Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
04/1996
04/11/1996CA2199621A1 Substituted aryl piperazines as neurokinin antagonists
04/10/1996EP0705830A1 2,3-Cyclic condensed 1,4-dihydropyridines, process for their preparation and their use as K-channel modulators
04/10/1996EP0705815A1 Process for the preparation of N-arylaminoacrylic acid derivatives and their use for preparing 4-quinolone-3-carboxylic acid derivatives
04/10/1996EP0705262A1 Process for asymmetric total synthesis of camptothecin
04/10/1996EP0705250A1 Bis-imide polycyclic and heterocyclic chromophores useful as tumoricidals
04/10/1996EP0705245A1 Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives
04/10/1996CN1120335A Photochromic naphthopyran compounds
04/10/1996CN1120313A Heart failure remedy
04/09/1996US5506239 Carbostyril derivative and platelets aggregation inhibitory agent
04/09/1996US5506192 Substituted phthalides and heterocyclic phthalides
04/04/1996WO1996010181A1 Compounds and methods for identifying activated platelets
04/04/1996WO1996004323A3 Gas phase production of polydienes
04/03/1996EP0704448A1 Heterocyclic substituted imidazolidines, process and intermediates for their preparation, their use as medicaments and pharmaceutical compositions containing them
04/03/1996EP0703916A1 14-substituted marcfortines and derivatives useful as antiparasitic agents
04/03/1996EP0703901A1 1-substituted isatin and oxindole derivatives as inhibitors of acetylcholinesterase
04/03/1996CN1031461C Resolution process of racemic semi-ester
04/02/1996US5504214 Fluorinated benzotriazoles
04/02/1996US5504210 Treatment for cardiovascular disorders
04/02/1996US5504204 Immunosuppressive, antiinflammatory, antifungal, antiproliferative and antitumor agents
04/02/1996US5504100 Synergistic combination of a 2-cyanobenzimidazole and an azole derivative
03/1996
03/30/1996CA2159425A1 New heterocycle substituted imidazolidines; process and intermediates for preparing them and their use as drugs; pharmaceutical compositions containing the same
03/28/1996WO1996009304A1 Benzopyranopyrazolyl derivatives for the treatment of inflammation
03/28/1996WO1996009058A1 Remedy and preventive for nervous system disorder
03/28/1996CA2202526A1 Therapeutic and prophylactic agent for nervous disturbances
03/27/1996EP0702681A1 Spiro-substituted azacycles as neurokinin antagonists
03/27/1996CN1119189A New benzopyran compounds, process for their preparation and the pharmaceutical compositions which contain them
03/26/1996US5502220 Process for the preparation of intermediates useful in the preparation of pyranyl cyanoguanidine derivatives
03/26/1996US5502193 2-substituted tertiary carbinol derivatives of 1,5-iminosugars
03/26/1996US5502189 Compounds formed from o-hydroxyphenyl-1,3,5-triazines and sterically hindered amines
03/26/1996US5502177 Pyrimidine derivatives for labeled binding partners
03/26/1996US5502072 Substituted oxindoles
03/26/1996US5502062 2-amino-4-quinolyl-dihydropyridines, processes for their preparation, and their use
03/26/1996CA1338190C 8,9-ANNELATED-ß-CARBOLINES AND 8,9-ANNELATED-3, 4-DIHYDRO-.BETA.-CAR BOLINES
03/21/1996DE4432970A1 New tetra:cyclic cpds., e.g. cyclo:alkyl:phenanthrene derivs.
03/20/1996EP0701559A1 Cephalostatin analogues and their use as anti-tumour agents
03/20/1996EP0701558A1 Process of making spirocycles and analogs thereof
03/20/1996EP0701439A1 Stable copper(i) complexes and methods related thereto
03/20/1996EP0638584B1 5-o-desosaminylerythronolide a derivative
03/19/1996US5500438 Arthropodicidal anilides
03/19/1996US5500432 Induction and inhibition of apoptosis
03/19/1996US5500430 Amidic derivatives of glutamic, aspartic and 2-amino adipic acids, a process for preparing same, and anti-gastrin composition containing the derivatives
03/14/1996WO1996007411A1 Novel antiarrhythmic agents
03/14/1996WO1996007409A1 Alkaloids and their antiviral agents
03/13/1996EP0700396A1 Piperidine derivatives, their preparation and use
03/12/1996USRE35177 N-fluoropyridinium salt and process for preparing same
03/12/1996US5498717 6,7-dialkoxy-3,4-diydroisoquinolin-8-yl compounds
03/12/1996US5498625 Substantially pure enantieners of 2-azabicyclo(2.2.1)hept-5-en-3-one
03/07/1996WO1996006610A1 Use of 5-substituted pyridine and hexahydroquinoline-3 carboxylic acid derivatives for treating diseases of the central nervous system
03/07/1996WO1996006606A1 Dihydro-2,3-benzodiazepine derivatives
03/07/1996DE4430639A1 Verwendung von 5-substituierten Pyridin- und Hexahydrochinolin-3-carbonsäurederivaten Use of 5-substituted pyridine and hexahydroquinoline-3-carboxylic acid derivatives
03/07/1996CA2198495A1 Use of 5-substituted pyridine and hexahydroquinoline-3 carboxylic acid derivatives for treating diseases of the central nervous system
03/06/1996EP0699678A1 Crystalline form of dihydro-2,3-benzodiazepine derivative
03/06/1996EP0699677A1 Stereoselective process for producing dihydro-2,3-benzodiazepine derivatives
03/06/1996EP0699676A1 Physical form of dihidro-2,3-benzodiazepine derivative
03/06/1996EP0699201A1 SUBSTITUTED METHYLENEDIOXY 3',4':6,7]INDOLIZINO- 1,2-$i(b)]QUINOLINONES
03/05/1996US5496952 Method of making asymmetric DE ring intermediates for the synthesis of camptothecin and camptothecin analogs
03/05/1996US5496727 Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
03/05/1996CA1338109C Pyridine derivatives and intermediates thereof
02/1996
02/29/1996WO1996006093A1 7-azabicyclo[2.2.1]-heptane and -heptene derivatives as cholinergic receptor ligands
02/29/1996WO1996006085A1 Process for preparing chiral tetracyclic dopaminergic compounds
02/29/1996CA2195676A1 Process for preparing chiral tetracyclic dopaminergic compounds
02/28/1996EP0698023A1 Fibrinogen receptor antagonists
02/27/1996US5495020 Chemical intermediate for bactericides, microbiocides, disinfectants; side effect reduction, absorption
02/27/1996US5494913 Antifungal compounds
02/27/1996US5494887 Ring annulated 5-alkoxy-n-aryl[1,2,4]triazolo[1,5-C]-pyrimidine-2-sulfonamide herbicides
02/26/1996CA2156672A1 2,3-bridged 1,4-dihydropyridines, processes for their preparation and their use as medicaments
02/22/1996DE4418691A1 3'-(4'-) nicht-radioaktiv markierte Nukleoside und Nukleotide mit Aminocarbonsäure-, Peptid- oder Carbonsäure-Spacer 3 '- (4') non-radioactively labeled nucleosides and nucleotides with aminocarboxylic acid, peptide or carboxylic acid-spacer
02/21/1996EP0697421A1 Gas phase polymerization process
02/21/1996EP0697412A1 Benzoxazolyl- and benzo-thiazolyl-oxazolidinones
02/20/1996US5492902 Biodegradable, nontoxic
02/15/1996WO1996004323A2 Gas phase production of polydienes
02/15/1996WO1996004322A1 Gas phase production of polydienes
02/15/1996WO1996004321A1 Gas phase polymerization process
02/15/1996WO1996004286A1 Process for making quinolonyl lactam antimicrobials and novel intermediate compounds
02/15/1996WO1996004284A1 Insecticidal polycyclic compounds
02/15/1996WO1996004283A1 New 3-substituted 3h-2,3-benzodiazepine derivatives, their preparation and use as medicaments
02/15/1996WO1996003987A1 Lactone compounds for treating patients with precancerous lesions
02/15/1996CA2196676A1 Gas phase production of polydienes
02/15/1996CA2196675A1 Gas phase polymerization process
02/15/1996CA2196664A1 Gas phase production of polydienes
02/15/1996CA2172710A1 Lactone compounds for treating patients with precancerous lesions
02/14/1996EP0696589A1 N-(substituted amino)imide derivatives, preparation process thereof, and herbicidal compositions
02/14/1996EP0696582A1 Polycyclic spirophthalimide derivatives, process for their preparation and their use as fulgimides
02/14/1996EP0696285A1 Water soluble derivatives of camptothecin and their use as antitumor agents
02/13/1996US5491237 Catalytic dehydroxylation, oxidation, enzymatic acylation, catalytic isomerization, cyclization, intramolecular heck reaction
02/13/1996EP0705262A4 Process for asymmetric total synthesis of camptothecin
02/08/1996WO1996003124A1 Dynemicin analogs
02/08/1996DE4428835A1 Neue 3-substituierte 3H-2,3-Benzodiazepinderivate, deren Herstellung und Verwendung als Arzneimittel New 3-substituted 3H-2,3-benzodiazepine derivatives, their preparation and use as medicaments
02/07/1996EP0695302A1 3-halo-3-heteroaryl carboxylic acid derivatives, methods of preparing them and intermediates used in their preparation
02/07/1996EP0695296A1 3-(hetero)aryloxy(thio) carboxylic acid derivatives, method of preparing them and intermediates used in their preparation
02/07/1996EP0695295A1 3-(hetero)aryl carboxylic acid derivatives, methods of preparing them and intermediates used in their preparation
02/07/1996EP0672029A4 SELECTIVE PRECIPITATION OF -g(a)-ARYL CARBOXYLIC ACID SALTS.
02/06/1996US5489691 Cyclization; decyclization; hydrolysis; neutralization; salt formation
02/06/1996US5489690 Process for trans-6[2-(substituted-pyrrol-1-yl)alkyl]pyran-2-one inhibitors of cholesterol synthesis
02/06/1996US5489689 Preparation of piperidine derivatives
02/06/1996US5489688 Process for preparing trans-piperidine-2,5-dicarboxylates
02/06/1996US5489685 Method of synthesizing furo[2,3-b]pyridine carboxylic acid esters
02/06/1996US5489680 Carbamates of rapamycin
02/06/1996US5489595 Carbamates of rapamycin
02/06/1996US5489593 Anti-aids piperazines