Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
02/2005
02/10/2005CA2534212A1 Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
02/10/2005CA2533820A1 Spatially-defined macrocycles incorporating peptide bond surrogates
02/10/2005CA2532382A1 N-sulfonylheterocyclopyrrolylalkylamine compounds as 5-hydroxytryptamine-6 ligands
02/10/2005CA2518950A1 Indazole derivatives
02/09/2005EP1505062A1 Heterocyclic derivatives and their use as antithrombotic agents
02/09/2005EP1504003A1 Nitrosated imidazopyridines
02/09/2005EP1503998A1 Heteroaryl substituted spirocyclic sufamides for inhibition of gamma secretase
02/09/2005EP1503994A1 Substituted (thioxo)carbonylamino phenyl uraciles
02/09/2005EP1503760A1 Camptothecin derivatives and polymeric conjugates thereof
02/09/2005EP1487795A4 Synthesis of enantiomerically pure amino-substituted fused bicyclic rings
02/09/2005EP1349839B1 Phenylethenyl or phenylethinyl derivatives as glutamate receptor antagonists
02/09/2005EP1204322B1 Fungicides
02/09/2005EP1044202B1 1'- 4- 1- (4-fluorophenyl)- 1h-indole-3-yl] -1-butyl]-spiro isobenzofuran- 1(3h),4'- piperidine] hydrohalogenides
02/09/2005EP0941093B1 Use of nk-1 receptor antagonists for treating major depressive disorders with anxiety
02/09/2005CN1578779A Small organic molecule regulators of cell proliferation
02/09/2005CN1578663A Inhibitors of histone deacetylase
02/09/2005CN1576277A New derivatives of benzo[a]pyrano[3, 2-h]acridin-7-one, a process for their preparation and pharmaceutical compounds containing them
02/09/2005CN1188403C Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
02/08/2005US6852860 Method for making piperidone ketals using polyphosphoric acid
02/08/2005US6852725 Imidazolyl derivatives
02/03/2005WO2005010063A1 Vinyl monomer, polymer derived from such monomer, and a light-emitting device using such polymer
02/03/2005WO2005010009A1 Thienopyridine and furopyridine kinase inhibitors
02/03/2005WO2005009969A1 Aminoquinoline derivatives and their use as adenosine a3 ligands
02/03/2005WO2005009398A2 Tetracyclic benzamide derivatives and methods of use thereof
02/03/2005WO2005009347A2 7-substituted camptothecin and camptothecin analogs and methods for preparing same
02/03/2005WO2003106450A8 Phenylaminopyrimidines and their use as rho-kinase inhibitors
02/03/2005WO2003063779A3 Selective analgesic agents
02/03/2005US20050027130 Rhodamine dye compounds for patterns with DNA sequences for kits
02/03/2005US20050027122 Compounds for modulators of chemokine activity
02/03/2005US20050026944 Thienopyridine and furopyridine kinase inhibitors
02/03/2005US20050026942 Chemokine receptor binding heterocyclic compounds
02/03/2005US20050026929 2-Phenyl-4-(piperidin-1-ylcarbonyl)-oxazole derivatives; capsase activators; cancer, autoimmune diseases, rheumatoid arthritis, inflammatory bowel disease, or psoriasis
02/03/2005US20050026915 As melanin concentrating hormone (MCH)receptor antagonists, for prevention or treatment of obesity or eating disorders; (2E)-3-(4-chlorophenyl)-N-[2-(dimethylamino)quinolin-6-yl]prop-2-enamide
02/03/2005CA2532982A1 Thienopyridine and furopyridine kinase inhibitors
02/03/2005CA2530046A1 7-substituted camptothecin and camptothecin analogs and methods for preparing same
02/03/2005CA2517260A1 Tetracyclic benzamide derivatives and methods of use thereof
02/02/2005EP1501841A2 Non nucleoside reverse transcriptase inhibitors
02/02/2005EP1501837A1 Cascade esters of camptothecins and methods of treating cancer using these compounds
02/02/2005EP1501836A1 Halo-alkyl esters of camptothecins and methods of treating cancer using these compounds
02/02/2005EP1501835A2 2-(quinolonyl)-fused heterocycles as androgen receptor modulators
02/02/2005EP1501831A1 Inhibitors of checkpoint kinases (wee1 and chk1)
02/02/2005EP1501803A2 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity
02/02/2005EP1501799A1 Compounds useful in preparing camptothecin derivatives
02/02/2005EP1137413B1 Non-peptide antagonists of glp-1 receptor and methods of use
02/02/2005CN1575292A Pharmaceutically acceptable salts of 20(s)-camptothecins
02/02/2005CN1575172A Substituted ideno[1, 2-c]isoquinoline derivatives and methods of use thereof
02/02/2005CN1572299A Agents for improving excretory potency of urinary bladder
02/02/2005CN1187355C Method for refining high-purity tetradoxin
02/01/2005US6849743 Synthesis of clasto-lactacystin β-lactone and analogs thereof
02/01/2005US6849629 Heteroaromatic substituted sulfonyl or sulfoxide or thio-pyridazinone derivatives, useful for treating diabetic complications and cardiovascular disorders
02/01/2005US6849627 Including interleukin-1 and Tumor Necrosis Factor; treating rheumatoid arthritis, osteoarthritis, inflammatory bowel disease, septic shock, cardiopulmonary dysfunction, acute respiratory disease, and cachexia
02/01/2005US6849622 May be useful for the prophylaxis and treatment of diabetes, particularly type 2 diabetes, and for prophylaxis and treatment of other diseases induced or exacerbated by impaired glucose tolerance
02/01/2005US6849620 N-(azabicyclo moieties)-substituted hetero-bicyclic aromatic compounds for the treatment of disease
01/2005
01/27/2005WO2005007652A2 Substituted quinolin-4-ylamine analogues
01/27/2005WO2005007629A1 Piperidine or 8-aza-bicyclo[3.2.1]oct-3-yl derivatives useful as modulators of chemokine receptor activity
01/27/2005WO2005007103A2 Use of parthenolide derivatives as antileukemic and cytotoxic agents
01/27/2005WO2005007099A2 Pkb inhibitors as anti-tumor agents
01/27/2005WO2005007084A2 Pancratistatin cyclic phosphate prodrugs an phenpanstatin cyclic phosphate prodrugs
01/27/2005WO2004110385A3 Modulators of the glucocorticoid receptor and method
01/27/2005US20050020644 Bicyclic fused pyridinyl amides and advantagesous compositons thereof for use as fungicides
01/27/2005US20050020619 Anticancer agents ; cardiovascular disorders; antiinflammatory agents;antiarthritic agents; Crohn's diseases; antiischemic agents
01/27/2005US20050020595 Compounds, methods and pharmaceutical compositions for inhibiting PARP
01/27/2005US20050020578 Oxidoreductase enzyme inhibitors such as (R)-1-[4-(2-methyl-4-phenyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-pyrimidin-2-yl-ethanol, used as antidiabetic agents
01/27/2005US20050020573 5HT2c receptor modulators
01/27/2005US20050020481 Ion channel modulating compounds and uses thereof
01/27/2005US20050019263 Conjugate for differentiating between healthy and unhealthy tissue
01/27/2005CA2532229A1 Use of parthenolide derivatives as antileukemic and cytotoxic agents
01/27/2005CA2531535A1 Substituted quinolin-4-ylamine analogues
01/26/2005EP1499619A1 Bicyclic heterocycles, medicaments containing these compounds, their use, and method for the production thereof
01/26/2005EP1499618A1 Furyl compounds
01/26/2005EP1499617A1 Camptothecin-taxoid conjugates as antimitotic and antitumor agents
01/26/2005EP1499616A1 Heterocyclic compounds
01/26/2005EP1499615A1 Thienyl compounds
01/26/2005EP1499609A2 Pesticidal heterocycles
01/26/2005EP1499305A2 Use of ep4 receptor ligands in the treatment of il-6 involved diseases
01/26/2005EP1427727B1 Compounds which inhibit the release of inflammatory cytokines
01/26/2005EP0975637B1 Amidino-camptothecin derivatives
01/26/2005EP0958514B1 Novel photochromic heterocyclic fused indenonaphthopyrans
01/26/2005CN1571789A Himbacine analogues as thrombin receptor antagonists
01/26/2005CN1569857A Method and technology for resin absorption purification of lycoris radiate galanthamine hydrobromide from alkaloid
01/26/2005CN1569856A Method and technology for acid water extracting of lycoris radiate galanthamine hydrobromide from alkaloid
01/26/2005CN1186324C Condensed heteroaryl derivatives
01/25/2005CA2309352C Heterocyclic-substituted tricyclics as thrombin receptor antagonists
01/25/2005CA2103383C Quinazoline derivatives
01/20/2005WO2005005600A2 Camptothecin analogs having an e-ring ketone
01/20/2005WO2005005431A2 7-polyaminoalkyl(oxy)iminomethylcamptothecins bearing protective groups
01/20/2005WO2005005430A2 Process for the preparation of furopyrroles
01/20/2005WO2005005397A1 5-substituted quinazolinone derivatives
01/20/2005WO2005004801A2 Indole, azaindole and related heterocyclic n-substituted piperazine derivatives
01/20/2005WO2004099124A3 Novel bioisosteres of actinonin
01/20/2005WO2004089926A8 Genipin derivatives and uses thereof
01/20/2005WO2004073601A3 Process for the preparation of hexacyclic camptothecin derivatives
01/20/2005WO2004069792A3 Quinoline-derived amide modulators of vanilloid vr1 receptor
01/20/2005WO2003076443A9 Spiro compounds with npy antagonistic activity
01/20/2005US20050014953 Method for the racemization of etodolic acid
01/20/2005US20050014802 Prevent reproduction of virus; antitumor agents
01/20/2005US20050014775 Anticancer agents
01/20/2005US20050014771 fused thienopyrimidine compounds useful as phosphatidylinositol 3-kinase inhibitors and carcinostatic agents
01/20/2005US20050014769 Anticancer agents; controlling apoptosis
01/20/2005DE10329860A1 Sulfonamidderivate polycyclischer Farbstoffe für analytische Anwendungen Sulfonamide derivatives of polycyclic dyes for analytical applications