Purpurin-18 anhydrides and imides as photosensitizers
11/30/1995WO1995032205A1 Tricyclic dicarbonyl derivatives
11/30/1995WO1995032187A1 Novel fused indan derivative and pharmaceutically acceptable salt thereof
11/30/1995WO1995027715A3 Method of manufacture of (-)galanthamine in high yield and purity substantially free of epigalanthamine
11/30/1995CA2189776A1 Tricyclic dicarbonyl derivatives
11/29/1995EP0684240A1 Hydroxamic acid derivatives with tricyclic substitution
11/29/1995EP0683782A1 Spiro (2h-1-benzopyran-2, 4' piperidine) class iii antiarrhythmics
11/28/1995US5470981 Process for trans-6-[2-(substituted-pyrrol-1-yl)alkyl]pyran-2-one inhibitors of cholesterol synthesis
11/28/1995US5470872 Muscle relaxants
11/28/1995CA2091986C Certain cycloalkyl and azacycloalkyl pyrrolopyrimidines; a new class of gaba brain receptor ligands
11/28/1995CA2023018C 2-oxo-3,8-diazaspiro /4,5/decane derivatives, pharmaceutical compositions containing them and process for preparing the same