Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
09/2003
09/24/2003CN1443766A Method for preparing cis-1,3-dibenzylimidazoline-2-ketone-2H-furano [3,4-d] imidazol-2,4,6-triuetone (I)
09/23/2003USRE38257 Piperdine derivatives and hypotensives containing the same
09/23/2003US6624187 Long wave length absorbing bacteriochlorin alkyl ether analogs
09/18/2003WO2003076938A1 Novel fluorescent label compounds
09/18/2003WO2003076443A1 Spiro compounds with npy antagonistic activity
09/18/2003WO2003076440A1 Condensed heterocyclic compounds as calcitonin agonists
09/18/2003WO2003076424A1 Macrocyclic compounds useful as pharmaceuticals
09/18/2003WO2003076398A2 Pyrrole-2, 5-dione derivatives and their use as gsk-3 inhibitors
09/18/2003WO2003048122A3 Inhibitors of cytosolic phospholipase a2
09/18/2003WO2003022848A3 Process for the preparation of diketopyrrolopyrroles
09/18/2003WO2003011851A3 Aromatic hydroxamic acid derivatives useful as hdac inhibitors
09/18/2003WO2002034745A8 Chemokine receptor binding heterocyclic compounds
09/18/2003US20030176702 N-(azabicyclo moieties)-substituted hetero-bicyclic aromatic compounds for the treatment of disease
09/18/2003US20030176697 Such as 2-(methylsulfanyl)-6-(3,5-dimethyoxyphenyl)-8-ethyl-8H-pyrido(2,3-d) -pyrimidine-7-one; antitumor agents; calcium channel blockers
09/18/2003US20030176520 4-cyanocoumarin derivatives and uses thereof
09/18/2003US20030176476 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
09/18/2003US20030176464 Phenyl substituted 4-hydroxy tetrahydroxypyridone
09/18/2003US20030176463 For therapy of disease states resulting from angiogenesis; can be administered orally
09/18/2003US20030176454 N-coating heterocyclic compounds
09/18/2003US20030176453 Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use therefor
09/18/2003US20030176433 For therapy and prophylaxis of hepatitis C virus (HCV) infection
09/18/2003US20030176432 Cyclic and heterocyclic N-substituted alpha-iminohydroxamic and -carboxylic acids
09/18/2003US20030176430 For therapy and prophylaxis of Tachykinin-mediated diseases
09/18/2003US20030176422 Pyridoarylphenyl oxazolidinone antibacterials, and related compositions and methods
09/18/2003US20030176370 Anti-viral pyrimidine nucleoside analogues
09/18/2003US20030176324 Derivatives of water insoluble drugs which exhibit good activity and water solubility
09/18/2003CA2482191A1 Spiro compounds with npy antagonistic activity
09/18/2003CA2478110A1 Novel fluorescent label compounds
09/18/2003CA2478065A1 Macrocyclic compounds useful as pharmaceuticals
09/18/2003CA2477984A1 Pyrrole-2, 5-dione derivatives and their use as gsk-3 inhibitors
09/17/2003EP1343827A1 N-alkoxy-4,4-dioxy-polyalkyl-piperidine compounds, their corresponding n-oxides and controlled radical polymerization therewith
09/17/2003EP1343796A2 Compounds and methods
09/17/2003EP1343789A1 Tricyclic derivatives of indole with antiangiogenic activity
09/17/2003EP1343767A2 Synthesis of pancratistatin
09/17/2003EP1343766A1 Cyclization process step in the making of quinolones and naphthyridines
09/17/2003EP1343753A2 Antimicrobial agents
09/17/2003EP1224174B1 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
09/17/2003EP1095021B1 Quinoline derivatives
09/17/2003EP0706526B1 Photochromic compounds
09/17/2003CN1443187A Fused cyclic compounds as modulators of nuclear hormone receptor function
09/17/2003CN1121398C Alicyclic acylated heterocyclic derivatives
09/17/2003CN1121391C Substituted 3-cyano quinolines
09/17/2003CN1121376C Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives and matrix metalloprotease inhibitors
09/16/2003US6620945 Squalene synthetase inhibitors; antilipemic agents, anticholesterol agents
09/16/2003US6620937 Intermediates in the synthesis of camptothecin and related compounds and synthesis thereof
09/16/2003US6620833 Coccidiosis treatment; 4,5-tetrafluoroethylenedioxybenzimidazole derivatives
09/16/2003US6620822 Synergistic mixtures comprising 5,7-dichloro-4-(4-fluoro-phenoxy)-quinoline
09/16/2003US6620546 Ionic composition comprising salt having conductivity of greater than 10-5 S.cm-1 between -30 and 150 degrees C; cation is proton, hydronium, hydroxonium, nitrosonium, ammonium or metal cation; anion is carbanion containing fluorine
09/16/2003CA2231025C Novel compounds of 2-aminoindane, process for their preparation and pharmaceutical compositions containing them
09/16/2003CA2047857C (quinolin-2-ylmethoxy)heterotetrahydrocarbazoles as inhibitors of the biosynthesis of leukotrienes
09/16/2003CA2046429C Imide derivatives, and their production and use
09/12/2003WO2003075091A1 Colour photographic recording material
09/12/2003WO2003074530A1 Bicyclic pyridine and pyrimidine p38 kinase inhibitors
09/12/2003WO2003074527A1 Crystalline polymorphic form of irinotecan hydrochloride
09/12/2003WO2003045942A3 Chemokine receptor antagonists and methods of use thereof
09/12/2003WO2003034987A3 Androgen receptor modulators and methods of use thereof
09/12/2003WO2002004443A3 Heterocycle carboxamides as antiviral agents
09/12/2003WO2001083800A9 Heterologous production of polyketides
09/12/2003CA2477926A1 Crystalline polymorphic form of irinotecan hydrochloride
09/12/2003CA2477721A1 Bicyclic pyridine and pyrimidine p38 kinase inhibitors
09/11/2003WO2003074046A1 Antidepressant
09/11/2003US20030171600 Diaminofluorescein derivatives
09/11/2003US20030171423 Enzyme inhibitor for treating HIV infections in mammals; viricides; patient is suffering from a multi-drug resistant HIV infection; AIDS therapy
09/11/2003US20030171418 Pyranoindazoles and their use for the treatment of glaucoma
09/11/2003US20030171394 Tricyclic dihydropyrazolone and tricyclic dihydroisoxazolone potassium channel openers
09/11/2003US20030171392 Substituted indeno[1,2-c]isoquinoline derivatives and methods of use thereof
09/11/2003US20030171219 2,4,5-trisubstituted phenylketo-enols for use as pesticides and herbicides
09/11/2003US20030170831 Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
09/10/2003EP1342723A1 Indole derivatives and use thereof in medicines
09/10/2003EP1341769A2 Bacterial gyrase inhibitors and uses thereof
09/10/2003EP1341763A2 N-alkoxy-4,4-dioxy-polyalkyl-piperidine compounds, with glycidyl or alkylcarbonyl groups as functional initiators for controlled radical polymerization
09/10/2003EP1341761A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-$g(g) BINDING AGENTS
09/10/2003EP1341540A2 Tyrosine kinase inhibitors
09/10/2003CN1441805A Antitumoral analogue of Et-743
09/10/2003CN1440973A Optical pure analog of camptothecine
09/10/2003CN1440972A Optical pure synthetic intermediate of camptothecine and its preparing method
09/09/2003US6617452 Liquid-liquid extraction being carried out in the first stage at a pH-value of about 4; treating narrow-angle glaucoma, Alzheimer's disease, as well as alcohol and nicotine dependence.
09/09/2003US6617437 Modified oligonucleotide of given formula; useful in diagnostics and therapeutics
09/09/2003US6617335 Multi-drug resistance reversal activities; sensitivity enhancers in cancer chemotherapy.
09/09/2003US6617327 For therapy of depression and other diseases such as obsessive compulsive disorder, panic attacks, generalized anxiety disorder, social anxiety disorder, sexual dysfunction, eating disorders, obesity, addictive disorders
09/09/2003CA2183155C Naphthylisoquinoline alkaloids, pharmaceutical compositions containing them and their use for the treatment of malaria
09/09/2003CA2138026C Novel 1,4-dihydroquinoxaline-2,3-diones and uses therefor as glycine receptor antagonists
09/04/2003WO2003072569A1 1,4-disubstituted benzofused cycloalkyl urea compounds useful in treating cytokine mediated diseases
09/04/2003WO2003072566A1 Fused tricyclic heterocycles useful for treating hyper-proliferative disorders
09/04/2003WO2003072561A1 Benzofuran and benzothiophene derivatives useful in the treatment of hyper-proliferative disorders
09/04/2003WO2003072027A2 Compositions and formulations of 9- nitrocamptothecin polymorphs and methods of use thereof
09/04/2003WO2003062209A3 Substituted quinazolin-4-ylamine analogues as modulators of capsaicin
09/04/2003WO2003047505A3 Topoisomerase poison agents
09/04/2003WO2003045313A3 2-aminoquinoline compounds
09/04/2003WO2002068387A8 Acylated piperidine derivatives as melanocortin-4 receptor agonists
09/04/2003US20030166935 Spiroazabicyclic heterocyclic compounds
09/04/2003US20030166929 Heterocyclic compounds useful as inhibitors of tyrosine kinases
09/04/2003US20030166693 Benzene derivatives and pharmaceutical use thereof
09/04/2003US20030166690 Use of compounds for decreasing activity of hormone-sensitive
09/04/2003US20030166689 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
09/04/2003US20030166671 Amorphous polymorphic forms by grinding or pulverizing; having a distinctive X-ray powder diffraction pattern; anti-tumor and -carcinogenic agents; administered by mouth, intravenous injection and inhalation
09/04/2003US20030166650 E.g., 3-(2-fluorophenyl)-N-(1-(3-morpholin-4-yl)phenyl)-propyl)acrylamide; disorders responsive to opening of KCNQ potassium channels; analgesics; migraine, bipolar disorders, anticonvulsants, antiepileptic, anxiolytic agents
09/04/2003US20030166649 E.g., 4-(2-(1-Benzhydryl-2-(2-((benzylsulfonyl)amino)ethyl)-5-chloro-1H-indol-3 -yl)ethoxy)benzoic acid; inhibitors of phospholipase enzymes, esp. phospholipase A2; antiarthritic and -inflammatory agents; analgesics; rheumatoid diseases
09/04/2003US20030166644 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
09/04/2003US20030166641 Heterocyclic amines such as 1-(3,4-methylenedioxyphenyl)-2-(5 -(3,4-dimethoxyphenyl)pyrimidin-2-yl)- 2,3,4,9-tetrahydro-1H-beta-carboline, used as enzyme inhibitors for prophylaxix of sexual disorders