Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
02/2006
02/23/2006WO2006019673A2 Jiadifenin analogs and uses thereof
02/23/2006WO2006018815A1 Piperazine derivatives as adrenergic receptor antagonists
02/23/2006WO2006018284A1 Compounds and compositions useful as cathepsin s inhibitors
02/23/2006WO2005003086A3 Sulfonic acid derivatives of polycyclic dyes used for analytical applications
02/23/2006US20060041136 alpha-(2-chlorophenyl)-6,7dihydrothieno[3,2-c]pyridine-5(4H)-acetic acid methyl ester (clopidogrel hydrogen sulphate); separating crystalline form out of a solution of clopidogrel in the form of the free base in a 2-propanol or n-butyl acetate solvent by adding sulphuric acid
02/23/2006US20060041129 Enantiomers of selected fused heterocyclics and uses thereof
02/23/2006US20060041128 Selected fused heterocyclics and uses thereof
02/23/2006US20060041123 Antibacterial agents
02/23/2006US20060040964 Eating disorders; psychological disorders; antidiabetic agents; cardiovascular disorders
02/23/2006US20060040961 N-isopropyl-5-phenyl-6-(4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)furo[2,3-d]pyrimidin-4-amine; inflammation, inhibition of T cell activation, proliferation, arthritis, organ transplant, ischemic or reperfusion injury, myocardial infarction, stroke, multiple sclerosis, inflammatory bowel disease, Crohn's
02/23/2006US20060040960 (3-amino-5,6,7,8-tetrahydrofuro[2,3-b]quinolin-2-yl)-(2,5-dimethoxyphenyl)methanone; antiproliferative agent; solid tumors: breast, respiratory tract, brain, reproductive organs, digestive tract, liver, skin, head and neck, thyroid, and their metastases; lymphomas, sarcomas, and leukemias
02/23/2006US20060040949 Treating antibiotic resistant bacterial infections; compounds based on quinoline rings; (3S)-2-(3-{[(Benzo[1,2,5]thiadiazol-5-ylmethyl)-amino]-methyl}-piperidin-1-yl)-(1RS)-(6-methoxy-quinolin-4-yl)-ethanol for example
02/23/2006US20060040948 Cognitive or neurodegenerative disease; Alzheimer's disease; HMG-CoA reductase inhibitors, gamma-secretase inhibitors, non-steroidal anti-inflammatory agents, N-methyl-D-aspartate receptor antagonists, cholinesterase inhibitors and anti-amyloid antibodies
02/23/2006US20060040930 Novel substituted [1,4] benzodioxino[2,3-e] isoindole derivatives, method for preparing and pharmaceutical compositions containing same
02/23/2006US20060040925 Aminocyclohexene quinolines and their azaisosteric analogues with antibacterial activity
02/23/2006US20060040918 Benzo d!azepine derivatives for the treatment of neurological disorders
02/23/2006US20060040900 R(-)-10-methoxy-11-O-acetyl-N-n-propyl-noraporphine; Parkinson's disease, sexual dysfunction, and depressive disorders
02/23/2006DE102004039382A1 Spirocyclische Cyclohexan-Derivate Spirocyclic cyclohexane derivatives
02/23/2006CA2577060A1 Substituted benzofused heterocycles
02/23/2006CA2576421A1 Inhibitors of hcv replication
02/23/2006CA2575826A1 Compounds and compositions useful as cathepsin s inhibitors
02/22/2006EP1627069A2 Methods for the isolation and purification of ansamitocins
02/22/2006EP1626970A1 Azabicycloalkane compounds as muscarinic receptor antagonists
02/22/2006EP1626967A1 Substituted pyrazoles
02/22/2006CN1738824A CCR1 antagonists for the treatment of I.A. demyelinating inflammatory disease
02/22/2006CN1738814A Indolyl pyrazinone derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis
02/22/2006CN1738799A Methods for preparing phenylalkyne derivatives
02/22/2006CN1243003C Aspertoxin P as compound with antineoplastic activity
02/22/2006CN1242995C Novel compounds, their use and preparation
02/21/2006US7001911 Fused cyclic modulators of nuclear hormone receptor function
02/21/2006US7001906 Pyrrolo (2,3-B) pyridine derivatives containing Pyran ring, useful as anticancer compounds
02/16/2006WO2006016203A1 An improved process for the preparation of irinotecan hydrochloride trihydrate
02/16/2006WO2005103057A8 6,7-dihydroxy-8-phenyl-3,6,7,8-tetrahydro-chromeno[7, 8-d]imidazole derivatives and their use as gastric acid secretion inhibitors
02/16/2006WO2005097107A8 Diphenyl - indol-2-on compounds and their use in the treatment of cancer
02/16/2006WO2004015119A3 Methods for the isolation and purification of ansamitocins
02/16/2006US20060036094 Method for producing zoanthamine alkaloid and intermediate used in same
02/16/2006US20060036091 synthetic metabolites of CCI-779; for detecting CCI-779 metabolites in samples; generating CCI-779 reduction and hydroxylation derivatives using a CYP3A4 isozyme system
02/16/2006US20060035945 Prevent reproduction, infection of virus; antitumor agents
02/16/2006US20060035935 Acylated piperidine derivatives as melanocortin-4 receptor agonists
02/16/2006US20060035925 Substituted 4h-chromenes and analogs as activators of caspases and inducers of apoptosis and the use thereof
02/16/2006US20060035919 4-[4-(4-Amino-phenyl)-3-oxo-3,5-dihydro-pyrazolo[4,3-c]quinolin-2-yl]-benzoic acid methyl ester; rheumatoid arthritis, multiple sclerosis, diabetes, asthma, transplantation, systemic lupus erythematosis and psoriasis; CD80 antagonists capable of inhibiting the interactions between CD80 and CD28
02/16/2006US20060035892 Nitrosated imidazopyridines
02/16/2006US20060035884 N-cyclic sulfonamido inhibitors of gamma secretase
02/16/2006US20060035883 Novel serotonin receptor ligands and their uses thereof
02/15/2006EP1626041A2 New materials useful as electolytic solutes
02/15/2006EP1624874A2 3-amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
02/15/2006CN1735619A Spirocyclic cyclohexane compounds
02/15/2006CN1735618A New tricyclic derivatives as LTD4 antagonists
02/15/2006CN1735617A Quinazoline derivatives as SRC tyrosine kinase inhibitors
02/15/2006CN1733725A Process for preparing 2-iminopyrrolidine derivatives
02/15/2006CN1733722A Bis-heterocyclic compounds with antitumour and chemosensitising activity
02/15/2006CN1241927C Efficient method for refining tetrodotoxin by liquid-phase method
02/15/2006CN1241926C Novel intermediate for preparing camptothecin derivative (CPT-11) and correlated compound and method thereof
02/15/2006CN1241925C New [3,4-a: 3.4-c] carbazole compound, its preparation method and drug composition containing them
02/15/2006CN1241924C Method for preparing enkephalinase and angiotensin-converting enzyme inhibitor intermediate and its intermediate
02/15/2006CN1241923C Method for extracting total alkaloid of corydalis rhizome and its new usage
02/14/2006US6998485 3a,8a-Bis-azidomethyl-3a,4,8a,9-tetrahydro-3H,8H-bis[1,2,3]triazolo[1,5-a;1'',5''-d]pyrazine; provides low molecular weight energetic compounds with multiple energetic groups
02/14/2006US6998406 Fluorenecarboxylic acid esters, process for the manufacture thereof, and use thereof as medicaments
02/14/2006US6998256 Methods of obtaining epothilone D using crystallization and /or by the culture of cells in the presence of methyl oleate
02/14/2006CA2209825C Heterocyclic-fused pyridines
02/14/2006CA2135926C Substituted hexahydrobenzo[a]phenanthridines
02/09/2006WO2006014135A1 Novel piperidine derivatives as histamine h3 receptor ligands for treatment of depression
02/09/2006WO2006013546A2 Process for the preparation of pure galantamine
02/09/2006WO2005095409A3 Tetrahydroquinoline derivatives and a process for preparing the same
02/09/2006WO2003090691A3 Method and compositions for identifying anti-hiv therapeutic compounds
02/09/2006US20060030616 Anhydride modified cantharidin analogues useful in the treatment of cancer
02/09/2006US20060030598 Thiazolyl inhibitors of Tec family tyrosine kinases
02/09/2006US20060030580 Contacting phenolic piperidines with opioid receptors; analgesics, anticonvulsants, antitussive agents; diarrhea, drug addiction
02/09/2006US20060030571 Ecteinascidins
02/09/2006US20060030557 Substituted pyridines having antiangiogenic activity
02/09/2006US20060030543 Multicyclic sulfonamide compounds as inhibitors of histone deacetylase for the treatment of disease
02/09/2006CA2576109A1 Novel piperidine derivatives as histamine h3 receptor ligands for treatment of depression
02/09/2006CA2575100A1 Heterocyclic compounds
02/08/2006EP1623987A1 Fused pyrido[3',2':4,5]thieno[3,2-d]pyrimidines and pyrido[3',2':4,5]furo[3,2-d]pyrimidines
02/08/2006EP1623986A1 Use of vinca alkaloid and its salt
02/08/2006EP1622913A1 Heterocyclic compounds for use in the treatment of viral infections
02/08/2006EP1622905A1 Imidazopyridine intermediates
02/08/2006EP1622876A1 Cannabinoid receptor ligands and uses thereof
02/08/2006EP1622865A2 Novel bioisosteres of actinonin
02/08/2006EP1622569A2 Aza spiro alkane derivatives as inhibitors of metallproteases
02/08/2006EP1318978B1 N-acylsulfonamide apoptosis promoters
02/08/2006CN1732163A Novel compounds as anti-inflammatory, immunomodulatory and anti-proliferatory agents
02/08/2006CN1732147A Novel compounds as anti-inflammatory, immunomodulatory and anti-proliferatory agents
02/08/2006CN1240702C Process for extracting tetrodosin with high output rate
02/08/2006CN1240700C Aromatic heterocyclic carboxylic acid derivative, preparing method and application in medicine
02/08/2006CN1240679C 2- and 2,5-substituted phenylketoenols
02/07/2006US6995174 for inhibiting proteases
02/07/2006US6995167 Arylkylamine spirofuropyridines useful in therapy
02/07/2006US6995163 having an excellent corticotrophin-releasing-factor receptor antagonistic activity; for treating or preventing depression, nerve system disorders, schizophrenia, peptic ulcer, irritable bowel syndrome
02/07/2006CA2200433C Phenyloxazolidinone antimicrobials
02/07/2006CA2119783C Substituted phenserines and phenylcarbamates of (-)-eseroline, (-)-n1-noreseroline, and (-)-n1-benzylnoreseroline; as specific inhibitors of acetylcholinesterase
02/02/2006WO2006012473A1 Dynamic knowledge-based networking system and method
02/02/2006WO2006012310A2 Carbazole derivatives for treating polycystic kidney disease
02/02/2006WO2006012173A1 Amido compounds and their use as pharmaceuticals
02/02/2006WO2006011040A1 Quinazolin-4-yl- piperidine and cinnolin-4-yl- piperidine derivatives as pde10 inhibitors for the treatment of cns disorders
02/02/2006US20060025603 A reactant/solvent dimethyl formamide is made slightly basic, heating the solution to reduce the water content, then cooling, adding the hexanitrostilbene, heating to a predetermined temperature, cooling and filtering to accumulate 2,4,7,9-tetranitro-10H-benzo[4,5]furo[3,2]indole product
02/02/2006US20060025600 Process for preparing zolmitriptan compounds
02/02/2006US20060025588 Directly hydrogenating a heteroaryl alpha-hydroxyacetamide in the presence of a strong acid, a halide and a catalyst; for example, the heteroaryl acetamide is zolpidem and the heteroaryl alpha-hydroxyacetamide is alpha-hydroxyzolpidem
02/02/2006US20060025435 Novel 4-phenyl substituted tetrahydroisoquinolines and therapeutic use thereof
02/02/2006US20060025428 Bicyclic heteroaromatic compounds as kinase inhibitors