Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
08/2005
08/09/2005US6927292 Pharmaceutical intermediates; nitrogen and oxygen fused heterocycles
08/09/2005US6927234 possessing anti-cancer activity, anti-inflammatory activity, anti-obesity activity, and/or hair growth promotion activity
08/09/2005US6927232 Phenylethynyl and styryl derivatives of imidazole and fused ring heterocycles
08/09/2005US6927226 Antidepressant azaheterocyclymethyl derivatives of 7,8-dihydro-3H-6,9-dioxa-1,3-diazacyclopenta[a]naphthalene
08/09/2005US6927221 Tricyclic fused heterocyclic compound, process for preparing it and medicament comprising it
08/09/2005US6927214 Non-peptide GLP-1 agonists
08/09/2005CA2095659C Heteroatoms-containing tricyclic compounds
08/04/2005WO2005070941A1 Rifamycin imino derivatives effective against drug-resistant microbes
08/04/2005WO2005070940A2 Rifamycin derivatives effective against drug-resistant microbes
08/04/2005WO2005070936A1 20-esterized camptothecin derivatives, their preparation and the pharmaceutical compositions and the use
08/04/2005WO2005070925A1 Aryl substituted heterocycles, method for production and use thereof as medicaments
08/04/2005WO2005070920A1 Amino-benzazoles as p2y1 receptor inhibitors
08/04/2005WO2005069981A2 Method of preparation of benzofuran-2-carboxylic acid {(s)-3-methyl-1-[(4s, 7r)-7methyl-3-oxo-1-(pyridine-2-sulfonyl)-azepan-4-ylcarbamoyl]-butyl}-amide
08/04/2005WO2005069865A2 Pyrrolopyrimidine derivatives and analogs and their use in the treatment and prevention of diseases
08/04/2005WO2005049735A3 A process for aqueous milling of quinacridone pigments
08/04/2005US20050171152 N-( alpha -ethylbenzyl)-3-hydroxy-2-phenylquinoline-4-carboxamide; neurokinin NK-3 receptor antagonists; chemical intermediates; efficient process with increased yields; coupling an ortho-hydroxy acid with an amine; easy conversion side-product to desired; CNC disorders; anxiolitic and antidepressant
08/04/2005US20050171140 Prevent cholesterol biosynthesis; moderating blood serum lipid ; antidiabetic agents; obesity; hypotensive agents; osteoporosis; Alzheimer's disease; cardiovascular disorders; hormone replacement therapy
08/04/2005US20050171135 1'-[4-[1-(4-fluorophenyl)-1H-indole-3-Y1]-spiro[isobenzofuran-1(3H), 4'-piperidine]hydrohalogenides
08/04/2005US20050171114 Antitumor agents; superior cytotoxic activity; bioavailability; 1,2-dihydroxy-6-methoxy-3,3,14-trimethyl-1,2,3,14-tetrahydro-7H-benzo[b]-chromeno[6,5-g][1,8]naphthyridin-7-one; adenocarcinomas and carcinomas, sarcomas, gliomas and leukaemias; Derivatives of acronycine
08/04/2005US20050171106 5'-((benzo)thiophen-1 or 2-yl)spiro[1-azabicyclo[2.2.2]octane-3,2'(3'H)-furo[2,3-b]pyridine] compounds, optionally tritium labeled; binding ligands for nicotinic acetylcholine receptors
08/04/2005US20050171096 Hydantoins and related heterocycles as inhibitors of matrix metalloproteinases and/or TNF-alpha converting enzyme (TACE)
08/04/2005US20050170475 Using actinomycetes to ferment maytansines
08/04/2005US20050170411 Genes and proteins involved in the biosynthesis of enediyne ring structures
08/04/2005US20050170363 For conjugation with biomolecules, drugs, and toxins
08/04/2005CA2554138A1 Aryl substituted heterocycles, method for production and use thereof as medicaments
08/03/2005EP1558618A1 5-(1 ,1 -CYCLOALKYL/ALKENYL)METHYLIDENE 1,2-DIHYDRO- 5H /-CHROMENO[3,4-f ] QUINOLINES AS SELECTIVE PROGESTERONE RECEPTOR MODULATOR COMPOUNDS
08/03/2005EP1558605A2 Process for making spirolactone compounds
08/03/2005EP1558585A1 Neurologically-active compounds
08/03/2005EP1558579A1 N-alkyl-4-methyleneamino-3-hydroxy-2-pyridones as antimicrobials
08/03/2005EP1558576A2 Piperidinyl cyclopentyl aryl benzylamide modulators of chemokine receptor activity
08/03/2005EP1558341A2 Transcription factor modulating compounds and methods of use thereof
08/03/2005EP1558252A2 Substituted furo 2,3-b] pyridine derivatives
08/03/2005EP1558243A2 Tetrahydropyranyl cyclopentyl benzylamide modulators of chemokine receptor activity
08/03/2005EP1558083A2 Compounds, compositions, and methods
08/03/2005EP1362051B1 Method for purifying 20(s)-camptothecin
08/03/2005EP1123293B1 Core-extended perylene bisimides
08/03/2005CN1649885A Cellular accumulation of phosphonate analogs of HIV protease inhibitor compounds and the compounds as such
08/03/2005CN1649873A Camptothecin-taxoid conjugates as antimitotic and antitumor agents
08/03/2005CN1648128A Aromatic heterocyclic carboxylic derivative, preparing method and use on medicine
08/03/2005CN1647816A Process for preparing decumbent corydalis tuber total alkaloid and its preparation and quality detecting method
08/03/2005CN1213050C Oxadicyclo [2.2.1] heptane derivative, its preparing method and use as pesticide
08/03/2005CN1213049C Alkylated imidazopyridine derivatives and medicine containing them and use
08/02/2005US6924292 Nitrogen compounds such as 2-(methylsulfinyl) N [3-(3,4,8,9-tetrahydro-6-methoxy-3,3,8,8-tetramethylfuro[2,3-h]isoquinolin-1-yl)phenyl]acetamide, used as phosphodiesterase inhibitors; antidiabetics; antiinflammatory agents
08/02/2005US6924291 Process for making spiro isobenzofuranone compounds
08/02/2005US6924285 Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them
08/02/2005US6924280 Dipeptide derivatives
08/02/2005CA2362339C Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives
08/02/2005CA2362337C Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives
08/02/2005CA2190087C Nitro compounds and their compositions having anti-inflammatory, analgesic and anti-thrombotic activities
07/2005
07/28/2005WO2005068473A1 Bicyclic pyrazolo-fused compounds as protein kinase modulators
07/28/2005WO2005068466A1 Compounds useful in therapy
07/28/2005WO2005068457A1 Cataltytic asymmetric hetero diels-alder reaction of a heteroaromatic c-nitroso dienophile: a novel method for synthesis of chiral non-racemic amino alcohols
07/28/2005WO2005068436A1 6-amino-5-cyano-pyrimidine-4-ones used for improving perception, power of concentration, learning efficiency, and/or memory power
07/28/2005WO2005067900A2 Azabenzofuran substituted thioureas as inhibitors of viral replication
07/28/2005WO2005067546A2 Pyrrolopyrimidine derivatives and analogs and their use in the treatment and prevention of diseases
07/28/2005WO2005033073A3 Spirocyclic heterocyclic derivatives and methods of their use
07/28/2005WO2005019224A3 Novel antiinfective compounds
07/28/2005US20050165114 Antiinflammatory agent, immunosuppressant, anticancer agents, antiarthritic agents; AP-1 activation inhibitor, NF-kappa B activation inhibitor
07/28/2005US20050165058 Oxybenzamide derivatives useful for inhibiting factor Xa or Vlla
07/28/2005US20050165045 Compounds and methods
07/28/2005US20050165042 Fused tricyclic heterocycles useful for treating hyper-proliferative disoroders
07/28/2005US20050165029 Pyrrolopyrimidine derivatives and analogs and their use in the treatment and prevention of diseases
07/28/2005US20050165022 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses
07/28/2005US20050165007 Benzimidazoles and analogs thereof as antivirals
07/28/2005US20050164885 Alkyl dihalogenated phenyl-substituted ketoenols useful as pesticides and herbicides
07/28/2005US20050164883 agronomically tolerable salts, isomers and enantiomers of those compounds, are suitable for use as herbicides
07/28/2005DE10360793A1 Spirocyclische Cyclohexan-Derivate Spirocyclic cyclohexane derivatives
07/28/2005DE10360792A1 Spirocyclische Cyclohexan-Derivate Spirocyclic cyclohexane derivatives
07/28/2005CA2554382A1 Compounds useful in therapy
07/28/2005CA2553200A1 6-amino-5-cyano-pyrimidine-4-ones used for improving perception, power of concentration, learning efficiency, and/or memory power
07/28/2005CA2552002A1 Azabenzofuran substituted thioureas as inhibitors of viral replication
07/28/2005CA2547703A1 Bicyclic pyrazolo-fused compounds as protein kinase modulators
07/27/2005EP1557424A1 Bi-cyclic nucleoside, nucleotide and oligonucleoide analogues
07/27/2005EP1557410A2 Bacterial gyrase inhibitors and uses thereof
07/27/2005EP1557409A1 5HT2C receptor modulators
07/27/2005EP1556362A2 Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
07/27/2005EP1556053A1 Antiinflammation agents
07/27/2005EP1556047A2 Pgd2 receptor antagonists for the treatment of inflammatory diseases
07/27/2005EP1379523B1 1,2,3,4-tetrahydroisoquinolines derivatives as urotensin ii receptor antagonists
07/27/2005EP1343766B1 Cyclization process step in the making of quinolones and naphthyridines
07/27/2005EP1313736B1 Condensed pyrazindione derivatives as inhibitors of pde5
07/27/2005EP1287004B1 Synthetic process for the manufacture of an ecteinascidin compound
07/27/2005CN1646536A Methods for producing norgalanthamine, as well as isomers, salts and hydrates thereof
07/27/2005CN1646530A Nitrosated imidazopyridines
07/27/2005CN1646528A Polycyclic compounds as potent alpha2-adrenoceptor antagonists
07/27/2005CN1646493A 5HT2C receptor modulators
07/27/2005CN1646491A Compounds used to prepare camptothecin derivatives
07/26/2005US6921772 Methods and compositions for the treatment of chronic lymphocytic leukemia
07/26/2005CA2324848C Method of making camptothecin and camptothecin analogs
07/26/2005CA2258548C Phenylamino-substituted tricyclic derivatives for treatment of hyperproliferative diseases
07/21/2005WO2005066183A1 Spirocyclic cyclohexane derivatives with affinity for the orl1-receptor
07/21/2005WO2005066181A1 Process for the preparation of 1,3-dioxolo [4,5-c] piperidin-7-ols and related compounds
07/21/2005WO2005066135A2 Pyrrole and pyrazole daao inhibitors
07/21/2005WO2005066126A1 Cb1 modulator compounds
07/21/2005WO2005065779A1 Calcitonin gene related peptide receptor antagonists
07/21/2005WO2005065050A2 Bicyclic compound
07/21/2005WO2005020911A3 Benzo[1, 3]dioxole compounds, pharmaceutical compositions thereof, and processes of making and using the same
07/21/2005WO2004055004A8 Carboxylic acid, phosphate or phosphonate substituted quinazolin-4-ylamine analogues as capsaicin receptor modulators
07/21/2005US20050159461 Treating cancer with a synergistic mixtures; anticarcinogenic agents; epothilone has secondary amide instead of an ester
07/21/2005US20050159438 Spirocyclic heterocyclic derivatives and methods of their use