Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
06/2004
06/30/2004CN1509291A Oxazolo-and-furopyrimidines and their use in medicaments against tumors
06/30/2004CN1509290A Process for synthesis of derivatives of 2,30dihydro-1,4-dioxino-[2,3-f]quinoline
06/30/2004CN1509183A Use of proteasome inhibitors to treat dry eye disorders
06/30/2004CN1509140A Pyridinyl fused bicyclic amide as fungicides
06/30/2004CN1508137A 2-phenyl-substituted imidazo-triazone used as phosphodiesterase inhibitor
06/30/2004CN1155578C Production of cyclic acid
06/29/2004US6756381 A purified antitumor agent is crystallized from acetone or dichloromethane
06/29/2004US6756378 VLA-4 inhibitor compounds
06/29/2004CA2205384C Dihydropyrimidines and uses thereof
06/24/2004WO2004052893A2 Substituted dihydropyrano indole-3,4-dione derivatives and 3-oxoacetic acid substituted 2-hydroxymethylindole derivatives as inhibitors of plasminogen activator inhibitor-1 (pai-1)
06/24/2004WO2004052864A1 Pyrazole and imidazole compounds and uses thereof
06/24/2004WO2004052847A2 Tricyclic steroid hormone nuclear receptor modulators
06/24/2004WO2004017922A3 Keto cannabinoids with therapeutic indications
06/24/2004WO2003105724A3 Novel maxi-k channel blockers, methods of use and process for making the same
06/24/2004WO2003092580B1 Methods and compositions for treatment of central and peripheral nervous system disorders and novel compounds useful therefor
06/24/2004WO2003090690A3 Cellular accumulation of phosphonate analogs of hiv protease inhibitor compounds and the compounds as such
06/24/2004WO2003051841A3 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
06/24/2004WO2002092594A8 Substituted 4h-chromenes and analogs as activators of caspases and inducers of apoptosis and the use thereof
06/24/2004US20040122230 Opiate analogs selective for the delta -opioid receptor
06/24/2004US20040122074 1-[5-(4-chloro-phenyl)-1-(2-chloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-2-piperidin-1-yl-ethanone,e.g. as antagonist or inverse agonists; nicotine partial agonist; an opioid antagonist; a dopaminergic agent; an attention deficit disorder agent
06/24/2004US20040122073 E.g., 1-[[7-(aminoiminomethyl)-2-naphthalenyl]methyl]-2,5-dioxo-4-phenyl-3-(phenylmethyl)-4-imidazolidineacetamide; enzme enzyme inhibitors of the blood Factor VIIa complex; myocardial infarction; antiischemic agents; brain disorders ,
06/24/2004US20040122050 Cyclohexyl sulphone derivatives as gamma-secretase inhibitors
06/24/2004US20040122034 Polymorph forms of n-(2,3-dimethyl-5,6,7,8-tetrahydrofuro[2,3-b]quinolin-4-yl)-2-(2-oxopyrrolidin-1-1yl)acetamide
06/24/2004US20040122017 Melanin concentrating hormone (MCH) modulators; metabolic and eating disorders
06/24/2004US20040121997 20-hydroxyeicosatetraenoic acid production inhibitors
06/24/2004US20040121911 Ketol fatty acid derivative and plant growth regulators
06/24/2004US20040121316 Method and compositions for identifying anti-HIV therapeutic compounds
06/24/2004CA2509242A1 Substituted dihydropyrano indole-3,4-dione derivatives and 3-oxoacetic acid substituted 2-hydroxymethylindole derivatives as inhibitors of plasminogen activator inhibitor-1 (pai-1)
06/24/2004CA2505887A1 Pyrazole and imidazole compounds and uses thereof
06/23/2004EP1431285A1 Reverse hydroxamic acid derivatives
06/23/2004EP1430903A1 Use of proteasome inhibitors for the treatment of viral infections
06/23/2004EP1430059A1 Pharmaceutically acceptable salts of 20(s)-camptothecins
06/23/2004EP1430048A1 3-(arylamino)methylene-1, 3-dihydro-2h-indol-2-ones as kinase inhibitors
06/23/2004EP1430042A2 Bicyclic heterocycles as rxr ligands
06/23/2004EP1429765A2 Inhibitors of histone deacetylase
06/23/2004CN1507446A Broadspectrum 2-amino-benzoxazole sulfonamide HIV protease inhibitors
06/23/2004CN1507445A Chromenylmethyl pyrimidinediamines as antibacterial agents
06/23/2004CN1507434A Novel 4-anilinoquinoline-3-carboxamides compound
06/23/2004CN1154646C Benzisozazoles and phenones as alpha antagonist
06/23/2004CN1154634C 2-phenyl-substituted heterocyclic 1,3-keonols as herbicides and pesticides
06/22/2004US6753430 Optically active quinoline carboxylic acid derivatives with 7-pyrrolidine substituents causing optical activity and a process for the preparation thereof
06/22/2004US6753429 1,4-disubstituted benzenes as insecticides
06/22/2004US6753342 2-(1h-indol-3-yl)-2-oxo-acetamides with antitumor activity
06/22/2004US6753331 Heterocyclic derivatives which inhibit factor Xa
06/17/2004WO2004050652A1 Novel azole derivatives
06/17/2004WO2004050629A2 The use of 4-phenyl substituted tetrahydroisoquinolines in the treatment of pain, migraine and urinary incontinence
06/17/2004WO2004050623A1 Methods for preparing phenylalkyne derivatives
06/17/2004WO2004050613A2 2-substituted-3-propenamide derivatives and methods of using the same
06/17/2004WO2004050035A2 Benzimidazoles and analogs thereof as antivirals
06/17/2004WO2004013282A3 Bis (amino acid) molecular scaffolds
06/17/2004US20040116706 Therapeutic ureas
06/17/2004US20040116469 Quinoline-4-carboxamide derivatives as NK-2 and NK-3 receptor antagonists
06/17/2004US20040116461 Immunomodulatory compounds
06/17/2004US20040116457 Agents for improving excretory potency of urinary bladder
06/17/2004US20040116456 Remedies for psychoneurosis
06/17/2004US20040116454 Pyrazole compounds useful as protein kinase inhibitors
06/17/2004US20040116417 Thiohydantoins and use thereof for treating diabetes
06/17/2004US20040116410 Diazepinones as antiviral agents
06/17/2004US20040116406 for the treatment of disorders of the central nervous system such as cerebral, central nervous or psychiatric symptoms, defunctionalization manifestations or disorders which occur as a result of unintentional or intentional intake of psychotropic
06/17/2004US20040116404 Sulphones which modulate the action of gamma secretase
06/17/2004US20040116328 Condensed imidazole derivatives
06/17/2004DE19742593B4 Neuer farbbildender Farbstoffvorläufer, Zusammensetzung, die denselben enthält und farbbildendes wärmeempfindliches Aufzeichnungsmaterial New color-forming dye precursor composition comprising the same and color-forming heat-sensitive recording material
06/17/2004DE10256405A1 New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
06/17/2004DE10247233A1 New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
06/17/2004CA2508311A1 The use of 4-phenyl substituted tetrahydroisoquinolines in the treatment of pain, migraine and urinary incontinence
06/17/2004CA2507875A1 Methods for preparing phenylalkyne derivatives
06/17/2004CA2507742A1 Novel azole derivatives
06/16/2004EP1428824A1 Heterocyclic substituted aminoazacycles useful as central nervous system agents
06/16/2004EP1427732A1 Spirocyclic-6,7-dihydro-5h-pyrazolo 1,2-a]pyrazol-1-ones which control inflammatory cytokines
06/16/2004EP1427728A1 6,7-DIHYDRO-5H-PYRAZOLO 1,2-A PYRAZOL-1-ONES WHICH CONTROL INFLAMMATORY cYTOKINES
06/16/2004EP1427727A1 Compounds which inhibit the release of inflammatory cytokines
06/16/2004EP1427722A2 Pyrrole-type compounds, compositions, and methods for treating cancer, treating viral diseases and causing immunosuppression
06/16/2004EP1427706A1 Substituted pyrazolo compounds for the treatment of inflammation
06/16/2004EP1427408A2 CYCLIC HYDROXAMIC ACIDS AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-$g(a) CONVERTING ENZYME (TACE)
06/16/2004EP1427407A2 Fatty amine drug conjugates
06/16/2004EP1427287A1 Pesticidal and parasitical di-and trifluorosubstituted alkene compounds
06/16/2004EP1341763B1 N-alkoxy-4,4-dioxy-polyalkyl-piperidine compounds, with glycidyl or alkylcarbonyl groups as functional initiators for controlled radical polymerization
06/16/2004EP1119570B1 Tricyclic delta3-piperidines as pharmaceuticals
06/16/2004CN1505626A Novel benzylpiperidine compound
06/16/2004CN1505613A Substituted indoles, pharmaceutical compositions containing such indoles and their use as ppar-gamma binding agents
06/16/2004CN1505607A Peptide-deformylase inhibitors
06/16/2004CN1505516A Utilization of galanthamine for the treatment of pathologies of the central nervous system owing to intoxications with psychotropic substances
06/16/2004CN1505514A Combinations of aldose reductase inhibitors and cyclooxygenase-2 inhibitors
06/16/2004CN1153771C Benzofuran-[3,4-f] quinoline derivatives, combination containing the same and application thereof
06/15/2004US6750357 Rhodamine-based fluorophores useful as labeling reagents
06/15/2004US6750346 Chromenes as terminal end groups
06/15/2004US6750233 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
06/15/2004US6750228 Uncontrolled breakdown of connective tissue by metalloproteases is a feature of many pathological conditions
06/15/2004US6750223 To inhibit the growth of a variety of tumor/cancer cells, especially leukemia, colon, melanoma, and breast cancer cells
06/15/2004US6750214 Quinoline and quinazoline compounds useful in therapy
06/15/2004CA2313302C New metalloprotease inhibitors, the process for preparing them and the pharmaceutical compounds containing them
06/15/2004CA2153195C New benzopyran derivatives; process for preparing the same and pharmaceutical compositions containing them
06/10/2004WO2004048378A1 Pyrazoloquinolines with immunomodulating activity
06/10/2004WO2004048332A1 Isoindoline derivative
06/10/2004WO2004047837A2 Beta-blockers having antioxidant and nitric oxide-donor activity
06/10/2004WO2004047755A2 Fused bicyclic nitrogen-containing heterocycles
06/10/2004WO2004032845A3 R-nsaid esters and their use
06/10/2004WO2004028445A3 Processes for preparing 1,3-dioxolane nucleosides
06/10/2004WO2003072027A3 Compositions and formulations of 9- nitrocamptothecin polymorphs and methods of use thereof
06/10/2004US20040110945 Very Late Antigen (Vla-4); such as 4-((4S)-fluoro-1-(2-phenylamino-6-benzoxazolylacetyl)-(2S)-pyrrolidinylmethoxy)benzoic acid; for treatment of inflammatory diseases, autoimmune diseases, metastasis, bronchial asthma, rhinostenosis, and diabetes