Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
02/2003
02/18/2003US6521666 Inhibitors of α4 mediated cell adhesion
02/18/2003US6521653 Microbicidal benzotriazoles
02/18/2003US6521620 Suppressing tumors, especially breast cancers; antiproli-ferative agents; arthritis, vascular restenosis, psoriasis and angiogenesis; extremely low cytotoxicity
02/13/2003WO2003011869A1 Radioligands and their use for identifying potassium channel modulators
02/13/2003WO2003011851A2 Aromatic hydroxamic acid derivatives useful as hdac inhibitors
02/13/2003WO2002088146A3 ANTIDEPRESSANT INDOLETETRAHYDROPYRIDINE DERIVATIVES OF 2,3-DIHYDRO-7H-[1,4]DIOXINO[2,3-e]INDOLE
02/13/2003WO2001072754A8 Alkylated imidazopyridine derivatives
02/13/2003US20030033089 Substituted quinazolines and analogs and the use thereof
02/13/2003US20030032652 Hydroxamic and carboxylic acid derivatives
02/13/2003US20030032644 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity
02/13/2003US20030032624 Esterifying camptothecin or a derivative with an aminoalkanoic acid or an imidoalkanoic acid and camptothecin; useful for treating cancer.
02/13/2003CA2449804A1 Aromatic hydroxamic acid derivatives useful as hdac inhibitors
02/12/2003EP1283043A1 Ophthalmic solution
02/12/2003EP1283042A1 Aqueous liquid preparation
02/12/2003EP1282630A1 Hydroxylamine esters as polymerization initiators
02/12/2003EP1003724B1 Substituted quinoline derivatives with antiviral action
02/12/2003EP0947514B1 Novel phenanethridinium derivatives
02/12/2003EP0926146B1 Chromene compounds
02/12/2003EP0863906B1 Heterocyclic dioxethane substrates, process for their preparation and their use
02/12/2003EP0793497B1 Novel enediyne quinone imines and methods of preparation and use thereof
02/11/2003US6518430 Process for the preparation of 5-(substituted)-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-F]quinolines and derivatives thereof
02/11/2003US6518427 Compounds are exceedingly water soluble which is useful in preparing pharmaceutical formulations of these compounds. They are also rapidly converted back to the parent amines in vivo, making them useful as prodrugs of the parent amines.
02/11/2003US6518426 Pyrimidine derivatives and methods of making and using these derivatives
02/11/2003US6518421 Process for the preparation of epothilone analogs
02/11/2003US6518294 Fused pyrazolyl compounds
02/11/2003US6518265 1H-imidazopyridine derivatives
02/11/2003CA2205274C Novel 2,3 disubstituted-(5,6)-heteroarylfused-pyrimidine-4-ones
02/06/2003WO2003010230A1 Method of mass-colouring synthetic materials
02/06/2003WO2003010175A2 Radiolabeled neuropeptide y y5 receptor antagonists
02/06/2003WO2003010169A1 Antidepressant azaheterocyclylmethyl derivatives of 7, 8-dihydro-6h-5-oxa-1-aza-phenanthrene
02/06/2003WO2003010158A1 Novel compounds
02/06/2003WO2003010141A2 Hepatitis c virus polymerase inhibitors with a heterobicyclic structure
02/06/2003WO2003010140A2 Hepatitis c virus polymerase inhibitors with heterobicyclic structure
02/06/2003WO2003010138A2 Piperidine derivatives as antibacterial agents
02/06/2003WO2003009852A1 Tyrosine kinase inhibitors
02/06/2003WO2002079146A3 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
02/06/2003WO2002059112A3 Pyrazole compounds useful as protein kinase inhibitors
02/06/2003US20030028026 Nitrate salts of Salbutamol, Cetirizine, Loratadine, Terfenadine, Emedastine, Ketotifen, Nedocromil, Ambroxol, Dextromethorphan, Dextorphan, Isoniazide, Erythromycin, and Pyrazinamide; respiratory system pathology treatment
02/06/2003US20030028022 Preferably tertiary amines comprising tetrahydroquinoline and benzimidazole; use treating human immunodeficiency virus (HIV) and Feline Immunodeficiency Virus (FIV)
02/06/2003US20030027842 Halogenobenzimidazoles
02/05/2003EP1280813A1 Anti-viral pyrimidine nucleoside analogues
02/05/2003EP1280809A1 Antitumoral ecteinascidin derivatives
02/05/2003EP1280798A1 Bicyclic heterocylces, medicaments containing said compounds, the use thereof and method for producing them
02/05/2003EP1280770A1 C 2? phenyl-substituted cyclic keto-enols used as pesticides and herbicides
02/05/2003EP1086078B1 Neuropeptide y5 receptor antagonists
02/05/2003EP0758334B1 Substituted (1,4)dioxino(2,3-f)benzoimidazole derivatives and their use in pest control
02/05/2003CN1395507A Catalysts comprising N-substituted cyclic imides and processes for prepairing organic compounds with catalysts
02/05/2003CN1100780C Process for preparing 2-chloro-beziidazole derivatives
02/04/2003US6515135 Aminoaryl oxazolidinone N-oxides
02/04/2003US6515126 Chemical synthesis of spirocyclic piperidines by double ring-closing metathesis
02/04/2003US6515027 Substituted benzanilides as CCR5 receptors ligands, antiinflammatory agents and antiviral agents
02/04/2003US6514984 Human non-pancreatic secretory phospholipase A2 inhibitors
02/04/2003US6514983 Inhibitors of the nucleic enzyme poly(adenosine 5'-diphospho-ribose)polymerase
01/2003
01/30/2003WO2003008421A1 Process for preparation of amidine derivatives
01/30/2003WO2003008420A1 2-(aminomethyl)-tetrahydro-9-oxa-1,3-diaza-cyclopenta[a]naphthalenyl derivatives with antipsychotic activity
01/30/2003WO2003008419A1 2-(AMINOMETHYL)-TETRAHYDRO-9-OXA-1,3-DIAZA-CYCLOPENTA[a]NAPHTHALENYL DERIVATIVES WITH ANTIPSYCHOTIC ACTIVITY
01/30/2003WO2003008410A2 Polypyrroles as agents for treating cancer, treating viral diseases and causing immunosuppression
01/30/2003WO2003007966A1 Active substance combination for medicamentous therapy of nicotine dependency
01/30/2003WO2002088079A3 Dual inhibitors of pde 7 and pde 4
01/30/2003WO2002012247A1 Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof
01/30/2003WO2002000617A3 Selective androgen receptor modulators and methods for their identification, design and use
01/30/2003US20030023082 Epothilone derivatives and methods for making and using the same
01/30/2003US20030022913 Novel immunomodulating compounds
01/30/2003US20030022905 Prevention and/or therapy of ischaemia and reperfusion damage; poly(ADP-ribose)-synthetase inhibitors
01/30/2003US20030022885 Pyrazole compounds useful as protein kinase inhibitors
01/30/2003CA2454545A1 2-(aminomethyl)-tetrahydro-9-oxa-1,3-diaza-cyclopenta[a]naphthalenyl derivatives with antipsychotic activity
01/30/2003CA2454543A1 2-(aminomethyl)-tetrahydro-9-oxa-1,3-diaza-cyclopenta[a]naphthalenyl derivatives with antipsychotic activity
01/30/2003CA2453664A1 Process for preparation of amidine derivatives
01/30/2003CA2453636A1 Polypyrroles as agents for treating cancer, treating viral diseases and causing immunosuppression
01/30/2003CA2417804A1 Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof
01/29/2003EP1278747A1 Pyrano, piperidino, and thiopyrano compounds and methods of use
01/29/2003EP1278746A2 Dihydropyridine compounds and methods of use
01/29/2003EP1278742A1 Chromenylmethylpyrimidinediamines as antibacterial agents
01/29/2003EP1278739A1 Amino substituted dibenzothiophene derivatives for the treatment of disorders mediated by the np y5 receptor
01/29/2003EP1278526A2 Treatment of cerebrovascular disease
01/29/2003EP1278502A2 Protease inhibitors
01/29/2003EP1161434B1 Pyridopyranoazepine derivatives, preparation and therapeutic use
01/29/2003EP1033369B1 5H-PYRANO [2,3-d:6,5-d']DIPYRIMIDINE DERIVATIVES HAVING AN ANTIBACTERIAL, ANTIVIRAL AND IMMUNO-MODULATING ACTIVITY
01/29/2003EP0835243B1 Dialkyl phenyl halide-substituted keto-enols for use as herbicides and pesticides
01/29/2003EP0754175B1 Alkoxy-alkyl-substituted 1-h-3-aryl-pyrrolidine-2,4-diones used as herbicides and pesticides
01/29/2003CN1393446A 稠合吡唑化合物 Fused pyrazole compounds
01/29/2003CN1100058C Novel intermediates and process for manufacture of camptothecin derivatives (CPT-11) and related compounds
01/29/2003CN1100057C Chromene compounds, process for their preparation and pharmaceutical compositions containing them
01/28/2003WO2002018372A1 Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
01/28/2003US6512120 Functionalized pyrrolidine compounds through the use of intramolecular Diels Alder reactions. further in situ and resin-bound synthetic generation of chemical libraries.
01/28/2003US6512112 Useful as prodrugs, easily convert to parent amine in vivo; antibiotic activity versus gram negative aerobic and anaerobic bacteria
01/28/2003US6511986 Method of treating estrogen receptor positive carcinoma
01/28/2003US6511977 For preventing or treating cardiac arrhythmia or atrial arrhythmia
01/28/2003US6511942 Animal husbandry, veterinary medicine
01/23/2003WO2003006563A1 A compressed fluid formulation
01/23/2003WO2003006060A1 Sh3 domain binding inhibitors
01/23/2003WO2002066475A3 Tricyclic androgen receptor modulator compounds
01/23/2003WO2002050066A3 Pyrazole compounds useful as protein kinase inhibitors
01/23/2003WO2002034760A3 Compounds and methods
01/23/2003WO2002017893A3 Sgk2 and sgk3 used as diagnostic and therapeutic targets
01/23/2003US20030018199 Process for preparing chiral diol sulfones and dihydroxy acid HMG CoA reductase inhibitors
01/23/2003US20030018046 Chemokine receptor binding heterocyclic compounds
01/23/2003US20030018042 Psychological disorders; Alzheimer's disease
01/23/2003CA2417156A1 3,4-dihydroisoquinoline derivative compound and a pharmaceutical agent comprising it as active ingredient
01/22/2003EP1277756A1 Ketol fatty acid derivatives and plant growth regulating agents