Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726) |
---|
08/09/2005 | US6927292 Pharmaceutical intermediates; nitrogen and oxygen fused heterocycles |
08/09/2005 | US6927234 possessing anti-cancer activity, anti-inflammatory activity, anti-obesity activity, and/or hair growth promotion activity |
08/09/2005 | US6927232 Phenylethynyl and styryl derivatives of imidazole and fused ring heterocycles |
08/09/2005 | US6927226 Antidepressant azaheterocyclymethyl derivatives of 7,8-dihydro-3H-6,9-dioxa-1,3-diazacyclopenta[a]naphthalene |
08/09/2005 | US6927221 Tricyclic fused heterocyclic compound, process for preparing it and medicament comprising it |
08/09/2005 | US6927214 Non-peptide GLP-1 agonists |
08/09/2005 | CA2095659C Heteroatoms-containing tricyclic compounds |
08/04/2005 | WO2005070941A1 Rifamycin imino derivatives effective against drug-resistant microbes |
08/04/2005 | WO2005070940A2 Rifamycin derivatives effective against drug-resistant microbes |
08/04/2005 | WO2005070936A1 20-esterized camptothecin derivatives, their preparation and the pharmaceutical compositions and the use |
08/04/2005 | WO2005070925A1 Aryl substituted heterocycles, method for production and use thereof as medicaments |
08/04/2005 | WO2005070920A1 Amino-benzazoles as p2y1 receptor inhibitors |
08/04/2005 | WO2005069981A2 Method of preparation of benzofuran-2-carboxylic acid {(s)-3-methyl-1-[(4s, 7r)-7methyl-3-oxo-1-(pyridine-2-sulfonyl)-azepan-4-ylcarbamoyl]-butyl}-amide |
08/04/2005 | WO2005069865A2 Pyrrolopyrimidine derivatives and analogs and their use in the treatment and prevention of diseases |
08/04/2005 | WO2005049735A3 A process for aqueous milling of quinacridone pigments |
08/04/2005 | US20050171152 N-( alpha -ethylbenzyl)-3-hydroxy-2-phenylquinoline-4-carboxamide; neurokinin NK-3 receptor antagonists; chemical intermediates; efficient process with increased yields; coupling an ortho-hydroxy acid with an amine; easy conversion side-product to desired; CNC disorders; anxiolitic and antidepressant |
08/04/2005 | US20050171140 Prevent cholesterol biosynthesis; moderating blood serum lipid ; antidiabetic agents; obesity; hypotensive agents; osteoporosis; Alzheimer's disease; cardiovascular disorders; hormone replacement therapy |
08/04/2005 | US20050171135 1'-[4-[1-(4-fluorophenyl)-1H-indole-3-Y1]-spiro[isobenzofuran-1(3H), 4'-piperidine]hydrohalogenides |
08/04/2005 | US20050171114 Antitumor agents; superior cytotoxic activity; bioavailability; 1,2-dihydroxy-6-methoxy-3,3,14-trimethyl-1,2,3,14-tetrahydro-7H-benzo[b]-chromeno[6,5-g][1,8]naphthyridin-7-one; adenocarcinomas and carcinomas, sarcomas, gliomas and leukaemias; Derivatives of acronycine |
08/04/2005 | US20050171106 5'-((benzo)thiophen-1 or 2-yl)spiro[1-azabicyclo[2.2.2]octane-3,2'(3'H)-furo[2,3-b]pyridine] compounds, optionally tritium labeled; binding ligands for nicotinic acetylcholine receptors |
08/04/2005 | US20050171096 Hydantoins and related heterocycles as inhibitors of matrix metalloproteinases and/or TNF-alpha converting enzyme (TACE) |
08/04/2005 | US20050170475 Using actinomycetes to ferment maytansines |
08/04/2005 | US20050170411 Genes and proteins involved in the biosynthesis of enediyne ring structures |
08/04/2005 | US20050170363 For conjugation with biomolecules, drugs, and toxins |
08/04/2005 | CA2554138A1 Aryl substituted heterocycles, method for production and use thereof as medicaments |
08/03/2005 | EP1558618A1 5-(1 ,1 -CYCLOALKYL/ALKENYL)METHYLIDENE 1,2-DIHYDRO- 5H /-CHROMENO[3,4-f ] QUINOLINES AS SELECTIVE PROGESTERONE RECEPTOR MODULATOR COMPOUNDS |
08/03/2005 | EP1558605A2 Process for making spirolactone compounds |
08/03/2005 | EP1558585A1 Neurologically-active compounds |
08/03/2005 | EP1558579A1 N-alkyl-4-methyleneamino-3-hydroxy-2-pyridones as antimicrobials |
08/03/2005 | EP1558576A2 Piperidinyl cyclopentyl aryl benzylamide modulators of chemokine receptor activity |
08/03/2005 | EP1558341A2 Transcription factor modulating compounds and methods of use thereof |
08/03/2005 | EP1558252A2 Substituted furo 2,3-b] pyridine derivatives |
08/03/2005 | EP1558243A2 Tetrahydropyranyl cyclopentyl benzylamide modulators of chemokine receptor activity |
08/03/2005 | EP1558083A2 Compounds, compositions, and methods |
08/03/2005 | EP1362051B1 Method for purifying 20(s)-camptothecin |
08/03/2005 | EP1123293B1 Core-extended perylene bisimides |
08/03/2005 | CN1649885A Cellular accumulation of phosphonate analogs of HIV protease inhibitor compounds and the compounds as such |
08/03/2005 | CN1649873A Camptothecin-taxoid conjugates as antimitotic and antitumor agents |
08/03/2005 | CN1648128A Aromatic heterocyclic carboxylic derivative, preparing method and use on medicine |
08/03/2005 | CN1647816A Process for preparing decumbent corydalis tuber total alkaloid and its preparation and quality detecting method |
08/03/2005 | CN1213050C Oxadicyclo [2.2.1] heptane derivative, its preparing method and use as pesticide |
08/03/2005 | CN1213049C Alkylated imidazopyridine derivatives and medicine containing them and use |
08/02/2005 | US6924292 Nitrogen compounds such as 2-(methylsulfinyl) N [3-(3,4,8,9-tetrahydro-6-methoxy-3,3,8,8-tetramethylfuro[2,3-h]isoquinolin-1-yl)phenyl]acetamide, used as phosphodiesterase inhibitors; antidiabetics; antiinflammatory agents |
08/02/2005 | US6924291 Process for making spiro isobenzofuranone compounds |
08/02/2005 | US6924285 Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them |
08/02/2005 | US6924280 Dipeptide derivatives |
08/02/2005 | CA2362339C Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives |
08/02/2005 | CA2362337C Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives |
08/02/2005 | CA2190087C Nitro compounds and their compositions having anti-inflammatory, analgesic and anti-thrombotic activities |
07/28/2005 | WO2005068473A1 Bicyclic pyrazolo-fused compounds as protein kinase modulators |
07/28/2005 | WO2005068466A1 Compounds useful in therapy |
07/28/2005 | WO2005068457A1 Cataltytic asymmetric hetero diels-alder reaction of a heteroaromatic c-nitroso dienophile: a novel method for synthesis of chiral non-racemic amino alcohols |
07/28/2005 | WO2005068436A1 6-amino-5-cyano-pyrimidine-4-ones used for improving perception, power of concentration, learning efficiency, and/or memory power |
07/28/2005 | WO2005067900A2 Azabenzofuran substituted thioureas as inhibitors of viral replication |
07/28/2005 | WO2005067546A2 Pyrrolopyrimidine derivatives and analogs and their use in the treatment and prevention of diseases |
07/28/2005 | WO2005033073A3 Spirocyclic heterocyclic derivatives and methods of their use |
07/28/2005 | WO2005019224A3 Novel antiinfective compounds |
07/28/2005 | US20050165114 Antiinflammatory agent, immunosuppressant, anticancer agents, antiarthritic agents; AP-1 activation inhibitor, NF-kappa B activation inhibitor |
07/28/2005 | US20050165058 Oxybenzamide derivatives useful for inhibiting factor Xa or Vlla |
07/28/2005 | US20050165045 Compounds and methods |
07/28/2005 | US20050165042 Fused tricyclic heterocycles useful for treating hyper-proliferative disoroders |
07/28/2005 | US20050165029 Pyrrolopyrimidine derivatives and analogs and their use in the treatment and prevention of diseases |
07/28/2005 | US20050165022 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses |
07/28/2005 | US20050165007 Benzimidazoles and analogs thereof as antivirals |
07/28/2005 | US20050164885 Alkyl dihalogenated phenyl-substituted ketoenols useful as pesticides and herbicides |
07/28/2005 | US20050164883 agronomically tolerable salts, isomers and enantiomers of those compounds, are suitable for use as herbicides |
07/28/2005 | DE10360793A1 Spirocyclische Cyclohexan-Derivate Spirocyclic cyclohexane derivatives |
07/28/2005 | DE10360792A1 Spirocyclische Cyclohexan-Derivate Spirocyclic cyclohexane derivatives |
07/28/2005 | CA2554382A1 Compounds useful in therapy |
07/28/2005 | CA2553200A1 6-amino-5-cyano-pyrimidine-4-ones used for improving perception, power of concentration, learning efficiency, and/or memory power |
07/28/2005 | CA2552002A1 Azabenzofuran substituted thioureas as inhibitors of viral replication |
07/28/2005 | CA2547703A1 Bicyclic pyrazolo-fused compounds as protein kinase modulators |
07/27/2005 | EP1557424A1 Bi-cyclic nucleoside, nucleotide and oligonucleoide analogues |
07/27/2005 | EP1557410A2 Bacterial gyrase inhibitors and uses thereof |
07/27/2005 | EP1557409A1 5HT2C receptor modulators |
07/27/2005 | EP1556362A2 Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes |
07/27/2005 | EP1556053A1 Antiinflammation agents |
07/27/2005 | EP1556047A2 Pgd2 receptor antagonists for the treatment of inflammatory diseases |
07/27/2005 | EP1379523B1 1,2,3,4-tetrahydroisoquinolines derivatives as urotensin ii receptor antagonists |
07/27/2005 | EP1343766B1 Cyclization process step in the making of quinolones and naphthyridines |
07/27/2005 | EP1313736B1 Condensed pyrazindione derivatives as inhibitors of pde5 |
07/27/2005 | EP1287004B1 Synthetic process for the manufacture of an ecteinascidin compound |
07/27/2005 | CN1646536A Methods for producing norgalanthamine, as well as isomers, salts and hydrates thereof |
07/27/2005 | CN1646530A Nitrosated imidazopyridines |
07/27/2005 | CN1646528A Polycyclic compounds as potent alpha2-adrenoceptor antagonists |
07/27/2005 | CN1646493A 5HT2C receptor modulators |
07/27/2005 | CN1646491A Compounds used to prepare camptothecin derivatives |
07/26/2005 | US6921772 Methods and compositions for the treatment of chronic lymphocytic leukemia |
07/26/2005 | CA2324848C Method of making camptothecin and camptothecin analogs |
07/26/2005 | CA2258548C Phenylamino-substituted tricyclic derivatives for treatment of hyperproliferative diseases |
07/21/2005 | WO2005066183A1 Spirocyclic cyclohexane derivatives with affinity for the orl1-receptor |
07/21/2005 | WO2005066181A1 Process for the preparation of 1,3-dioxolo [4,5-c] piperidin-7-ols and related compounds |
07/21/2005 | WO2005066135A2 Pyrrole and pyrazole daao inhibitors |
07/21/2005 | WO2005066126A1 Cb1 modulator compounds |
07/21/2005 | WO2005065779A1 Calcitonin gene related peptide receptor antagonists |
07/21/2005 | WO2005065050A2 Bicyclic compound |
07/21/2005 | WO2005020911A3 Benzo[1, 3]dioxole compounds, pharmaceutical compositions thereof, and processes of making and using the same |
07/21/2005 | WO2004055004A8 Carboxylic acid, phosphate or phosphonate substituted quinazolin-4-ylamine analogues as capsaicin receptor modulators |
07/21/2005 | US20050159461 Treating cancer with a synergistic mixtures; anticarcinogenic agents; epothilone has secondary amide instead of an ester |
07/21/2005 | US20050159438 Spirocyclic heterocyclic derivatives and methods of their use |