Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
07/2005
07/07/2005US20050148578 1H-8-oxa-1-aza-dibenzo[e,h]azulene; dual inhibitors of tumour necrosis factor(alpha) and interleukin 1; antiinflammatory, analgesics
07/07/2005US20050148572 2-(2,4-difluorophenyl)-2-[(3R,6R)-3-(2,3-dihydro-1H-inden-2-yl)-6-isobutyl-2,5-dioxopiperazin-1-yl]-N,N-dimethylethanamide; to suppress uterine contractions; cyclization of leucine analogs
07/07/2005CA2550888A1 Vinylogous 4h-pyrones and their use in promoting plant growth
07/07/2005CA2550643A1 1,2,3,4-tetrahydroisoquinoline derivatives, preparations thereof and uses thereof
07/07/2005CA2549651A1 Benzenesulfonylamino-pyridin-2-yl derivatives and related compounds as inhibitors of 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-hsd-1) for the treatment of diabetes and obesity
07/07/2005CA2548518A1 Biaryl sulfonamides as mmp inhibitors
07/07/2005CA2548494A1 Novel tricyclic spiroderivatives as modulators of chemokine receptor activity
07/06/2005EP1550655A1 Bicyclic intermediates
07/06/2005EP1549641A1 Antimicrobial 3.1.0 bicyclic oxazolidinone derivatives
07/06/2005EP1549156A1 Denatured carob flour (dcf) with a low content of soluble tannins and sugars, meant for human consumption and process to obtain it
07/06/2005EP1280809B1 Antitumoral ecteinascidin derivatives
07/06/2005CN1634921A Crystalline anti-cholinergic tiotropium crystal
07/06/2005CN1634894A Spiro[benzocyclo-4'-piperidine-2'-one] template compound and method for preparing same
07/06/2005CN1209107C Carbazolyl alkaloid anticarcinogen and its prepn
07/05/2005CA2220509C Fused polycyclic heterocycle derivatives
07/05/2005CA2183972C Oxazolidinone derivatives and pharmaceutical compositions containing them
06/2005
06/30/2005WO2005058912A1 Process for preparing amide acetals
06/30/2005WO2005058910A1 The method of manufacturing of 7-ethyl-10-hydroxycamptothecin
06/30/2005WO2005058893A1 Tricyclic benzimidazoles
06/30/2005WO2005058843A1 Substituted 6-cyclohexylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitors
06/30/2005WO2005058325A1 Tricyclic imidazopyridines for use as gastric secretion inhibitors
06/30/2005WO2005058231A2 Rifamycin analogs and uses thereof
06/30/2005WO2005033113A3 Indole derivatives
06/30/2005WO2004089926A3 Genipin derivatives and uses thereof
06/30/2005US20050143443 4-substituted pyrrole-2-carboxylic acidsand 5-substituted pyrazole-3-carboxylic acids/esters/salts; increase D-Serine level; reduce level of toxic products of D-Serine oxidation; activate N-methyl-D-aspartate NMDA-glutamate receptors; neuropathic agent, schizophrenia, Alzheimer's, anaxia
06/30/2005US20050143436 N-acylamino with fused nitrogen heterocyclic ring compound; capase enzyme inhibitors; antiinflammatory agents; oral bioavailability; autoimmune diseases, destructive bone disorders, proliferative disorders, infectious diseases, degenerative diseases, and necrotic diseases
06/30/2005US20050143422 N-({4'-[(1-benzofuran-2-ylcarbonyl)amino]-1,1'-biphenyl-4-yl}sulfonyl)glycine; metalloproteinase inhibitors; arthritis, macular degeneration, graft versus host disease, cancer, osteoarthritis
06/30/2005US20050143421 Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy
06/30/2005US20050143418 Pesticidal heterocycles
06/30/2005US20050143382 Heterocyclic compounds as pharmaceutically active compounds
06/30/2005US20050143373 Benzodioxole derivatives
06/30/2005US20050143372 Compounds, pharmaceutical compositions and methods of use therefor
06/30/2005US20050142601 Nucleic acids encoding an enediyne polyketide synthase complex
06/30/2005US20050142322 Optical recording media and dipyrrpomethene-metal chelate compounds
06/30/2005US20050139814 Benzofuran and benzothiophene derivatives useful in the treatmint of hyper-proliferative disorders
06/30/2005DE10354629A1 2-Ethyl-4,6-dimethyl-phenyl substituierte spirocyclische Tetramsäure-Derivate 2-ethyl-4,6-dimethyl-phenyl substituted spirocyclic tetramic acid derivatives
06/30/2005CA2549042A1 Tricyclic benzimidazoles
06/30/2005CA2549030A1 Tricyclic imidazopyridines for use as gastric secretion inhibitors
06/30/2005CA2549001A1 Rifamycin analogs and uses thereof
06/30/2005CA2548273A1 Substituted 6-cyclohexylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitors
06/30/2005CA2547519A1 Process for preparing amide acetals
06/29/2005EP1546391A2 Energy transfer dyes, terminators and use thereof
06/29/2005EP1546151A1 Antidepressant cycloalkylamine derivatives of heterocycle-fused benzodioxans
06/29/2005EP1546143A1 Heterocyclic substituted piperazines for the treatment of schizophrenia
06/29/2005EP1546137A1 Benzimidazol-1-yl-thiophene compounds for the treatment of cancer
06/29/2005EP1546125A2 Fluorescent labeling reagents with multiple donors and acceptors
06/29/2005EP1545545A2 COMPOUNDS WITH THE BICYCLO 4.2.1 NONANE SYSTEM FOR THE TREATMENT OF i FLAVIVIRIDAE /i INFECTIONS
06/29/2005EP1545502A2 Keto cannabinoids with therapeutic indications
06/29/2005EP1545211A1 Nodulisporic acid derivative spot-on formulations for combating parasites
06/29/2005CN1633434A Imidazo[1, 2-a]pyridine derivative
06/29/2005CN1633413A 20-hydroxyeicosatetraenoic acid production inhibitors
06/29/2005CN1633297A Acylated piperidine derivatives as melanocortin-4 receptor agonists
06/29/2005CN1631879A Substituted phenyl keto enols as pesticides and herbicides
06/29/2005CN1631878A C2 phenyl-substituted cyclic keto-enols used as pesticides and herbicides
06/28/2005US6912470 Nucleotide sequences coding enzymatic polypeptide for use in the production of anticarcinogenic and infection agents
06/28/2005US6911543 Azabicyclic-substituted fused-heteroaryl compounds for the treatment of disease
06/28/2005US6911445 For reatment of depression, childhood depression, dysthymia, anxiety, panic disorder, post-traumatic stress disorder, premenstrual dysphoric disorder, attention deficit disorder, obsessive-compulsive disorder, cocaine and alcohol addiction
06/23/2005WO2005057207A1 Trityl derivatives for enhancing mass spectrometry
06/23/2005WO2005056554A2 Azepinoindole derivatives as pharmaceutical agents
06/23/2005WO2005056524A2 Therapeutic agents useful for treating pain
06/23/2005WO2005033930A3 Process for upgrading naphtha
06/23/2005WO2005030333A3 Novel derivatives of 4a,5,9,10,11,12-hexahydrobenzofuro[3a,3,2] [2]- benzazepine, method for the production thereof and use thereof in the production of medicaments
06/23/2005WO2004089307A8 Acylated spiropiperidine derivatives as melanocortin-4 receptor agonists
06/23/2005US20050137221 Keratinocyte-proliferative diseases; inhibitor of solubilization of Epidermal Growth Factor; 3,4,5-trihydroxy-1-(4'-methoxybenzenesulfonyl)-piperidine-2-carboxylic acid hydroxamide; 7-acetoxy-5-(4'-methoxybenzenesulfonyl)-2,2-dimethyl-h exahydro-[1,3]dioxolo[4,5-c]pyridine-6-carboxy ester intermediate
06/23/2005US20050137219 alzheimer's disease; schizophrenia
06/23/2005US20050137215 Antiarthritic and antiinflammatory agents; analgesics; the proline derivatives do not displace gabapentin from alpha-2-delta receptors
06/23/2005US20050137201 Compositions useful as inhibitors of protein kinases
06/23/2005US20050137191 Nitrate esters and their use for mitigating cellular damage
06/23/2005US20050137189 For therapy of Gram-positive bacterial infection
06/23/2005US20050137187 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor
06/22/2005EP1543011A2 Thienopyrrolyl and furanopyrrolyl compounds and their use as histamine h4 receptor ligands
06/22/2005EP1542674A1 Chondropsin-class antitumor v-atpase inhibitor compounds, compositions and methods of use thereof
06/22/2005EP1525265A4 Chiral indole intermediates and their fluorescent cyanine dyes containing functional groups
06/22/2005EP1007533B1 Bioconjugates and delivery of bioactive agents
06/22/2005CN1630653A Pyrazolyl-substituted heterocycles and their use as phytosanitary products
06/22/2005CN1630639A Novel pyridine- and quinoline-derivatives
06/22/2005CN1629145A Condensed heteroaryl derivatives
06/21/2005WO2005066180A1 Cysteine protease inhibitors
06/21/2005US6909001 Cyclization of salicaldehyde with 3-(2-furyl)-3-oxopropane-nitrile, to form 2-amino-4-(2-furyl)-5H-chromeno(2,3-b) pyridine-3-carbonitrile, used as mitogen activated protein kinase inhibitors
06/21/2005US6908927 Reduction physical cigarette smoking
06/21/2005US6908922 Linear cyclic ureas
06/21/2005CA2108068C Carbamates of rapamycin
06/16/2005WO2005054251A1 New cartharidic amine, demethyl cartharidic amine derivatives and their medicinal use
06/16/2005WO2005054249A1 Novel compounds
06/16/2005WO2005054234A2 Substituted piperidino phenyloxazolidinones having antimicriobial activity with improved in vivo efficacy
06/16/2005WO2005054205A1 Protein modifier production inhibitor
06/16/2005WO2005054203A1 Quinoline derivatives substituted by aliphatic amino groups, the preparation and the pharmaceutical use thereof
06/16/2005WO2005054183A2 Quinolinone based protein kinase inhibitors
06/16/2005WO2005053692A1 Advanced quinolinone based protein kinase inhibitors
06/16/2005WO2005053688A1 Substituted furo[2,3-g] indazoles for the treatment of glaucoma
06/16/2005WO2005016255A3 Substituted tetrahydroquinolines, phenylacetic acids and benzoic acids as hepatocyte nuclear factor 4 (hnf-4 ) modulator compounds
06/16/2005WO2005005430A3 Process for the preparation of furopyrroles
06/16/2005WO1990000853A8 Method of treating neurological disorders
06/16/2005US20050131177 1-Alkoxy-polyalkyl-piperidine derivatives and their use as polymerization regulators
06/16/2005US20050131164 Dehydration mixture of oxyamides; reacting acid or ester with dialkanolamine
06/16/2005US20050131051 2-3-disubstituted quinuclidiness as modulators of monoamine transporters and theraperutic and diagnostic methods based thereon
06/16/2005US20050131043 Phenylethynyl and styryl derivatives of imidazole and fused ring heterocycles
06/16/2005US20050131007 Process for preparing new tiotropium salts, new tiotropium salts as such and pharmaceutical compositions thereof
06/16/2005US20050131003 Heterocyclic compounds
06/16/2005US20050130979 2,3-dihydroxy-6-nitro-7-sulfamoyl-benzo(F)quinoxaline (NBQX) or the quinoxalinedione is 9-methyl-amino-6-nitro-hexahydro-benzo(F) quinoxalinedione (PNQX) for treating demyelinating disorders