Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726) |
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11/20/2003 | WO2003095459A2 Alkaloid-derived compounds and use thereof in cancer and malaria treatment |
11/20/2003 | WO2003095447A1 Process for the preparation of a hydrate of an anthranilic acid derivative |
11/20/2003 | WO2003095427A1 Spiro-ring compound |
11/20/2003 | WO2003057173A3 Broad spectrum inhibitors |
11/20/2003 | WO2002102315A3 QUINAZOLINE AND PYRIDO[2,3-d]PYRIMIDINE INHIBITORS OF PHOSPHODIESTERASE (PDE) 7 |
11/20/2003 | WO2002100860A3 Heterocyclic compounds, method for preparing same and use thereof as medicines, in particular as anti-bacterial agents |
11/20/2003 | US20030216494 Free radical catalyst for addition polymer |
11/20/2003 | US20030216421 Cascade esters of camptothecins and methods of treating cancer using these compounds |
11/20/2003 | US20030216419 Isomeric fused pyrrolocarbazoles and isoindolones |
11/20/2003 | US20030216399 A dipeptide containing bi or tri-heterocylic ring with nitrogen atom which forms amide with carbonyl group of dipeptide chain; useful for treating osteoporosis, congestive heart failure and accelerates wound healing |
11/20/2003 | US20030216397 A compound having a fused ecteinascidin five ring system with a 1,4 bridge; anticarcinogenic agent |
11/20/2003 | US20030216378 Azepino[4,5-b]pyrano[3,2-e]indoles |
11/20/2003 | US20030216373 Activity against both Gram-positive and Gram-negative pathogens are generally regarded as having a broad spectrum of activity |
11/20/2003 | US20030216324 Five-member heterocyclic compounds substituted with an alpha-amino carbonyl group; antiasthma agents |
11/20/2003 | US20030216260 Preparation by intramolecular cyclization |
11/20/2003 | CA2484815A1 Cascade esters of camptothecins and methods of treating cancer using these compounds |
11/19/2003 | EP1362052A1 Inhibitors of cruzipain and other cysteine proteases |
11/19/2003 | EP1362051A2 Method for purifying 20(s)-camptothecin |
11/19/2003 | EP1361877A1 Pharmaceutical dosage forms of epothilones for oral administration |
11/19/2003 | EP0984970B1 Spiro-quinuclidine derivatives, their preparation and use |
11/19/2003 | EP0973392B1 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds |
11/19/2003 | EP0898571B1 Thieno-pyridine sulfonamides, derivatives thereof and related compounds that modulate the activity of endothelin |
11/19/2003 | CN1457339A Chemokine receptor binding heterocyclic compounds |
11/19/2003 | CN1456154A Method for curing sepsis |
11/18/2003 | US6649763 Optically active quinoline carboxylic acid derivatives with 7-pyrrolidine substituents causing optical activity and a process for the preparation thereof |
11/18/2003 | US6649647 Trioxane derivatives |
11/18/2003 | US6649626 Stimulants of gamma -aminobutyric acid receptors; psychological disorders |
11/18/2003 | US6649624 Useful as neuropeptide Y receptor antagonists and as agents for therapy of cardiovascular disorders, central nervous system disorders, metabolic diseases |
11/18/2003 | US6649622 Treating diabetes, especially Type II diabetes |
11/18/2003 | US6649618 Substituted amidoalkyl-uracils and their use |
11/18/2003 | US6649608 Cyclin-dependent serine/threonine and focal adhesion kinase inhibitors |
11/18/2003 | US6649589 Blocking tumor necrosis factor activity with soluble cytokine receptor, monoclonal antibody or tetracycline derivative |
11/13/2003 | WO2003093274A1 Camptothecin-taxoid conjugates as antimitotic and antitumor agents |
11/13/2003 | WO2003093252A1 Heteroaryl substituted spirocyclic sulfamides for inhibition of gamma secretase |
11/13/2003 | WO2003093244A1 Substituted (thioxo)carbonylamino phenyl uraciles |
11/13/2003 | WO2003093231A2 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity |
11/13/2003 | WO2003092580A2 Methods and compositions for treatment of central and peripheral nervous system disorders and novel compounds useful therefor |
11/13/2003 | WO2003092374A2 Pesticidal heterocycles |
11/13/2003 | WO2003032897A3 Azabicyclic compounds for the treatment of fibromyalgia syndrome |
11/13/2003 | WO2003029213A9 Spirocyclic 3-phenyl-3-substituted 4-ketolactams and 4-ketolactones |
11/13/2003 | WO2003024448A3 Inhibitors of histone deacetylase |
11/13/2003 | WO2002099077A3 Methods and compositions related to tagging of membrane surface proteins |
11/13/2003 | US20030212271 Reacting dialkyl malonate ester with trifluoroacetic acid; cyclization, controlling temperature |
11/13/2003 | US20030212115 Remedies for inflammatory bowel diseases |
11/13/2003 | US20030212101 Respiratory system disorders; antiinflammatory agents; psychological disorders |
11/13/2003 | US20030212094 Novel cyclic amide derivatives |
11/13/2003 | US20030212089 Arylindenopyridines and related therapeutic and prophylactic methods |
11/13/2003 | US20030212087 Plant extracts; antitumor, anticancer agents; topoisomerase inhibitor |
11/13/2003 | CA2484599A1 Methods and compositions for treatment of central and peripheral nervous system disorders and novel compounds useful therefor |
11/13/2003 | CA2484280A1 Substituted (thioxo)carbonylamino phenyl uraciles |
11/13/2003 | CA2483843A1 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity |
11/12/2003 | EP1361225A1 Compounds substituted with bicyclic amino groups |
11/12/2003 | EP1359908A1 Quinolines and nitrogenated derivatives thereof substituted in 4-position by a piperidine-containing moiety and their use as antibacterial agents |
11/12/2003 | EP1280813B1 Anti-viral pyrimidine nucleoside analogues |
11/12/2003 | EP1206265B1 Src kinase inhibitor compounds |
11/12/2003 | EP1058549A4 THROMBIN OR FACTOR Xa INHIBITORS |
11/12/2003 | EP0975599B1 Subtituted isoquinolines as ultra short acting neuromuscular blockers |
11/11/2003 | US6645999 Lactacystin analogs |
11/11/2003 | US6645990 For prophylaxis and therapy of diseases, such as cell proliferation or apoptosis mediated diseases |
11/11/2003 | US6645983 Pharmaceutical compositions comprising 4-quinolones for treating cancers |
11/11/2003 | US6645980 Ligands for biological receptors such as opiate receptors or G-protein coupled receptors used for treating pain, drug dependence or tinnitus in mammals |
11/11/2003 | US6645975 Process for the preparation of dinaposoline |
11/11/2003 | US6645973 Heterocyclic amines such as 1-carboxymethyl-4-(4-chlorophenyl) spiro(2H-1-benzopyran-2,4'-piperidine)hydrochloride used for therapy of nervous system disorders; Alzheimer's, Parkinson's and Huntington's disease |
11/11/2003 | CA2290332C Optically pure androgen mediator |
11/06/2003 | WO2003091264A2 Non nucleoside reverse transcriptase inhibitors |
11/06/2003 | WO2003091257A1 [1,4]DIAZOCINO [7,8,1-hi]INDOLE DERIVATIVES AS ANTIPSYCHOTIC AND ANTIOBESITY AGENTS |
11/06/2003 | WO2003091255A1 Inhibitors of checkpoint kinases (wee1 and chk1) |
11/06/2003 | WO2003091253A1 Nitrosated imidazopyridines |
11/06/2003 | WO2003090691A2 Method and compositions for identifying anti-hiv therapeutic compounds |
11/06/2003 | WO2003090690A2 Cellular accumulation of phosphonate analogs of hiv protease inhibitor compounds and the compounds as such |
11/06/2003 | WO2003090680A2 Novel phenyl derivatives as inducers of apoptosis |
11/06/2003 | WO2003090672A2 2-(quinolonyl)-fused heterocycles as androgen receptor modulators |
11/06/2003 | WO2003039539A3 Use of endothelin receptor antagonists in the treatment of tumour diseases |
11/06/2003 | WO2002076979A8 1,2,3,4-tetrahydroisoquinolines derivatives as urotensin ii receptor antagonists |
11/06/2003 | WO2002076375A3 Process for the preparation of benazepril |
11/06/2003 | US20030208082 Nitrogen compounds such as 4,5-diisopropyl-1-methyl-2-styryl -1H-imidazole, used as glutamate receptor antagonists, for prophylaxis of psychological disorders, as anxiolytic agents and analgesics |
11/06/2003 | US20030208076 Preparation of fused polycyclic alkaloids by ring closure of azomethine ylides, novel compounds thereof and their use as chemotherapeutic agents |
11/06/2003 | US20030208066 4-((4-But-2-ynyloxy-benzenesulfonyl)-methyl-amino)-1,3-dimethy l-1H- pyrazolo(3,4-b)and dericatives; bioavailability; no pharmacokinetic problems; bioselectiveity; rheumatoid arthritis, osteoarthritis, sepsis, AIDS, ulcerative colitis |
11/06/2003 | US20030207900 2-substituted amino-bicyclic pyridine and pyrimidine compounds; for treatment of inflammation, inflammatory bowel disease, Alzheimer's disease, Crohn's disease, multiple sclerosis and asthma |
11/06/2003 | US20030207894 1,4-Disubstituted benzenes as insecticides |
11/06/2003 | US20030207883 Indazole benzimidazole compounds |
11/06/2003 | US20030207824 Pyrimidine derivatives for labeled binding partners |
11/06/2003 | CA2484090A1 Nitrosated imidazopyridines |
11/06/2003 | CA2483496A1 Inhibitors of checkpoint kinases (wee1 and chk1) |
11/06/2003 | CA2481449A1 Method and compositions for identifying anti-hiv therapeutic compounds |
11/06/2003 | CA2481324A1 [1,4]diazocino [7,8,1-hi]indole derivatives as antipsychotic and antiobesity agents |
11/06/2003 | CA2481285A1 Non nucleoside reverse transcriptase inhibitors |
11/05/2003 | EP1359152A2 Diazabicyclic derivatives as nicotinic acetylcholine receptor ligands |
11/05/2003 | EP1359146A2 8-substituted-2,6-methano-3-benzazocines and 3-substituted morphinanes as opioid receptor binding agents |
11/05/2003 | EP1359139A1 Terphenyl compounds bearing substituted amino groups |
11/05/2003 | EP1358185A2 Pyridoarylphenyl oxazolidinone antibacterials, and related compositions and methods |
11/05/2003 | EP1358178A2 Sulfonamide lactam inhibitors of factor xa |
11/05/2003 | EP1220858B1 Oxazinoquinolones useful for the treatment of viral infections |
11/05/2003 | EP0971930B1 Process for preparing single enantiomer narwedine |
11/05/2003 | EP0946566B1 Pro-drugs and counterparts of camptothecin, their application as medicines |
11/05/2003 | EP0861842B1 Novel water-soluble fluoroethylcamptothecin derivative and process for production thereof |
11/05/2003 | CN1454083A Selective androgen receptor modulators and methods for their identification design and use |
11/05/2003 | CN1453279A Plant extractive and alkaloid with cough-relieving activity |
11/05/2003 | CN1126737C Novel pyrrole compound, its preparation and pharmaceutical composition containing the same |
11/04/2003 | US6642249 3-Oxo-pyrazolo(4,3-c) -quinolin-2-yl, -thiochroman-2-yl, or -chromen-2-yl derivatives; CD80 antagonists |