Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
01/2005
01/20/2005CA2530450A1 5-substituted quinazolinone derivatives
01/19/2005EP1497296A1 1,4 DIAZOCINO 7,8,1-hi INDOLE DERIVATIVES AS ANTIPSYCHOTIC AND ANTIOBESITY AGENTS
01/19/2005EP1496910A1 Kinase inhibitors
01/19/2005EP0777492B1 Combinatorial libraries of substrate-bound cyclic organic compounds
01/19/2005CN1566116A Process for preparing wedelia lactone and application thereof
01/19/2005CN1566100A Aporphine and ketone group aporphine compound and medicinal use thereof
01/19/2005CN1185214C Novel indeno indolone compound, its preparation method and drug composition comprising the same
01/18/2005US6844445 Central nervous system disorders; psychological disorders
01/18/2005US6844352 1′-[4-[1-(4-fluorophenyl)-1H-indole-3-yl]-1-butyl]-spiro[isobenzofuran-1(3H),4′-piperidine] hydrohalogenides
01/18/2005US6844350 Febrifugine, isofebrifugine and method for producing the same
01/13/2005WO2005003137A1 Salinosporamides and methods for use thereof
01/13/2005WO2005003132A1 Perylenetetracarboxylic acid dibenzimidazole sulfoderivatives containing oxo-groups in the perylene core which form part of a para-quinoid system of bonds, lyotropic liquid crystal systems and anisotropic films containing the same, and methods for making the same
01/13/2005WO2005003128A1 Thiazolylpiperidine derivatives as mtp inhibitors
01/13/2005WO2005003097A1 Cis-2,4,5-triaryl-imidazolines
01/13/2005WO2005003086A2 Sulfonic acid derivatives of polycyclic dyes used for analytical applications
01/13/2005WO2005002577A1 Dual nk1/nk3 antagonists for treating schizophrenia
01/13/2005WO2005002503A2 Asymmetric benzimidazoles and related compounds as potassium channel modulators
01/13/2005WO2004096805A3 Lyotropic liquid crystal systems based on sulfonated perylenetetracarboxylic acid dibenzimidazoles
01/13/2005WO2004050035A3 Benzimidazoles and analogs thereof as antivirals
01/13/2005US20050010046 Topoisomerase poison agents
01/13/2005US20050009898 New substituted indolinones, their manufacture and their use as medicaments
01/13/2005US20050009894 Benzimidazole derivatives and their use as KDR kinase protein inhibitors
01/13/2005US20050009855 1-(hydroxy, oxo, or epoxy)-3-oxo-3'-benzaminocarbonyl-4'-(carboxy or carboxylate)-1,2,3-trihydroindene-2-spiro-2'-tetrahydrofuran derivatives; these compounds interfere with the E1-E2-DNA complex during initiation of DNA replication
01/13/2005US20050009830 Fused ring cinnoline derivatives including naphthocinnolines, quinollinocinnolines and naphthopyridinopyridines, e.g., 2,3-Dimethoxydibenzo[ch]cinnoline and 2,3-Dimethoxy-8,9-methylenedioxy-dibenzo[c,h]cinnoline; treatment of anticancer agnets, fungicides and bactericides
01/13/2005US20050009826 5,6,13-trizaza- or 6,13-diazachryseno[2,3-d]-[1,3]dioxole derivatives; enzyme inhibitors; anticarcinogenic, antiproliferative agents; bactericides, fungicides
01/13/2005US20050009825 Cytotoxic agents
01/13/2005US20050009824 Solubilized topoisomerase poisons
01/13/2005US20050009823 E.g., derivatives of pyrazolo[1,5-a]pyrimidines; [1,2,3]triazolo[4,5-b]pyridines; and pyrrolo[3,2-d]pyrimidines and their use as corticotropin releasing factor antagonists
01/13/2005US20050009820 Thiochromenones used to combat painful conditions and neurodegenerative diseases
01/13/2005US20050009755 (74)(3S)-3-amino-1-(1-benzyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-4-yl)-5-methyl-2-heptanone for example; cysteine protease inhibitors; treating bone resorption diseases such as osteoporosis
01/13/2005CA2530886A1 Dual nk1/nk3 antagonists for treating schizophrenia
01/13/2005CA2530215A1 Salinosporamides and methods for use thereof
01/13/2005CA2528119A1 Cis-2,4,5-triaryl-imidazolines
01/13/2005CA2525580A1 Asymmetric benzimidazoles and related compounds as potassium channel modulators
01/12/2005EP1496060A1 Antitumoral analogs of ET-743
01/12/2005EP1495022A1 Diazabicyclo alkane derivatives with nk1 antagonistic activity
01/12/2005EP1495014A2 Novel flavanoids and chalcones as chemotherapeutic, chemopreventive, and antiangiogenic agents
01/12/2005EP1495000A1 Alpha, omega-dicarboximide derivatives as useful uro-selective a1a adrenoceptor blockers
01/12/2005EP1494672A1 Aminocarbonyl substituted pyridines, pyridazines, pyrimidines, pyrazines and triazines having antiangiogenic activity
01/12/2005EP1494670A1 Medicine for treating cancer
01/12/2005CN1564818A Process for stereoselective synthesis of 2-hydroxymethyl chromans
01/11/2005US6841304 Dissolves other salts, in particular metallic salts, such as lithium salts, to give highly conductive solutions
01/11/2005CA2215351C Process for isolating galanthamine
01/06/2005WO2005000842A1 Benzothiazole derivatives as adenosine receptor ligands
01/06/2005WO2005000250A2 Imaging agents and methods of imaging alpha 7-nicotinic cholinergic receptor
01/06/2005WO2004103967A3 Thiocarbamate inhibitors of alpha-4 integrins
01/06/2005WO2004071382A3 Substituted heterocycles
01/06/2005US20050004204 2-Iminopyrrolidine derivatives
01/06/2005US20050004197 Thrombin receptors antagonists; oral efficacy
01/06/2005US20050004159 for example, 8-(1-ethylpropyl)-3-mesityl-2,5-dimethyl-8H-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidine; having an excellent corticotrophin-releasing-factor receptor antagonistic activity
01/06/2005US20050004157 Serotonin uptake inhibitors and 5-HT1A receptor antagonists; antidepressants; psychological disorders
01/06/2005US20050004147 Tricyclic fused heterocyclic compound, process for preparing it and medicament comprising it
01/06/2005US20050004143 Bi-cyclic pyrimidine inhibitors of TGFbeta
01/06/2005US20050004142 furo(2,3-d)pyrimidine and thieno(2,3-d)pyrimidine compounds for treating cancer and hyperproliferative diseases; receptor tyrosine kinase inhibitors
01/06/2005US20050004133 Inhibiting ligand gated ion channel vanilloid receptor (VR1); pain relievers; such as 6-(3,4-dichloro-phenyl)-N-(2-oxo-2,3-dihydro-1H-benzoimidazol-5-yl)-nicotinamide
01/06/2005US20050004130 New metabotropic glutamate receptor compounds
01/06/2005US20050004124 Synergistic mixture; antidiabetic agents; antiischemic agents
01/06/2005US20050004112 C-fms kinase inhibitors
01/06/2005US20050004110 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease
01/06/2005US20050004099 Spiroazabicyclic heterocyclic compounds
01/06/2005US20050004039 Selective analgesic agents
01/06/2005US20050001202 Perylenetetracarboxylic acid dibenzimidazole sulfoderivatives containing oxo-groups in the perylene core which form part of a para-quinoid system of bonds, lyotropic liquid crystal systems and anisotropic films containing the same, and methods for making the same
01/06/2005CA2672071A1 Process for preparing 3-acylaminobenzofuran-2-carboxylic acid derivative
01/05/2005EP1493738A1 Epothilone derivatives
01/05/2005EP1493057A1 Colour photographic recording material
01/05/2005EP1492571A2 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands
01/05/2005EP1492539A1 Statin therapy for enhancing cognitive maintenance
01/05/2005EP1492536A1 4-(n-phenylamino)-quinazolines / quinolines as tyrosine kinase inhibitors
01/05/2005CN1561215A Salts of substituted 1, 2, 3, 4-tetrahydroquinoline-2-carboxylic acid compounds used as nmda antagonist
01/05/2005CN1183138C Process for promoting generation of 10-hydroxycamptothecin in the bud of camptotheca seed
01/05/2005CN1183137C Synthesis method of [3aS, 6aR]-1,3-dibenzyl-tetrahydro-4H-fruo [3,4-d]-imidazolyl-2,4[1H}-diketone [I]
01/04/2005US6838559 Such as 2-((6-(((4-(3,4-dimethoxyphenyl)methyl)amino)-7-ethyl-7H-purin-2-yl)amino) -4,5-methyl-N-phenyl-5-thiazole-carboxamide for treatment of lymphocyte mediated diseases such as transplant rejection and graft versus host disease
01/04/2005US6838527 Polymer-immobilized α-iminoester
01/04/2005US6838477 Lactacystin analogs
01/04/2005US6838471 Inhibition of inflammatory cytokine production by cholinergic agonists and vagus nerve stimulation
01/04/2005US6838457 Fused heteroaryl derivatives
01/04/2005US6838291 For identifying compounds that bind to ion channel and may have antiarrhythmic activity
01/04/2005CA2242015C New chromene derivatives, the procedure for preparing them and the pharmaceutical compounds that contain them
01/04/2005CA2186015C Nicotinic acid derivatives and herbicides
01/04/2005CA2093076C 2- and 3-amino and azido derivatives of 1,5-iminosugars
12/2004
12/30/2004US20040266840 Inhibits replication and/or proliferation of Hepatitis C virus (HCV)
12/30/2004US20040266821 Obesity, diabetes, sexual dysfunction
12/30/2004US20040266804 Camptothecin analogs having an E-ring ketone
12/30/2004US20040266803 7-Substituted camptothecin and camptothecin analogs and methods for producing the same
12/30/2004US20040266759 Possess antithrombotic and anticoagulant properties; example compound: 1-(5-Chlorobenzo[b]furan-2-ylsulphonyl)-4-[4-(4-pyridyl)benzoyl]piperazine
12/30/2004US20040266758 Modulators of the glucocorticoid receptor and method
12/30/2004US20040266753 Benzo[a]pyrano[3,2-h]acridin-7-one compounds
12/30/2004DE10326386A1 N-Heterocyclyl-phenylsubstituierte cyclische Ketoenole N-heterocyclyl-substituted cyclic ketoenols
12/29/2004WO2004113394A2 Living radical polymerization initiator comprising a functional group capable of reacting with polypeptides or the like, comb polymer obtained therewith, polypeptide conjugates and drugs obtained therefrom
12/29/2004WO2004113345A1 Fused pyrrole compound and medicinal use thereof
12/29/2004WO2004075853A3 Halogenated triptolide derivatives as immunomodulators and anticancer agents
12/29/2004EP1491544A1 Benzo[a]pyrano[3,2-h]acridin-7-one derivatives, processes for their preparation and pharmaceutical compositions thereof
12/29/2004EP1491541A1 Pyridazinone aldose reductase inhibitors
12/29/2004EP1491540A1 Pyridazinone aldose reductase inhibitors
12/29/2004EP1491353A1 Optical recording media and dipyrromethene-metal chelate compounds
12/29/2004EP1490361A1 Polycyclic compounds as potent alpha2-adrenoceptor antagonists
12/29/2004EP1490356A1 (3z)-3-(3-hydro-isobenzofuran-1-ylidene)-1,3-dihydro-2h-indol-2-ones as kinase inhibitors
12/29/2004EP1490058A1 Peroxisome proliferator activated receptor modulators
12/29/2004EP1490047A2 Certain pharmaceutically useful substituted aminoalkyl heterocycles
12/29/2004EP1373259B1 Pyridazinone aldose reductase inhibitors