Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726) |
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03/13/2003 | CA2422135A1 Urea derivatives and adhesion molecule inhibitors containing the same as effective ingredients |
03/12/2003 | EP1289999A1 Antitumoral analogs of et-743 |
03/12/2003 | EP1289985A2 Beta-carboline derivatives useful as inhibitors of phosphodiesterase |
03/12/2003 | EP1289525A2 Tricyclic pyrazole derivatives as protein kinase inhibitors |
03/12/2003 | EP1075477B1 Novel Benzonaphthyridine-N-oxides |
03/12/2003 | CN1402721A Benzoimidazole derivs. useful as antiproliferative agents |
03/12/2003 | CN1402643A Integrin-mediated drug targeting |
03/12/2003 | CN1102932C Novel water-soluble analogues of 20(S)-camptothecin, preparing method and use thereof |
03/07/2003 | WO2002020481A2 Substituted 4-phenyl-1-(1-phenyl-cyclohexyl)-1,2,3,6-tetrahydropyridine |
03/07/2003 | CA2421835A1 Substituted 4-phenyl-1-(1-phenyl-cyclohexyl)-1,2,3,6-tetrahydropyridines |
03/06/2003 | WO2003018589A1 Novel 4-aminofuropyrimidines and the use thereof |
03/06/2003 | WO2003018559A2 Intermediates and preparation thereof for the enantioselective synthesis of (20r) homocamptothecins |
03/06/2003 | WO2003017764A1 Substituted propargylamines |
03/06/2003 | WO2003000240A3 Stable powder inhalation dosage formulation |
03/06/2003 | US20030045719 And optionally resolving mixture to obtain the desired enantiomer; antitumor agents |
03/06/2003 | US20030045717 Suitable as fluorescent dyes (fluorophores) for used in optical determination and demonstration methods in medicine, pharmacology and biological and environmental sciences; photostability, storage stability |
03/06/2003 | US20030045714 Photochromic sections being 2H-pyrans and/ or spirooxazines; use in ophthalmic lenses or sun-protection roofs |
03/06/2003 | US20030045711 Epothilone derivatives and methods for making and using the same |
03/06/2003 | US20030045542 Antidepressant azaheterocyclylmethyl derivatives of 2,3-dihydro-1,4-dioxino[2,3-f]quinoline |
03/06/2003 | US20030045540 Nicotinic acetylcholine receptors antagonists; central nervous system disorder treatments |
03/06/2003 | US20030045537 4-(Phenylamino)-[1,4]dioxano[2,3-g]quinazoline derivatives and process for preparing the same |
03/06/2003 | US20030045526 Antipsychotic aminomethyl derivatives of 1,3,7,8-tetrahydro-6,9-dioxa-1,3-diaza-cyclopenta[a]-naphthalen-2-one |
03/06/2003 | US20030045516 Chemokine receptor antagonists and methods of use therefor |
03/06/2003 | US20030045432 Phenyl-substituted cyclic ketoenols |
03/06/2003 | US20030044399 Method of treatment |
03/05/2003 | EP1288203A1 Cyclic nitrones and pharmaceutical compositions containing them |
03/05/2003 | EP1287004A1 Synthetic process for the manufacture of an ecteinascidin compound |
03/05/2003 | EP1287002A1 Crf receptor antagonists |
03/05/2003 | EP1286999A1 PYRANO[2,3-c]IMIDAZO[1,2-a]PYRIDINE DERIVATIVES FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS |
03/05/2003 | EP1286998A1 Oxazolidinone derivatives with antibiotic activity |
03/05/2003 | EP1286994A1 Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity |
03/05/2003 | EP1286978A1 Cyclohexyl derivatives and their use as therapeutic agents |
03/05/2003 | EP1286973A2 Novel carbamates and carbamides, production and use thereof as endothelin receptor antagonists |
03/05/2003 | EP1286967A1 Cyclohexane derivatives and their use as therapeutic agents |
03/05/2003 | EP0792273B1 Bicyclic oxazine and thiazine oxazolidinone antibacterials |
03/05/2003 | EP0690863B1 Tetracyclic compounds as dopamine agonists |
03/05/2003 | CN1400969A Fused imidazolium derivatives |
02/27/2003 | WO2003016310A1 Alkyl-substituted imidazopyridines for the treatment of gastrointestinal disorders |
02/27/2003 | WO2002098865A3 Cyclic nucleotide phosphodiesterase inhibitors, preparation and uses thereof |
02/27/2003 | WO2002098350A3 Pyranoindazoles and their use for the treatment of glaucoma |
02/27/2003 | WO2002096881A8 Method for preparation of 10,11-dihydro-10-hydroxy-5h-dibenz/b,f/azepine-5-carboxamide and 10,11-dihydro-10-0x0-5h-dibenz/b,f/azepine-5-carboxamide |
02/27/2003 | WO2002092602A3 PROCESSES FOR THE SYNTHESIS OF DERIVATIVES OF 2,3-DIHYDRO-1,4-DIOXINO-[2,3-f] QUINOLINE |
02/27/2003 | WO2002092588A3 Aromatic sulfone hydroxamates and their use as protease inhibitors |
02/27/2003 | WO2002089782A3 Dioxanes and uses thereof |
02/27/2003 | WO2002086878A3 Optical data carrier whose information layer contains a light-absorbing compound having a number of chromophoric centers |
02/27/2003 | WO2002060904A3 A process for the preparation of epothilone analogs |
02/27/2003 | US20030040630 Method for producing sulfonyl imidazole derivatives |
02/27/2003 | US20030037701 2-(aminomethyl)-tetrahydro-9-oxa-1,3-diaza-cyclopenta[a]-naphthalenyl derivatives with antipsychotic activity |
02/27/2003 | CA2452801A1 Alkyl-substituted imidazopyridines for the treatment of gastrointestinal disorders |
02/26/2003 | EP1112456B1 Tube for lining pipes and channels, and a method and device for the production thereof |
02/26/2003 | EP0754040B1 Rapamycin derivatives |
02/26/2003 | CN1398863A Benzo [b] pyran-[3,2-h] acridinyl-7-one compounds, their prepn and medicine composition containing them |
02/25/2003 | US6525197 Producing chemical intermediates for such as epothilone or epothilone analogues synthesis |
02/25/2003 | US6525193 Aminoaryl oxazolidinone N-oxides |
02/25/2003 | US6525047 Which are growth hormone secretogogues and increase the level of endogenous growth hormone; treating osteoporosis, congestive heart failure, frailty associated with aging, obesity; accelerating bone fracture repair |
02/20/2003 | WO2003014124A1 Substituted 5,6,6a,11b-tetrahydro-7-oxa-5-aza-benzo[c]fluorene-6-carboxylic acid derivatives serving as nmda antagonists |
02/20/2003 | WO2003014123A1 Tricyclic imidazopyridines |
02/20/2003 | WO2003014120A1 Amino-substituted imidazopyridines for the treatment of gastrointestinal diseases |
02/20/2003 | WO2003014119A1 Tricyclic epoxides |
02/20/2003 | WO2003014083A1 Spiro compounds |
02/20/2003 | WO2003014069A1 Fluoro linkers and their use as linkers for enzyme-activated drug conjugates |
02/20/2003 | WO2003013537A2 Irinotecan for treatment of cancer |
02/20/2003 | WO2003013536A2 Methods for treatment of cancer using irinotecan based on ugt1a1 |
02/20/2003 | WO2003013535A2 Use of irinotecan for improved treatment of cancer based on mdr1 |
02/20/2003 | WO2003013534A2 Methods for the treatment of cancer with irinotecan based on cyp3a5 |
02/20/2003 | WO2003013533A2 Methods for improved treatment of cancer with irinotecan based on mrp1 |
02/20/2003 | WO2003013530A2 Salts of substituted 1, 2, 3, 4-tetrahydroquinoline-2-carboxylic acid derivatives as nmda antagonists |
02/20/2003 | WO2003013522A1 Preventives/remedies for cholinergic neuropathy |
02/20/2003 | WO2003013430A2 Benzoquinone ansamycins |
02/20/2003 | WO2002070525A3 Nitrogen-based camptothecin derivatives |
02/20/2003 | WO2002068387A3 Acylated piperidine derivatives as melanocortin-4 receptor agonists |
02/20/2003 | US20030036652 Spiro[isobenzofuran-1,4'-piperidin]-3-ones and 3H-spiroisobenzofuran-1,4'-piperidines |
02/20/2003 | US20030036543 Especially as inhibitors of Aurora-2 and GSK-3, for treating diseases such as cancer, diabetes and Alzheimer's disease. |
02/20/2003 | CA2456599A1 Spiro compounds |
02/20/2003 | CA2456594A1 Preventives/remedies for cholinergic neuropathy |
02/20/2003 | CA2456175A1 Benzoquinone ansamycins |
02/20/2003 | CA2456124A1 Substituted 5,6,6a,11b-tetrahydro-7-oxa-5-aza-benzo[c]fluorene-6-carboxylic acid derivatives serving as nmda antagonists |
02/20/2003 | CA2456103A1 Salts of substituted 1, 2, 3, 4-tetrahydroquinoline-2-carboxylic acid derivatives |
02/20/2003 | CA2454648A1 Irinotecan for treatment of cancer |
02/20/2003 | CA2454643A1 Methods for the treatment of cancer with irinotecan based on cyp3a5 |
02/20/2003 | CA2454640A1 Methods for treatment of cancer using irinotecan based on ugt1a1 |
02/20/2003 | CA2454637A1 Use of irinotecan for improved treatment of cancer based on mdr1 |
02/20/2003 | CA2454627A1 Methods for improved treatment of cancer with irinotecan based on mrp1 |
02/20/2003 | CA2453245A1 Fluoro linkers and their use as linkers for enzyme-activated drug conjugates |
02/20/2003 | CA2452803A1 Tricyclic imidazopyridines |
02/20/2003 | CA2452802A1 Tricyclic epoxides |
02/19/2003 | EP1283855A1 Stable near-infrared (nir) marker dyes based on benzopyrylium-polymethines |
02/19/2003 | EP1283834A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
02/19/2003 | EP1283833A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
02/19/2003 | EP1283832A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
02/19/2003 | EP1283831A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
02/19/2003 | EP1119571B1 Tricyclic delta3-piperidines as alpha2-antagonists |
02/19/2003 | EP0931083B1 Process for producing ecteinascidin compounds |
02/19/2003 | EP0920429B1 Substituted pyrido- or pyrimido-containing 6,6- or 6,7-bicyclic derivatives |
02/19/2003 | EP0817786B1 Substituted tetronic acids useful for treating hiv and other retroviruses |
02/19/2003 | EP0799218B1 Diaryl-2-(5h)-furanones as cox-2 inhibitors |
02/19/2003 | EP0750618B1 Oxazolidinone derivatives and pharmaceutical compositions containing them |
02/19/2003 | CN1101818C Novel water-soluble c-ring analogues of 20(s)-campothecin |
02/18/2003 | US6521757 Preparation of fused polycyclic alkaloids by ring closure of azomethine ylides, novel compounds thereof and their use as chemotherapeutic agents |
02/18/2003 | US6521753 Indolinospiropyran compounds and methods for their manufacture |